公开(公告)号：EP0812317A1

公开(公告)日：1997-12-17

申请号：EP96916056.0

申请日：1996-05-13

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： GRAMMENOS, Wassilios ,  MÜLLER, Bernd ,  SAUTER, Hubert ,  OBERDORF, Klaus ,  KÖNIG, Hartmann ,  GÖTZ, Norbert ,  RACK, Michael ,  LORENZ, Gisela ,  AMMERMANN, Eberhard ,  STRATHMANN, Siegfried

IPC: A01N43 ,  C07D249 ,  C07D271 ,  C07D285 ,  C07D401 ,  C07D521

CPC classification number: C07D271/07 ,  A01N43/653 ,  A01N43/82 ,  C07D249/12 ,  C07D271/113 ,  C07D285/13 ,  C07D401/04

Abstract: Compounds of general formula (I) in which R is cyano, halogen, alkyl or alkoxy; n is 0, 1 or 2, in which the components R may be different if n is 2; Het is a 5-membered heteroaromatic substance containing three nitrogen atoms or two nitrogen atoms and one oxygen or sulphur atom bearing a possibly substituted 6-membered aromatic or heteroaromatic substance; process for their production and their use as pesticides and fungicides.

公开(公告)号：EP1819668A2

公开(公告)日：2007-08-22

申请号：EP05810670.9

申请日：2005-11-24

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： VON DEYN, Wolfgang ,  BASTIAANS, Henricus, Maria, Martinus ,  POHLMAN, Matthias ,  RACK, Michael ,  BAUMANN, Ernst ,  PUHL, Michael ,  HOFMANN, Michael ,  TEDESCHI, Livio ,  KORDES, Markus ,  KORADIN, Christopher ,  ANSPAUGH, Douglas, D. ,  CULBERTSON, Deborah, L. ,  COTTER, Henry, Van Tuyl ,  OLOUMI-SADEGHI, Hassan

IPC: C07C311/16 ,  C07C311/29 ,  C07C311/39 ,  C07C323/32 ,  C07C319/20 ,  A01N41/06

CPC classification number: C07C319/20 ,  A01N41/06 ,  C07C311/29 ,  C07C323/62

Abstract: The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds (I), where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to: the use of compounds (I) and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula (I) and/or at least one agriculturally useful salt of (I) and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula (I) and/or at least one agriculturally acceptable salt thereof; a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula (I).

Abstract translation: 本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物（I），其中变量Alk和R1-R5如权利要求1中所定义，和/或其可农用盐。 此外，本发明涉及：化合物（I）和/或其盐用于对抗动物害虫的用途; 包含这种量的至少一种通式（I）的化合物和/或至少一种（I）的农业上有用的盐和至少一种惰性液体和/或固体农艺上可接受的载体的农业组合物，其具有杀虫作用 和如果需要的话，至少一种表面活性剂; 以及防治动物害虫的方法，其包括使动物害虫，其习性，繁殖场，食物供应，植物，种子，土壤，面积，动物害虫正在生长或可能生长的材料或环境，或材料，植物 （I）的至少一种2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上受到保护的种子，土壤，表面或空间免于动物攻击或侵染 其可接受的盐; 一种用于保护种子免受土壤昆虫以及所得植物的根和茎由土壤和叶面昆虫引起的方法，包括在播种之前和/或在萌芽后使种子与2-氰基-3-（卤代）烷氧基 - 苯磺酰胺 通式（I）的化合物。

公开(公告)号：EP1819224A1

公开(公告)日：2007-08-22

申请号：EP05810640.2

申请日：2005-11-30

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HOFMANN, Michael ,  RACK, Michael ,  KUHN, David, G. ,  CULBERTSON, Deborah, L. ,  ANSPAUGH, Douglas

IPC: A01N37/28 ,  A01N37/30 ,  C07C243/18 ,  C07C243/42

CPC classification number: C07C243/38 ,  A01N37/28 ,  A01N43/10 ,  A01N43/12 ,  A01N43/40 ,  C07D213/81 ,  C07D213/82 ,  C07D261/20 ,  C07D307/68 ,  C07D307/81 ,  C07D317/50 ,  C07D333/38 ,  C07D405/12

Abstract: The present invention relates to new hydrazide compounds which are useful for combating animal pests, in particular insects, arachnids and nematodes and to the salts thereof. The invention also relates to a method for combating insects, nematodes and arachnids. The hydrazide compounds of the invention are described by the general formula (I) wherein ..… is absent or a covalent bond; A is an optionally substituted cyclic radical selected from phenyl, naphthyl and a 5- or 6-membered heterocyclic radical with 1 to 4 heteroatoms which are selected, independently of one another, from O, N and S, the 5- or 6-membered heterocyclic radical may have a carbonyl group as ring member; Q is selected from the group consisting of a single bond, C1-C4 alkylidene, O-C1-C4 alkylidene, S-C1-C4 alkylidene and NR9-C1-C4 alkylidene, wherein the alkylidene group in the last four mentioned radicals is unsubstituted or carries 1, 2, 3 or 4 substituents selected from OH, =O, halogen, C1-C4 haloalkyl and C1-C4 alkoxy; or A-Q may together be C1-C10-alkyl, which may be substituted by 1 or 2 substituents selected from the group consisting of =O, OH, C1-C4-alkoxy, C1-C4-alkylthio, halogen or C1-C4-alkylcarbonyloxy, X is C=O, C=S or SO2; Ar is an optionally substituted aromatic radical selected from phenyl, naphthyl, pyridyl, pyrimidyl, furyl and thienyl; and R1 to R6 and R9 are as described in the claims and the specification.

公开(公告)号：EP1732927A2

公开(公告)日：2006-12-20

申请号：EP05716387.5

申请日：2005-03-26

Applicant: BASF Aktiengesellschaft

Inventor： BLETTNER, Carsten ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GROTE, Thomas ,  HÜNGER, Udo ,  MÜLLER, Bernd ,  NIEDENBRÜCK, Matthias ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  WAGNER, Oliver ,  RACK, Michael ,  NAVE, Barbara ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich ,  STIERL, Reinhard

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to the 6-(2-fluorophenyl)-triazolopyrimidines of formula (I), wherein the substituents are defined as follows: R1 represents C4-C8 alkyl, C4-C8 halogen alkyl, substituted C3-C8 cycloalkyl, C3-C8 halogen cycloalkyl, C5-C8 alkenyl, C2-C8 halogen alkenyl, C3-C6 cycloalkenyl, C3-C6 halogen cycloalkenyl, C2-C8 alkinyl, C2-C8 halogen alkinyl or phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group including O, N or S; R2 represents hydrogen, C1-C3 alkyl or one of the groups mentioned for R1, R1 and R2, together with the nitrogen atom to which they are bound, may form a five-membered or six-membered heterocyclyl or heteroaryl which is bound via N, and may contain one to three additional heteroatoms from the group including O, N and S as a ring member, whereby piperidino-1-yl which is optionally substituted by methyl groups is exempt; R1 and/or R2 may be substituted according to the description; L1 represents chlorine or fluorine; L2 represents hydrogen, if L1 represents fluorine, L2 additionally represents fluorine; X represents alkyl. The invention also relates to a method for producing the aforementioned compounds, to agents containing them and to their use for controlling phytopathogenic parasitic fungi.

公开(公告)号：EP1699763A1

公开(公告)日：2006-09-13

申请号：EP04804216.2

申请日：2004-12-22

Applicant: BASF Aktiengesellschaft

Inventor： GEWEHR, Markus ,  RACK, Michael ,  MÜLLER, Bernd ,  GROTE, Thomas ,  GRAMMENOS, Wassilios ,  TORMO I BLASCO, Jordi ,  SCHWÖGLER, Anja ,  RHEINHEIMER, Joachim ,  BLETTNER, Carsten ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  WAGNER, Oliver ,  SPEAKMAN, John-Bryan ,  STRATHMANN, Siegfried ,  STIERL, Reinhard ,  RETHER, Jan

IPC: C07D213/81 ,  A01N43/40

CPC classification number: C07D213/81 ,  A01N43/40 ,  A01N47/22

Abstract: The invention relates to 3-trifluoromethyl picolinic acid anilides of general formula (I), wherein X represents oxygen, sulfur, or a direct bond, W represents oxygen or sulfur, n represents 0, 1, 2, 3, or 4, and the substituents have the meaning indicated in the claims, as well as the agriculturally useful salts of (I). The invention further relates to the use of said 3-trifluoromethyl picolinic acid anilides of general formula (I) and the agriculturally acceptable salts thereof as fungicides as well as plant protection agents containing the same.

Abstract translation: 本发明涉及通式（I）的3-三氟甲基吡啶甲酸N-酰苯胺，其中X表示氧，硫或直接键，W表示氧或硫，n表示0,1,2,3或4，并且 取代基具有权利要求中所指的含义以及（I）的农业上有用的盐。 本发明进一步涉及所述通式（I）的3-三氟甲基吡啶甲酸N-酰苯胺及其农业上可接受的盐作为杀真菌剂以及含有其的植物保护剂的用途。

公开(公告)号：EP1648890A2

公开(公告)日：2006-04-26

申请号：EP04763272.4

申请日：2004-07-15

Applicant: BASF Aktiengesellschaft

Inventor： WAGNER, Oliver ,  GROTE, Thomas ,  BLETTNER, Carsten ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GYPSER, Andreas ,  MÜLLER, Bernd ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  TORMO I BLASCO, Jordi ,  AKERS, Alan ,  SPEAKMAN, John-Bryan ,  RACK, Michael ,  STIERL, Reinhard ,  SCHERER, Maria ,  STRATHMANN, Siegfried ,  SCHÖFL, Ulrich

IPC: C07D471/04 ,  A01N43/90

CPC classification number: C07D471/04 ,  A01N43/90

Abstract: The invention relates to bicyclic compounds of general formula I, wherein X, Y independently represent N or C-R4; n stands for 1, 2, 3, 4 or 5; Ra represents halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl, C1-C6-halogenalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8 cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8; R2 denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8, and R3 represents hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl or C3-C6-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen. Said invention also relates to the agriculturally-acceptable salts of said compounds (I), plant protection agents, containing at least one compound of general formula (I) and/or one agriculturally-acceptable salt of (I) and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.

Abstract translation: 本发明涉及通式I的双环化合物，其中X，Y独立地代表N或C-R4; n代表1,2,3,4或5; R 1表示卤素，氰基，C 1 -C 6烷基，C 1 -C 6烷氧基，C 1 -C 6卤代烷基，C 1 -C 6卤代烷氧基，C 2 -C 6烯基，C 2 -C 6烯氧基或C R 1表示任选被烷基和/或卤素单取代或多取代的卤素，氰基，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 2 -C 6烯基，C 2 -C 6炔基，C 3 -C 8环烷基， C8环烯基，任选被烷基和/或卤素单取代或多取代，OR6，SR6或NR7R8; R 2表示任选被烷基和/或卤素单取代或多取代的卤素，氰基，C 1 -C 6烷基，C 1 -C 6卤代烷基，C 2 -C 6烯基，C 2 -C 6炔基，C 3 -C 8环烷基， 任选被烷基和/或卤素，OR 6，SR 6或NR 7 R 8单取代或多取代的C 8 - 环烯基，且R 3表示氢，C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基， 通过烷基和/或卤素。 本发明还涉及含有至少一种通式（I）的化合物和/或（I）的一种农业上可接受的盐和至少一种液体的所述化合物（I）的农业上可接受的盐，植物保护剂或 固体载体物质，以及防治植物病原性真菌的方法。

公开(公告)号：EP1633755A1

公开(公告)日：2006-03-15

申请号：EP04735002.0

申请日：2004-05-27

Applicant: BASF Aktiengesellschaft

Inventor： WAGNER, Oliver ,  GROTE, Thomas ,  BLETTNER, Carsten ,  GEWEHR, Markus ,  GRAMMENOS, Wassilios ,  GYPSER, Andreas ,  MÜLLER, Bernd ,  RHEINHEIMER, Joachim ,  SCHÄFER, Peter ,  SCHIEWECK, Frank ,  SCHWÖGLER, Anja ,  TORMO I BLASCO, Jordi ,  AKERS, Alan ,  SPEAKMAN, John-Bryan ,  RACK, Michael ,  STIERL, Reinhard ,  SCHERER, Maria ,  SCHÖFL, Ulrich ,  STRATHMANN, Siegfried

IPC: C07D487/04 ,  A01N43/90

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The invention relates to substituted pyrazolopyrimidines of formula (I) wherein the substituents have the following designations: L represents halogen, alkyl, halogenalkyl, alkenyl, alkoxy, amino, NHR, NR2, cyano, S(=O)nA1 or C(=O)A2, R representing alkyl or alkylcarbonyl, A1 representing hydrogen, hydroxy, alkyl, alkylamino or dialkylamino, n representing 0, 1 or 2, and A2 representing alkenyl, alkoxy, halogenalkoxy or one of the groups cited for A1; m represents 0 or 1 to 5; R1 represents alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, alkadienyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, phenyl, naphthyl, or a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; and R2 represents hydrogen or one of the groups cited for R1. Together with the nitrogen atom to which they are bonded, R1 and R2 can form a five-membered to six-membered ring that can be interrupted by an atom from the groups O, N and S, and R1 and/or R2 can also be substituted according to the description. Furthermore, in formula (I): X represents halogen, cyano, OH, alkyl, alkoxy or halogenalkoxy; Y represents a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle according to the description, or a group X or another group according to the description; p represents 1 or 2, the groups Y being potentially different when p = 2; and p represents 0, when X is according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing the same, and the use thereof for controlling phytopathogenic fungi.

公开(公告)号：EP1578198A1

公开(公告)日：2005-09-28

申请号：EP03782439.8

申请日：2003-12-18

Applicant: BASF Aktiengesellschaft

Inventor： STEINER, Gerd ,  SCHMIDT, Thomas ,  KORDES, Markus ,  VON DEYN, Wolfgang ,  GÖTZ, Norbert ,  HOFMANN, Michael ,  DE KRAMER, Jacobus Jan ,  HEFFERNAN, Gavin ,  CULBERTSON, Deborah L. ,  TREACY, Michael, F. ,  OLOUMI-SADEGHI, Hassan ,  EBUENGA, Cecille ,  TEDESCHI, Livio ,  BUCCI, Toni ,  PARRA RAPADO, Liliana ,  RACK, Michael ,  BAUMANN, Ernst ,  PUHL, Michael

IPC: A01N43/72 ,  A01N43/62 ,  A01N43/34 ,  C07D223/20 ,  C07D281/14 ,  C07D267/18 ,  C07D243/38

CPC classification number: C07D267/20 ,  A01N43/72 ,  C07D223/20 ,  C07D243/38 ,  C07D267/18 ,  C07D281/14 ,  C07D281/16 ,  C07D413/12

Abstract: Use of compounds of formula (I): wherein X is S, O, S=O, SO2, NRa, or CRbRc;R1,R2 are halogen, OH, SH, NH2, CN, NO2, alkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkenyl, alkenyloxy, alkenylamino, alkenylthio, alkynyl, alkynyloxy, alkynylamino, alkynylthio, alkylsulfonyl, alkylsulfoxyl, alkenylsulfonyl, alkynylsulfoxyl, formyl, alkylcarbonyl, hydroxycarbonyl, alkoxycarbonyl, carbonyloxy, alkylcarbonyloxy, phenyloxy, alkylcarbonylamino, C(O)NRdRe, or (SO2)NRdRe, or C=NORf)-Gp-Rf', ora mono- or bicyclic 5- to 10-membered aromatic or heteroaromatic ringsystem, optionally substituted, which is unfused or fused to the aromatic group to which it is bonded and which, when unfused, is bonded directly or through an O, S, alkyl, or alkoxy linkage, or cycloalkyl, wherein the carbon atoms in these groups may be substituted.R3,R4 are each independently H, alkyl, haloalkyl, alkylamino, alkoxy, cycloalkyl, wherein the carbon atoms in these groups may be substituted, or R3 and R4 together with the nitrogen atom to which they are attached form a saturated or partially saturated mono- or bicyclic 5- to 10-membered ringsystem or 5-membered hetaryl, phenyl or benzyl, wherein the rings are optionally sub-stituted, or R3 and R4 together form the chains -(CH2)2N+(O-)(CH2)2- or -(CH2)3N+(O-)(CH2)2-;and Ra, Rb, Rc, Rd, Re, Rf', Rf, G, and p are as defined in the description;m is 0, 1, 2, 3 or 4;n is 0, 1, 2, 3 or 4;or the enantiomers or diastereomers, salts or esters thereof for combatting insects, arachnids, or nematodes, methods for the control of these pests and of protecting growing plants from attack or infestation by these pests by applying a pesticidally effective amount of compounds of formula ( I), compounds of formula (I), processes for preparing them, and compositions comprising them.

公开(公告)号：EP1556346A1

公开(公告)日：2005-07-27

申请号：EP03758015.6

申请日：2003-10-17

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： REINHARD, Robert ,  HAMPRECHT, Gerhard ,  PUHL, Michael ,  SEITZ, Werner ,  PARRA RAPADO, Liliana ,  SCANNELL-LANSKY, Annegret ,  GROSSMANN, Klaus ,  SCHIFFER, Helmut ,  WITSCHEL, Matthias ,  ZAGAR, Cyrill ,  LANDES, Andreas ,  RACK, Michael

IPC: C07D207/26 ,  C07D207/24 ,  A01N43/34

CPC classification number: C07D207/277 ,  A01N43/36 ,  C07D207/24 ,  C07D403/06 ,  C07D405/04 ,  C07D409/04

Abstract: The invention relates to 1-phenylpyrrolidine-2-one-3-carboxamides of general formula (I), wherein variables R1, R2, R3, X, Y, A, n, Ra, Rb, Rc, Rd and Re have the meanings as cited in Claim 1, and to agriculturally usable salts thereof. The invention also relates to: the use of compounds I and/or the salts thereof as herbicides; plant protection products containing, as active substances, at least one 1-phenylpyrrolidine-2-one-3-carboxamide of formula (I) and/or at least one agriculturally usable salt of formula (I), and; a method for controlling unwanted plant growth during which a herbicidally effective amount of at least one 1-phenylpyrrolidine-2-one-3-carboxamide of formula (I) or of an agriculturally usable salt of formula (I) is permitted to act upon plants, the habitat thereof or upon seeds.

公开(公告)号：EP1501361A1

公开(公告)日：2005-02-02

申请号：EP03725066.9

申请日：2003-04-22

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： WAGNER, Oliver ,  RACK, Michael ,  WITSCHEL, Matthias ,  ZAGAR, Cyrill ,  LANDES, Andreas

IPC: A01N43/80 ,  C07D413/04 ,  C07D417/04

CPC classification number: C07D413/04 ,  A01N43/80 ,  C07D261/08 ,  C07D413/14 ,  C07D417/04

Abstract: The invention relates to 3-heteroaryl substituted isoxazolines of formula (I), or to their salts that can be used for agricultural purposes. In said formula, the variables are defined as follows: X represents a substituted 5-membered heteroaryl comprising between one and four nitrogen atoms, or between one and three nitrogen atoms and one oxygen or sulphur atom, or one oxygen or sulphur atom, or represents a substituted 6-membered heteroaryl comprising between one and four nitrogen atoms, whereby the aforementioned 5-membered heteroaryl is not pyrazolyl or thienyl; R1 - R7 represent hydrogen, alkyl or haloalkyl; Y represents an optionally substituted aryl, or benzo[1,4]dioxonyl, benzo[1,3]dioxolanyl, 2,3-dihydrobenzofuranyl or benzimidazole, or an optionally substituted 5- to 6-membered heteroaryl. The invention also relates to methods and intermediate products for the production of said compounds, in addition to the use thereof or of agents containing the compounds for controlling undesired plants.