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11.发明授权3- 또는 5-아미노 4-이미다졸릴 피라졸 유도체, 그의 제조방법 및 그를 포함하는 농원예용 살균제 조성물 失效3-또는5-아미노4-이미다졸릴피라졸유도체，그의제조방법및그를포함하는농원예용살균제조성물
公开(公告)号：KR100383099B1
公开(公告)日：2003-05-12
申请号：KR1020000041639
申请日：2000-07-20
Applicant: 한국화학연구원
IPC: C07D403/04
Abstract: PURPOSE: Provided is 3- or 5-amino 4-imidazolyl pyrazole derivatives which has selective bacteriocidal effect on plants. And method of preparing them and an antifungal composition comprising them for agriculture are also provided. CONSTITUTION: 3- or 5-amino 4-imidazolyl pyrazole derivatives are represented by the formula(1), wherein X is hydrogen, chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings and C-C3 alkoxy group having 1-3 benzene cycles, nitro group, or phenyl group substituted or unsubstituted trihaloalkyl group; Y is C1-C3 alkyl group; hydrogen; chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings, C1-C3 alkoxy group having 1-3 benzene rings, nitro group,or trihaloalkyl group substituted or unsubstituted benzyl group; or chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings, C1-C3 alkoxy group having 1-3 benzene rings, nitro group,or trihaloalkyl group substituted or unsubstituted penethyl group; and R is C1-C4 alkyl group; hydrogen; or chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings, C1-C3 alkyl group having 1-3 benzene rings, C-C4 alkoxy group having 1-3 benzene rings, nitro group,or trihaloalkyl group substituted or unsubstituted phenyl group.
Abstract translation: 用途：提供对植物具有选择性杀菌效果的3-或5-氨基-4-咪唑基吡唑衍生物。 还提供了它们的制备方法和包含它们的用于农业的抗真菌组合物。 构成：3-或5-氨基-4-咪唑基吡唑衍生物由式（1）表示，其中X是氢，具有1-3个苯环的氯基，具有1-3个苯环的氟基和C 1 -C 3烷氧基 具有1-3个苯环，硝基或苯基取代或未取代的三卤代烷基; Y是C1-C3烷基; 氢; 具有1-3个苯环的氯基，具有1-3个苯环的氟基，具有1-3个苯环的C1-C3烷氧基，硝基或三卤代烷基取代或未取代的苄基; 或具有1-3个苯环的氯基，具有1-3个苯环的氟基，具有1-3个苯环的C1-C3烷氧基，硝基或三卤代烷基取代或未取代的苯甲基; 和R是C1-C4烷基; 氢; 或具有1-3个苯环的氯基，具有1-3个苯环的氟基，具有1-3个苯环的C1-C3烷基，具有1-3个苯环的C-C4烷氧基，硝基或三卤代烷基取代 或未被取代的苯基。
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公开(公告)号：KR1020030017213A
公开(公告)日：2003-03-03
申请号：KR1020010051413
申请日：2001-08-24
Applicant: 한국화학연구원
IPC: A01N37/10
CPC classification number: A01N37/10 , A01N25/06 , A01N25/08 , A01N25/14 , A01N2300/00
Abstract: PURPOSE: A new methoxy acrylate compound introduced by an unsaturated carbonylthioenol group is provided which exhibits excellent germicidal activity against various plant pathogenic bacteria and is useful as an agricultural or horticultural fungicide. CONSTITUTION: The agricultural or horticultural fungicide contains a methoxy acrylate derivative represented by the formula(1). In formula, R1 represents a phenyl, substituted phenyl, naphthyl, substituted naphthyl, pyridyl, substituted pyridyl, furanyl, substituted furanyl, pyrrolyl, substituted pyrrolyl, thiopheneyl, substituted thiophenyl, indolinyl or substituted indolinyl group, in which the substituted group is selected from halogen, cyclo, C1-3 alkyl, C1-3 haloalkyl and C1-3 alkoxy group and can be substituted in the range of 1 to 4, two adjacent substituted groups can combine to form -OCH2CH2O-; R2 represents H or C1-3 alkyl; R3 represents C1-3 alkyl; X represents S or NH; Y represents CH or N.
Abstract translation: 目的：提供由不饱和羰基硫醇烯基引入的新的甲氧基丙烯酸酯化合物，对各种植物病原菌具有优异的杀菌活性，可用作农业或园艺杀真菌剂。 构成：农业或园艺杀菌剂含有式（1）表示的甲氧基丙烯酸酯衍生物。 在式中，R 1表示苯基，取代的苯基，萘基，取代的萘基，吡啶基，取代的吡啶基，呋喃基，取代的呋喃基，吡咯基，取代的吡咯基，噻吩基，取代的噻吩基，二氢吲哚基或取代的二氢吲哚基，其中取代基选自 卤素，环，C 1-3烷基，C 1-3卤代烷基和C 1-3烷氧基，并且可以在1至4的范围内被取代，两个相邻的取代基可以结合形成-OCH 2 CH 2 O-; R2代表H或C1-3烷基; R3表示C1-3烷基; X表示S或NH; Y表示CH或N.
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13.发明公开3- 또는 5-아미노 4-이미다졸릴 피라졸 유도체, 그의 제조방법 및 그를 포함하는 농원예용 살균제 조성물 失效3-或5-氨基-4-咪唑烷基吡唑衍生物，其制备方法和包含农业的抗真菌组合物
公开(公告)号：KR1020020008242A
公开(公告)日：2002-01-30
申请号：KR1020000041639
申请日：2000-07-20
Applicant: 한국화학연구원
IPC: C07D403/04
Abstract: PURPOSE: Provided is 3- or 5-amino 4-imidazolyl pyrazole derivatives which has selective bacteriocidal effect on plants. And method of preparing them and an antifungal composition comprising them for agriculture are also provided. CONSTITUTION: 3- or 5-amino 4-imidazolyl pyrazole derivatives are represented by the formula(1), wherein X is hydrogen, chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings and C-C3 alkoxy group having 1-3 benzene cycles, nitro group, or phenyl group substituted or unsubstituted trihaloalkyl group; Y is C1-C3 alkyl group; hydrogen; chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings, C1-C3 alkoxy group having 1-3 benzene rings, nitro group,or trihaloalkyl group substituted or unsubstituted benzyl group; or chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings, C1-C3 alkoxy group having 1-3 benzene rings, nitro group,or trihaloalkyl group substituted or unsubstituted penethyl group; and R is C1-C4 alkyl group; hydrogen; or chloro group having 1-3 benzene rings, fluoro group having 1-3 benzene rings, C1-C3 alkyl group having 1-3 benzene rings, C-C4 alkoxy group having 1-3 benzene rings, nitro group,or trihaloalkyl group substituted or unsubstituted phenyl group.
Abstract translation: 目的：提供对植物具有选择性杀菌作用的3-或5-氨基-4-咪唑基吡唑衍生物。 还提供了制备它们的方法和包含它们用于农业的抗真菌组合物。 构成：3-或5-氨基-4-咪唑基吡唑衍生物由式（1）表示，其中X是氢，具有1-3个苯环的氯基，具有1-3个苯环的氟基和C-C3烷氧基 具有1-3个苯环，硝基或苯基取代或未取代的三卤代烷基; Y为C1-C3烷基; 氢; 具有1-3个苯环的氯基团，具有1-3个苯环的氟基团，具有1-3个苯环的C1-C3烷氧基，硝基或三卤代烷基取代或未取代的苄基; 或具有1-3个苯环的氯基，具有1-3个苯环的氟基，具有1-3个苯环的C1-C3烷氧基，硝基或三卤代烷基取代或未取代的乙基; 并且R是C 1 -C 4烷基; 氢; 或具有1-3个苯环的氯基，具有1-3个苯环的氟基，具有1-3个苯环的C1-C3烷基，具有1-3个苯环的C-C4烷氧基，硝基或三卤代烷基取代的 或未取代的苯基。
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14.发明公开옥심기를 가교로 하는, 불소화 비닐기가 치환된 프로페노익 에스테르 및 아미드 화합물, 이의 제조방법 및 이를 포함하는 살균제 조성물 有权由氟族基团交联并由氟化乙烯基团取代的新型丙烯酸酯和酰胺化合物，其制备方法和包括其的双酚A的组合物
公开(公告)号：KR1020010017960A
公开(公告)日：2001-03-05
申请号：KR1019990033722
申请日：1999-08-16
Applicant: 한국화학연구원
IPC: C07C207/00
Abstract: PURPOSE: Provided is a novel propenoic ester and amide compound being cross-linked by an oxime group and substituted by a fluorinated vinyl group. The novel compound has excellent sterilizability and a broad antibacterial activity. Also, its preparation method and a bactericide composition including these are provided. CONSTITUTION: A novel propenoic ester compound being cross-linked by an oxime group and substituted by a fluorinated vinyl group is represented by the formula (1), wherein X is CH or N ; Y is O or NH ; R1 is hydrogen, C1-4 alkyl or C1-4 alkyl substituted with halogen ; and R2 is phenyl, C1-4 alkyl,, C1-4 alkyl substituted with halogen, C1-4 alkoxy, methylenedioxy, phenyl in which more than one group is substituted with halogen or naphthalene. The novel propenoic ester compound is prepared by reacting a brominated compound of the formula (2) and an oxime compound of the formula (3) in the presence of a base, to obtain compound of the formula (4); debenzylating the resultant compound, to obtain phenolic ester compound of the formula (5); and reacting the resultant compound with a fluorinated vinyl compound of the formula (6) in the presence of a base.
Abstract translation: 目的：提供一种新的丙烯酸酯和酰胺化合物，通过肟基交联并被氟化乙烯基取代。 该新型化合物具有优异的灭菌性和广泛的抗菌活性。 此外，还提供了其制备方法和包括这些的杀菌剂组合物。 构成：通过肟基交联并被氟代乙烯基取代的新型丙烯酸酯化合物由式（1）表示，其中X为CH或N; Y是O或NH; R1是氢，C1-4烷基或被卤素取代的C1-4烷基; 和R 2是苯基，C 1-4烷基，被卤素取代的C 1-4烷基，C 1-4烷氧基，亚甲二氧基，其中多于一个基团被卤素或萘取代的苯基。 通过使式（2）的溴化化合物与式（3）的肟化合物在碱的存在下反应制备新的丙烯酸酯化合物，得到式（4）的化合物; 将所得化合物脱苄化，得到式（5）的酚酯化合物; 并使所得化合物与式（6）的氟化乙烯基化合物在碱的存在下反应。
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15.发明授权
公开(公告)号：KR100270599B1
公开(公告)日：2000-11-01
申请号：KR1019980041817
申请日：1998-10-07
Applicant: 한국화학연구원
IPC: C07C251/48
Abstract: 본 발명은 메톡시아크릴레이트 또는 메톡시이미노 아세테이트 유도체, 그의 제조 방법 및 그를 이용한 살균제 조성물에 관한 것이다. 이 유도체 화합물은 하기 화학식 1을 갖고, 아미노산이 치환된 옥심을 갖는다. 이 화합물을 포함하는 살균제 조성물은 내성균을 비롯한 식물 병원균에 대해 광범위한 살균효과를 가지고, 식물에 침투 효과 뿐만 아니라 질병 예방 및 치료 효과가 뛰어나며, 기타 성분과 함께 광범위한 식물 병원균에 대해 사용될 수 있다.
[화학식 1]
상기 식에서,
R
1 는 수소, C
1 -C
3 알킬기, C
1 -C
3 알킬티오- 또는 알킬설폰-치환된 알킬기, 페닐기, 또는 벤질기이고; R
2 은 C
1 -C
5 알킬기이고; X는 벤질옥시, C
1 -C
3 알콕시, C
1 -C
3 알킬기, 1 내지 3개의 클로로 또는 플루오로, C
1 -C
3 트리할로알킬기, 또는 C
1-3 알킬 또는 알콕시-치환되거나 치환되지 않은 페녹시기이고; Z는 CH 또는 N 이다.-
Patent Agency Ranking
公开(公告)号：KR100124946B1
公开(公告)日：1997-12-08
申请号：KR1019930011382
申请日：1993-06-22
Applicant: 한국화학연구원
IPC: C07D215/42 , C07D215/20 , C07H17/04
CPC classification number: C07D401/12 , A01N43/42 , A01N43/50 , A01N43/90 , A01N55/00 , C07D215/42 , C07D221/10 , C07D405/12 , C07D409/12 , C07D491/04 , C07F7/0812
Abstract: 4-Alkylsulfoxy-2-quinolinon(ii) and HNR6R7(iii) were reacted in the presence of inactive solvent such as diethylether, diisopropylether, tetrahydrofurane, benzene, toluene, dichloroethane, chloroform,ethylacetate, ethylpropionate, chlorobenzene at 0-260 deg.C for 0.5-24hr to give(I) which is useful for herbicide and insecticide.In formula R1-4=h, allyl or allyloxy, C1-10 aralkyl or alkyl, R6=H or C1-5 alkyl, alkoxyalkyl, phenylacetyl or (R19)Si, R17-18=H or C1-5 alkyl,or-T-(CH2)-T Y=O,S Z=hetero ring, T=O,S, R20=C1-3 alkyl, m,n,p,q,r=1-4, R21=C1-3 alkyl.
Abstract translation: 在惰性溶剂如乙醚，二异丙基醚，四氢呋喃，苯，甲苯，二氯乙烷，氯仿，乙酸乙酯，丙酸乙酯，氯苯在0-260度的存在下，使4-烷基亚磺酰基-2-喹啉酮（ⅱ）和HNR6R7（ⅲ） 在式R1-4 = h中，烯丙基或烯丙氧基，C 1-10芳烷基或烷基，R 6 = H或C 1-5烷基，烷氧基烷基，苯乙酰基或 （R19）Si，R17-18 = H或C1-5烷基或-T-（CH2）-TY = O，SZ =杂环，T = O，S，R20 = C1-3烷基，m， p，q，r = 1-4，R 21 = C 1-3烷基。
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公开(公告)号：KR1020100123937A
公开(公告)日：2010-11-26
申请号：KR1020090042909
申请日：2009-05-18
Applicant: 원광대학교산학협력단 , 한국화학연구원
Abstract: PURPOSE: An insecticide composition containing 4-quinolinone derivative compound is provided to ensure high insecticidal effect against Bursaphelenchus xylophilus. CONSTITUTION: An insecticide composition for preventing pest contains 4-quinolinone derivative compound of general formula I as an active ingredient. The pest is Bursaphelenchus xylophilus, Bursaphelenchus mucronatus, Bursaphelenchus fraudulentus Ruhm or Bursaphelenchus kolymensis Korenchenko. The insecticide composition is treated to insects or habitat of insects by spraying.
Abstract translation: 目的：提供含有4-喹啉酮衍生物化合物的杀虫剂组合物，以确保木麻黄的杀虫效果。 构成：用于防治害虫的杀虫剂组合物含有作为活性成分的通式I的4-喹啉酮衍生物化合物。 害虫是Bursaphelenchus xylophilus，Bursaphelenchus mucronatus，Bursaphelenchus fraudulentus Ruhm或Bursaphelenchus kolymensis Korenchenko。 杀虫剂组合物通过喷雾处理昆虫或昆虫栖息地。
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