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公开(公告)号:AT361910T
公开(公告)日:2007-06-15
申请号:AT03721841
申请日:2003-04-23
Applicant: AVENTIS PHARMA INC
Inventor: MERRIMAN GREGORY , WEINTRAUB PHILIP , SABOL JEFFREY , DHARANIPRAGADA RAMALINGA , HRIB NICHOLAS , JURCAK JOHN , GROSS ALEXANDRE , WHITELEY BRIAN , MUSICK KWON , KLEIN JOSEPH
IPC: C07D209/42 , A61K31/40 , A61K31/404 , A61K31/405 , A61K31/4436 , A61K31/4439 , A61K31/454 , A61K31/4545 , A61K31/506 , A61K31/5377 , A61P11/02 , A61P11/06 , A61P17/00 , A61P27/16 , A61P29/00 , A61P31/04 , A61P31/12 , A61P35/00 , A61P37/08 , A61P43/00 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D409/12 , C07D417/12 , C07D417/14
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公开(公告)号:AU2003225131A1
公开(公告)日:2003-11-10
申请号:AU2003225131
申请日:2003-04-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN G , GROSS ALEXANDRE , WHITELEY BRIAN , MUSICK KWON YON , KLEIN JOSEPH T , MERRIMAN GREGORY H , WEINTRAUB PHILIP M , SABOL JEFFREY S , DHARANIPRAGADA RAMALINGA , HRIB NICHOLAS J
IPC: A61K31/40 , A61K31/404 , A61K31/405 , A61K31/4436 , A61K31/4439 , A61K31/454 , A61K31/4545 , A61K31/506 , A61K31/5377 , A61P11/02 , A61P11/06 , A61P17/00 , A61P27/16 , A61P29/00 , A61P31/04 , A61P31/12 , A61P35/00 , A61P37/08 , A61P43/00 , C07D209/42 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D409/12 , C07D417/12 , C07D417/14
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公开(公告)号:CA2483091A1
公开(公告)日:2003-11-06
申请号:CA2483091
申请日:2003-04-23
Applicant: AVENTIS PHARMA INC
Inventor: HRIB NICHOLAS J , JURCAK JOHN G , GROSS ALEXANDRE , MUSICK KWON YON , WEINTRAUB PHILIP M , MERRIMAN GREGORY H , SABOL JEFFREY S , DHARANIPRAGADA RAMALINGA , KLEIN JOSEPH T , WHITELEY BRIAN
IPC: A61K31/40 , A61K31/404 , A61K31/405 , A61K31/4436 , A61K31/4439 , A61K31/454 , A61K31/4545 , A61K31/506 , A61K31/5377 , A61P11/02 , A61P11/06 , A61P17/00 , A61P27/16 , A61P29/00 , A61P31/04 , A61P31/12 , A61P35/00 , A61P37/08 , A61P43/00 , C07D209/42 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D409/12 , C07D417/12 , C07D413/14 , C07D403/14
Abstract: This inventions discloses and claims 3-substituted amino-1H-indole-2- carboxylic acid and 3-substituted amino-benzothiophene-2-carboxylic acid derivatives for use in treating allergy, asthma, rhinitis, dermatitis, B-cel l lymphomas, tumors and diseases associated with bacterial, rhinovirus or respiratory syncytial virus (RSV) infections. It has now been found that the compounds of this invention are capable of modulating T helper (Th) cells, Th1/Th2, and thereby capable of inhibiting the transcription of interieukin- 4(IL-4) message, IL-4 release or IL-4 production.
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公开(公告)号:AT468341T
公开(公告)日:2010-06-15
申请号:AT04779049
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN , BARRAGUE MATTHIEU , GILLESPY TIMOTHY , EDWARDS MICHAEL , MUSICK KWON , WEINTRAUB PHILIP , DU YAN , DHARANIPRAGADA RAMALINGA , PARKAR ASHFAQ
IPC: C07D495/04 , C07D519/00
Abstract: Thienopyrazoles of formula I, their preparation, pharmaceutical compositions comprising these compounds, and their pharmaceutical uses in the treatment of disease states capable of being modulated by the inhibition of the protein kinases, in particular interleukin-2 inducible tyrosine kinase (ITK).
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公开(公告)号:RS20060162A
公开(公告)日:2008-06-05
申请号:YUP20060162
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , DU YAN , DHARANIPRAGADA RAMALINGA , PARKAR ASHFAQ AHMED , WEINTRAUB PHILIP MARVIN
IPC: C07D495/04 , C07D519/00
Abstract: Tienopirazoli, njihova priprema, farmaceutski preparati koji sadrže ova jedinjenja, i njihova farmaceutsko upotreba u lečenju bolesnih stanja koja se mogu menjati inhibicijom protein kinaze, naročito tirozin kinaze koja se može indukovati interleukinom-2.
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公开(公告)号:DE60313769T2
公开(公告)日:2008-03-06
申请号:DE60313769
申请日:2003-04-23
Applicant: AVENTIS PHARMA INC
Inventor: MERRIMAN GREGORY H , WEINTRAUB PHILIP M , SABOL JEFFREY S , DHARANIPRAGADA RAMALINGA , HRIB NICHOLAS J , JURCAK JOHN G , GROSS ALEXANDRE , WHITELEY BRIAN , MUSICK KWON YON , KLEIN JOSEPH T
IPC: C07D209/42 , A61K31/40 , A61K31/404 , A61K31/405 , A61K31/4436 , A61K31/4439 , A61K31/454 , A61K31/4545 , A61K31/506 , A61K31/5377 , A61P11/02 , A61P11/06 , A61P17/00 , A61P27/16 , A61P29/00 , A61P31/04 , A61P31/12 , A61P35/00 , A61P37/08 , A61P43/00 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D409/12 , C07D417/12 , C07D417/14
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公开(公告)号:DE60313769D1
公开(公告)日:2007-06-21
申请号:DE60313769
申请日:2003-04-23
Applicant: AVENTIS PHARMA INC
Inventor: MERRIMAN GREGORY H , WEINTRAUB PHILIP M , SABOL JEFFREY S , DHARANIPRAGADA RAMALINGA , HRIB NICHOLAS J , JURCAK JOHN G , GROSS ALEXANDRE , WHITELEY BRIAN , MUSICK KWON YON , KLEIN JOSEPH T
IPC: C07D209/42 , A61K31/40 , A61K31/404 , A61K31/405 , A61K31/4436 , A61K31/4439 , A61K31/454 , A61K31/4545 , A61K31/506 , A61K31/5377 , A61P11/02 , A61P11/06 , A61P17/00 , A61P27/16 , A61P29/00 , A61P31/04 , A61P31/12 , A61P35/00 , A61P37/08 , A61P43/00 , C07D401/12 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D409/12 , C07D417/12 , C07D417/14
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