N-(2-NITROPHENYL)-2-AMINOPYRIMIDINE DERIVATIVES

    公开(公告)号:CA1218372A

    公开(公告)日:1987-02-24

    申请号:CA484416

    申请日:1985-06-19

    Applicant: CIBA GEIGY AG

    Abstract: Pesticidal compositions The invention discloses novel N-(2-nitrophenyl)-2-aminopyrimidine derivatives of the general formula I (I) wherein R1 and R2 are hydrogen, NO2 or CF3, with the proviso that only R1 or R2 can be NO2; R4 is hydrogen or the -C(O)R' group, in which R' is C1-C4alkyl which is unsubstituted or substituted by halogen, C1-C3alkoxy or C1-C3 alkylthio; R5, R6 and R7 are each independently halogen, nitro, cyano, thiocyano, C1-C12alkyl, C3-C8cycloalkyl, C1-C9alkylthio, C1-C6alkylsulfonyl, C1-C6alkylsulfoxyl, C3-C6alkenyl, C3-C6haloalkenyl, C3-C6alkynyl, C3-C6haloalkynyl, C3-C6alkenyloxy, C3-C6haloalkanyloxy, C3-C6alkenylthio, C3-C6alkynyloxy, C3-C6haloalkynyloxy, C1-C8alkyl which is substituted by halogen, cyano and/or C1-C4alkoxy, or are unsubstituted C1-C8alkoxy or halogen-substituted C1-C8alkoxy, the alkyl moiety of which may be interrupted by one or more single oxygen atoms, or are the Q-(E)n-(X)m group, in which n is 0 or 1, m is 0 or 1, Q is phenyl which is unsubstituted or substituted by halogen, nitro, C1-C3alkyl, CF3 and/or C1-C3alkoxy, or is a saturated or unsaturated heterocyclic radical containing one or more hetero atoms, E is a C1-C3alkylene bridge, and X is oxygen or sulfur, and R6 and/or one of the radicals R5 or R7 can also be hydrogen. Also disclosed are methods of preparing these compounds, and agrochemical compositions which contain one such compound as active ingredient. The invention further relates to the use of the novel compounds, or compositions containing them, in agriculture and related fields.

    25.
    发明专利
    未知

    公开(公告)号:BR8504584A

    公开(公告)日:1986-07-15

    申请号:BR8504584

    申请日:1985-09-19

    Applicant: CIBA GEIGY AG

    Abstract: There are described novel, microbicidally active 5-(arylmethylimino)-pyrimidines of the formula I (I) wherein Rn-A- is an unsubstituted or substituted phenyl, naphthyl, biphenyl, phenoxyphenyl or phenylthiophenyl, and R1 is an ether, thioether or amino function, these substances being produced according to the invention by substitution of the halogen atom in the claimed intermediates of the formula II (II) The use of these substances in plant protection, and also further important intermediates, are likewise described.

Patent Agency Ranking