6.
    发明专利
    未知

    公开(公告)号:DE19756115A1

    公开(公告)日:1999-06-24

    申请号:DE19756115

    申请日:1997-12-17

    Applicant: BASF AG

    Abstract: The invention relates to substituted phenylpyrazolones of formula (I) in which the substituents have the following meanings: Y represents halogen, alkyl, halogen alkyl or alkoxyl; n represents 0, 1 or 2, whereby the radical Y can be different when n = 2; E represents a group A (A), whereby # characterizes the bond with the phenyl ring; R represents halogen, cyano, alkyl or halogen alkyl; R represents hydrogen or alkyl; R represents alkyl or halogen alkyl; T represents a direct bond, oxygen or CH2O; Z represents a) when T represents oxygen or oxymethylene, a group X, N=CWR or N=C(R )-C(R )=NOR , whereby X represents optionally substituted heterocyclyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted arylmethylene or optionally substituted heteroarylmethylene; W represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkinyl, optionally substituted cycloalkyl, optionally substituted cycloalkenyl, optionally substituted heterocyclyl, optionally substituted aryl or optionally substituted heteroaryl; R represents hydrogen, cyano, alkyl, halognealkyl, alkoxyl, alkoxyl alkyl, cycloalkyl; R represents hydrogen, cyano, halogen, C(R )=NOR or W, OW, SW or NR W, whereby R represents hydrogen, alkyl, alkenyl or alkinyl; R represents hydrogen or alkyl; R represents hydrogen, optionally substituted alkyl, optionally substituted alkenyl or optionally substituted alkinyl, and b) when T represents a direct bond, Z represents a group W, CH2-CH2-W, CH=CH-W, CC-W, S-W, CH2-S-W, CH=N-O-CH2-W, CH2-O-C(=O)-W or CH2-O-C(CH3)=N-N=C(CH3)-W. The invention also relates to a method and intermediate products for the production of said phenylpyrazolones used for combating parasitic fungi and animal parasites.

    New phenyl carbamate derivatives
    8.
    发明专利

    公开(公告)号:DE19745650A1

    公开(公告)日:1999-04-22

    申请号:DE19745650

    申请日:1997-10-16

    Applicant: BASF AG

    Abstract: Substituted oxy- or oxymethylenephenyl-oxazolidine and -oxazolidinedione derivatives (I) are new. They are prepared from new activated phenyl-oxazolidine derivatives (IIA) and activated phenyl-oxazolidinedione derivatives (IVB), which in turn are obtained via new substituted nitrobenzene and aniline derivatives (1), phenyl isocyanates (2) and substituted anilides (3). Substituted oxy- or oxymethylenephenyl-oxazolidine and -oxazolidinedione derivatives (I) are new: Y = halo; 1-4C alkyl; 1-4C haloalkyl; or 1-4C alkoxy; n = 0-2; E = group of formula (a) or (b): Ra = halo; CN; 1-4C alkyl or 1-4C alkoxy optionally substituted by halo; 3-6C alkenyloxy, 3-6C alkynyloxy; 3-6C cycloalkyl; S(O)m-1-4C alkyl; or NRaRb; m = 0-2; Ra and Rb = H; 1-4C alkyl; 3-6C alkenyl; or 3-6C alkynyl; Rb = 1-4C alkyl; 1-4C haloalkyl; 3-6C cycloalkyl; or optionally substituted arylmethylene; T = O or oxymethylene; Z' = X; N=CWR ; or N=C(R )-C(R )=NOR ; X = optionally substituted heterocyclyl, aryl, heteroaryl, arylmethylene or heteroarylmethylene; W = optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, heterocyclyl, aryl or heteroaryl; R = H; CN; 1-4C alkyl; 1-4C haloalkyl; 1-4C alkoxy; 1-4C alkoxy-1-4C alkyl; or 3-6C cycloalkyl; R = H; CN; halo; C(Rd)=NOR3; W; OW; SW or NRcW; Rc = H; alk yl; alkenyl; or alkynyl; Rd = H or alkyl; R = H; or optionally substituted alkyl, alkenyl or alkynyl. Independent claims are also included for: (A) activated phenyl-oxazolidine derivatives of formula (IIA); (B) activated phenyl-oxazolidinedione derivatives of formula (IVB); (C) substituted nitrobenzene and aniline derivatives of formula (1); (D) phenyl isocyanates of formula (2); and (E) Substituted anilides (3). L = OH; CH3; CH2L'; or L'; L' = nucleophilic leaving group; La = CH3; CH2L'; NO2; alkylsulphonate; or arylsulphonate; Q = NH2 or NO2; T' = OZ'; CH2O-X; or CH2O-N=C(R )-C(R )=NOR ; Z' = N=CWR or N=C(R )-C(R )=NOR ; E asterisk = NH-C(O)-NH-OH; NH-C(O)-O-NH-C(O)-OR; NH-C(S)-R'; or NH-C(NOH)-R'; R = 1-4C alkyl; R' = 1-4C alkyl; 1-4C haloalkyl; or 3-6C cycloalkyl.

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