New 7-amino-6-phenyl-triazolopyrimidine derivatives are broad-spectrum fungicides useful in protection of plants or materials such as wood

    公开(公告)号:DE10257394A1

    公开(公告)日:2004-06-24

    申请号:DE10257394

    申请日:2002-12-06

    Applicant: BASF AG

    Abstract: 2,5-Disubstituted-7-amino-6-phenyl-(1,2,4)-triazolo(1,5-a)pyrimidine derivatives (I) are new. 2,5-Disubstituted-7-amino-6-phenyl-(1,2,4)-triazolo(1,5-a)pyrimidine derivatives of formula (I) are new. L = halogen, CN, NO2, alkyl, 2-10C alkenyl, 2-10C alkynyl, 2-10C alkynyl, haloalkyl, 2-10C haloalkenyl, alkoxy, 2-10C alkenyloxy, 2-10C alkynyloxy, haloalkoxy, C(O)A or S(O)pA'; A = H, OH, 1-8C alkyl, 2-8C alkenyl, 1-8C alkoxy, haloalkoxy or mono- or di-(1-8C alkyl)amino; A' = H, 1-8C alkyl or haloalkyl; m = 0-5; X = CN, 1-4C alkyl, 1-4C haloalkyl, 1-4C alkoxy or 1-2C haloalkoxy; R1, R2 = H or 1-8C alkyl, 1-8C haloalkyl, cycloalkyl, halocycloalkyl, 2-8C alkenyl, 4-10C alkadienyl, 2-8C haloalkenyl, cycloalkenyl, 2-8C alkynyl, 2-8C haloalkynyl, cycloalkynyl, phenyl, naphthyl, 5- or 6-membered heteroaryl or 5-10 membered saturated, partially unsaturated or aromatic heterocyclyl (containing 1-4 of O, N and/or S), all optionally substituted (os) by 1-4 Ra; or NR1R2 = 5 or 6 membered heterocycle optionally containing an additional O, N or S heteroatom, os by one or more halogen, alkyl, haloalkyl or 1-3C alkylenedioxy and/or optionally having an N and an adjacent C linked by a 1-4C alkylene chain; Ra = halogen, CN, NO2, OH, alkyl, haloalkyl, alkylcarbonyl, cycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, alkoxycarbonyl, alkenyl, alkenyloxy, 3-6C alkynyloxy, cycloalkyl, phenyl, naphthyl or 5-10 membered saturated, partially unsaturated or aromatic heterocyclyl containing 1-4 of O, N and/or S, where cyclic residues are optionally partially or completely halogenated and os by 1-3 Rb; Rb = halogen, CN, NO2, OH, SH, NH2, COOH, C(O)NH2, C(S)NH2, alkyl, haloalkyl, 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, alkoxy, haloalkoxy, alkylthio, mono- or dialkylamino, CHO, alkylcarbonyl, alkylsulfonyl, alkylsulfoxyl, alkylcarbonyl, alkylcarbonyloxy, mono- or dialkylaminocarbonyl, mono- or dialkylaminothiocarbonyl, 3-10C cycloalkyl, 3-10C cycloalkoxy, 3-10 membered heterocyclyl, 3-10 membered heterocyclyloxy, aryl, aryloxy, arylthio, arylalkoxy, arylalkyl (where all aryl moieties are preferably 6-10 membered), 5 or 6 membered heteroaryl, 5 or 6 membered heteroaryloxy or 5 or 6 membered heteroarylthio (where all rings are optionally partially or completely halogenated and os by alkyl or haloalkyl (for which no C-numbers are specified)); R3 = CN, OH, 1-8C alkoxy, 3-8C alkenyloxy, 1-8C haloalkoxy, 3-8C haloalkenyloxy, NR1R2 or S(O)nR31; n, p = 0-2; and R31 = H, OH, 1-8C alkyl, 2-8C alkenyl or C(O)A. Unless specified otherwise alkyl moieties have 1-6C, alkenyl moieties 2-6C and cycloalkyl, cycloalkenyl or cycloalkynyl moieties 3-6C. Independent claims are included for the preparation of (I).

Patent Agency Ranking