公开(公告)号：AU2004266783A1

公开(公告)日：2005-03-03

申请号：AU2004266783

申请日：2004-07-03

Applicant: BASF AG

Inventor： SCHWOGLER ANJA ,  GRAMMENOS WASSILIOS ,  SCHOFL ULRICH ,  WAGNER OLIVER ,  SCHAFER PETER ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED ,  BLASCO JORDI TORMO I ,  MULLER BERND ,  BLETTNER CARSTEN ,  RHEINHEIMER JOACHIM ,  STIERL REINHARD ,  SCHIEWECK FRANK ,  GEWEHR MARKUS ,  GYPSER ANDREAS ,  SCHERER MARIA

IPC: C07D239/42

Abstract: The invention relates to 2-substituted pyrimidines of the formula I in which the index n and these substituents R 1 , R 2 and R 3 are as defined in the description and R 4 is as defined below: R 4 corresponds to one of the formulae where R a is hydrogen, C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 3 -C 6 -cycloalkyl or C 1 -C 4 -alkoxy and R 5 is hydrogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 1 -C 4 -alkyloxy-C 1 -C 2 -alkyl, phenyl-C 1 -C 2 -alkyl or phenyloxy-C 1 -C 2 -alkyl, to processes for preparing these compounds, to compositions comprising these compounds and to their use as pesticides.

公开(公告)号：ZA200400914B

公开(公告)日：2005-02-04

申请号：ZA200400914

申请日：2004-02-04

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  LORENZ GISELA ,  MUELLER BERND ,  RACK MICHAEL ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SAUTER HUBERT ,  SCHIEWECK FRANK ,  SCHAEFER PETER ,  STIERL REINHARD ,  STRATHMANN SIEGFIED ,  BLASCO JORDI TORMO I

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N

Abstract: 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines (I) are new. 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines of formula (I) are new. [Image] n : 0-5; R : halo, CN, OH or OCN, or alkyl, alkenyl, alkynyl, T', haloalkenyl, OT, alkenyloxy, alkynyloxy, OT', cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, CONH 2, mono- or dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); T : 1-6C alkyl; T' : 1-6C haloalkyl; Het : 5-10 membered, saturated, partially unsaturated or aromatic heterocycle containing 1-4 of O, N and/or S heteroatoms; R 11-10C alkyl, alkenyl, alkynyl, 3-12C cycloalkyl, 3-10C cycloalkenyl, phenyl, naphthyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); R ahalo, CN, NO 2, OH, T, T', COT, cycloalkyl, OT, OT', COOT, NHT, NT 2, 2-6C alkenyl, 2-6C alkenyloxy, 3-6C alkynyloxy, alkoximino, alkenyloximino, alkynyloximino, aralkoximino, alkynyl, alkynyloxycarbonyl, phenyl, naphthyl or Het (where all aliphatic, alicyclic or aromatic groups are optionally partially or completely halogenated and optionally substituted by 1-3 R aand/or 1-3 R c); R bhalo, CN, NO 2, OH, SH, NH 2, COOH, CONH 2, CSNH 2, T, T', 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, OT, OT', ST, NHT, NT 2, CHO, COT, SO 2T, SOT, COOT, OCOT, CONHT, CONT 2, CSNHT or CSNT 2; R ccycloalkyl, -O-cycloalkyl, heterocyclyl, -O-heterocyclyl, aryl, -O-aryl, -S-aryl, -O-T-aryl, -T-aryl, heteroaryl, -O-heteroaryl or -S-heteroaryl (where cycloalkyl or heterocyclyl rings are 3-10 membered, aryl rings are preferably 6-10 membered and heteroaryl rings are preferably 5-6 membered; and all rings are optionally partially or completely halogenated and optionally substituted by alkyl or haloalkyl); and R 21-4C alkyl, 2-4C alkynyl or 2-4C alkynyl (all optionally substituted by halo, CN, NO 2, OMe, OEt or 1-4C alkoxycarbonyl; Unless specified otherwise alkyl moieties have 1-8C, alkenyl or alkynyl moieties 2-10C and cycloalkyl or cycloalkenyl moieties 3-6C. Independent claims are also included for: (1) preparation of (I); and (2) dicarbonyl compound intermediates of formula (III), provided that n is not 0 and R 1and R 2are not both Me. [Image] ACTIVITY : Fungicide. 7-Cyclohexyl-5-methyl-6-(2-chloro-6-fluorophenyl)-1,2,4-triazolo[1,5-a]pyrimidine (Ia) at a concentration of 63 ppm gave at least 90 % protection of tomato plants against Alternaria solani. MECHANISM OF ACTION : None given.

公开(公告)号：MA27198A1

公开(公告)日：2005-01-03

申请号：MA27909

申请日：2004-10-15

Applicant: BASF AG

Inventor： SCHOEFL ULRICH ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHILEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C255/57 ,  C07D487/04

公开(公告)号：HU0401746A2

公开(公告)日：2004-12-28

申请号：HU0401746

申请日：2002-07-08

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

公开(公告)号：DE60015817D1

公开(公告)日：2004-12-16

申请号：DE60015817

申请日：2000-12-11

Applicant: BASF AG

Inventor： PEES KLAUS-JUERGEN ,  TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  CULLMANN DR ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL DR

IPC: A01N43/90 ,  C07D487/04 ,  A01N43/56

公开(公告)号：AT275340T

公开(公告)日：2004-09-15

申请号：AT01964978

申请日：2001-06-13

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  GOETZ NORBERT ,  VOLK THORSTEN ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

IPC: A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22 ,  C07C233/69

Abstract: Use of phenethylacrylamides of the formula I:in which the substituents have the following meanings:X is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and -O-C(R ,R )-C=C-R ;R ,R and R have the meanings given in the description;m,n independently of one another are 1 to 4, it being possible for the radicals X or Y to be different if m or n is greater than 1;Y is halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl;R ,R independently of one another are hydrogen, halogen, alkyl, alkoxy, haloalkoxy and CF3;R ,R ,R ,R independently of one another are hydrogen, halogen, alkyl, alkoxy, orR and R together form a cyclopropyl ring, it being possible for the C-R - and C-R bonds can be in the E- or Z-position relative to each other;for controlling phytopathogenic fungal pests, novel phenethylacrylamides, their preparation, and compositions comprising them.

公开(公告)号：AU2003293894A1

公开(公告)日：2004-07-09

申请号：AU2003293894

申请日：2003-12-16

Applicant: BASF AG

Inventor： GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD ,  MULLER BERND ,  BLASCO JORDI TORMO I

IPC: C07D487/04 ,  A01N43/653

Abstract: Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R 1 is C 1 -C 10 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -alkynyl, C 3 -C 10 -cycloalkyl, C 3 -C 10 -cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R 2 is C 1 -C 4 -alkyl which may be substituted by halogen, cyano, nitro or C 1 -C 2 -alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SO m -R x , NR x R y or NR x -(C-O)-R y ; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

公开(公告)号：EE200200685A

公开(公告)日：2004-06-15

申请号：EEP200200685

申请日：2001-06-13

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  MUELLER BERND ,  BLASCO JORDI TORMO I ,  GOETZ NORBERT ,  VOLK THORSTEN ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

IPC: A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22 ,  C07C233/69

Abstract: Use of phenethylacrylamides of the formula I:in which the substituents have the following meanings:X is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and -O-C(R ,R )-C=C-R ;R ,R and R have the meanings given in the description;m,n independently of one another are 1 to 4, it being possible for the radicals X or Y to be different if m or n is greater than 1;Y is halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl;R ,R independently of one another are hydrogen, halogen, alkyl, alkoxy, haloalkoxy and CF3;R ,R ,R ,R independently of one another are hydrogen, halogen, alkyl, alkoxy, orR and R together form a cyclopropyl ring, it being possible for the C-R - and C-R bonds can be in the E- or Z-position relative to each other;for controlling phytopathogenic fungal pests, novel phenethylacrylamides, their preparation, and compositions comprising them.

公开(公告)号：AU2003283348A1

公开(公告)日：2004-06-07

申请号：AU2003283348

申请日：2003-11-04

Applicant: BASF AG

Inventor： BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04

Abstract: The invention relates to 5-alkyl-7-aminotriazolopyrimidines of the formula (I) and to the salts thereof. In said formula substituents have the following meanings: R1 and R2 each is a hydrogen atom or a group of alkyl, alcenyl, haloalkyl, cycloalky, phenyl or naphtyle, saturated, unstaturated or aromatic heterocycle having from five to six members which contain from one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can from together with a connecting them nitrogen atom a cycle of 5 to 6 members containing from one to four nitrogen atoms or from one to three nitrogen atoms and one sulfur or oxygen atom, R3 is a cycloalkyl or bicycloalkyl group, R1, R2 and R3 can be substituted in conformity with a description, and X is an alkyl or alkyl halide group. The inventive methods and intermediary products necessary for producing said compounds, agents containing them and the use therefore for fighting against harmful mushroom are also disclosed.

公开(公告)号：AU2003214116A1

公开(公告)日：2003-09-22

申请号：AU2003214116

申请日：2003-03-12

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  GYPSER ANDREAS ,  MULLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHWOGLER ANJA ,  BLASCO JORDI TORMO I ,  GOTZ NORBERT ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  BLETTNER CARSTEN

IPC: A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07B61/00 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34

Abstract: Z-substituted acrylamides of formula (I), where the substituents have the following meanings: X=H, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, with X in the 3- or 4-position, n=1 or 2, where X can be different if n=2, R 1 =alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, aziridine and oxirane and R 2 =H, alkyl, haloalkyl, allyl, propargyl or CH 2 C≡C-alkyl. Methods for production thereof, agents comprising the above and the use thereof for the treatment of plant-pathogenic fungal pests.