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    4.
    发明专利
    未知

    公开(公告)号：DE19756115A1

    公开(公告)日：1999-06-24

    申请号：DE19756115

    申请日：1997-12-17

    Applicant: BASF AG

    Inventor： MUELLER BERND DR ,  SAUTER HUBERT DR ,  BAYER HERBERT DR ,  GEWEHR MARKUS DR ,  GRAMMENOS WASSILIOS DR ,  GROTE THOMAS DR ,  GYPSER ANDREAS DR ,  PTOCK ARNE DR ,  ROEHL FRANZ DR ,  GOETZ NORBERT DR ,  GOETZ ROLAND DR ,  HARRIES VOLKER DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR ,  STRATHMANN SIEGFRIED DR

    IPC: A01N43/48 ,  C07C243/22 ,  C07D231/22 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  A01N43/56

    Abstract: The invention relates to substituted phenylpyrazolones of formula (I) in which the substituents have the following meanings: Y represents halogen, alkyl, halogen alkyl or alkoxyl; n represents 0, 1 or 2, whereby the radical Y can be different when n = 2; E represents a group A (A), whereby # characterizes the bond with the phenyl ring; R represents halogen, cyano, alkyl or halogen alkyl; R represents hydrogen or alkyl; R represents alkyl or halogen alkyl; T represents a direct bond, oxygen or CH2O; Z represents a) when T represents oxygen or oxymethylene, a group X, N=CWR or N=C(R )-C(R )=NOR , whereby X represents optionally substituted heterocyclyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted arylmethylene or optionally substituted heteroarylmethylene; W represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkinyl, optionally substituted cycloalkyl, optionally substituted cycloalkenyl, optionally substituted heterocyclyl, optionally substituted aryl or optionally substituted heteroaryl; R represents hydrogen, cyano, alkyl, halognealkyl, alkoxyl, alkoxyl alkyl, cycloalkyl; R represents hydrogen, cyano, halogen, C(R )=NOR or W, OW, SW or NR W, whereby R represents hydrogen, alkyl, alkenyl or alkinyl; R represents hydrogen or alkyl; R represents hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkinyl, and b) when T represents a direct bond, Z represents a group W, CH2-CH2-W, CH=CH-W, CC-W, S-W, CH2-S-W, CH=N-O-CH2-W, CH2-O-C(=O)-W or CH2-O-C(CH3)=N-N=C(CH3)-W. The invention also relates to a method and intermediate products for the production of said phenylpyrazolones used for combating parasitic fungi and animal parasites.

    New phenyl carbamate derivatives
    5.
    发明专利
    New phenyl carbamate derivatives 未知

    公开(公告)号：DE19745650A1

    公开(公告)日：1999-04-22

    申请号：DE19745650

    申请日：1997-10-16

    Applicant: BASF AG

    Inventor： BAYER HERBERT DR ,  GEWEHR MARKUS DR ,  GROTE THOMAS DR ,  MUELLER BERND DR ,  SAUTER HUBERT DR ,  GRAMMENOS WASSILIOS DR ,  GYPSER ANDREAS DR ,  PTOCK ARNE DR ,  GOETZ ROLAND DR ,  RACK MICHAEL DR ,  AMMERMANN EBERHARD DR ,  HARRIES VOLKER DR ,  LORENZ GISELA DR ,  STRATHMANN SIEGFRIED DR ,  ROEHL FRANZ DR

    IPC: A01N43/82 ,  A01N43/836 ,  C07C259/14 ,  C07C265/12 ,  C07D271/06 ,  C07D271/07 ,  C07D413/12 ,  C07C251/40 ,  C07D413/04 ,  C07D413/14

    Abstract: Substituted oxy- or oxymethylenephenyl-oxazolidine and -oxazolidinedione derivatives (I) are new. They are prepared from new activated phenyl-oxazolidine derivatives (IIA) and activated phenyl-oxazolidinedione derivatives (IVB), which in turn are obtained via new substituted nitrobenzene and aniline derivatives (1), phenyl isocyanates (2) and substituted anilides (3). Substituted oxy- or oxymethylenephenyl-oxazolidine and -oxazolidinedione derivatives (I) are new: Y = halo; 1-4C alkyl; 1-4C haloalkyl; or 1-4C alkoxy; n = 0-2; E = group of formula (a) or (b): Ra = halo; CN; 1-4C alkyl or 1-4C alkoxy optionally substituted by halo; 3-6C alkenyloxy, 3-6C alkynyloxy; 3-6C cycloalkyl; S(O)m-1-4C alkyl; or NRaRb; m = 0-2; Ra and Rb = H; 1-4C alkyl; 3-6C alkenyl; or 3-6C alkynyl; Rb = 1-4C alkyl; 1-4C haloalkyl; 3-6C cycloalkyl; or optionally substituted arylmethylene; T = O or oxymethylene; Z' = X; N=CWR ; or N=C(R )-C(R )=NOR ; X = optionally substituted heterocyclyl, aryl, heteroaryl, arylmethylene or heteroarylmethylene; W = optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, heterocyclyl, aryl or heteroaryl; R = H; CN; 1-4C alkyl; 1-4C haloalkyl; 1-4C alkoxy; 1-4C alkoxy-1-4C alkyl; or 3-6C cycloalkyl; R = H; CN; halo; C(Rd)=NOR3; W; OW; SW or NRcW; Rc = H; alk yl; alkenyl; or alkynyl; Rd = H or alkyl; R = H; or optionally substituted alkyl, alkenyl or alkynyl. Independent claims are also included for: (A) activated phenyl-oxazolidine derivatives of formula (IIA); (B) activated phenyl-oxazolidinedione derivatives of formula (IVB); (C) substituted nitrobenzene and aniline derivatives of formula (1); (D) phenyl isocyanates of formula (2); and (E) Substituted anilides (3). L = OH; CH3; CH2L'; or L'; L' = nucleophilic leaving group; La = CH3; CH2L'; NO2; alkylsulphonate; or arylsulphonate; Q = NH2 or NO2; T' = OZ'; CH2O-X; or CH2O-N=C(R )-C(R )=NOR ; Z' = N=CWR or N=C(R )-C(R )=NOR ; E asterisk = NH-C(O)-NH-OH; NH-C(O)-O-NH-C(O)-OR; NH-C(S)-R'; or NH-C(NOH)-R'; R = 1-4C alkyl; R' = 1-4C alkyl; 1-4C haloalkyl; or 3-6C cycloalkyl.

    New 3-aryl-methyl-uracil derivatives
    9.
    发明专利
    New 3-aryl-methyl-uracil derivatives 未知

    公开(公告)号：DE19738084A1

    公开(公告)日：1999-03-04

    申请号：DE19738084

    申请日：1997-09-01

    Applicant: BASF AG

    Inventor： MENKE OLAF DR ,  GOETZ ROLAND DR ,  RACK MICHAEL DR ,  HAMPRECHT GERHARD DR ,  MENGES MARKUS DR ,  REINHARD ROBERT DR ,  SCHAEFER PETER DR ,  ZAGAR CYRILL DR ,  WESTPHALEN KARL-OTTO DR ,  WALTER HELMUT DR ,  MISLITZ ULF DR

    IPC: A01N43/80 ,  C07D405/06 ,  C07D413/06 ,  C07D417/06 ,  C07F9/6584 ,  C07D239/54 ,  A01N43/54 ,  A01N43/84 ,  A01N57/02 ,  C07D403/06 ,  C07F9/6564 ,  C07F9/6571

    Abstract: 3-Arylmethyluracil derivatives (I.1)-(I.4) are new, where A = H, 1-4C alkyl, NH2, 1-4C alkylamino or di-(1-4C alkyl)amino; X = O or S; n = not defined; R1 = 1-4C haloalkyl; R2 = H, halo or 1-3C alkyl; R3-R5 = H, CN, thiocyanato, halo, 1-4C haloalkyl, 1-4C haloalkoxy, 1-4C haloalkylthio, 1-4C alkyl or 1-4C alkoxy; R6, R7 = 1-4C alkyl, NH2, 1-4C alkylamino or di(1-4C alkyl)amino, or R6 and R7 together form =O; R8 may be in position alpha or beta and R3 is in the other position; R8 = (1) H, halo, amino, 1-4C alkylsulphonylamino or di(1-4C alkyl)amino; (2) 1-6C alkoxy, 1-6C alkylthio, 3-6C cycloalkoxy, 3-6C cycloalkylthio, 2-6C alkenyloxy, 5-7C cycloalkenyloxy, 2-6C alkenylthio, 2-6C alkynyloxy, 2-6C alkynylthio, (1-6C alkyl)carbonyloxy, (1-6C alkyl)carbonylthio, (1-6C alkoxy)carbonyloxy, (2-6C alkenyl)carbonyloxy, (2-6C alkenyl)carbonylthio, (2-6C alkynyl)carbonyloxy, (2-6C alkynyl)carbonylthio, 1-6C alkylsulphonyloxy or 1-6C alkylsulphonyl, where the last 18 groups may contain 1-4 substituents; (3) CT-R11, C(R11)(Y1R12)(Y2R13), C(R11)=C(R14)CN, C(R11)=C(R14)CO-R15, CH(R11)-CH(R14)CO-R15, C(R11)=C(R14)-CH2-CO-R15, C(R11)=C(R14)-C(R16)=C(R17)-CO-R15, C(R11)=C(R14)-CH2-CH(R18)CO-R15, CO-OR19, CO-SR19, CO-N(R19)-OR20, C?=C-CO-NH-OR20, C?=C-CO-N(R19)-OR20, , C?=C-CS-NH-OR20, C?=C-CS-N(R19)-OR20, C(R11)=C(R14)-CO-NH-OR20, C(R11)=C(R14)-CO-N(R19)-OR20, C(R11)=C(R14)-CS-NH-OR20, C(R11)=C(R14)-CS-N(R19)-OR20, C(R11)=C(R14)-C(R21)=N-OR20, C(R21)=N-OR20, C?=C-C(R21)=N-OR20, C(Y1R12)(Y2R13)-OR19, C(Y1R12)(Y2R13)-SR19, C(Y1R12)(Y2R13)-N(R23)(R24), N(R23)(R24), CO-N(R23)(R24), or groups of formula (i), (ii), -C?=C-(i), -C?=C-(ii), -C(R11)=C(R14)-(i) or -C(R11)=C(R14 )-(ii); Y1, Y2 = S or O; theta = 1-3C alkylene optionally substituted by 1-6C alkyl; R11 = H, CN, 1-6C alkyl, 1-6C haloalkyl, 2-6C alkenyl, 2-6C alkynyl, 3-6C cycloalkyl, 1-6C alkoxy-(1-6C alkyl) or (1-6C alkoxy)carbonyl; R12, R13 = 1-6C alkyl, 1-6C haloalkyl, 3-6C alkenyl, 3-6C alkynyl or 1-6C alkoxy-(1-6C alkyl) or R12 and R13 together form a 2-4 membered carbon chain which is optionally substituted and can contain non-adjacent O, S or N atoms instead of C atoms or be condensed or form a spiro attachment with a 3-7 membered ring; R14 = H, CN, halo, 1-6C alkyl, 1-6C haloalkyl, 1-6C alkoxy, (1-6C alkyl)carbonyl or (1-6C alkoxy)carbonyl; R15 = H, OR22, SR22, 1-6C alkyl (optionally substituted by one or two 1-6C alkoxy groups), 2-6C alkenyl, 2-6C alkynyl, 1-6C haloalkyl, 3-6C cycloalkyl, 1-6C alkylthio-(1-6C alkyl), 1-6C alkyliminooxy, N(R23)(R24) or optionally substituted phenyl; R22 has the same meanings as R19; R16 = H, CN, halo, 1-6C alkyl, 3-6C alkenyl, 3-6C alkynyl, 1-6C alkoxy-(1-6C alkyl), (1-6C alkyl)carbonyl, (1-6C alkoxy)carbonyl, N(R25)(R26) or optionally substituted phenyl; R25, R26 have the same meanings as R23 and R24; R17 = H, halo, CN, 1-6C alkyl, 1-6C alkoxy, 1-6C haloalkyl, (1-6C alkyl)carbonyl or (1-6C alkoxy)carbonyl; R18 = H, CN, 1-6C alkyl or (1-6C alkoxy)carbonyl; R19 = H, 1-6C alkyl, 1-6C haloalkyl, 2-6C alkenyl or 2-6C alkynyl (where the latter four groups are optionally substituted), (1-6C alkyl)carbonyl, (1-6C haloalkyl)carbonyl, (1-6C alkoxy)carbonyl, 1-6C alkylaminocarbonyl, di-(1-6C alkyl)aminocarbonyl, 1-6C alkoxyimino-(1-6C alkyl), 3-6C cycloalkyl, phenyl or phenyl-(1-6C alkyl), where the phenyl ring is optionally substituted; R20 = H, 1-6C alkyl, 1-6C haloalkyl, 3-6C cycloalkyl, 3-6C alkenyl, 3-6C alkynyl, hydroxy-(1-6C alkyl), 1-6C alkoxy-(1-6C alkyl), 1-6C alkylthio-(1-6C alkyl), cyano-(1-6C alkyl), (1-6C alkyl)carbonyl-(1-6C alkyl), (1-6C alkoxy)carbonyl-(1-6C alkyl), (1-6C alkoxy)carbonyl-(2-6C alkenyl), (1-6C alkyl)carbonyloxy-(1-6C alkyl) or phenyl-(1-6C alkyl), where the phenyl ring may contain 1-3 substituents; R

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