公开(公告)号：JP2012006936A

公开(公告)日：2012-01-12

申请号：JP2011160861

申请日：2011-07-22

Applicant: Basf Se ,  ビーエーエスエフ ソシエタス・ヨーロピアBasf Se

Inventor： LOEHR SANDRA ,  GEBHARDT JOACHIM ,  MAYER GUIDO ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WOLF BERND

IPC: C07D239/54 ,  C07C307/06

CPC classification number: C07D239/54

Abstract: PROBLEM TO BE SOLVED: To provide a process for preparing 3-phenyl(thio)uracils and -dithiouracils.SOLUTION: In the process for preparing 3-phenyl(thio)uracils and -dithiouracils, carbamates having X, X, Ar, and A in formula and enamines having X, R, R, and Rare made to react with each other (in formula, X, X, and Xrepresent oxygen or sulfur, Ar represents a phenyl residue, A represents an amino residue, and R, R, and Rrepresent hydrogen or the like).

Abstract translation: 待解决的问题：提供制备3-苯基（硫代）尿嘧啶和二硫尿嘧啶的方法。 解决方案：在制备3-苯基（硫代）尿嘧啶和二硫尿嘧啶的方法中，具有X 1 的氨基甲酸酯，X ，Ar和A在具有X 2 ，R 1 ，R 2 ，并且使R 3 彼此反应（在公式中，X 1 ，X < SP POS =“POST”> 2 ，X 3 表示氧或硫，Ar表示苯基，A表示氨基残基，R 1 ，R 2 ，R 3 表示氢等。 版权所有（C）2012，JPO＆INPIT

公开(公告)号：BRPI0719209A2

公开(公告)日：2014-06-10

申请号：BRPI0719209

申请日：2007-10-12

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

IPC: C07D239/54 ,  A01N43/48

Abstract: The present invention relates to a crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)pyrimidinyl]-4-fluoro-N-[[methyl(1-methylethyl)-amino]sulfonyl]benzamide. The invention also relates to a process for the preparation of this crystalline form and to plant protection formulations which comprise this crystalline form of the phenyluracil.

公开(公告)号：ZA200903231B

公开(公告)日：2010-07-28

申请号：ZA200903231

申请日：2009-05-11

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND ,  SAXELL HEIDI EMILIA ,  MICHEL ALFRED

IPC: A01N20100101 ,  C07D20100101

Abstract: The present invention relates to a crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)pyrimidinyl]-4-fluoro-N-[[methyl(1-methylethyl)-amino]sulfonyl]benzamide. The invention also relates to a process for the preparation of this crystalline form and to plant protection formulations which comprise this crystalline form of the phenyluracil.

公开(公告)号：MX2009003497A

公开(公告)日：2009-04-14

申请号：MX2009003497

申请日：2007-10-12

Applicant: BASF SE

Inventor： MICHEL ALFRED ,  WEVERS JAN HENDRIK ,  ZAGAR CYRILL ,  SIEVERNICH BERND ,  KEIL MICHAEL ,  REINHARD ROBERT ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  WOLF BERND ,  GEBHARDT JOACHIM ,  MAYER GUIDO ,  ERK PETER ,  SCHMIDT THOMAS ,  COX GERHARD ,  LOEHR SANDRA ,  SAXELL HEIDI EMILIA

IPC: C07D239/54 ,  A01N43/48

Abstract: Forma cristalina de 2-cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(tr ifluorometil)-1-(2H)pirimidinil]-4-fluoro-N-[[metil(1-metiletil)a mino]sulfonil]benzamida. También un proceso para la preparación de esta forma cristalina y formulaciones fitoprotectoras que comprenden esta forma cristalina del feniluracilo.

公开(公告)号：BRPI0609798B1

公开(公告)日：2015-01-27

申请号：BRPI0609798

申请日：2006-05-18

Applicant: BASF SE

Inventor： GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WEVERS JAN HENDRIK ,  ZECH HELMUT ,  HAEBERLE RUDOLF

IPC: C07D239/54

Abstract: The present invention relates to a process for preparing 1-alkyl-3-phenyluracils of the formula I where the variables R1 to R7 are as defined in the description by reacting 3-phenyluracils of the formula II and alkylating agents of the formula III R1-L1  III, with one another, wherein during the entire reaction the pH is kept in a range from 1 to 6 by adding base a little at a time.

公开(公告)号：BRPI0619760A2

公开(公告)日：2012-02-22

申请号：BRPI0619760

申请日：2006-11-23

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

IPC: C07C303/38 ,  C07C201/12 ,  C07C205/58 ,  C07C303/40 ,  C07C311/51

Abstract: A process for preparing sulfonamides I where the variables are each as defined in the description, by reacting m-nitrobenzoyl chlorides II with amino sulfones III, under the influence of B equivalents of base IV, wherein, in step a), the amino sulfone III is reacted with B1 equivalents of base IV, and, in step b), the reaction mixture resulting from step a) is reacted with m-nitrobenzoyl chlorides II and B2 equivalents of base IV; where B, B1 and B2 are each as defined in the description.

公开(公告)号：MX2009003431A

公开(公告)日：2009-04-14

申请号：MX2009003431

申请日：2007-10-12

Applicant: BASF SE

Inventor： MICHEL ALFRED ,  WEVERS JAN HENDRIK ,  ZAGAR CYRILL ,  SIEVERNICH BERND ,  KEIL MICHAEL ,  REINHARD ROBERT ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  WOLF BERND ,  GEBHARDT JOACHIM ,  MAYER GUIDO ,  ERK PETER ,  SCHMIDT THOMAS ,  COX GERHARD ,  LOEHR SANDRA ,  SAXELL HEIDI EMILIA

IPC: C07D239/54 ,  A01N43/48

Abstract: Hidratos de 2-cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(trifluorom etil)-1-(2H)-pirimidinil]-4-flúor-N-[[metil-(1-metiletil)amino]su lfonil]benzamida. También un proceso para la preparación de estos hidratos y formulaciones destinadas a la fitoprotección que comprenden hidratos del feniluracilo I.

公开(公告)号：AT408604T

公开(公告)日：2008-10-15

申请号：AT06755248

申请日：2006-05-18

Applicant: BASF SE

Inventor： GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WEVERS JAN HENDRIK ,  ZECH HELMUT ,  HAEBERLE RUDOLF

IPC: C07D239/54

Abstract: The present invention relates to a process for preparing 1-alkyl-3-phenyluracils of the formula I where the variables R1 to R7 are as defined in the description by reacting 3-phenyluracils of the formula II and alkylating agents of the formula III R1-L1  III, with one another, wherein during the entire reaction the pH is kept in a range from 1 to 6 by adding base a little at a time.

公开(公告)号：UA97498C2

公开(公告)日：2012-02-27

申请号：UAA200904967

申请日：2007-11-02

Applicant: BASF SE

Inventor： RACK MICHAEL ,  SMIDT SEBASTIAN PEER ,  LOEHR SANDRA ,  KEIL MICHAEL ,  DIETZ JOCHEN ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  ZIERKE THOMAS ,  LOHMANN JAN KLAAS ,  SUKOPP MARTIN

IPC: C07D237/04 ,  C07F7/04

Abstract: Данноеизобретениекасаетсяспособаполучениядифторметилзамещенныхпиразол-4-илкарбоксилатовформулы I, (I)вкоторойRозначает C-C-алкил, С-С-циклоалкил, С-С-алкокси-С-С-алкили т.п.; иRозначаетводород, С-С-алкил, бензилилифенил,причема) соединениеобщейформулы II, (II)вкоторой X означаетфтор, хлорилибром, Rимеетодноизприведенныхпреждезначенийи RозначаетС-С-циклоалкил, С-С-алкенил, бензилилифенил,взаимодействуетс силановымсоединениемобщейформулы RSiCl, вкоторой n означает 1, 2 или 3 изаместители R, независимодруготдругавыбраныизС-С-алкилаилифенила, ис металлом, которыйвыбранизметаллов 1, 2, 3, 4 и 12 группыПериодическойсистемыэлементови имеетокислительно-восстановительныйпотенциалменьшечем-0,7 V, вперечислениинанормальныйводородныйэлектро

公开(公告)号：ES2361206T3

公开(公告)日：2011-06-14

申请号：ES07821246

申请日：2007-10-12

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

IPC: C07D239/54 ,  A01N43/48

Abstract: Forma cristalina II de 2-cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(trifluormetil)-1-(2H)-pirimidinil]-4-fluor-N-[[metil-(1metiletil)amino]sulfonil]-benzamida, en la que la porción de solvente en la red cristalina se encuentra por debajo de 10 % molar respecto de 2-Cloro-5-[3,6-dihidro-3-metil-2,6-dioxo-4-(trifluormetil)-1-(2H)-pirimidinil]-4-fluor-N-[[metil-(1metiletil)amino]sulfonil]benzamida.