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公开(公告)号:AT16282T
公开(公告)日:1985-11-15
申请号:AT82104542
申请日:1982-05-25
Applicant: HOECHST AG
Inventor: HERTENSTEIN ULRICH DR , MILDENBERGER HILMAR DR , SACHSE BURKHARD DR , HARTZ PETER DR
IPC: A01N43/653 , A01P3/00 , A61K31/41 , A61K31/415 , C07D231/12 , C07D233/56 , C07D233/58 , C07D233/60 , C07D233/64 , C07D233/68 , C07D233/91 , C07D235/06 , C07D249/08 , C07D521/00
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公开(公告)号:DE3121676A1
公开(公告)日:1982-12-16
申请号:DE3121676
申请日:1981-06-01
Applicant: HOECHST AG
Inventor: HERTENSTEIN ULRICH DIPL CHEM D , MILDENBERGER HILMAR DIPL CHEM , SACHSE BURKHARD , HARTZ PETER DR
IPC: A01N43/653 , A01P3/00 , A61K31/41 , A61K31/415 , C07D231/12 , C07D233/56 , C07D233/58 , C07D233/60 , C07D233/64 , C07D233/68 , C07D233/91 , C07D235/06 , C07D249/08 , C07D521/00 , C07D235/04 , C07D233/06
Abstract: Substituted ethanols of the general formula in which Ar1 is a carbocyclic or heterocyclic ring and Az is a triazolyl, benzimidazolyl, pyrazolyl or imidazolyl radical, are reacted with aryl hydrocarbons Ar2-H, in which Ar2 has the same meaning as Ar1, in the presence of an acidic catalyst, to give 1,1-diaryl-2-azolylethanes. The substances, which, apart from the imidazolyl derivatives, are new, can be used as biocides, in particular fungicides.
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公开(公告)号:DE3020500A1
公开(公告)日:1982-01-21
申请号:DE3020500
申请日:1980-05-30
Applicant: HOECHST AG
Inventor: EHRHARDT HEINZ DIPL CHEM DR , MILDENBERGER HILMAR DIPL CHEM , SACHSE BURKHARD , HARTZ PETER DR
IPC: A01N43/653 , C07D249/08 , C07D521/00 , A01N43/64
Abstract: 1-(3-Oxopropyl)-1,2,4-triazole derivs. (Ia) and their metal complexes with group Ib, IIb, IVb or VIII metals, as well as their salts and quaternisation prods (Ib) are new. In the formulae R is H, phenyl opt. substd. by halogen and/or 1-4C alkyl, or 1-18C alkyl opt. substd. by halogen, CN or a gp. OR1 in which R1 is 1-4C alkyl, phenyl or phenyl substd. by halogen or 1-4C alkyl; Z is 1- or 2-naphthyl or one of the groups (A), (B) or (C) in which R2 is H, halogen, NO2, CN, OH, 1-6C alkyl, 5-6C cycloalkyl, 1-6C alkoxy, 2-6C alkenyloxy, -(CH2)3-, -(CH2)4- or opt halo-substd. phenyl or phenoxy, R3 is H, 1-4C alkyl or halogen, n is 1, 2, 3 or 4 and m is 1, 2 or 3; R4 is H, 1-18C alkyl, oxoalkyl or alkenyl, or opt. halo-substd. phenacyl; and Y is the anion of an organic or inorganic acid. (I) are fungicides and bactericides esp. useful against rusts and mildews of plants, some cpds. (I) have systemic activity. (I) are also suitable for use in the technical sector, e.g. in timber preservatives, in paints, and as antifungal and antibacterial preservatives.
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公开(公告)号:DE3402166A1
公开(公告)日:1985-07-25
申请号:DE3402166
申请日:1984-01-23
Applicant: HOECHST AG
Inventor: SCHAPER WOLFGANG DR , BLUME ERNST DR , RAETHER WOLFGANG DR , DITTMAR WALTER DR , ALPERMANN HANS GEORG DR , SACHSE BURKHARD DR , HARTZ PETER DR
IPC: A01N43/50 , A01N43/653 , A61K31/41 , A61K31/415 , A61P25/00 , A61P25/24 , A61P25/26 , A61P31/04 , B27K3/38 , C07C45/60 , C07C49/84 , C07D233/60 , C07D249/08 , C07D295/096 , C07D295/185 , C07D333/00 , C07D401/06 , C07D401/12 , C07D401/14 , C07D405/06 , C07D409/06 , C07D521/00 , C09D5/14 , C07D403/10
Abstract: Azolyl derivatives of the formula I where A = CH or N; n = 2 - 12; Ar = aromatic; R = alkyl, alkenyl, alkynyl or benzyl; and Q = -S(O)1-3R or -OR (R = alkyl, cycloalkyl, alkenyl and some aromatics; R = saturated or unsaturated alkyl, cycloalkyl, cycloalkylalkyl, aromatics) and processes for their preparation are described. They are antimicrobial agents active against fungal infections. The intermediates of the formula VIIa have antidepressive properties.
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公开(公告)号:GR850174B
公开(公告)日:1985-05-13
申请号:GR850100174
申请日:1985-01-22
Applicant: HOECHST AG
Inventor: SCHAPER WOLFGANG DR , BLUME ERNST DR , RAETHER WOLFGANG DR , DITTMAR WALTER DR , ALPERMANN HANS GEORG DR , SACHSE DURKARD DR , HARTZ PETER DR
IPC: A01N43/50 , A01N43/653 , A61K31/41 , A61K31/415 , A61P25/00 , A61P25/24 , A61P25/26 , A61P31/04 , B27K3/38 , C07C45/60 , C07C49/84 , C07D233/60 , C07D249/08 , C07D295/096 , C07D295/185 , C07D333/00 , C07D401/06 , C07D401/12 , C07D401/14 , C07D405/06 , C07D409/06 , C07D521/00 , C09D5/14
Abstract: Azolyl derivatives of the formula I where A = CH or N; n = 2 - 12; Ar = aromatic; R = alkyl, alkenyl, alkynyl or benzyl; and Q = -S(O)1-3R or -OR (R = alkyl, cycloalkyl, alkenyl and some aromatics; R = saturated or unsaturated alkyl, cycloalkyl, cycloalkylalkyl, aromatics) and processes for their preparation are described. They are antimicrobial agents active against fungal infections. The intermediates of the formula VIIa have antidepressive properties.
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公开(公告)号:DE2918591A1
公开(公告)日:1980-11-20
申请号:DE2918591
申请日:1979-05-09
Applicant: HOECHST AG
Inventor: KNORR HARALD DIPL CHEM DR , MILDENBERGER HILMAR DIPL CHEM , SALBECK GERHARD DIPL CHEM DR , SACHSE BURGHARD , HARTZ PETER DR
IPC: A01N43/42 , A01N43/653 , A01N43/78 , A01N47/12 , A01N47/18 , A01N47/20 , C07D215/36 , C07D215/42 , C07D215/48 , C07D219/10 , C07D215/16 , A61K31/47 , C07D219/04
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公开(公告)号:DE2918590A1
公开(公告)日:1980-11-13
申请号:DE2918590
申请日:1979-05-09
Applicant: HOECHST AG
Inventor: KNORR HARALD DIPL CHEM DR , MILDENBERGER HILMAR DIPL CHEM , SALBECK GERHARD DIPL CHEM DR , SACHSE BURGHARD , HARTZ PETER DR
IPC: A01N43/42 , A01N47/06 , C07D215/18 , C07D215/22 , C07D215/233 , C07D215/36 , C07D215/48 , C07D219/04 , C07D215/16 , A61K31/47
Abstract: derivs. of formula (I) are new. R1 is H, 1-12C alkyl, benzyl, phenyl (opt. substd. by 1 or 2 Cl or by CF3 or 1-4C alkyl), -16C alkoxy-carbonyl, aryl-aminocarbonyl (in which aryl is opt. substd. by halogen, CF3, NO2 or 1-5C alkyl) N-alkyl-aryl aminocarbonyl (where alkyl has 1-3C and aryl is opt. substd. by halogen, CF3, or 1-4C alkyl), aminocarbonyl, 1-10C alkylaminocarbonyl, or di-(1-10C) alkylaminocarbonyl; R2 is H, opt. branched 1-12C alkyl, benzyl, phenyl (opt. substd. by 2 Cl or CF3, NO2 or 1-4C alkyl), 1-6C alkoxycarbonyl, phenylthio morpholino, piperidino, arylamino (in which aryl is substd. by halogen or 1-4C alkyl), di (1-6C) alkylaminomethyl morpholinomethyl or piperidinomethy; or R1 and R2 are together -CH2CH2CH2CH2-;R3 is H or 1-4C alkyl;R4 is H or opt. branched 1-12C alkyl;R5 is H or 1-4C alkyl;R6 is H or 1-6C alkyl;A is SH, Cl or -OR7;R7 is -SO2NR8R9 or -COOR10;R8 is opt. branched 1-10C alkyl, Ph or H and R9 is H or opt. branched 1-10C alkyl, or R8 and R9 together are -(CH2)-n, -CH2CH2OCH2CH2- or -CH2CH2N-(Me)CH2CH2- where n = 4 or 5; and R10 is 1-10C alkyl or Ph opt. substd. by halogen or NO2. (I) are biocides with a relatively broad spectrum of activity against fungi and bacteria, and are esp. useful for treating diseases of leaves. (I) are effective e.g. against phytopathogenic fungi and bacteria such as Botrytic cinerea and Xanthomonas oryltae, as well as against non-phytopathogenic fungi and bacteria such as Penicillium funiculosum and E. coli.
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公开(公告)号:MY8700827A
公开(公告)日:1987-12-31
申请号:MY8700827
申请日:1987-12-30
Applicant: HOECHST AG
Inventor: HERTENSTEIN ULRICH DR , MILDENBERGER HILMAR DR , SACHSE BURKHARD DR , HARTZ PETER DR
IPC: A01N43/653 , A01P3/00 , A61K31/41 , A61K31/415 , C07D231/12 , C07D233/56 , C07D233/58 , C07D233/60 , C07D233/64 , C07D233/68 , C07D233/91 , C07D235/06 , C07D249/08 , C07D521/00
Abstract: Substituted ethanols of the general formula in which Ar1 is a carbocyclic or heterocyclic ring and Az is a triazolyl, benzimidazolyl, pyrazolyl or imidazolyl radical, are reacted with aryl hydrocarbons Ar2-H, in which Ar2 has the same meaning as Ar1, in the presence of an acidic catalyst, to give 1,1-diaryl-2-azolylethanes. The substances, which, apart from the imidazolyl derivatives, are new, can be used as biocides, in particular fungicides.
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公开(公告)号:DE3527334A1
公开(公告)日:1987-02-05
申请号:DE3527334
申请日:1985-07-31
Applicant: HOECHST AG
Inventor: SCHALLER RAINER DR , MILDENBERGER HILMAR DR , HANDTE REINHARD DR , HARTZ PETER DR , SACHSE BURKHARD DR
IPC: A01N35/04 , A01N37/12 , A01N37/34 , A01N37/36 , A01N37/38 , A01N37/42 , A01N43/06 , A01N43/10 , A01N43/40 , C07C323/25 , C07D213/34 , C07D295/088 , C07D295/10 , C07D333/18 , C07D333/22 , C09D5/14 , C09D15/00 , C10M129/24 , C07C149/273 , C07C149/34 , C07D265/30
Abstract: 1,2-Diarylpropanones of the formula (I) in which Ar denotes 1- or 2-naphthyl, (substituted) thienyl, (substituted) furyl, (substituted) pyridyl or (substituted) phenyl, Ar denotes a radical as indicated for Ar with the exception of (substituted) pyridyl, Z denotes O or S(O)r, R denotes H or alkyl, p denotes 0, 1, 2, 3 or 4 and Q denotes a radical of the formulae -OR , -SR , -NR R , -CHR R or -COR , in which R denotes H, (substituted) alkyl, cycloalkyl or substituted phenyl, R and R denote alkyl, alkenyl, alkynyl, (substituted) cycloalkyl or (substituted) aryl, (substituted) aryl(C1-C2)alkyl, or one of the radicals R and R denotes a 5- to 7-membered (substituted) heterocycle having 1 to 3 hetero atoms, or R and R together with the nitrogen atom to which they are bonded denote a 5- to 7-membered (substituted) heterocycle having 1 to 3 hetero atoms, R and R denote H, alkyl, alkoxy, (substituted) phenyl, or (substituted) phenoxy, or R and R together with the C atom to which they are bonded denote a 5- to 9-membered saturated or unsaturated hydrocarbon ring in which 1 to 3 ring members can be replaced by hetero atoms and which can be substituted by one to three alkyl groups, and R denotes alkyl, alkoxy or a radical as indicated for Ar , have advantageous fungicidal activities, in particular against fungal pests in agriculture.
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公开(公告)号:DE2948095A1
公开(公告)日:1981-06-19
申请号:DE2948095
申请日:1979-11-29
Applicant: HOECHST AG
Inventor: BAUER KLAUS DR , BIERINGER HERMANN DR , FRISCH GERHARD DIPL CHEM DR , GORBACH SIEGBERT DIPL CHEM DR , HARTZ PETER DR , HOERLEIN GERHARD DIPL CHEM DR , KNORR HARALD DIPL CHEM DR
IPC: A01N39/02 , A01N43/40 , A01N43/52 , A01N43/54 , A01N43/74 , A01N47/44 , C07C233/46 , C07C255/32 , C07D213/64 , C07D213/643 , C07D239/34 , C07D263/56 , C07D263/58 , C07D277/62 , C07D277/64 , C07D277/68 , C07C103/48 , A01N37/18 , C07C103/46 , C07C121/66 , C07C149/20 , C07C149/23
Abstract: Amides of formula (I) are new, (where A is a (R)n-substd. phenyl, 2-pyridyl, 2-pyrimidyl, benzoxazol-2-yl, benzothiazol-2-yl or 1-methylbenzimidazol-2-yl gp.; where R is halogen, CF3, CN, NO2, halomethoxy or Me and n is 0-3. X is O, OCH2 or CH2. R2 is H, halogen, CF3 or Me. R1 is Me or methoxymethyl. B is a direct bond, CH2CH2 or CH=CH. R3 is H and E is 1-3C alkylene opt. substd. by a Ph, PhCH2, MeS, CONH2 or guanidyl gp. and/or by one or two 1-4C alkyl gps., or R3 is a 1,3-propylene gp. linked to E and E is CH. G is CN, COOH or COOR4, where R4 is 1-4C alkyl; with the proviso that E-G is not CH2CH2CN, CH(Me)COOR4 or CH(Et)COOR4 when A is (R)n-substd. phenyl, X is O or CH2, R1 is Me, B is a direct bond and R3 is H). (I) are useful as (a) herbicides, esp. for selective control of annual and perennial grasses in wheat, sugar beet, soya and cotton crops, (b) agricultural fungicides, esp. active against Botrytis cinerea, Piricularia oryzae and Pythium ultimum, and (c) technical biocides with fungicidal, bactericidal and algicidal activity.
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