-
公开(公告)号:MY162396A
公开(公告)日:2017-06-15
申请号:MYPI2013000767
申请日:2011-09-02
Applicant: UCB PHARMA SA
Inventor: PARTON ANDREW HARRY , ALI MEZHER HUSSEIN , BROOKINGS DNIEL CHRISTOPHER , BROWN JULIEN ALISTAR , FORD DANIEL JAMES , FRANKLIN RICHARD JEREMY , LANGHAM BARRY JOHN , NEUSS JUDI CHARLOTTE , QUINCEY JOANNA RACHEL
IPC: C07D471/04 , A61K31/519 , A61P9/00 , A61P25/28 , A61P29/00
Abstract: A SERIES OF QUINOLONE AND QUINOXALINE DERIVATIVES COMPRISING A FLUORINATED ETHYL SIDE-CHAIN, BEING SELECTIVE INHIBITORS OF PI3 KINASE ENZYMES, ARE ACCORDINGLY OF BENEFIT IN MEDICINE, FOR EXAMPLE IN THE TREATMENT OF INFLAMMATORY, AUTOIMMUNE, CARDIOVASCULAR, NEURODEGENERATIVE, METABOLIC, ONCOLOGICAL, NOCICEPTIVE OR OPHTHALMIC CONDITIONS.