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公开(公告)号:SG10201505951VA
公开(公告)日:2015-08-28
申请号:SG10201505951V
申请日:2011-07-28
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: MATSUO YO , HISADA SHOJI , NAKAMURA YUSUKE , AHMED FERYAN , HUNTLEY RAYMOND , WALKER JOEL R , DECORNEZ HELENE
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公开(公告)号:MX2014008780A
公开(公告)日:2014-10-23
申请号:MX2014008780
申请日:2012-12-21
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: NAKAMURA YUSUKE , WALKER JOEL R , MATSUO YO , HISADA SHOJI , AHMED FERYAN , HUNTLEY RAYMOND
IPC: A61K31/4745 , C07D471/04
Abstract: La presente invención está dirigida a un compuesto representado por la fórmula (I), que comprende un derivado de 1,5-naftiridina; en una modalidad, el derivado de 1,5-naftiridina de fórmula (I) tiene actividad inhibitoria contra la cinasa de cierre de leucina embrionaria materna (MELK); la presente invención también incluye un método para preparar el derivado de 1,5-naftiridina de fórmula (I); la presente invención también incluye una composición farmacéutica que contiene el derivado de 1,5-naftiridina de fórmula (I) como ingrediente activo.
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53.
公开(公告)号:ZA201103964B
公开(公告)日:2012-02-29
申请号:ZA201103964
申请日:2011-05-30
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: MATSUO YO , LI YINGFU , WALKER JOEL R , AHMED FERYAN , OHSAWA RYUJI , HISADA SHOJI
IPC: A01N20060101 , A61K20060101
Abstract: 7-Hydroxy-benzoimidazole-4-yl-methanone Derivatives, which are useful for PBK inhibitors, are provided.
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公开(公告)号:CO6361935A2
公开(公告)日:2012-01-20
申请号:CO11061830
申请日:2011-05-19
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: MATSUO YO , AHSAWA RYUJI , HISADA SHOJI
IPC: A61K31/4184
Abstract: Se proporcionan inhibidores GSK-3beta que comprenden derivados de 7-hidroxi-benzoimidazol-4-il-metanona. Por ejemplo los inhibidores que tienen la siguiente fórmula general (I)
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55.
公开(公告)号:CA2741988A1
公开(公告)日:2010-05-06
申请号:CA2741988
申请日:2009-07-30
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: MATSUO YO , LI YINGFU , WALKER JOEL R , AHMED FERYAN , OHSAWA RYUJI , HISADA SHOJI
IPC: C07D409/14 , A61K31/4184 , A61K31/454 , A61P35/00 , C07D235/04 , C07D401/12 , C07D403/12 , C07D409/04
Abstract: 7-Hydroxy-benzoimidazole-4-yl-methanone Derivatives, which are useful for PBK inhibitors, are provided.
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56.1,5-NAPHTHYRIDINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME 有权
Title translation: 1,5-Naphthyridine抑制剂和Melk抑制剂公开(公告)号:EP2753329A4
公开(公告)日:2015-11-25
申请号:EP12865937
申请日:2012-12-21
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: MATSUO YO , HISADA SHOJI , NAKAMURA YUSUKE , AHMED FERYAN , WALKER JOEL R , HUNTLEY RAYMOND
IPC: C07D471/04 , A61K31/4745 , A61P35/00
CPC classification number: A61K31/5377 , A61K31/4375 , A61K31/496 , A61K31/506 , C07D471/04
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57.GLYCOGEN SYNTHASE KINASE-3 BETA INHIBITORS CONTAINING 7-HYDROXY-BENZOIMIDAZOLE-4-YL-METHANONE DERIVATIVES 审中-公开
Title translation: GLYCOGEN-SYNTHASE-KINASE-3-BETA-HEMMER MIT 7-羟基苯并咪唑-4-甲酰胺公开(公告)号:EP2358365A4
公开(公告)日:2012-05-30
申请号:EP09827294
申请日:2009-09-29
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: MATSUO YO , OHSAWA RYUJI , HISADA SHOJI
IPC: A61K31/4184 , A61K31/454 , A61K31/496 , A61P3/10 , A61P25/06 , A61P25/24 , A61P25/28 , A61P43/00 , C07D235/08 , C07D235/18 , C07D401/12 , C07D409/04 , C07D409/06 , C07D409/14
CPC classification number: C07D409/04 , C07D235/08 , C07D235/18 , C07D401/12 , C07D403/12 , C07D409/06 , C07D409/14
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58.
公开(公告)号:EP2597955A4
公开(公告)日:2014-02-19
申请号:EP11813209
申请日:2011-07-28
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: MATSUO YO , HISADA SHOJI , NAKAMURA YUSUKE , AHMED FERYAN , HUNTLEY RAYMOND , WALKER JOEL R , DECORNEZ HELENE
IPC: C07D215/46 , C07D215/54 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D409/04 , C07D409/06 , C07D409/14
CPC classification number: C07D215/54 , A61K31/4709 , C07D215/46 , C07D401/04 , C07D401/10 , C07D401/12 , C07D401/14 , C07D409/04 , C07D409/06 , C07D409/14 , C07D413/06 , C07D453/02 , C07D471/04
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59.
公开(公告)号:EP2552206A4
公开(公告)日:2013-08-14
申请号:EP11763307
申请日:2011-03-29
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: NAKAMURA YUSUKE , MATSUO YO , HISADA SHOJI , AHMED FERYAN , HUNTLEY RAYMOND , SAJJADI-HASHEMI ZOHREH , JENKINS DAVID M , KARGBO ROBERT B , CUI WENGE , GAUUAN POLIVINA JOLICIA F , WALKER JOEL R , DECORNEZ HELENE , GURRAM MAHENDER
IPC: A01N43/42 , C07D221/06 , C07D487/04 , C07D495/04 , C07D513/04
CPC classification number: C07D495/04 , C07D213/64 , C07D221/06 , C07D221/16 , C07D401/04 , C07D401/10 , C07D487/04 , C07D513/04 , C07D519/00
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60.BENZOIMIDAZOLE DERIVATIVES AND GLYCOGEN SYNTHASE KINASE-3 BETA INHIBITORS CONTAINING THE SAME 审中-公开
Title translation: 为了BENZOIMIDAZOLDERIVATE和糖原合酶激酶3 BETA抑制剂公开(公告)号:EP2309855A4
公开(公告)日:2012-06-27
申请号:EP09803582
申请日:2009-07-30
Applicant: ONCOTHERAPY SCIENCE INC
Inventor: OHTANI MITSUAKI , MATSUO YO , LI YINGFU , WALKER JOEL R , JENKINS DAVID M , AHMED FERYAN , OHSAWA RYUJI , HISADA SHOJI
IPC: A01N43/30
CPC classification number: C07D409/04 , C07D235/18 , C07D405/04 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14
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