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公开(公告)号:AU2002304642B2
公开(公告)日:2008-02-07
申请号:AU2002304642
申请日:2002-05-17
Applicant: BASF AG
Inventor: GYPSER ANDREAS , SCHAFER PETER , LORENZ GISELA , AMMERMANN EBERHARD , ROSE INGO , RHEINHEIMER JOACHIM , SCHIEWECK FRANK , SPEAKMAN JOHN-BRYAN , STRATHMANN SIEGFRIED , GROTE THOMAS
IPC: C07D265/24 , A01N43/86 , A01N43/90 , C07D498/04 , C07D513/04
Abstract: Oxazin(ethi)one compounds of the formula I: in which the variables Z, R 1 , R 2 , R 3 and n are as defined in claim 1 and A is a 5- or 6-membered carbocycle or a 5- or 6-membered heterocycle having 1, 2 or 3 heteroatoms selected from the group consisting of N, O and S, each of which cycles is attached via two carbon atoms to the oxazin(ethi)one ring, and the agriculturally useful salts of the oxazin(ethi)one compounds I are described. Moreover, the invention describes the use of compounds I and their salts for controlling phytopathogenic fungi, compositions which comprise the compounds I and/or their salts in a fungicidally effective amount and a method for controlling phytopathogenic fungi which comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula I as claimed in claim 1 and/or a salt of I.
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公开(公告)号:SI1414302T1
公开(公告)日:2007-08-31
申请号:SI200230527
申请日:2002-07-16
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , SAUTER HUBERT , MULLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAFER PETER , SCHIEWECK FRANK , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD , KRUMMEL GUNTER
IPC: A01N43/90 , A01N43/00 , C07D487/00 , C07D487/04
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公开(公告)号:EA008889B1
公开(公告)日:2007-08-31
申请号:EA200401164
申请日:2003-03-19
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , BLETTNER CARSTEN , MULLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHAFER PETER , SCHIEWECK FRANK , SCHWOGLER ANJA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD , SCHOFL ULRICH
IPC: C07D487/04 , A01N43/90 , C07C255/57 , C07C323/62 , C07D239/00 , C07D249/00
Abstract: Триазолопиримидиныформулы Iвкоторойзаместителиимеютследующиезначения: Lозначаетциано, S(=O)AилиС(=O)А, гдеАозначаетводород, гидрокси, С-Салкил, С-Салкиламиноилиди-(С-Салкил)амино; АозначаетС-Салкокси, C-СгалогеналкоксиилиоднуизприведенныхдляАгрупп; n равно 0, 1 или 2; L, Lозначаетводородилигалоген; L, Lозначаетводород, галогенили C-Салкил; X означаетгалоген, циано, С-Салкил, С-Сгалогеналкил, С-СалкоксиилиС-С-галогеналкокси; RС-Салкил, С-Сгалогеналкил, С-Сциклоалкил, С-С-галогенциклоалкил, С-Салкенил, С-Салкадиенил, С-С-галогеналкенил, С-Сциклоалкенил, С-Салкинил, С-С-галогеналкинилилиС-Сциклоалкинил, фенил, нафтил, илиотпяти- додесятичленныйнасыщенный, частичноненасыщенныйилиароматическийгетероцикл, содержащийотодногодочетырехгетероатомовизгруппы, включающейО, N или S; Rозначаетводородили R, Rи Rмогутобразовыватьвместес атомомазота, скоторымонисвязаны, пяти- илишестичленноекольцо, котороеможетбытьпрерваноодниматомомизгруппы, включающейО, N и S и/илиможетбытьзамещено; причем Rи/или Rможетбытьзамещенсогласноописанию. Способи промежуточныепродуктыдляполученияэтихсоединений, содержащиеихсрдства, атакжеихприменениедляборьбыс фитопатогеннымигрибами.
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公开(公告)号:DE50209786D1
公开(公告)日:2007-05-03
申请号:DE50209786
申请日:2002-07-16
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , SAUTER HUBERT , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD , KRUMMEL GUENTER
IPC: A01N43/90 , C07D487/04
Abstract: The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R 1 , R 2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R 1 and R 2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R 3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R 3 and R 2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by R a . The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.
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公开(公告)号:AT357142T
公开(公告)日:2007-04-15
申请号:AT02790165
申请日:2002-07-16
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , SAUTER HUBERT , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD , KRUMMEL GUENTER
IPC: A01N43/90 , C07D487/04
Abstract: The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R 1 , R 2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R 1 and R 2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R 3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R 3 and R 2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by R a . The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.
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公开(公告)号:AT353901T
公开(公告)日:2007-03-15
申请号:AT02758297
申请日:2002-07-03
Applicant: BASF AG
Inventor: MUELLER BERND , SAUTER HUBERT , GEWEHR MARKUS , GRAMMENOS WASSILIOS , TORMO I BLASCO JORDI , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , RACK MICHAEL , LORENZ GISELA , STRATHMANN SIEGFRIED , AMMERMANN EBERHARD , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines (I) are new. 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines of formula (I) are new. [Image] n : 0-5; R : halo, CN, OH or OCN, or alkyl, alkenyl, alkynyl, T', haloalkenyl, OT, alkenyloxy, alkynyloxy, OT', cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, CONH 2, mono- or dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); T : 1-6C alkyl; T' : 1-6C haloalkyl; Het : 5-10 membered, saturated, partially unsaturated or aromatic heterocycle containing 1-4 of O, N and/or S heteroatoms; R 11-10C alkyl, alkenyl, alkynyl, 3-12C cycloalkyl, 3-10C cycloalkenyl, phenyl, naphthyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); R ahalo, CN, NO 2, OH, T, T', COT, cycloalkyl, OT, OT', COOT, NHT, NT 2, 2-6C alkenyl, 2-6C alkenyloxy, 3-6C alkynyloxy, alkoximino, alkenyloximino, alkynyloximino, aralkoximino, alkynyl, alkynyloxycarbonyl, phenyl, naphthyl or Het (where all aliphatic, alicyclic or aromatic groups are optionally partially or completely halogenated and optionally substituted by 1-3 R aand/or 1-3 R c); R bhalo, CN, NO 2, OH, SH, NH 2, COOH, CONH 2, CSNH 2, T, T', 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, OT, OT', ST, NHT, NT 2, CHO, COT, SO 2T, SOT, COOT, OCOT, CONHT, CONT 2, CSNHT or CSNT 2; R ccycloalkyl, -O-cycloalkyl, heterocyclyl, -O-heterocyclyl, aryl, -O-aryl, -S-aryl, -O-T-aryl, -T-aryl, heteroaryl, -O-heteroaryl or -S-heteroaryl (where cycloalkyl or heterocyclyl rings are 3-10 membered, aryl rings are preferably 6-10 membered and heteroaryl rings are preferably 5-6 membered; and all rings are optionally partially or completely halogenated and optionally substituted by alkyl or haloalkyl); and R 21-4C alkyl, 2-4C alkynyl or 2-4C alkynyl (all optionally substituted by halo, CN, NO 2, OMe, OEt or 1-4C alkoxycarbonyl; Unless specified otherwise alkyl moieties have 1-8C, alkenyl or alkynyl moieties 2-10C and cycloalkyl or cycloalkenyl moieties 3-6C. Independent claims are also included for: (1) preparation of (I); and (2) dicarbonyl compound intermediates of formula (III), provided that n is not 0 and R 1and R 2are not both Me. [Image] ACTIVITY : Fungicide. 7-Cyclohexyl-5-methyl-6-(2-chloro-6-fluorophenyl)-1,2,4-triazolo[1,5-a]pyrimidine (Ia) at a concentration of 63 ppm gave at least 90 % protection of tomato plants against Alternaria solani. MECHANISM OF ACTION : None given.
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公开(公告)号:DE502004002570D1
公开(公告)日:2007-02-15
申请号:DE502004002570
申请日:2004-07-15
Applicant: BASF AG
Inventor: SCHWOEGLER ANJA , GEWEHR MARKUS , MUELLER BERND , GROTE THOMAS , GRAMMENOS WASSILIOS , TORMO I BLASCO JORDI , GYPSER ANDREAS , RHEINHEIMER JOACHIM , BLETTNER CARSTEN , SCHAEFER PETER , SCHIEWECK FRANK , WAGNER OLIVER , STIERL REINHARD , SCHOEFL ULRICH , STRATHMANN SIEGFRIED , SCHERER MARIA
IPC: C07D239/42
Abstract: The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R 1 to R 3 and L are as defined in the description and R 4 corresponds to one of the formulae in which R a , X and R b are as defined in the description; and also to processes for preparing these compounds, to pesticidal compositions comprising these compounds and to their use as pesticides.
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公开(公告)号:ECSP066295A
公开(公告)日:2006-10-25
申请号:ECSP066295
申请日:2006-01-19
Applicant: BASF AG
Inventor: STIERL REINHARD , SCHERER MARIA , TORMO I BLASCO JORDI , GROTE THOMAS , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , BLETTNER CARSTEN , GEWEHR MARKUS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , MULLER BERND , GRAMMENOS WASSILIOS
IPC: C07D239/42
Abstract: . La invención se refiere a pirimidinas 2-sustituidas de la fórmula I, en la que el índice y los sustituyentes R1, R2 y R3 tienen las definiciones indicadas en la descripción y R4 tiene el significado siguiente:R4 corresponde a las fórmulas donde X es un enlace directo, -(C=O)-, -(C=O)-NH-, -(C=O)-O-, -O-, -NRc-, donde la parte de molécula izquierda está unida cada vez con el átomo de nitrógeno;Ra significa hidrógeno, metilo, bencilo, trifluorometilo, alilo, propargilo o metoximetilo; Rb es hidrógeno, alquilo C1-C6, alquinilo C2-C6;Rc es hidrógeno, metilo o acilo C1-C4Z es S o NRb;pudiendo los grupos alifáticos de las definiciones de los radicales Ra, Rb y/o Rc a su vez llevar uno o dos grupos RwRw significa halógeno, ORx, NHRx, alquilo C1-C6, alcoxicarbonyilo C1-C4-, acilamino C1-C4, [1,3]dioxolano -alquilo-C1-C4, [1,3]dioxano -alquilo-C1-C4, significandoRx es hidrógeno, metilo, alilo o propargilo.Procedimiento para la obtención de estos compuestos, productos que contienen estos compuestos y el uso de los mismos como pesticidas.
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公开(公告)号:DE50304232D1
公开(公告)日:2006-08-24
申请号:DE50304232
申请日:2003-04-30
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: C07D487/04 , A01N43/90 , C07C69/612 , C07C69/65 , C07C69/738 , C07D239/00 , C07D249/00
Abstract: Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (1), in which the substituents have the following meaning: L 1 represents alkyl; L 2 represents halogen; L 3 represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R 1 , R 2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S. R 1 and R 2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R 1 and/or R 2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi.
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公开(公告)号:ECSP066278A
公开(公告)日:2006-07-28
申请号:ECSP066278
申请日:2006-01-11
Applicant: BASF AG
Inventor: STIERL REINHARD , SCHERER MARIA , TORMO I BLASCO JORDI , GROTE THOMAS , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , BLETTNER CARSTEN , GEWEHR MARKUS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , MULLER BERND , SCHAFER PETER , GRAMMENOS WASSILIOS
IPC: C07D239/42
Abstract: La invención se refiere a pirimidinas 2-sustituidas de la fórmula I Ien la que el índice n y los sutituyentes R1 hasta R3, así como L tienen las definiciones indicadas en la descripción y R4 corresponde a una de las fórmulas donde Ra, X y Rb tienen las definiciones indicadas en la descripción;así como procedimientos para su obtención, productos pesticidas que las contienen y el uso de las mismas como pesticidas.
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