公开(公告)号：PL366463A1

公开(公告)日：2005-02-07

申请号：PL36646302

申请日：2002-03-13

Applicant: BASF AG

Inventor： GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00

Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.

公开(公告)号：CA2532917A1

公开(公告)日：2005-02-03

申请号：CA2532917

申请日：2004-07-15

Applicant: BASF AG

Inventor： STIERL REINHARD ,  SCHERER MARIA ,  GYPSER ANDREAS ,  SPEAKMAN JOHN-BRYAN ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  RACK MICHAEL ,  GRAMMENOS WASSILIOS ,  GEWEHR MARKUS ,  WAGNER OLIVER ,  BLETTNER CARSTEN ,  GROTE THOMAS ,  SCHAEFER PETER ,  SCHOEFL ULRICH ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  STRATHMANN SIEGFRIED ,  SCHWOEGLER ANJA ,  SCHIEWECK FRANK

IPC: C07D471/04 ,  A01N43/90

Abstract: The invention relates to bicyclic compounds of general formula I, wherein X, Y independently represent N or C-R4; n stands for 1, 2, 3, 4 or 5; Rarepresent s halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl, C1-C6- halogenalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 denotes halogen , cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8- cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5- C8 cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8; R2 denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalky l, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl, optionally mono - or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8, and R3 represents hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl or C3-C6-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen. Said invention also relates to the agriculturally-acceptable salts of said compounds (I), plant protection agents, containing at least one compound of general formula (I) and/or one agriculturally-acceptable salt of (I) and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.

公开(公告)号：BR0308443A

公开(公告)日：2005-01-18

申请号：BR0308443

申请日：2003-03-19

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  FL ULRICH SCH ,  STRATHMANN SIEGFRIED ,  SCHELBERGER KLAUS ,  CHRISTEN THOMAS

IPC: A01N43/42 ,  A01N33/18 ,  A01N35/04 ,  A01N35/06 ,  A01N37/34 ,  A01N37/46 ,  A01N37/52 ,  A01N43/24 ,  A01N43/28 ,  A01N43/32 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/653 ,  A01N43/78 ,  A01N47/14 ,  A01N47/18 ,  A01N47/34 ,  B60Q1/50

Abstract: A new fungicidal mixture contains synergistic amounts of (1) prothioconazole (I) and (2) at least one of 20 other specific fungicides, e.g. boscalid, carboxine, metrafenone, quinoxyfen, fenoxanil, carbendazim, metalaxyl, prochloraz or anthraquinone. A fungicidal mixture contains synergistic amounts of the following active components: (1) prothioconazole (I) or its salt or adduct; and (2) one or more of boscalid, carboxine, metrafenone, N-(alpha -cyclopropoxyimino)-(2,3-difluoro-6-trifluoromethyl-benzyl)-phenylacetamide, N-(alpha -cyclopropoxyimino)-2,3-difluoro-6-difluoromethyl-benzyl)-phenylacetamide, quinoxyfen, dithianon, thiram, mepiquat chloride, cyazofamid, fenoxanil, 6-fluoro-2-(1-(2-(isopropoxycarbonylamino)-isovaleramido)-ethyl)-benzothiazole, thiophanate methyl, carbendazim, metalaxyl, fludioxonil, thiabendazole, quintozen, prochloraz and/or anthraquinone. Independent claims are included for: (a) a harmful fungus control method involving application of the mixture of (1) and (2) to the fungi, their habitat or plants, seeds, soil, surfaces, materials or regions to be protected ((1) and (2) being applied simultaneously, separately or successvely); and (b) a fungicidal composition comprising the (1)/(2) mixture together with a solid or liquid carrier. ACTIVITY : Fungicide. In tests for protective action against Blumeria graminis f. sp. triciti (mildew) in wheat, prothioconazole (I) at 1 ppm alone or boscalid (II) at 4 ppm alone gave no (0%) control, whereas a combination of 1 ppm (I) and 4 ppm (II) gave 92% control. MECHANISM OF ACTION : None given in the source material.

公开(公告)号：PL365819A1

公开(公告)日：2005-01-10

申请号：PL36581902

申请日：2002-01-19

Applicant: BASF AG

Inventor： PTOCK ARNE ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  REDDIG ACHIM

IPC: A01N43/50 ,  A01N43/80 ,  A01N47/12

Abstract: Fungicidal mixtures, comprising A) imidazole derivatives of the formula I in which R 1 and R 2 are halogen or phenyl, which may be substituted by halogen or alkyl, or R 1 and R 2 together with the bridging C-C double bond form a 3,4-difluoromethylenedioxyphenyl group; R 3 is cyano or halogen, and R 4 is dialkylamino or isoxazol-4-yl, which may carry two alkyl radicals; and B) valinamides of the formula II, in which R' is phenyl, which is substituted in the 4-position by halogen, C 1 -C 4 -alkyl or C 1 -C 4 -alkoxy, is 1- or 2-naphthyl, or is benzothiazol-2-yl, which is substituted in the 6-position by halogen; and R'' is C 3 -C 4 -alkyl; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II and the use of the compounds I and the compounds II for preparing such mixtures are described.

公开(公告)号：AU2004251016A2

公开(公告)日：2005-01-06

申请号：AU2004251016

申请日：2004-06-19

Applicant: BASF AG

Inventor： SCHOFL ULRICH ,  STIERL REINHARD ,  GROTE THOMAS ,  BLASCO JORDI TORMO I ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED

IPC: A01N43/90

Abstract: Fungicidal mixtures for controlling rice pathogens, comprising, as active components, 1) the triazolopyrimidine derivative of the formula I, and 2) an acryloylmorpholide of the formula II, in which X is chlorine or fluorine, in a synergistically effective amount, methods for controlling rice pathogens using mixtures of the compound I with the compounds II, the use of the compound I and the compounds II for preparing such mixtures and compositions comprising these mixtures are described.

公开(公告)号：AU2004251015A1

公开(公告)日：2005-01-06

申请号：AU2004251015

申请日：2004-06-19

Applicant: BASF AG

Inventor： STIERL REINHARD ,  GROTE THOMAS ,  HADEN EGON ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  HAMPEL MANFRED ,  BLASCO JORDI TORMO I ,  SCHOFL ULRICH

IPC: A01N43/90

Abstract: Fungicidal mixtures, comprising, as active components 1) the triazolopyrimidine derivative of the formula I, and 2) dithianon of the formula II, in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with the compound II and the use of the compound I with the compound II for preparing such mixtures and compositions comprising these mixtures are described.

公开(公告)号：HRP20040985A2

公开(公告)日：2004-12-31

申请号：HRP20040985

申请日：2004-10-20

Applicant: BASF AG

Inventor： BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  C07C255/57 ,  C07D487/04 ,  C07C323/62

Abstract: The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L 1 represents cyano, S(-O) n A 1 or C(-O)A 2 , wherein A 1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A 2 stands for C 1 -C 8 alkoxy, C 1 -C 6 haloalkoxy or one of the groups named in A 1 ; and n stands for 0, 1 or 2; L 2 , L 3 represent hydrogen or halogen; L 4 , L 5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R 1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R 2 represents hydrogen or R 1 ; R 1 and R 2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R 1 and/or R 2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.

公开(公告)号：BR0307912A

公开(公告)日：2004-12-21

申请号：BR0307912

申请日：2003-02-26

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  SCHELBERGER KLAUS ,  SPADAFORA V JAMES ,  CHRISTEN THOMAS

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/40 ,  A01N43/653 ,  A01N43/84

Abstract: A fungicidal mixture comprising (1) 2-[2-(1-chlorocyclopropyl)-3-(2-chlorophenyl)-2-hydroxy-propyl]-2,4-dihydro-[1,2,4]-triazole-3-thione (prothioconazole) of the formula I or a salt or adduct thereof and at least one further fungicide or a salt or adduct thereof selected from the group consisting of (2) fenpropimorph of the formula II and (3) tridemorph of the formula III n=10, 11, 12 (60-70%) or 13 and (4) fenpropidin of the formula IV in a synergistically effective amount is described.

公开(公告)号：CA2527136A1

公开(公告)日：2004-12-09

申请号：CA2527136

申请日：2004-05-27

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  RHEINHEIMER JOACHIM ,  SPEAKMAN JOHN-BRYAN ,  BLETTNER CARSTEN ,  RACK MICHAEL ,  GROTE THOMAS ,  WAGNER OLIVER ,  GRAMMENOS WASSILIOS ,  STRATHMANN SIEGFRIED ,  MUELLER BERND ,  SCHERER MARIA ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  AKERS ALAN ,  TORMO I BLASCO JORDI ,  SCHAEFER PETER ,  GYPSER ANDREAS ,  SCHWOEGLER ANJA ,  SCHIEWECK FRANK

IPC: C07D487/04 ,  A01N43/90

Abstract: The invention relates to substituted pyrazolopyrimidines of formula (I) wherein the substituents have the following designations: L represents halogen, alkyl, halogenalkyl, alkenyl, alkoxy, amino, NHR, NR2, cyano, S(=O)nA1 or C(=O)A2, R representing alkyl or alkylcarbonyl, A1 representing hydrogen, hydroxy, alkyl, alkylamino or dialkylamino, n representing 0, 1 or 2, and A2 representing alkenyl, alkoxy, halogenalkoxy or one of the groups cited for A1; m represents 0 or 1 to 5; R1 represents alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, alkadienyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, phenyl, naphthyl, or a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; and R2 represents hydrogen or one of the groups cited for R1. Together wi th the nitrogen atom to which they are bonded, R1 and R2 can form a five-member ed to six-membered ring that can be interrupted by an atom from the groups O, N and S, and R1 and/or R2 can also be substituted according to the description . Furthermore, in formula (I): X represents halogen, cyano, OH, alkyl, alkoxy or halogenalkoxy; Y represents a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle according to the description, or a group X or another group according to the description; p represents 1 or 2 , the groups Y being potentially different when p = 2; and p represents 0, whe n X is according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing the same, and the use thereof for controlling phytopathogenic fungi.

公开(公告)号：CA2526155A1

公开(公告)日：2004-12-02

申请号：CA2526155

申请日：2004-05-15

Applicant: BASF AG

Inventor： HADEN EGON ,  SCHERER MARIA ,  STIERL REINHARD ,  GROTE THOMAS ,  HAMPEL MANFRED ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  TORMO I BLASCO JORDI

IPC: A01N43/90 ,  A01N37/50

Abstract: The invention relates to fungicidal mixtures containing the following as active components: 1) dimoxystrobin of formula (I) and 2) the compound of formula (II) in synergistically active quantities. The invention also relate s to a method for controlling harmful fungi using a mixture of compounds (I) a nd (II), to the use of the compounds (I) and (II) for producing mixtures of thi s type and to agents containing said mixtures.