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    4.
    发明专利
    未知

    公开(公告)号：AT337317T

    公开(公告)日：2006-09-15

    申请号：AT03767889

    申请日：2003-11-04

    Applicant: SERVIER LAB

    Inventor： RAULT SYLVAIN ,  LANCELOT JEAN-CHARLES ,  KOPP MARINA ,  CAIGNARD DANIEL-HENRI ,  PFEIFFER BRUNO ,  RENARD PIERRE ,  BIZOT-ESPIARD JEAN-GUY

    IPC: A61P3/04 ,  A61P3/06 ,  A61P3/10 ,  A61P9/10 ,  C07D471/04 ,  A61K31/44 ,  C07D235/00 ,  C07D221/00

    Abstract: Imidazopyridine derivatives (I) are new. Imidazopyridine derivatives of formula (I), their enantiomers, diastereoisomers, and their salts with acids and bases are new. R1 = H, halogen, alkyl, polyhaloalkyl, CN, NO2, hydroxycarbonyl, alkoxycarbonyl, aminocarbonyl, or dialkylaminocarbonyl; R2 = H, alkyl, aryl (optionally substituted), heteroaryl (optionally substituted) or a group of formula R20-C(X)-; R20 = alkyl, alkoxy, amino, alkylamino, dialkylamino, aryl (optionally substituted), or heteroaryl (optionally substituted); X = O, S, or NR21; R21, R3 = H or alkyl; n = 1-6; and N = pyrido ring with the N atom in the 1, 2, 3, or 4 positions. Alkyl and alkoxy groups have 1-6 C atoms, aryl is phenyl or naphthyl, polyhaloalkyl groups having 1-3 C atoms and 1-7 halogen atoms, heteroaryl groups may be mono or bicyclic of 5 - 11 ring atoms, at least one ring being aromatic, and having 2 or 3 heteroatoms (O, N, S) and may be substituted by 1-3 alkyl groups. Optional substituents on aryl groups may be 1 or 2 substituents selected from halogens, alkyl, alkoxy, polyhaloalkyl, hydroxy, CN, NO2, amino, alkylamino, dialkylamino, carboxyl, amido, and -COO-alkyl groups, and heteroaryl groups having a non-aromatic ring may be further substituted on this non-aromatic ring by oxo.

    5.
    发明专利
    未知

    公开(公告)号：DK1560826T3

    公开(公告)日：2006-08-14

    申请号：DK03767886

    申请日：2003-11-04

    Applicant: SERVIER LAB

    Inventor： RENARD PIERRE ,  RAULT SYLVAIN ,  KOPP MARINA ,  CAIGNARD DANIEL-HENRI ,  LANCELOT JEAN-CHARLES ,  PFEIFFER BUNO

    IPC: C07D471/04 ,  A61K31/505 ,  A61P3/04 ,  A61P3/10 ,  A61P9/10 ,  A61P9/12 ,  A61P19/02 ,  A61P35/00

    Abstract: Pyridopyrimidone derivatives (I), their enantiomers, diastereoisomers, tautomers, and their salts with acids and bases are new. Pyridopyrimidone derivatives of formula (I), their enantiomers, diastereoisomers, tautomers, and their salts with acids and bases are new. R1, R2 = H or alkyl; R3 = halogen, alkoxy, aryl (optionally substituted by 1-3 R33), or NR'1R'2; R'1, R'2 = H, alkyl, or R'1-N-R'2 is a heterocycle; R4 = H or NR''1R''2; R''1, R''2 = H or alkyl; R1+R2, R'1+R'2, R''1+R''2 = mono or bicyclic of 5 - 11 C heterocycle optionally containing a further 1 or 2 heteroatoms (O, N, S), optionally substituted by 1-3 alkyl groups; R33 = halogens, alkyl, alkoxy, polyhaloalkyl (containing 1 - 3 C atoms and 1 - 7 halogen atoms) and hydroxy; provided that: (1) alkyl and alkoxy groups have 1 - 8 C atoms, aryl is phenyl or naphthyl; and An Independent claim is also included for the preparation of (I).

    6.
    发明专利
    未知

    公开(公告)号：BR0315996A

    公开(公告)日：2005-09-27

    申请号：BR0315996

    申请日：2003-11-04

    Applicant: SERVIER LAB

    Inventor： RAULT SYLVAIN ,  LEFLEMME NICOLAS ,  DALLEMAGNE PATRICK ,  LESTAGE PIERRE ,  LOCKHART BRIAN ,  DANOBER LAURENCE ,  PFEIFFER BRUNO ,  RENARD PIERRE

    IPC: A61P25/04 ,  A61P25/28 ,  C07D211/86 ,  C07D401/04 ,  C07D409/04 ,  A61K31/44

    Abstract: 2,3-Dihydro-4(1H)-pyridinone derivatives (I), their enantiomers, diastereoisomers, and acid addition salts are new. 2,3-Dihydro-4(1H)-pyridinone derivatives (I), their enantiomers, diastereoisomers, and acid addition salts are new. R1 = H, 1-6C alkyl, acyl, alkoxycarbonyl, aralkyl aralkoxycarbonyl, or trifluoroacetyl; R2 = 1-6C alkyl; X = O or NOR3; R3 = H, 1-6C alkyl (optionally substituted by OH, amino, alkylamino, dialkylamino and alkoxy); Ar = aryl or heteroaryl where aryl groups may be phenyl, biphenylyl, naphthyl, or tetrahydronaphthyl, all of which are optionally substituted by halogens, alkyl, OH, alkoxy, trihalomethyl, nitro, amino, alkylamino and dialkylamino groups, and heteroaryl groups may be mono or bicyclic and may be substituted by halogens, alkyl, OH, alkoxy, trihalomethyl, nitro, amino, alkylamino and dialkylamino groups.

    8.
    发明专利
    未知

    公开(公告)号：FR2846656B1

    公开(公告)日：2004-12-24

    申请号：FR0213802

    申请日：2002-11-05

    Applicant: SERVIER LAB

    Inventor： RAULT SYLVAIN ,  LANCELOT JEAN CHARLES ,  KOPP MARINA ,  CAIGNARD DANIEL HENRI ,  PFEIFFER BRUNO ,  RENARD PIERRE ,  BIZOT ESPIARD JEAN GUY

    IPC: A61P3/04 ,  A61P3/06 ,  A61P3/10 ,  A61P9/10 ,  C07D471/04 ,  A61K31/437

    Abstract: Imidazopyridine derivatives (I) are new. Imidazopyridine derivatives of formula (I), their enantiomers, diastereoisomers, and their salts with acids and bases are new. R1 = H, halogen, alkyl, polyhaloalkyl, CN, NO2, hydroxycarbonyl, alkoxycarbonyl, aminocarbonyl, or dialkylaminocarbonyl; R2 = H, alkyl, aryl (optionally substituted), heteroaryl (optionally substituted) or a group of formula R20-C(X)-; R20 = alkyl, alkoxy, amino, alkylamino, dialkylamino, aryl (optionally substituted), or heteroaryl (optionally substituted); X = O, S, or NR21; R21, R3 = H or alkyl; n = 1-6; and N = pyrido ring with the N atom in the 1, 2, 3, or 4 positions. Alkyl and alkoxy groups have 1-6 C atoms, aryl is phenyl or naphthyl, polyhaloalkyl groups having 1-3 C atoms and 1-7 halogen atoms, heteroaryl groups may be mono or bicyclic of 5 - 11 ring atoms, at least one ring being aromatic, and having 2 or 3 heteroatoms (O, N, S) and may be substituted by 1-3 alkyl groups. Optional substituents on aryl groups may be 1 or 2 substituents selected from halogens, alkyl, alkoxy, polyhaloalkyl, hydroxy, CN, NO2, amino, alkylamino, dialkylamino, carboxyl, amido, and -COO-alkyl groups, and heteroaryl groups having a non-aromatic ring may be further substituted on this non-aromatic ring by oxo.

    IMIDAZOPYRIDINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
    10.
    发明专利
    IMIDAZOPYRIDINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME 未知

    公开(公告)号：AU2003292323A1

    公开(公告)日：2004-06-03

    申请号：AU2003292323

    申请日：2003-11-04

    Applicant: SERVIER LAB

    Inventor： BIZOT-ESPIARD JEAN-GUY ,  RAULT SYLVAIN ,  LANCELOT JEAN-CHARLES ,  KOPP MARINA ,  CAIGNARD DANIEL-HENRI ,  PFEIFFER BRUNO ,  RENARD PIERRE

    IPC: A61P3/04 ,  A61P3/06 ,  A61P3/10 ,  A61P9/10 ,  C07D471/04 ,  A61K31/44

    Abstract: Imidazopyridine derivatives (I) are new. Imidazopyridine derivatives of formula (I), their enantiomers, diastereoisomers, and their salts with acids and bases are new. R1 = H, halogen, alkyl, polyhaloalkyl, CN, NO2, hydroxycarbonyl, alkoxycarbonyl, aminocarbonyl, or dialkylaminocarbonyl; R2 = H, alkyl, aryl (optionally substituted), heteroaryl (optionally substituted) or a group of formula R20-C(X)-; R20 = alkyl, alkoxy, amino, alkylamino, dialkylamino, aryl (optionally substituted), or heteroaryl (optionally substituted); X = O, S, or NR21; R21, R3 = H or alkyl; n = 1-6; and N = pyrido ring with the N atom in the 1, 2, 3, or 4 positions. Alkyl and alkoxy groups have 1-6 C atoms, aryl is phenyl or naphthyl, polyhaloalkyl groups having 1-3 C atoms and 1-7 halogen atoms, heteroaryl groups may be mono or bicyclic of 5 - 11 ring atoms, at least one ring being aromatic, and having 2 or 3 heteroatoms (O, N, S) and may be substituted by 1-3 alkyl groups. Optional substituents on aryl groups may be 1 or 2 substituents selected from halogens, alkyl, alkoxy, polyhaloalkyl, hydroxy, CN, NO2, amino, alkylamino, dialkylamino, carboxyl, amido, and -COO-alkyl groups, and heteroaryl groups having a non-aromatic ring may be further substituted on this non-aromatic ring by oxo.

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