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公开(公告)号：WO0160319A3
公开(公告)日：2002-03-21
申请号：PCT/US0104915
申请日：2001-02-15
Applicant: ARCH DEV CORP , LIAO SHUTSUNG , HIIPAKKA RICHARD A , KAO YUNG HSI
Inventor： LIAO SHUTSUNG , HIIPAKKA RICHARD A , KAO YUNG-HSI
IPC: A61K31/045 , A61K31/05 , A61K31/175 , A61K31/351 , A61K31/353 , A61K31/397 , A61K31/50 , A61K31/549 , A61P3/10 , A61P29/00 , A61P35/00 , A61K31/35
CPC classification number: A61K31/549 , A61K31/045 , A61K31/05 , A61K31/175 , A61K31/351 , A61K31/353 , A61K31/397 , A61K31/50
Abstract: A method for reducing food intake in a subject and a method for reducing the levels of an endocrine in a subject. The methods include administering to the subject in need thereof an effective amount of a compound of the formula (I). Also disclosed is a liposomal preparation which includes a liposome and a compound entrapped therein. The entrapped compound is of the formula shown above.
Abstract translation: 用于减少受试者的食物摄入的方法和降低受试者内分泌水平的方法。 所述方法包括向有需要的受试者施用有效量的式（I）化合物。 还公开了一种脂质体制剂，其包括脂质体和包埋在其中的化合物。 包埋的化合物具有如上所示的式子。
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2.发明申请
公开(公告)号：WO9637201A3
公开(公告)日：1997-01-03
申请号：PCT/US9607137
申请日：1996-05-16
Applicant: ARCH DEV CORP , LIAO SHUTSUNG , LIANG THEMING
Inventor： LIAO SHUTSUNG , LIANG THEMING
IPC: C07D311/62 , A61K8/36 , A61K8/37 , A61K8/49 , A61K8/67 , A61K31/19 , A61K31/20 , A61K31/202 , A61K31/216 , A61K31/235 , A61K31/335 , A61K31/35 , A61K31/352 , A61K31/353 , A61K31/565 , A61K36/00 , A61K45/06 , A61P3/00 , A61P3/04 , A61P13/02 , A61P15/00 , A61P17/00 , A61P35/00 , A61P43/00 , A61Q7/00 , A61Q19/00 , A61Q19/06 , C07C53/21 , C07C57/52 , C07C57/56 , C07C61/16 , C07C61/40 , C07C69/88 , A61K31/38 , A61K31/395
CPC classification number: A61K8/361 , A61K8/37 , A61K8/498 , A61K8/67 , A61K31/216 , A61K31/353 , A61K31/565 , A61K45/06 , A61K2800/782 , A61Q7/00 , A61Q19/00 , A61Q19/06 , C07C53/21 , C07C57/52 , C07C57/56 , C07C61/16 , C07C61/40 , C07C69/88 , A61K31/35 , A61K31/235 , A61K31/20 , A61K31/19 , A61K2300/00
Abstract: Disclosed are a novel class of antiandrogenic compounds including saturated and unsaturated fatty acids, catechin gallates, their derivatives, and synthetic analogs, their method of synthesis, and their use in treating disorders associated with androgenic activities. Also disclosed is the use of known compounds not previously known for their antiandrogenic activity in treating disorders related to androgenic activities and cancers.
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公开(公告)号：WO9003979A3
公开(公告)日：1990-05-17
申请号：PCT/US8904312
申请日：1989-10-02
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , PATAKI JOHN , HARVEY RONALD G
IPC: A61K31/045 , A61K31/05 , A61K31/12 , A61K31/22 , C07C39/17 , C07C45/51 , C07C49/657 , C07C49/665 , C07C49/747 , C07C49/753 , C07C49/792 , C07J1/00 , C07J63/00
CPC classification number: C07J63/008 , A61K31/045 , A61K31/05 , A61K31/12 , A61K31/22 , C07C39/17 , C07C45/513 , C07C45/516 , C07C49/657 , C07C49/665 , C07C49/747 , C07C49/753 , C07C49/792 , C07C2603/26 , C07J1/0055 , C07J1/0059 , C07J1/007 , C07J1/0088
Abstract: Disclosed are novel classes of anti-androgens including dihydrophenanthrene derivatives, their method of synthesis and their use in treating disorders associated with excessive androgenic activities.
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公开(公告)号：EP0652749A4
公开(公告)日：1997-04-09
申请号：EP93910950
申请日：1993-04-30
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , LIANG TEHMING
IPC: G01N33/74 , A61K8/00 , A61K8/14 , A61K8/30 , A61K8/35 , A61K8/36 , A61K8/368 , A61K8/37 , A61K8/49 , A61K8/67 , A61K9/127 , A61K31/19 , A61K31/20 , A61K31/23 , A61K31/353 , A61K31/38 , A61K31/40 , A61K31/557 , A61K31/565 , A61K45/06 , A61K47/42 , A61P3/06 , A61P13/02 , A61P15/00 , A61P17/00 , A61P35/00 , A61Q5/00 , A61Q7/00 , A61Q19/00 , C07C53/00 , C07C53/21 , C07C57/03 , C07C57/26 , C07C57/30 , C07C57/46 , C07C57/52 , C07C57/56 , C07C61/16 , C07C61/40 , C07C69/63 , C07C69/65 , C07C69/675 , C07C69/716 , C07C69/738 , C07C69/88 , C07D209/48 , C07D225/02 , C07D313/00 , C07D317/64 , C07D331/00 , C07D337/00 , C12N9/99 , A61K31/275 , A61K31/33 , A61K31/335 , A61K31/695
CPC classification number: C07D337/00 , A61K8/361 , A61K8/37 , A61K8/4906 , A61K8/4973 , A61K8/67 , A61K31/20 , A61K31/23 , A61K31/353 , A61K31/565 , A61K45/06 , A61K2800/782 , A61Q5/00 , A61Q19/00 , C07C53/21 , C07C57/52 , C07C57/56 , C07C61/16 , C07C61/40 , C07C69/63 , C07C69/65 , C07C69/675 , C07C69/716 , C07C69/738 , C07C69/88 , C07D209/48 , C07D225/02 , C07D313/00 , A61K2300/00
Abstract: Disclosed are a novel class of anti-androgenic compounds including saturated and unsaturated fatty acids, their derivatives, and synthetic analogs, according to the following formula: CH3-(CH2)a-(CR1R2CH=CH)b-(CH2)c-COOH, wherein R1 and R2 are each either hydrogen or a halogen; wherein a and c are integers from 0-9; wherein b is an integer from 1-6, provided that 12
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5.发明公开METHODS AND COMPOSITIONS FOR REGULATION OF 5-ALPHA REDUCTASE ACTIVITY 审中-公开ZUSAMMENSTELLUNGEN ZUR REGELIERUNG DES S-ALPHA-REDUKTASEAKTIVITÄT
公开(公告)号：EP1027045A4
公开(公告)日：2004-12-08
申请号：EP98956358
申请日：1998-10-30
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , HIIPAKKA RICHARD A
IPC: A61K31/00 , A61K31/047 , A61K31/075 , A61K31/12 , A61K31/135 , A61K31/165 , A61K31/235 , A61K31/24 , A61K31/35 , A61K31/352 , A61K31/353 , A61K31/44 , A61P3/04 , A61P13/08 , A61P17/00 , A61P17/14 , A61P35/00 , A61P43/00 , C07C49/105 , C07C49/248 , C07C49/255 , C07D311/30 , C07D311/36 , C07D311/62 , C07D311/82 , C07D311/92 , C07C49/76 , C07D311/04
CPC classification number: A61K31/44 , A61K31/00 , A61K31/075 , A61K31/12 , A61K31/35 , C07C49/248 , C07C49/255 , C07D311/62
Abstract: Compounds that inhibit 5alpha-reductase are provided. The compounds are used to treat prostate cancer, breast cancer, obesity, skin disorders and baldness.
Abstract translation: 提供抑制5α-还原酶的化合物。 该化合物用于治疗前列腺癌，乳腺癌，肥胖，皮肤病和秃发。
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Patent Agency Ranking
公开(公告)号：EP1189922A4
公开(公告)日：2002-08-14
申请号：EP00928431
申请日：2000-04-27
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , SONG CHING
IPC: A61K31/165 , A61K31/215 , A61K31/255 , A61K31/40 , A61K31/445 , A61K31/56 , A61K31/565 , A61K31/568 , A61K31/57 , A61K31/575 , A61K31/585 , A61P1/16 , A61P3/10 , A61P7/06 , A61P9/10 , A61P25/28 , A61P29/00 , A61P35/00 , A61P35/02 , A61P43/00 , C07J1/00 , C07J3/00 , C07J9/00 , C07J17/00 , C07J19/00 , C07J41/00 , C07J31/00
CPC classification number: C07J17/00 , A61K31/565 , A61K31/57 , A61K31/575 , A61K31/585 , C07J3/00 , C07J9/00 , C07J41/00
Abstract: Steroid derivatives of this invention interact with nuclear liver X receptor (LXR) and ubiquitous receptor (UR) and can be used to treat a variety of LXR- or UR-mediated disorders.
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公开(公告)号：EP1214070A4
公开(公告)日：2008-07-16
申请号：EP01910769
申请日：2001-02-15
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , HIIPAKKA RICHARD A , KAO YUNG-HSI
IPC: A61K31/045 , A61K31/05 , A61K31/175 , A61K31/351 , A61K31/353 , A61K31/397 , A61K31/50 , A61K31/549 , A61P3/10 , A61P29/00 , A61P35/00 , A61K31/35
CPC classification number: A61K31/549 , A61K31/045 , A61K31/05 , A61K31/175 , A61K31/351 , A61K31/353 , A61K31/397 , A61K31/50
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公开(公告)号：ZA200109793B
公开(公告)日：2003-02-28
申请号：ZA200109793
申请日：2001-11-28
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , SONG CHING
IPC: A61K20060101 , C07J20060101 , C07J , A61K
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公开(公告)号：CA1338667C
公开(公告)日：1996-10-22
申请号：CA614576
申请日：1989-09-29
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , PATAKI JOHN , HARVEY RONALD G
IPC: G01N33/50 , A61K31/00 , A61K31/045 , A61K31/05 , A61K31/12 , A61K31/22 , A61K31/565 , A61P5/26 , C07C22/04 , C07C33/18 , C07C35/42 , C07C35/44 , C07C39/12 , C07C39/17 , C07C45/51 , C07C49/115 , C07C49/225 , C07C49/657 , C07C49/665 , C07C49/747 , C07C49/753 , C07C49/792 , C07C69/00 , C07J1/00 , C07J63/00 , C07C33/00 , A61K31/56
Abstract: Disclosed are novel classes of anti-androgens including dihydrophenanthrene derivatives, their method of synthesis and their use in treating disorders associated with excessive androgenic activities. Preferred derivatives include 1-¢2-(9,10-dihydrophenanthryl)!-1-ethanol; 6,7,16,17-tetrahydro-15H-cyclopenta¢a!-phenanthren-17-ol; 1-¢2-(9(or 10)-methyl-9,10-dihydrophenanthryl)!-1-ethanol; 2-hydroxy-9,10-dihydrophenanthrene; 6,7,16,17-tetrahydro-15H-cyclopenta¢a!pehanthren-17-one; 4'-oxo-7,8-cyclohexeno-9,10-dihydrophenanthren-1-ol; and 4'-oxo-7,8-cyclohexeno-phenanthren-1-ol. Also provided by the invention are the corresponding derivatives wherein a free hydroxyl group has been replaced with an acetate or a propionate moiety.
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公开(公告)号：DK54791A
公开(公告)日：1991-05-22
申请号：DK54791
申请日：1991-03-26
Applicant: ARCH DEV CORP
Inventor： LIAO SHUTSUNG , PATAKI JOHN , HARVEY RONALD G
IPC: G01N33/50 , A61K31/00 , A61K31/045 , A61K31/05 , A61K31/12 , A61K31/22 , A61K31/565 , A61P5/26 , C07C22/04 , C07C33/18 , C07C35/42 , C07C35/44 , C07C39/12 , C07C39/17 , C07C45/51 , C07C49/115 , C07C49/225 , C07C49/657 , C07C49/665 , C07C49/747 , C07C49/753 , C07C49/792 , C07C69/00 , C07J1/00 , C07J63/00 , C07C33/34 , C07C33/36 , C07C69/157
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