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公开(公告)号:WO2013006634A3
公开(公告)日:2013-05-10
申请号:PCT/US2012045431
申请日:2012-07-03
Applicant: VERTEX PHARMA , TANOURY GERALD J , JUNG YOUNG CHUN , MAGDZIAK DEREK , LOOKER ADAM , KLINE BILLIE J , JURCIK VACLAV , DOMINGUEZ OLMO BEATRIZ
Inventor: TANOURY GERALD J , JUNG YOUNG CHUN , MAGDZIAK DEREK , LOOKER ADAM , KLINE BILLIE J , JURCIK VACLAV , DOMINGUEZ OLMO BEATRIZ
IPC: C07D471/04
CPC classification number: C07D471/04 , C07B2200/13 , C07D239/42 , C07F5/025 , C07F5/04
Abstract: The present invention relates to processes and intermediates for the preparation of compounds useful as inhibitors of Janus kinases (JAK).
Abstract translation: 本发明涉及制备可用作Janus激酶(JAK)抑制剂的化合物的方法和中间体。
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公开(公告)号:CA2839937A1
公开(公告)日:2013-01-10
申请号:CA2839937
申请日:2012-07-03
Applicant: VERTEX PHARMA
Inventor: TANOURY GERALD J , JUNG YOUNG CHUN , MAGDZIAK DEREK , LOOKER ADAM , KLINE BILLIE J , JURCIK VACLAV , DOMINGUEZ OLMO BEATRIZ
IPC: C07D471/04
Abstract: The present invention relates to processes and intermediates for the preparation of compounds useful as inhibitors of Janus kinases (JAK).
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公开(公告)号:AU2012279046B2
公开(公告)日:2017-08-31
申请号:AU2012279046
申请日:2012-07-03
Applicant: VERTEX PHARMA
Inventor: TANOURY GERALD J , JUNG YOUNG CHUN , MAGDZIAK DEREK , LOOKER ADAM , KLINE BILLIE J , JURCIK VACLAV , DOMINGUEZ OLMO BEATRIZ
IPC: C07D471/04
Abstract: The present invention relates to processes and intermediates for the preparation of compounds useful as inhibitors of Janus kinases (JAK).
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公开(公告)号:CA2839937C
公开(公告)日:2020-11-03
申请号:CA2839937
申请日:2012-07-03
Applicant: VERTEX PHARMA
Inventor: TANOURY GERALD J , JUNG YOUNG CHUN , MAGDZIAK DEREK , LOOKER ADAM , KLINE BILLIE J , JURCIK VACLAV , DOMINGUEZ OLMO BEATRIZ
IPC: C07D471/04
Abstract: The present invention relates to processes and intermediate for the preparation of compounds of Formula l (see formula I) useful as inhibitors of Janus Kinases (JAK).
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公开(公告)号:AU2012279046A1
公开(公告)日:2014-01-23
申请号:AU2012279046
申请日:2012-07-03
Applicant: VERTEX PHARMA
Inventor: TANOURY GERALD J , JUNG YOUNG CHUN , MAGDZIAK DEREK , LOOKER ADAM , KLINE BILLIE J , JURCIK VACLAV , DOMINGUEZ OLMO BEATRIZ
IPC: C07D471/04
Abstract: The present invention relates to processes and intermediates for the preparation of compounds useful as inhibitors of Janus kinases (JAK).
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公开(公告)号:ZA201400049B
公开(公告)日:2015-04-29
申请号:ZA201400049
申请日:2014-01-06
Applicant: VERTEX PHARMA
Inventor: TANOIRY GERALD J , JUNG YOUNG CHUN , MAGDZIAK DEREK , LOOKER ADAM , KLINE BILLIE J , JURCIK VACLAV , DOMINGUEZ OLMO BEATRIZ
Abstract: The present invention relates to processes and intermediates for the preparation of compounds useful as inhibitors of Janus kinases (JAK).
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