公开(公告)号：NO992770A

公开(公告)日：1999-06-08

申请号：NO992770

申请日：1999-06-08

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  M LLER ACHIM ,  TREIBER HANS-J RG

IPC: A61K31/403 ,  A61K31/4035 ,  A61K31/405 ,  A61K31/4439 ,  A61K31/496 ,  A61K31/517 ,  A61K31/519 ,  A61K31/5377 ,  A61P9/00 ,  A61P25/00 ,  A61P25/08 ,  A61P25/14 ,  A61P25/28 ,  A61P35/00 ,  A61P35/04 ,  A61P43/00 ,  C07D209/48 ,  C07D209/66 ,  C07D239/70 ,  C07D239/96 ,  C07D401/12 ,  C07D471/04 ,  C07D475/02 ,  A61K31/40

CPC classification number: C07D471/04 ,  C07D209/66 ,  C07D239/70 ,  C07D239/96 ,  C07D475/02

公开(公告)号：AU9748498A

公开(公告)日：1999-05-17

申请号：AU9748498

申请日：1998-10-05

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  DULLWEBER UTA ,  STARCK DOROTHEA ,  STEINER GERD ,  BACH ALFRED ,  EMLING FRANZ ,  GARCIA-LADONA XAVIER ,  TESCHENDORF HANS-JURGEN ,  WICKE KARSTEN

IPC: A61K31/519 ,  A61P1/00 ,  A61P1/14 ,  A61P3/04 ,  A61P5/00 ,  A61P9/12 ,  A61P15/00 ,  A61P25/00 ,  A61P25/22 ,  A61P25/24 ,  A61P25/28 ,  A61P43/00 ,  C07D471/00 ,  C07D471/04

Abstract: 3-substituted tetrahydropyridopyrimidinone derivatives of the formula (I) wherein the radicals have the meanings given in the Description, to a method for producing said derivatives and, to their use for producing active ingredients for drugs.

公开(公告)号：CA2305258A1

公开(公告)日：1999-05-06

申请号：CA2305258

申请日：1998-10-05

Applicant: BASF AG

Inventor： STEINER GERD ,  STARCK DOROTHEA ,  DULLWEBER UTA ,  BACH ALFRED ,  LUBISCH WILFRIED ,  EMLING FRANZ ,  GARCIA-LADONA XAVIER ,  TESCHENDORF HANS-JURGEN ,  WICKE KARSTEN

IPC: A61K31/519 ,  A61P1/00 ,  A61P1/14 ,  A61P3/04 ,  A61P5/00 ,  A61P9/12 ,  A61P15/00 ,  A61P25/00 ,  A61P25/22 ,  A61P25/24 ,  A61P25/28 ,  A61P43/00 ,  C07D471/00 ,  C07D471/04

Abstract: The invention relates to 3-substituted tetrahydropyridopyrimidinone derivatives of formula (I) wherein the radicals have the meanings given in the Description, to a method for producing said derivatives, and to their use as selective 5HT1B-and 5HT1A antagonists.

公开(公告)号：ZA979175B

公开(公告)日：1999-04-14

申请号：ZA979175

申请日：1997-10-14

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  MOELLER ACHIM ,  DELZER JUERGEN

IPC: A61K31/445 ,  A61K31/4523 ,  A61K31/4545 ,  A61K31/4709 ,  A61K31/498 ,  A61K31/5355 ,  A61P9/10 ,  A61P25/14 ,  A61P25/28 ,  A61P35/00 ,  A61P43/00 ,  C07D211/62 ,  C07D213/40 ,  C07D295/04 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D409/06 ,  C07D413/12 ,  C07D413/14 ,  C07D ,  A61K

Abstract: Piperidineketocarboxylic acid derivatives of the general formula Iand their tautomeric and isomeric forms, and physiologically tolerable salts thereof, where the variables have the meanings given in the description, preparation of these compounds and their use as drugs.

公开(公告)号：ZA9709175B

公开(公告)日：1999-04-14

申请号：ZA9709175

申请日：1997-10-14

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  MOELLER ACHIM ,  DELZER JUERGEN

IPC: A61K31/445 ,  A61K31/4523 ,  A61K31/4545 ,  A61K31/4709 ,  A61K31/498 ,  A61K31/5355 ,  A61P9/10 ,  A61P25/14 ,  A61P25/28 ,  A61P35/00 ,  A61P43/00 ,  C07D211/62 ,  C07D213/40 ,  C07D295/04 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D409/06 ,  C07D413/12 ,  C07D413/14 ,  C07D ,  A61K

CPC classification number: C07D401/06 ,  C07D211/62 ,  C07D401/12

公开(公告)号：NO991761L

公开(公告)日：1999-04-14

申请号：NO991761

申请日：1999-04-14

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  M LLER ACHIM ,  DELZER J RGEN

IPC: A61K31/445 ,  A61K31/4523 ,  A61K31/4545 ,  A61K31/4709 ,  A61K31/498 ,  A61K31/5355 ,  A61P9/10 ,  A61P25/14 ,  A61P25/28 ,  A61P35/00 ,  A61P43/00 ,  C07D211/62 ,  C07D213/40 ,  C07D295/04 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D409/06 ,  C07D413/12 ,  C07D413/14

Abstract: Piperidineketocarboxylic acid derivatives of the general formula Iand their tautomeric and isomeric forms, and physiologically tolerable salts thereof, where the variables have the meanings given in the description, preparation of these compounds and their use as drugs.

公开(公告)号：AU4777097A

公开(公告)日：1998-05-11

申请号：AU4777097

申请日：1997-09-23

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  MOLLER ACHIM ,  DELZER JURGEN

IPC: A61K31/445 ,  A61K31/4523 ,  A61K31/4545 ,  A61K31/4709 ,  A61K31/498 ,  A61K31/5355 ,  A61P9/10 ,  A61P25/14 ,  A61P25/28 ,  A61P35/00 ,  A61P43/00 ,  C07D211/62 ,  C07D213/40 ,  C07D295/04 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D409/06 ,  C07D413/12 ,  C07D413/14

Abstract: Piperidineketocarboxylic acid derivatives of the general formula Iand their tautomeric and isomeric forms, and physiologically tolerable salts thereof, where the variables have the meanings given in the description, preparation of these compounds and their use as drugs.

公开(公告)号：AU3032397A

公开(公告)日：1998-01-14

申请号：AU3032397

申请日：1997-06-05

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  BEHL BERTHOLD ,  HOFMANN HANS-PETER ,  SZABO LASZLO

IPC: C07D403/04 ,  A61K31/495

公开(公告)号：BG101407A

公开(公告)日：1997-09-30

申请号：BG10140797

申请日：1997-04-11

Applicant: BASF AG

Inventor： LUBISCH WILFRIED ,  VIERLING MICHAEL ,  BEHL BERTHOLD ,  HOFMANN HANS P

IPC: A61K31/495 ,  A61P25/00 ,  A61P43/00 ,  C07D403/04

Abstract: Pyrrolyl-tetrahydrobenzoquinoxaline diodes having the formula are disclosed, as well as their tautomeric and isomeric forms, their physiologically compatible salts and their preparation. In the formula, the variables have the meanings given in the description. These new compounds are glutamate antagonists useful in the therapy of neurodegenerative diseases.

公开(公告)号：MX9702226A

公开(公告)日：1997-06-28

申请号：MX9702226

申请日：1995-09-19

Applicant: BASF AG

Inventor： TREIBER HANS-JORG ,  LUBISCH WILFRIED ,  BEHL BERTHOLD ,  HOFMANN HANS PETER

IPC: C07D487/04 ,  A61K31/495

Abstract: Se describen imidazoloquinoxalinonas de la formula (Ver Formula) donde R1-R5, A y B tienen los significados establecidos en la descripcion, y la preparacion de las mismas. Las sustancias novedosas son adecuadas para el control de enfermedades.