公开(公告)号：CA2467683C

公开(公告)日：2011-09-27

申请号：CA2467683

申请日：2002-11-15

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  SCHWOEGLER ANJA ,  RHEINHEIMER JOACHIM ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  ROSE INGO ,  SCHAEFER PETER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: C07D239/46 ,  A01N43/54 ,  C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D401/06 ,  C07D401/14 ,  C07D403/12

Abstract: 5-Phenylpyrimidines of formula (I), where the substituents and the indices have the following meanings: R1, R2 = H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkinyl or haloalkinyl, where R1 and R2 together with the nitrogen atom to which they are bonded may form a saturated or unsaturated ring, interrupted by an ether, thio, sulphoxy or sulphonyl group and which can be substituted by one to four groups Ra and/or Rb, R3 = H, halo, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy, R4 = H, halo, cyano, hydroxy, mercapto, azido, alkyl, alkenyl, alkinyl, haloalkyl, alkoxy, alkenyloxy, alkinyloxy, haloalkoxy, alkylthio, alkenylthio, alkinylthio, haloalkylthio, -ON=CRaRb, -CRc=NORa, -NRcN=CRaRb, -NRaRb, -NRcNRaRb, -NORa, -NRcC (=NRc') NRaRb, -NRcC (=0) NRaRb, -NRaC (=0) Rc, -NRaC (=NORc)Rc', -OC (=0) Rc, -C (=NORc) NRaRb, -CRc (=NNRaRb), -C (=0) NRaRb or -C (=0) Rc, where Ra,Rb,Rc are as defined in the description, X = halo, alkyl, alkoxy or haloalkyl and m = a whole number from 1 to 5. The invention further relates to methods for production of the above compounds, agents containing the same and use thereof for the treatment of noxious mycoses.

公开(公告)号：CA2434664C

公开(公告)日：2010-05-04

申请号：CA2434664

申请日：2002-01-17

Applicant: BASF AG

Inventor： EICKEN KARL ,  ROSE INGO ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  HADEN EGON

IPC: A01N35/04 ,  A01N25/02 ,  A01N25/08 ,  A01N37/52 ,  A01N43/08 ,  A01N43/10 ,  A01N43/36 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/78

Abstract: Fungicidal mixtures, comprising a) benzophenones of the formula I (see formula I) in which R1 is chlorine, methyl, methoxy, acetoxy, pivaloyloxy or hydroxyl; R2 is chlorine or methyl; R3 is hydrogen, halogen or methyl; and R4 is C1-C6-alkyl or benzyl, where the phenyl moiety of the benzyl radical may carry a halogen or methyl substituent, and b) oxime ether derivatives of the formula II (see formula II) where the substituents X1 to X5 and Y1 to Y4 are as defined in the description; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II and compositions comprising them are described.

公开(公告)号：AU2002352015B2

公开(公告)日：2008-07-31

申请号：AU2002352015

申请日：2002-11-15

Applicant: BASF AG

Inventor： SCHIEWECK FRANK ,  STRATHMANN SIEGFRIED ,  GYPSER ANDREAS ,  MULLER BERND ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  SCHAFER PETER ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  ROSE INGO ,  SCHWOGLER ANJA ,  STIERL REINHARD ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  RHEINHEIMER JOACHIM

IPC: C07D239/46 ,  A01N43/54 ,  C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D401/06 ,  C07D401/14 ,  C07D403/12

Abstract: 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, -ON-CRaRb, -CRc-NORa, -NRcN-CRaRb, -NRaRb, -NRcNRaRb, -NORa, -NRcC(-NRc')NRaRb, -NRcC(-O)NRaRb, -NRaC(-O)Rc, -NRaC(-NORc)Rc', -OC(-O)Rc, -C(-NORc)NRaRb, -CRc(-NNRaRb), -C(-O)NRaRb or -C(-O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

公开(公告)号：SK286039B6

公开(公告)日：2008-01-07

申请号：SK14002003

申请日：2002-05-17

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  ROSE INGO ,  GROTE THOMAS ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N43/00 ,  A01N43/86 ,  A01N43/90 ,  C07D265/00 ,  C07D265/24 ,  C07D498/00 ,  C07D498/04 ,  C07D513/00 ,  C07D513/04

Abstract: The invention relates to oxazin(thi)one compounds of formula (1) in which the A represents a 5 or 6 membered carbocycle or a 5 or 6 membered heterocycle comprising 1, 2 or 3 heteroatoms, selected from N, O and S, each of which cycles is fused to the oxazin(thi)one ring via two carbon atoms, and the agriculturally useful salts of the same. The invention further relates to the use of compounds of formula (1) and their salts to combat phytopathogenic fungi, as well as agents containing a fungicidally effective amount of said compounds (1) and/or salts thereof, and a method for combating phytopathogenic fungi, according to which said fungi, materials, plants, seeds and soil, which risk being attacked by fungi are treated with a fungicidally effective amount of at least one compound of formula (1) and /or a salt thereof.

公开(公告)号：AU2002302420B2

公开(公告)日：2007-12-06

申请号：AU2002302420

申请日：2002-03-13

Applicant: BASF AG

Inventor： SCHAFER PETER ,  BLASCO JORDI TORMO I ,  STIERL REINHARD ,  AMMERMANN EBERHARD ,  SCHIEWECK FRANK ,  GEWEHR MARKUS ,  RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  LORENZ GISELA ,  SAUTER HUBERT ,  MULLER BERND ,  ROSE INGO ,  STRATHMANN SIEGFRIED ,  GROTE THOMAS

IPC: C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00

Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.

公开(公告)号：PT1414302E

公开(公告)日：2007-05-31

申请号：PT02790165

申请日：2002-07-16

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  GEWEHR MARKUS ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  ROSE INGO ,  STIERL REINHARD ,  LORENZ GISELA ,  MUELLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  SCHAEFER PETER ,  BLASCO JORDI TORMO I ,  SAUTER HUBERT ,  SCHIEWECK FRANK ,  KRUMMEL GUENTER

IPC: A01N43/90 ,  C07D487/04

公开(公告)号：NZ529280A

公开(公告)日：2006-04-28

申请号：NZ52928002

申请日：2002-05-17

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  ROSE INGO ,  GROTE THOMAS ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N43/86 ,  A01N43/90 ,  C07D265/24 ,  C07D498/04 ,  C07D513/04

Abstract: An oxazin (ethi) one compound of the formula (I) and its agriculturally useful salts used in a method for controlling phytopathogenic fungi that comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula (I) and/or a salt thereof.

公开(公告)号：ES2247335T3

公开(公告)日：2006-03-01

申请号：ES02732728

申请日：2002-05-17

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  ROSE INGO ,  GROTE THOMAS ,  SCHAFER PETER ,  SCHIEWECK FRANK

IPC: A01N43/86 ,  A01N43/90 ,  C07D265/24 ,  C07D498/04 ,  C07D513/04

Abstract: Compuestos de oxazin(ti)ona de la **fórmula**, en la que las variables Z, A, n, R1, R2 y R3 tienen los significados siguientes: Z significa oxígeno o azufre, A significa un carbociclo con 5 o 6 miembros o un heterociclo con 5 o 6 miembros con 1, 2 o 3 heteroátomos, elegidos entre N, O y S, anillados a través de dos átomos de carbono con el anillo de oxazin(ti)ona; n significa un número desde 0 hasta 4; R1 significa hidrógeno, alquilo con 1 a 6 átomos de carbono, alquenilo con 2 a 6 átomos de carbono, alquinilo con 2 a 6 átomos de carbono, que estén substituidos respectivamente, en caso dado, por O- R4, por C(O)O-R5, por NR6R7, por C(O)NR6R7, por S- R8, por cicloalquilo con 3 a 8 átomos de carbono, por fenilo o por heterociclilo con 5 o 6 miembros, saturado o insaturado, con 1 hasta 3 heteroátomos, elegidos entre N, O y S, estando substituidos el fenilo y el heterociclilo, en caso dado, una, dos o tres veces, halógenoalquilo con 1 a 6 átomos de carbono, halógenoalquenilo con 2 a 6 átomos decarbono o halógenoalquinilo con 2 a 6 átomos de carbono.

公开(公告)号：EA006634B1

公开(公告)日：2006-02-24

申请号：EA200301173

申请日：2002-05-17

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  ROSE INGO ,  GROTE THOMAS ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRIAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N43/86 ,  A01N43/90 ,  C07D265/24 ,  C07D498/04 ,  C07D513/04

Abstract: Визобретенииописываютсяоксазин(ти)оновыесоединенияформулы Iвкоторойпеременные Z, A, n, R, Rи Rимеютследующиезначения:Z обозначаеткислород,Аобозначаетаннелированноебензольноекольцо,n обозначает 0 или 1,Rобозначает C-Салкил, необязательнозамещенныйС-Салкоксигруппойили C-Сциклоалкилом, C-Салкенил, C-Сгалогеналкилили C-Сгалогеналкенил,Rобозначает C-Салкилилициклопропилметил,Rобозначаетгалоген, C-Салкилили C-Салкоксигруппу,атакжеприемлемыедлясельскогохозяйствасолиэтихоксазин(ти)оновыхсоединенийформулы I.Крометого, взаявкеописываютсяприменениесоединенийформулы (I) иихсолейдляборьбыс фитопатогеннымигрибами, средства, содержащиесоединенияформулы (I) и/илиихсолив фунгицидноэффективномколичестве, атакжеспособборьбыс фитопатогеннымигрибами, заключающийсяв том, чтогрибыилиподвергаемыеопасностипоражениягрибамиматериалы, растения, семенаилипочвуобрабатываютфунгицидноэффективнымколичествомпоменьшеймереодногосоединенияформулы (I) поп.1 и/илисолисоединенияформулы (I).

公开(公告)号：NZ528409A

公开(公告)日：2005-11-25

申请号：NZ52840902

申请日：2002-03-13

Applicant: BASF AG

Inventor： GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MULLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD ,  GYPSER ANDREAS

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00 ,  C07D473/00

Abstract: Disclosed are compounds of the formula (I), wherein; R1 is pyrrole, pyrazole, imidazole, 1,2,4-triazole, 1,2,3-triazole, tetrazole, 1,2,3-triazine, 1,2,4-triazine, oxazole, isoxazole, 1,3,4-oxadiazole, furan, thiophene, thiazole, isothiazole, it being possible for the heterocycle to be bonded to the pyramidine ring via C or N, pyridazine, pyrimidine or pyrazine, it being possible for R1 to be substituted by one to three identical or different groups Ra; processes for their synthesis and intermediates therein. Further disclosed is a method for controlling harmful fungi, which comprises treating the fungi or the materials, plants, soil or seeds to be protected against fungal infection with an effective amount of a compound of the formula (I).