公开(公告)号：CA2520718A1

公开(公告)日：2004-10-14

申请号：CA2520718

申请日：2004-03-30

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GYPSER ANDREAS ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  STRATHMANN SIEGFRIED ,  RHEINHEIMER JOACHIM ,  SCHERER MARIA ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  SCHIEWECK FRANK

IPC: A01N43/90 ,  C07D487/04

Abstract: 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L = halogen, alkyl, halogenalkyl, alkoxy, amino , NHR, NR2, cyano, S(O)nA1 or C(O)A2; R = alkyl or alkylcarbonyl; A1 = hydroge n, hydroxy, alkyl, alkylamino or aialkylamino; n = 0, 1 or 2; A2 = alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A1; m = 1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond wit h the triazolopyrimidine skeleton; X = halogen, cyano, alkyl, halogenalkyl or alkoxy; R1 = hydrogen or alkyl; R2 = alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compoun ds and the use thereof to combat harmful phytopathogenic fungi.

公开(公告)号：AU2004226233A1

公开(公告)日：2004-10-14

申请号：AU2004226233

申请日：2004-03-24

Applicant: BASF AG

Inventor： MULLER BERND ,  SCHIEWECK FRANK ,  GRAMMENOS WASSILIOS ,  BLETTNER CARSTEN ,  SCHERER MARIA ,  GYPSER ANDREAS ,  SCHWOGLER ANJA ,  STIERL REINHARD ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  BLASCO JORDI TORMO I ,  SCHOFL ULRICH ,  GEWEHR MARKUS ,  STRATHMANN SIEGFRIED ,  SCHAFER PETER

IPC: A01N43/90 ,  C07D487/04

Abstract: 7-(Alkenylamino)triazolopyrimidines of the formula I wherein the substituents have the following meanings: L is halogen, alkyl, haloalkyl, alkoxy, amino, NHR or NR 2 ; R is alkyl or alkyl-carbonyl; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl or alkoxy; R 1 is alkyl or haloalkyl; R 2 is hydrogen, alkyl or haloalkyl; R 3 is alkenyl, which can be unsubstituted or partially or completely halogenated or can be substituted according to the Description; R 4 is hydrogen or alkyl, R 3 and R 4 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered unsaturated ring which can be interrupted by an atom from the group consisting of O, N and S and/or can carry one or more sub-stituents. Processes for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.

公开(公告)号：DE60013188D1

公开(公告)日：2004-09-23

申请号：DE60013188

申请日：2000-12-06

Applicant: BASF AG

Inventor： PEES KLAUS-JUERGEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL RHEINHARD

IPC: A01N43/90 ,  C07D487/04

公开(公告)号：DE10257394A1

公开(公告)日：2004-06-24

申请号：DE10257394

申请日：2002-12-06

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

Abstract: 2,5-Disubstituted-7-amino-6-phenyl-(1,2,4)-triazolo(1,5-a)pyrimidine derivatives (I) are new. 2,5-Disubstituted-7-amino-6-phenyl-(1,2,4)-triazolo(1,5-a)pyrimidine derivatives of formula (I) are new. L = halogen, CN, NO2, alkyl, 2-10C alkenyl, 2-10C alkynyl, 2-10C alkynyl, haloalkyl, 2-10C haloalkenyl, alkoxy, 2-10C alkenyloxy, 2-10C alkynyloxy, haloalkoxy, C(O)A or S(O)pA'; A = H, OH, 1-8C alkyl, 2-8C alkenyl, 1-8C alkoxy, haloalkoxy or mono- or di-(1-8C alkyl)amino; A' = H, 1-8C alkyl or haloalkyl; m = 0-5; X = CN, 1-4C alkyl, 1-4C haloalkyl, 1-4C alkoxy or 1-2C haloalkoxy; R1, R2 = H or 1-8C alkyl, 1-8C haloalkyl, cycloalkyl, halocycloalkyl, 2-8C alkenyl, 4-10C alkadienyl, 2-8C haloalkenyl, cycloalkenyl, 2-8C alkynyl, 2-8C haloalkynyl, cycloalkynyl, phenyl, naphthyl, 5- or 6-membered heteroaryl or 5-10 membered saturated, partially unsaturated or aromatic heterocyclyl (containing 1-4 of O, N and/or S), all optionally substituted (os) by 1-4 Ra; or NR1R2 = 5 or 6 membered heterocycle optionally containing an additional O, N or S heteroatom, os by one or more halogen, alkyl, haloalkyl or 1-3C alkylenedioxy and/or optionally having an N and an adjacent C linked by a 1-4C alkylene chain; Ra = halogen, CN, NO2, OH, alkyl, haloalkyl, alkylcarbonyl, cycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, alkoxycarbonyl, alkenyl, alkenyloxy, 3-6C alkynyloxy, cycloalkyl, phenyl, naphthyl or 5-10 membered saturated, partially unsaturated or aromatic heterocyclyl containing 1-4 of O, N and/or S, where cyclic residues are optionally partially or completely halogenated and os by 1-3 Rb; Rb = halogen, CN, NO2, OH, SH, NH2, COOH, C(O)NH2, C(S)NH2, alkyl, haloalkyl, 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, alkoxy, haloalkoxy, alkylthio, mono- or dialkylamino, CHO, alkylcarbonyl, alkylsulfonyl, alkylsulfoxyl, alkylcarbonyl, alkylcarbonyloxy, mono- or dialkylaminocarbonyl, mono- or dialkylaminothiocarbonyl, 3-10C cycloalkyl, 3-10C cycloalkoxy, 3-10 membered heterocyclyl, 3-10 membered heterocyclyloxy, aryl, aryloxy, arylthio, arylalkoxy, arylalkyl (where all aryl moieties are preferably 6-10 membered), 5 or 6 membered heteroaryl, 5 or 6 membered heteroaryloxy or 5 or 6 membered heteroarylthio (where all rings are optionally partially or completely halogenated and os by alkyl or haloalkyl (for which no C-numbers are specified)); R3 = CN, OH, 1-8C alkoxy, 3-8C alkenyloxy, 1-8C haloalkoxy, 3-8C haloalkenyloxy, NR1R2 or S(O)nR31; n, p = 0-2; and R31 = H, OH, 1-8C alkyl, 2-8C alkenyl or C(O)A. Unless specified otherwise alkyl moieties have 1-6C, alkenyl moieties 2-6C and cycloalkyl, cycloalkenyl or cycloalkynyl moieties 3-6C. Independent claims are included for the preparation of (I).

公开(公告)号：AU2003289871A1

公开(公告)日：2004-06-15

申请号：AU2003289871

申请日：2003-11-14

Applicant: BASF AG

Inventor： SCHOFL ULRICH ,  STIERL REINHARD ,  BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED

IPC: A01N43/90 ,  C07D487/04

Abstract: 2-Mercapto-substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy or -C(-O)-A; A is hydrogen, hydroxyl, alkyl, alkenyl, alkoxy, haloalkoxy, alkylamino or dialkylamino; m is 0, 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R 1 , R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four hetero atoms from the group consisting of O, N and S; R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S; where R 1 and/or R 2 may be substituted as stated in the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

公开(公告)号：AU2003279353A1

公开(公告)日：2004-06-07

申请号：AU2003279353

申请日：2003-11-04

Applicant: BASF AG

Inventor： BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C69/65 ,  C07C69/76 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R1 and R2 radicals may be substituted as defined in the description, R2 denote hydrogen, or a group mentioned for R1; or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L1, L3 independently denote hydrogen, halogen, or alkyl; L2 is hydrogen, halogen, haloalkyl, or NH2, NHRb, or N(Rb)2, wherein Rb is as defined in the description, wherein at least one from L1, L2, and L3 is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy. processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

公开(公告)号：DE59908820D1

公开(公告)日：2004-04-15

申请号：DE59908820

申请日：1999-10-01

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  SAUTER HUBERT ,  BAYER HERBERT ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  CULLMANN OLIVER ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/72 ,  A01N43/88 ,  A61K31/539 ,  A61P31/10 ,  C07D273/00 ,  C07D273/01

公开(公告)号：CZ20033153A3

公开(公告)日：2004-02-18

申请号：CZ20033153

申请日：2002-05-17

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  ROSE INGO ,  GROTE THOMAS ,  SCHAFER PETER ,  SCHEIWECK FRANK ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N43/86 ,  A01N43/90 ,  C07D265/24 ,  C07D498/04 ,  C07D513/04 ,  C07D495/04

Abstract: Oxazin(ethi)one compounds of the formula I: in which the variables Z, R 1 , R 2 , R 3 and n are as defined in claim 1 and A is a 5- or 6-membered carbocycle or a 5- or 6-membered heterocycle having 1, 2 or 3 heteroatoms selected from the group consisting of N, O and S, each of which cycles is attached via two carbon atoms to the oxazin(ethi)one ring, and the agriculturally useful salts of the oxazin(ethi)one compounds I are described. Moreover, the invention describes the use of compounds I and their salts for controlling phytopathogenic fungi, compositions which comprise the compounds I and/or their salts in a fungicidally effective amount and a method for controlling phytopathogenic fungi which comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula I as claimed in claim 1 and/or a salt of I.

公开(公告)号：AU2003216893A1

公开(公告)日：2003-10-13

申请号：AU2003216893

申请日：2003-03-27

Applicant: BASF AG

Inventor： STRATHMANN SIEGFRIED ,  STIERL REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GYPSER ANDREAS ,  MULLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHWOGLER ANJA ,  BLASCO JORDI TORMO I ,  GOTZ NORBERT ,  LORENZ GISELA ,  AMMERMANN EBERHARD

IPC: C07D213/56 ,  C07D213/61 ,  C07D263/10 ,  C07D213/26

Abstract: The present invention relates to novel phenethylacrylamides of the formula I in which the substituents R 1 , R 2 , R 3 and R 4 have the following meanings: R 1 is hydrogen, halogen, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, C 3 -C 8 -cycloalkyl, C 1 -C 4 -haloalkoxy or C 1 -C 4 -haloalkyl; R 2 is hydrogen, halogen, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, C 3 -C 10 -cycloalkyl, C 1 -C 4 -haloalkoxy or C 1 -C 4 -haloalkyl; R 3 is C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, propargyl, C 3 -C 4 -alkenyl or a radical of the formula -H 2 C-C≡C-C(R a , R a )-R c , wherein R a , R b independently of one another are hydrogen or methyl and R c is hydrogen or C 1 -C 4 -alkyl; R 4 is methyl or C 1 -haloalkyl; and Het is a 5- or 6-membered heteroaromatic ring, to processes for their preparation, and to the use of phenethylacrylamides of the formula I for controlling phytopathogenic harmful fungi.

公开(公告)号：AU2003215664A1

公开(公告)日：2003-10-08

申请号：AU2003215664

申请日：2003-03-19

Applicant: BASF AG

Inventor： SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD ,  SCHOFL ULRICH ,  BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM

IPC: A01N43/90 ,  C07C255/57 ,  C07D487/04 ,  C07C323/62

Abstract: The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L 1 represents cyano, S(-O) n A 1 or C(-O)A 2 , wherein A 1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A 2 stands for C 1 -C 8 alkoxy, C 1 -C 6 haloalkoxy or one of the groups named in A 1 ; and n stands for 0, 1 or 2; L 2 , L 3 represent hydrogen or halogen; L 4 , L 5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R 1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R 2 represents hydrogen or R 1 ; R 1 and R 2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R 1 and/or R 2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.