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公开(公告)号:BRPI0408864A
公开(公告)日:2006-04-11
申请号:BRPI0408864
申请日:2004-03-30
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L=halogen, alkyl, halogenalkyl, alkoxy, amino, NHR, NR 2 , cyano, S(O) n A 1 or C(O)A 2 ; R=alkyl or alkylcarbonyl, A 1 =hydrogen, hydroxy, alkyl, alkylamino or aialkylamino; n=0, 1 or 2; A 2 =alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A 1 ; m=1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond with the triazolopyrimidine skeleton; X=halogen, cyano, alkyl, halogenalkyl or alkoxy; R 1 =hydrogen or alkyl; R 2 =alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compounds and the use thereof to combat harmful phytopathogenic fungi.
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公开(公告)号:BR0317448A
公开(公告)日:2005-11-16
申请号:BR0317448
申请日:2003-12-17
Applicant: BASF AG
Inventor: MUELLER BERND , BLASCO JORDI TORMO I , GROTE THOMAS , BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: Triazolopyrimidines of the formula I in which the index n and the substituents R 1 , R 2 and R 3 are as defined in the description, and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
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公开(公告)号:BR0316033A
公开(公告)日:2005-09-13
申请号:BR0316033
申请日:2003-11-14
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: 2-Mercapto-substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy or -C(-O)-A; A is hydrogen, hydroxyl, alkyl, alkenyl, alkoxy, haloalkoxy, alkylamino or dialkylamino; m is 0, 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R 1 , R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four hetero atoms from the group consisting of O, N and S; R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S; where R 1 and/or R 2 may be substituted as stated in the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.
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公开(公告)号:BR0211180A
公开(公告)日:2004-08-10
申请号:BR0211180
申请日:2002-07-08
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , SAUTER HUBERT , LLER BERND M , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHOFER PETER , SCHIEWECK FRANK , RACK MICHAEL , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.
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公开(公告)号:BR0210858A
公开(公告)日:2004-06-29
申请号:BR0210858
申请日:2002-07-03
Applicant: BASF AG
Inventor: MUELLER BERND , SAUTER HUBERT , GEWEHR MARKUS , GRAMMENOS WASSILIOS , BLASCO JORDI TORMO I , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHOFER PETER , SCHIEWECK FRANK , RACK MICHAEL , LORENZ GISELA , STRATHMANN SIEGFRIED , AMMERMANN EBERHARD , STIERL REINHARD
IPC: A01N43/90 , C07D487/04 , A01N43/653
Abstract: 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines (I) are new. 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines of formula (I) are new. [Image] n : 0-5; R : halo, CN, OH or OCN, or alkyl, alkenyl, alkynyl, T', haloalkenyl, OT, alkenyloxy, alkynyloxy, OT', cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, CONH 2, mono- or dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); T : 1-6C alkyl; T' : 1-6C haloalkyl; Het : 5-10 membered, saturated, partially unsaturated or aromatic heterocycle containing 1-4 of O, N and/or S heteroatoms; R 11-10C alkyl, alkenyl, alkynyl, 3-12C cycloalkyl, 3-10C cycloalkenyl, phenyl, naphthyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); R ahalo, CN, NO 2, OH, T, T', COT, cycloalkyl, OT, OT', COOT, NHT, NT 2, 2-6C alkenyl, 2-6C alkenyloxy, 3-6C alkynyloxy, alkoximino, alkenyloximino, alkynyloximino, aralkoximino, alkynyl, alkynyloxycarbonyl, phenyl, naphthyl or Het (where all aliphatic, alicyclic or aromatic groups are optionally partially or completely halogenated and optionally substituted by 1-3 R aand/or 1-3 R c); R bhalo, CN, NO 2, OH, SH, NH 2, COOH, CONH 2, CSNH 2, T, T', 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, OT, OT', ST, NHT, NT 2, CHO, COT, SO 2T, SOT, COOT, OCOT, CONHT, CONT 2, CSNHT or CSNT 2; R ccycloalkyl, -O-cycloalkyl, heterocyclyl, -O-heterocyclyl, aryl, -O-aryl, -S-aryl, -O-T-aryl, -T-aryl, heteroaryl, -O-heteroaryl or -S-heteroaryl (where cycloalkyl or heterocyclyl rings are 3-10 membered, aryl rings are preferably 6-10 membered and heteroaryl rings are preferably 5-6 membered; and all rings are optionally partially or completely halogenated and optionally substituted by alkyl or haloalkyl); and R 21-4C alkyl, 2-4C alkynyl or 2-4C alkynyl (all optionally substituted by halo, CN, NO 2, OMe, OEt or 1-4C alkoxycarbonyl; Unless specified otherwise alkyl moieties have 1-8C, alkenyl or alkynyl moieties 2-10C and cycloalkyl or cycloalkenyl moieties 3-6C. Independent claims are also included for: (1) preparation of (I); and (2) dicarbonyl compound intermediates of formula (III), provided that n is not 0 and R 1and R 2are not both Me. [Image] ACTIVITY : Fungicide. 7-Cyclohexyl-5-methyl-6-(2-chloro-6-fluorophenyl)-1,2,4-triazolo[1,5-a]pyrimidine (Ia) at a concentration of 63 ppm gave at least 90 % protection of tomato plants against Alternaria solani. MECHANISM OF ACTION : None given.
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公开(公告)号:BR0209835A
公开(公告)日:2004-06-15
申请号:BR0209835
申请日:2002-05-17
Applicant: BASF AG
Inventor: RHEINHEIMER JOACHIM , GYPSER ANDREAS , ROSE INGO , GROTE THOMAS , SCHOFER PETER , SCHIEWECK FRANK , AMMERMANN EBERHARD , SPEAKMAN JOHN-BRYAN , STRATHMANN SIEGFRIED , LORENZ GISELA
IPC: A01N43/86 , A01N43/90 , C07D265/24 , C07D498/04 , C07D513/04
Abstract: Oxazin(ethi)one compounds of the formula I: in which the variables Z, R 1 , R 2 , R 3 and n are as defined in claim 1 and A is a 5- or 6-membered carbocycle or a 5- or 6-membered heterocycle having 1, 2 or 3 heteroatoms selected from the group consisting of N, O and S, each of which cycles is attached via two carbon atoms to the oxazin(ethi)one ring, and the agriculturally useful salts of the oxazin(ethi)one compounds I are described. Moreover, the invention describes the use of compounds I and their salts for controlling phytopathogenic fungi, compositions which comprise the compounds I and/or their salts in a fungicidally effective amount and a method for controlling phytopathogenic fungi which comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula I as claimed in claim 1 and/or a salt of I.
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公开(公告)号:BR0207975A
公开(公告)日:2004-06-15
申请号:BR0207975
申请日:2002-03-13
Applicant: BASF AG
Inventor: GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHOFER PETER , SCHIEWECK FRANK , SAUTER HUBERT , GEWEHR MARKUS , MUELLER BERND , BLASCO JORDI TORMO I , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/647 , A01N43/653 , A01N43/713 , A01N43/90 , C07D239/42 , C07D401/14 , C07D403/04 , C07D471/04 , C07D473/06 , C07D487/04 , C07D521/00 , C07D473/00
Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.
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公开(公告)号:BR9813613A
公开(公告)日:2000-10-10
申请号:BR9813613
申请日:1998-12-11
Applicant: BASF AG
Inventor: REINHARD ROBERT , HAMPRECHT GERHARD , MENGES MARKUS , MENKE OLAF , SCHOFER PETER , ZAGAR CYRILL , HEISTRACHER ELISABETH , OTTEN MARTINA , WALTER HELMUT , WESTPHALEN KARL-OTTO
IPC: C07D239/54 , A01N43/54 , A01N43/647 , A01N43/707 , A01N43/74 , A01N43/76 , A01N43/78 , C07D403/04 , C07D413/04 , C07D417/04 , C07F9/6558
Abstract: The invention relates to 3-(benzazol-4-yl)pyrimidine-dione-derivatives of formula (I) and the salts thereof, whereby X = O, S; R = H, NH2, C1-C6-alkyl, C1-C6-alkyl halide; R = H, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkylthio, C1-C6-alkylsulfinyl, C1-C6-alkylsulfonyl; R = H, halogen, C1-C6-alkyl; R = H, halogen; R = CN, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkoxyl, C1-C6-alkoxyl halide; =Y- = a group =N-N(R )-, =C(ZR )-N(R )-, =C(ZR )-O-, =C(ZR )-S-; R = C1-C6-alkyl, C1-C4-alkyl halide, C3-C6-cycloalkyl, C3-C6-alkenyl, C3-C6-alkynyl, C1-C6-alkyl-SO2, C1-C6-alkyl-CO, C1-C6-alkyl halide-CO, C1-C6-alkyl-CS, C1-C6-alkoxyl-CO, C1-C6-alkoxyl-CS or optionally substituted C1-C6-alkyl; Z = chemical bond, O, S, -S(O)-, -SO2-, -NH-, -N(R )-; R , R = C1-C6-alkyl, C1-C6-alkyl halide, hydroxy-C1-C4-alkyl, cyano-C1-C4-alkyl, C1-C4-alkoxyl-C1-C4-alkyl, C1-C4-alkoxyl halide-C1-C4-alkyl, C3-C4-alkenyloxyl-C1-C4-alkyl, C3-C4-alkynyloxyl-C1-C4-alkyl, C3-C8-cycloalkoxyl-C1-C4-alkyl, amino-C1-C4-alkyl, C1-C4-alkylamino-C1-C4-alkyl, di(C1-C4-alkyl)amino-C1-C4-alkyl, C1-C4-alkylthio-C1-C4-alkyl, C1-C4-alkylthio halide-C1-C4-alkyl, C3-C4-alkenylthio-C1-C4-alkyl, C3-C4-alkynylthio-C1-C4-alkyl, C1-C4-alkylsulfinyl-C1-C4-alkyl, C1-C4-alkylsulfinyl halide-C1-C4-alkyl, C3-C4-alkenylsulfinyl-C1-C4-alkyl, C3-C4-alkynylsulfinyl-C1-C4-alkyl, C3-C6-alkenyl, cyano-C3-C6-alkenyl, C3-C6-alkenyl halide, C3-C6-alkynyl, cyano-C3-C6-alkynyl, C3-C6-alkynyl halide, HO-CO-C1-C4-alkyl, (C1-C4-alkoxyl)CO-C1-C4-alkyl, (C1-C4-alkyl)CS-C1-C4-alkyl, H2N-CO-C1-C4-alkyl, C1-C4-alkyl-NHCO-C1-C4-alkyl, di(C1-C4-alkyl)NCO-C1-C4-alkyl, di(C1-C4-alkyl)phosphonyl-C1-C4-alkyl, optionally substituted C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, phenyl, phenyl-C1-C4-alkyl, 3- to 7-linked heterocyclyl or heterocyclyl-C1-C4-alkyl, whereby each heterocyclyl ring can contain a CO-ring link or CS-ring link, or provided that Z = chemical bond, R also H, OH, CN, SH, NH2, halogen, -CH(OH)-CH2-R , -CH(halogen)-CH2-R , -CH2-CH(halogen)-R , -CH=CH-R or -CH=C(halogen)-R , whereby R = COOH, (C1-C4-alkoxyl)carbonyl, (C1-C4-alkylthio)carbonyl, CONH2, C1-C4-alkyl-NHCO or di(C1-C4-alkyl)NCO, or R + R = an optionally substituted 1,3-propylene-, tetramethylene-, pentamethylene- or ethylene oxyethylene-chain.
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公开(公告)号:NO992924A
公开(公告)日:1999-08-13
申请号:NO992924
申请日:1999-06-15
Applicant: BASF AG
Inventor: ZAGAR CYRILL , HAMPRECHT GERHARD , MENGES MARKUS , MENKE OLAF , SCHOFER PETER , WESTPHALEN KARL-OTTO , MISSLITZ ULF , WALTER HELMUT
IPC: A01N43/56 , A01N43/74 , C07D413/04 , C07D417/04 , C07D471/00
CPC classification number: C07D413/04 , A01N43/74 , C07D417/04
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公开(公告)号:NO992924D0
公开(公告)日:1999-06-15
申请号:NO992924
申请日:1999-06-15
Applicant: BASF AG
Inventor: ZAGAR CYRILL , HAMPRECHT GERHARD , MENGES MARKUS , MENKE OLAF , SCHOFER PETER , WESTPHALEN KARL-OTTO , MISSLITZ ULF , WALTER HELMUT
IPC: A01N43/56 , A01N43/74 , C07D413/04 , C07D413/10 , C07D417/04 , C07D417/10 , C07D
Abstract: Substituted Pyrazol-3-ylbenzazoles Isalts thereof, and their use as herbicides or for the desiccation/defoliation of plants.
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