公开(公告)号：DE3842798A1

公开(公告)日：1990-06-21

申请号：DE3842798

申请日：1988-12-20

Applicant: HOECHST AG

Inventor： STARK HERBERT DR ,  SALBECK GERHARD DR ,  BONIN WERNER DR

IPC: A61K31/415 ,  A61P33/00 ,  C07D233/20 ,  C07D233/22 ,  C07D233/24

Abstract: The present invention relates to agents for systemic combating of ectoperasites in host animals, containing a compound of the formul I (I) in which R1 denotes hydrogen, (C1-C5)-alkyl, (C1-C3)-halogenoalkyl or halogen; R2 and R3 independently of one another denote (c1-C5)-alkyl, (C2-C5)-alkenyl, (C2-C5)-alkynyl, (C3-C7)-cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl, halogen, cyano, nitro, (C1-C5)-alkoxy, (C1 -C3)-alkoxy-C1-C3)-alkyl, (C1-C3)-halogenoalkoxy or (C1-C3)-alkylthio, or R2 and R3 together form a polymethylene chain having 2 to 5 carbon atoms: R4 denotes hydrogen, (c1-C10)-alkyl, (C2-C5)-alkenyl or (C3-C7)-cycloalkyl; R5 denotes hydrogen, (C1-C10)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)- cycloalkyl, (C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C hd 1-C3)-alkyl; X denotes oxygen, sulfur or an -NR6-group; and R6 denotes hydrogen, (C1-C5)-alkyl, (C3-C5)-alkenyl, C3-C5)-alkynyl, (C3-C7)-cycloalkyl, C3-C7)-cycloalkenyl, (C1-C3)-halogenoalkyl or (C1-C3)-alkoxy-(C1 -C3)-alkyl, or biologically tolerated acid addition salts thereof. The compounds of the formulas I are novel in some cases and are likewise included in the invention.

公开(公告)号：DE3040488A1

公开(公告)日：1982-06-03

申请号：DE3040488

申请日：1980-10-28

Applicant: HOECHST AG

Inventor： WELTER WOLFGANG DIPL CHEM DR ,  MILDENBERGER HILMAR DIPL CHEM ,  KNAUF WERNER ,  WALTERSDORFER ANNA ,  BONIN WERNER DR

IPC: C07C69/007 ,  A01N37/10 ,  A01N37/34 ,  A01N53/00 ,  A01N53/08 ,  C07C67/00 ,  C07C69/753 ,  C07C253/00 ,  C07C255/38 ,  C07C121/75 ,  C07C69/743 ,  C07C69/612 ,  C07C69/62 ,  C07C69/74 ,  A01N37/12

Abstract: Compounds of the formula wherein R1 denotes H, halogen, alkyl or CF3, R2 denotes H, halogen, alkyl or CF3, R3 denotes H, halogen, CN or alkyl, R4 denotes H, halogen, alkyl, phenyl or halogenophenyl, R5 denotes H, alkyl, alkynyl or CN and R6 denotes substituted dimethylcyclopropyl or 2-phenylisobutyl radicals, are effective insecticides and acaricides of the pyrethroid type.

公开(公告)号：DE3014097A1

公开(公告)日：1981-11-05

申请号：DE3014097

申请日：1980-04-12

Applicant: HOECHST AG

Inventor： SINHARAY AKHILESWAR DIPL CHEM ,  STAEHLER GERHARD DIPL CHEM DR ,  BONIN WERNER DR

IPC: A01N37/52 ,  C07C123/00 ,  A01N37/32

Abstract: Ni(2-Alkoxy carbonyl-2-cyano vinyl)-N1-methyl-N2- aryl-formamidines (I) are new, (where n is 0, 1, 2 or 3; R1 is H, halogen, 1-4C alkyl, 1-4C alkoxy, 1-4C alkylthio, CF3, NO2, CN, phenoxy, halophenoxy, phenylthio and/or halophenylthis; and R2 is 7-8C alkyl or 3-6C cycloalkyl). Prepn. consists of reacting N1-methyl N2 aryl formamidine (II) with alkoxymethylene cyano alkyl ester (IV), (where R3 is lower alkyl). (I) are pesticides, esp. insecticides and acaricides. They are particularly useful against ectoparasitic ticks.

公开(公告)号：DE2907090A1

公开(公告)日：1980-09-04

申请号：DE2907090

申请日：1979-02-23

Applicant: HOECHST AG

Inventor： SINHARAY AKHILESWAR DIPL CHEM ,  STAEHLER GERHARD DIPL CHEM DR ,  BONIN WERNER DR

IPC: A01N37/52 ,  C07C67/00 ,  C07C239/00 ,  C07C257/12 ,  C07C313/00 ,  C07C323/36 ,  C07C123/00 ,  A01N9/06

Abstract: New formamidine derivs. are cpds. of formula (I). In (I) n is 0, 1, 2 or 3; R1 is H, halogen, 1-4C alkyl, 1-4C alkoxy, 1-4C alkylthio, CF CF3, NO2, CN, phenoxy, halophenoxy, phenylthio and/or halophenylthio; and R2 is 1-6C alkyl or alkoxyalkyl. (I) have pesticidal properties and are partic. useful as insecticides and acaricides, esp. ectoparasiticides (e.g. against parasitic ticks). Effect of (I) is manifested as a strong inhibition of fertility and as 'detaching' effect particularly useful in host animals (e.g. cattle already infested by ticks.

公开(公告)号：DE4208254A1

公开(公告)日：1993-09-16

申请号：DE4208254

申请日：1992-03-14

Applicant: HOECHST AG

Inventor： SCHAPER WOLFGANG DR ,  PREUSS RAINER DR ,  SALBECK GERHARD DR ,  BRAUN PETER DR ,  KNAUF WERNER DR ,  SACHSE BURKHARD DR ,  WALTERSDORFER ANNA DR ,  KERN MANFRED DR ,  LUEMMEN PETER ,  BONIN WERNER DR

IPC: A01N43/54 ,  A01N43/90 ,  A01P3/00 ,  A01P7/02 ,  A01P7/04 ,  C07D239/34 ,  C07D239/42 ,  C07D239/46 ,  C07D239/52 ,  C07D239/60 ,  C07D239/88 ,  C07D239/94 ,  C07D401/12 ,  C07D405/12 ,  C07D491/048 ,  C07D495/04

Abstract: Substituted 4-amino and 4-alkoxy cycloalkylpyrimidines, a method of producing them and their use as pesticides and fungicides. The invention concerns compounds of formula (I) wherein R , R , R and Q are defined as per the description, X represents NH or oxygen, and E represents a bond or a 1-4 member C-chain; a method of producing them, agents containing them and their use in combatting vermin and as a fungicide.

公开(公告)号：DE3044010A1

公开(公告)日：1982-06-24

申请号：DE3044010

申请日：1980-11-22

Applicant: HOECHST AG

Inventor： HUETTELMAIER THOMAS DR ,  MILDENBERGER HILMAR DR ,  MATTERSTOCK KARL DR ,  BONIN WERNER DR ,  KNAUF WERNER DR ,  WALTERSDORFER ANNA DR

IPC: A01N37/10 ,  A01N37/38 ,  A01N53/00 ,  C07D213/65 ,  C07D277/68 ,  C07C121/75 ,  A01N43/06 ,  A61K31/22 ,  A61K31/275 ,  A61K31/34 ,  A61K31/38 ,  A61K31/425 ,  A61K31/44 ,  C07C69/612 ,  C07C69/635 ,  C07C69/747

Abstract: Aryl-substd. phenoxybenzyl carboxylic acid esters (I) are new: (where R is open-chain or cyclic 1-6C alkyl opt. mono- or polysubstd. by halogen, 1-3C alkyl, 3-6C cycloalkyl, 2-3C alkenyl or phenyl (opt. in turn substd. by halogen, 1-3C alkyl, 1-3C alkoxy, 1-3C alkylthio, halo-(1-2C alkyl), halo-(1-2C alkoxy), halo-(1,2C alkylthio) or methylenedioxy), or R is a spirocyclically linked 7-8C cycloalkenyl residue opt. fused with a benzene ring; R1 is halogen, CN, NO2, 1-6C alkyl, 3-6C cycloalkyl, 1-6C alkoxy, 1-6C alkylthio, halo-(1-2C alkyl) or methylenedioxy; R2 is an aromatic residue of formula (Ia), (Ib), (Ic) or (Id). R3 is H, halogen, CN, NO2, 1-6C alkyl, 1-6C alkoxy, 1-6C alkylthio or halo-(1-2C alkyl); or R2 and R3 together represent a saturated or unsaturated 4C carbon chain which may contain an N-atom instead of a -CH:group; X is H, CN, halogen, 1-6C alkyl, 1-6C haloalkyl, 3-6C cycloalkyl, 2-6C alkenyl or 2-6C alkynyl; R4 is halogen, CN, NO2, 1-6C alkyl, 3-6C cycloalkyl, phenyl, 1-6C alkoxy, 1-6C alkylthio, halo-(1-2C alkyl), halo-(1-2C alkoxy) or methylenedioxy; R5 is H, 1-6C alkyl or 3-6C cycloalkyl; Y is O, S, SO, SO2, OCH2, CH2O, CH2, SCH2, CH2S, CO, CH:CH, N(R5) or a direct chemical bond; Z is O or S; m is 0,1,2,3 or 4; and n is 0,1,2,3,4 or 5). The new cpds. are insecticides and acaricides. They are well tolerated by plants and are suitable for use in plant protection as well as in the stored products and hygiene sectors. In addition, the cpds. are useful in the veterinary sector against parasitic insects, mites and ticks.

公开(公告)号：DE2717437A1

公开(公告)日：1978-10-26

申请号：DE2717437

申请日：1977-04-20

Applicant: HOECHST AG

Inventor： SINHARAY AKHILESWAR DIPL CHEM ,  BONIN WERNER DR

IPC: A01N37/52 ,  C07C67/00 ,  C07C239/00 ,  C07C251/34 ,  C07C259/14 ,  C07C313/00 ,  C07C323/36 ,  C07C323/37 ,  C07C131/00 ,  A01N9/12 ,  A01N9/20

公开(公告)号：DE2334356A1

公开(公告)日：1975-01-30

申请号：DE2334356

申请日：1973-07-06

Applicant: HOECHST AG

Inventor： DRANSCH GUENTHER DR ,  HOERLEIN GERHARD DR ,  EMMEL LUDWIG DR ,  BONIN WERNER DR

IPC: A01N43/78 ,  C07D277/74 ,  C07D277/72 ,  A01N9/12

公开(公告)号：DE2229634A1

公开(公告)日：1974-01-31

申请号：DE2229634

申请日：1972-06-19

Applicant: HOECHST AG

Inventor： HOERLEIN GERHARD DR ,  SALBECK GERHARD DR ,  BONIN WERNER DR

IPC: C07F9/6553 ,  C07F9/6571 ,  A01N9/36

Abstract: Title cpds. of formula (I):- (where R1 = (1-4C) alkyl, (1-6C) O alkyl, or OPh; R2 = (1-6C) Oalkyl, NH2 opt. substd. by (1-6C) alkyl or (3-6C) NH alkenyl; R3-R7 = H or (1-4C) alkyl, at is not 3 gps being H; R8 and R9 = H, hal, (1-4C) alkyl, or (1-4C) Oalkyl; and X = O or S. are prepd. by condensing a 4-halothiochromanyl deriv. with an acid R1R2P(=X)SH.

公开(公告)号：DE3903404A1

公开(公告)日：1990-08-09

申请号：DE3903404

申请日：1989-02-06

Applicant: HOECHST AG

Inventor： KRATT GUENTER DR ,  SALBECK GERHARD DR ,  BONIN WERNER DR ,  DUEWEL DIETER DR

IPC: C07D239/557 ,  A01N43/54 ,  A01N57/36 ,  C07C217/84 ,  C07C265/12 ,  C07C323/36 ,  C07D239/54 ,  C07D239/545 ,  C07D239/553 ,  C07D239/60 ,  C07D239/62 ,  C07D319/12 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07F9/6584