公开(公告)号：DE19804486A1

公开(公告)日：1999-08-12

申请号：DE19804486

申请日：1998-02-05

Applicant: BASF AG

Inventor： PTOCK ARNE DR ,  SAUTER HUBERT DR ,  KIRSTGEN REINHARD DR ,  GRAMMENOS WASSILIOS DR ,  GROTE THOMAS DR ,  GYPSER ANDREAS DR ,  BAYER HERBERT DR ,  GEWEHR MARKUS DR ,  CULLMANN OLIVER DR RER NAT ,  MUELLER BERND DR ,  GOETZ ROLAND DR ,  ROEHL FRANZ DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR ,  HARRIES VOLKER DR ,  STRATHMANN SIEGFRIED DR

IPC: A01N43/48 ,  A01N43/56 ,  C07D401/12 ,  C07D401/14 ,  A61K31/44

Abstract: The present invention relates to compounds of the general formula (I) and to the salts thereof, wherein the substituents and the n index have the following values: Q represents -C(=CHCH3)-COOCH3, -C(=CHOCH3)-COOCH3, -C(=NOCH3)-COOCH3 or -C(=NOCH3)-CONH(CH3); R represents hydrogen, halogen, C1-C4 alkyl, C1-C2 halogenalkyl, C1-C4 alkoxy or C1-C2 halogenalkoxy; R represents halogen, C1-C4 alkyl, C1-C2 halogenalkyl or C1-C4 alkoxy; n is 0, 1 or 2, wherein the R substituents can be different when n = 2; and R represents phenyl, pyridyle or pyrimidyle. This invention also relates to agents containing these compounds as well as to the use of said compounds (I) and agents against noxious fungi and animal parasites.

公开(公告)号：DE19756115A1

公开(公告)日：1999-06-24

申请号：DE19756115

申请日：1997-12-17

Applicant: BASF AG

Inventor： MUELLER BERND DR ,  SAUTER HUBERT DR ,  BAYER HERBERT DR ,  GEWEHR MARKUS DR ,  GRAMMENOS WASSILIOS DR ,  GROTE THOMAS DR ,  GYPSER ANDREAS DR ,  PTOCK ARNE DR ,  ROEHL FRANZ DR ,  GOETZ NORBERT DR ,  GOETZ ROLAND DR ,  HARRIES VOLKER DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR ,  STRATHMANN SIEGFRIED DR

IPC: A01N43/48 ,  C07C243/22 ,  C07D231/22 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  A01N43/56

Abstract: The invention relates to substituted phenylpyrazolones of formula (I) in which the substituents have the following meanings: Y represents halogen, alkyl, halogen alkyl or alkoxyl; n represents 0, 1 or 2, whereby the radical Y can be different when n = 2; E represents a group A (A), whereby # characterizes the bond with the phenyl ring; R represents halogen, cyano, alkyl or halogen alkyl; R represents hydrogen or alkyl; R represents alkyl or halogen alkyl; T represents a direct bond, oxygen or CH2O; Z represents a) when T represents oxygen or oxymethylene, a group X, N=CWR or N=C(R )-C(R )=NOR , whereby X represents optionally substituted heterocyclyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted arylmethylene or optionally substituted heteroarylmethylene; W represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkinyl, optionally substituted cycloalkyl, optionally substituted cycloalkenyl, optionally substituted heterocyclyl, optionally substituted aryl or optionally substituted heteroaryl; R represents hydrogen, cyano, alkyl, halognealkyl, alkoxyl, alkoxyl alkyl, cycloalkyl; R represents hydrogen, cyano, halogen, C(R )=NOR or W, OW, SW or NR W, whereby R represents hydrogen, alkyl, alkenyl or alkinyl; R represents hydrogen or alkyl; R represents hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkinyl, and b) when T represents a direct bond, Z represents a group W, CH2-CH2-W, CH=CH-W, CC-W, S-W, CH2-S-W, CH=N-O-CH2-W, CH2-O-C(=O)-W or CH2-O-C(CH3)=N-N=C(CH3)-W. The invention also relates to a method and intermediate products for the production of said phenylpyrazolones used for combating parasitic fungi and animal parasites.

公开(公告)号：CZ9801686A3

公开(公告)日：1998-09-16

申请号：CZ168698

申请日：1996-12-11

Applicant: BASF AG

Inventor： OBERDORF KLAUS DR ,  GRAMMENOS WASSILIOS DR ,  SAUTER HUBERT DR ,  GROTE THOMAS DR ,  KIRSTGEN REINHARD DR ,  MULLER RUTH DR ,  MULLER BERND DR ,  ROHL FRANZ DR ,  RACK MICHAEL DR ,  BAYER HERBERT DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR ,  STRATHMANN SIEGFRIED DR ,  HARRIES VOLKER DR

IPC: C07D239/26 ,  A01N43/54 ,  A01N47/20 ,  A01N47/24 ,  A01P3/00 ,  C07D239/28 ,  C07D239/34 ,  C07D239/38

CPC classification number: C07D239/34 ,  A01N43/54

公开(公告)号：CZ176598A3

公开(公告)日：1998-09-16

申请号：CZ176598

申请日：1996-12-16

Applicant: BASF AG

Inventor： GROTE THOMAS DR ,  SAUTER HUBERT DR ,  KIRSTGEN REINHARD DR ,  BAYER HERBERT DR ,  MULLER RUTH DR ,  MULLER BERND DR ,  OBERDORF KLAUS DR ,  GRAMMENOS WASSILIOS DR ,  GOTZ NORBERT DR ,  RACK MICHAEL DR ,  HARREUS ALBRECHT DR ,  ROHL FRANZ DR ,  AMMERMANN EBERHARD DR ,  HARRIES VOLKER DR ,  LORENZ GISELA DR ,  STRATHMANN SIEGFRIED DR

IPC: C07C249/04 ,  A01N37/50 ,  A01N43/40 ,  A01P3/00 ,  A01P7/00 ,  C07C251/50 ,  C07C251/56 ,  C07C251/58 ,  C07C251/60 ,  C07C255/40

公开(公告)号：CZ9801099A3

公开(公告)日：1998-07-15

申请号：CZ109998

申请日：1996-09-30

Applicant: BASF AG

Inventor： BAYER HERBERT DR ,  SAUTER HUBERT DR ,  OBERDORF KLAUS DR ,  GRAMMENOS WASSILIOS DR ,  GROTE THOMAS DR ,  KIRSTGEN REINHARD DR ,  MULLER BERND DR ,  MULLER RUTH DR ,  ROHL FRANZ DR ,  AMMERMANN EBERHARD DR ,  HARRIES VOLKER DR ,  LORENZ GISELA DR ,  STRATHMANN SIEGFRIED DR ,  GOTZ NORBERT DR ,  RACK MICHAEL DR

IPC: C07C249/16 ,  A01N35/10 ,  A01N37/50 ,  A01N43/40 ,  A01N43/80 ,  A01N59/12 ,  C07C251/88 ,  C07D213/53 ,  C07D261/08

CPC classification number: C07D213/53 ,  A01N37/50 ,  C07C251/88 ,  C07D261/08

公开(公告)号：DE59209319D1

公开(公告)日：1998-06-10

申请号：DE59209319

申请日：1992-01-24

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS DR ,  HARREUS ALBRECHT DR ,  SAUTER HUBERT DR ,  HELLENDAHL BEATE DR ,  DOETZER REINHARDT DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N37/50 ,  A01N43/54 ,  A01N43/58 ,  A01N43/76 ,  A01N43/836 ,  C07C69/65 ,  C07C69/653 ,  C07C69/734 ,  C07C69/738 ,  C07C251/48 ,  C07C251/50 ,  C07C251/52 ,  C07C251/54 ,  C07C251/56 ,  C07C251/58 ,  C07C251/60 ,  C07C251/86 ,  C07C255/15 ,  C07C255/57 ,  C07C255/58 ,  C07C255/62 ,  C07D213/77 ,  C07D239/42 ,  C07D241/20 ,  C07D263/32 ,  C07D333/28

Abstract: Iminoalkyl-phenylacrylic acid derivs. (I) ar new: R = H or 1-6C alkyl; R = H; 1-4C alkyl opt. substd. by halo; or opt. substd. aryl; Z ,Z = H; halo; CN; NO2;etc.;Y = O; NH; or NR ; and R = H; 1-4C alkoxycarbonyl-1-4C alkyl; or opt. substd. alkyl, cycloalkyl, etc.; or Y+R form a ring which is opt. substd. when Y = NH or NR ; R = 1-6C alkyl; X = CH-1-4C alkoxy or CH-1-4C alkylthio (also 1-4C alkylidene and 1-4C alkoxyimino in the description).

公开(公告)号：DE19620392A1

公开(公告)日：1997-11-27

申请号：DE19620392

申请日：1996-05-21

Applicant: BASF AG

Inventor： OBERDORF KLAUS DR ,  GRAMMENOS WASSILIOS DR ,  SAUTER HUBERT DR ,  GROTE THOMAS DR ,  KIRSTGEN REINHARD DR ,  MUELLER RUTH DR ,  MUELLER BERND DR ,  ROEHL FRANZ DR ,  RACK MICHAEL DR ,  BAYER HERBERT DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR ,  STRATHMANN SIEGFRIED DR ,  HARRIES VOLKER DR

IPC: C07D239/34 ,  A01N37/18 ,  A01N43/54

Abstract: 2-(pyrimidin-4-yloxy)methyl)phenylacetic acid derivatives of formula (I) and their salts and N-oxides are new. R1 = H or 1-4C alkyl; R2 = halo, CH3, CH2CH3, halomethyl or haloethyl; R3 = phenyl, phenoxy, phenoxymethyl, benzyloxy or heteroaryl, (all optionally ring-substituted), H, amino, OH, SH, halo, 1-8C alkyl (optionally substituted by Ar or halo), alkoxy-(1-4C alkyl), alkoxy, mono- or di- alkylamino, alkylthio, alkylsulphoxy, alkylsulphonyl, 3-8C cycloalkyl, trialkylsilyloxy; Ar = phenyl (optionally mono- or di-substituted by halo, CN, NO2, 1-4C alkyl, 1-4C haloalkyl or 1-4C alkoxy); R4 = H, CN, halo, 1-4C alkyl, 1-4C haloalkyl or 1-4C alkoxy; Q = C(=NOCH3)CONHCH3, C(=NOCH3)COOCH3 or N(OCH3)COOCH3; alkyl, alkoxy have 1-8 C unless specified otherwise.

公开(公告)号：DE59403764D1

公开(公告)日：1997-09-25

申请号：DE59403764

申请日：1994-04-13

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS DR ,  SIEGEL WOLFGANG DR ,  OBERDORF KLAUS DR ,  MUELLER BERND DR ,  SAUTER HUBERT DR ,  DOETZER REINHARD DR

IPC: C07B61/00 ,  C07C45/46 ,  C07C45/48 ,  C07C49/84 ,  C07C65/40 ,  C07C67/313 ,  C07C69/734 ,  C07C69/736 ,  C07C235/34 ,  C07C235/80 ,  C07C251/48 ,  C07C255/54 ,  C07D213/50

Abstract: The process is characterised in that 4-alkanoylaryl benzyl ethers of the general formula I where the variables have the following meaning: R is hydrogen, halogen, cyano; alkyl, alkoxy; X is CH2, CH-CH3, CH-CH2-CH3, CH-OCH3, N-OCH3; Y is oxygen, sulphur, a direct bond or nitrogen; m is 0, 1, 2 or 3; R is hydrogen; alkyl, alkenyl, alkynyl, alkoxy; R is cyano, halogen, alkyl, alkoxy, haloalkyl; R is alkyl, haloalkyl; cycloalkyl; or an optionally substituted mono- to trinuclear aromatic system, are prepared by reacting an aryl benzyl ether of the general formula II where X, Y, R, R , R and m have the abovementioned meaning, with a carboxylic acid halide or with a carboxylic anhydride or with a carboxylic - sulphonic anhydride in the presence of an acid and optionally in the presence of a diluent.

公开(公告)号：DE59108832D1

公开(公告)日：1997-09-25

申请号：DE59108832

申请日：1991-12-10

Applicant: BASF AG

Inventor： WINGERT HORST DR ,  WOLF BERND DR ,  BENOIT REMY DR ,  SAUTER HUBERT DR ,  HEPP MICHAEL DR ,  GRAMMENOS WASSILIOS DR ,  KUEKENHOEHNER THOMAS DR

IPC: C07C69/736 ,  C07C20060101 ,  C07C51/09 ,  C07C51/367 ,  C07C59/68 ,  C07C65/21 ,  C07C65/24 ,  C07C67/22 ,  C07C69/738 ,  C07C69/76 ,  C07C235/34 ,  C07C235/78 ,  C07C249/08 ,  C07C251/48 ,  C07C253/14 ,  C07C255/17 ,  C07C255/40 ,  C07C317/24

Abstract: Prepn. of 2-phenoxymethyl benzoic acid derivs. of formula (I) comprises (a) converting a phenol of formula (II) to the phenolate in the presence of a basic diluent; (b) mixing the mixt. with a lactone of formula (III); (c) distilling off the diluent; (d) reacting the mixt. at 50-250 degrees C in the melt; and (e) dissolving the liq. melt with water and acidifying. X, Y = halogen, 1-4C alkyl, 1-4C alkoxy or CF3; m = 0-4; n = 0-3.

公开(公告)号：DK0621264T3

公开(公告)日：1997-09-15

申请号：DK94105661

申请日：1994-04-13

Applicant: BASF AG

Inventor： SIEGEL WOLFGANG DR ,  SAUTER HUBERT DR ,  OBERDORF KLAUS DR ,  MUELLER BERND DR ,  GRAMMENOS WASSILIOS DR ,  DOETZER REINHARD DR

IPC: C07B61/00 ,  C07C45/46 ,  C07C45/48 ,  C07C49/84 ,  C07C65/40 ,  C07C67/313 ,  C07C69/734 ,  C07C69/736 ,  C07C235/34 ,  C07C235/80 ,  C07C251/48 ,  C07C255/54 ,  C07D213/50

Abstract: The process is characterised in that 4-alkanoylaryl benzyl ethers of the general formula I where the variables have the following meaning: R is hydrogen, halogen, cyano; alkyl, alkoxy; X is CH2, CH-CH3, CH-CH2-CH3, CH-OCH3, N-OCH3; Y is oxygen, sulphur, a direct bond or nitrogen; m is 0, 1, 2 or 3; R is hydrogen; alkyl, alkenyl, alkynyl, alkoxy; R is cyano, halogen, alkyl, alkoxy, haloalkyl; R is alkyl, haloalkyl; cycloalkyl; or an optionally substituted mono- to trinuclear aromatic system, are prepared by reacting an aryl benzyl ether of the general formula II where X, Y, R, R , R and m have the abovementioned meaning, with a carboxylic acid halide or with a carboxylic anhydride or with a carboxylic - sulphonic anhydride in the presence of an acid and optionally in the presence of a diluent.