-
公开(公告)号:DE3205638A1
公开(公告)日:1983-08-25
申请号:DE3205638
申请日:1982-02-17
Applicant: HOECHST AG
Inventor: HUMBURG GERHARD DR , MILDENBERGER HILMAR DR , BOSSE DIETER DR , SACHSE BURKHARD DR
IPC: A01N43/54 , A01N43/78 , C07D239/30 , C07D239/34 , C07D239/38 , C07D239/42 , C07D239/46 , C07D239/48 , C07D239/50 , C07D239/58 , C07D239/60 , C07D401/12 , C07D417/12 , C07D239/28 , A01N43/48 , C07D401/00 , C07D403/00
Abstract: The invention relates to novel 2,4,6-trisubstituted pyrimidine-5-carboxylic acids and their derivatives of the general formula I in which R = OH, (C1-C12)-alkoxy, (C5-C8)-cycloalkoxy, optionally substituted phenoxy or NR R , R = H, (C1-C4)-alkyl, and R = optionally substituted phenyl, X, Y and Z, which can be identical or different, denote Cl, Q(C1-C4)-alkyl, Q-CH2-phenyl, Q-CH2-COO-(C1-C4)-alkyl, optionally substituted Q-phenyl where Q represents O, S, SO or SO2, or NR R where R5 = H, (C1-C4)-alkyl, optionally substituted phenyl, benzyl or diphenylmethyl, or R and R together with the adjacent N atom form a heterocyclic 5-7-membered ring and X furthermore denotes -S-heteroaryl, and to processes for their preparation, and to their use as pesticides.
-
公开(公告)号:CH626777A5
公开(公告)日:1981-12-15
申请号:CH759377
申请日:1977-06-21
Applicant: HOECHST AG
Inventor: HOERLEIN GERHARD DR , BECKER WERNER , LANGELUEDDEKE PETER DR , KOECHER HELMUT DR , SACHSE BURKHARD DR
IPC: C07C69/712 , A01N31/14 , A01N37/40 , A01N39/02 , A01P13/00 , C07C67/00 , C07C69/67 , C07C69/68 , C07C69/90 , C07C201/00 , C07C205/38 , C07C205/57 , C07C205/61 , C07C231/00 , C07C235/20 , C07C253/00 , C07C255/14 , C07C313/00 , C07C319/20 , C07C323/17 , C07C323/20 , C07C325/00 , C07C327/22 , C07D213/63
-
公开(公告)号:DE3779738D1
公开(公告)日:1992-07-16
申请号:DE3779738
申请日:1987-12-21
Applicant: HOECHST AG
Inventor: HAMMANN PETER DR , GRABLEY SUSANNE DR , VOELSKOW HARTMUT DR , SACHSE BURKHARD DR , RAETHER WOLFGANG DR , GIANI CARLO DR , SEIBERT GERHARD PROF DR
IPC: C12P17/08 , A01N47/44 , A01N63/02 , A61K20060101 , A61K31/365 , A61P31/00 , A61P31/10 , C07D313/00 , C07D493/04 , C07D493/08 , C12N20060101 , C12P20060101 , C12P1/02 , C12P1/06 , C12P17/16 , C12P17/18 , C12R1/465
Abstract: Macrolide antibiotics of formula (I) are new: A = a gp. of formula A1-A4 R = R4 when A = A1 or A2, or R2 when A = A3 or A4; R1 and R2 = H or malonyl, not more than one R2 being malonyl; R3 and R4 = H, 1-6C alkyl or allyl; excluding those cpds. (I; A = A1) where (a) R1 = malonyl and all R2, R3 and R4 = H, (b) R1 = malonyl, all R2 and R4 = H and R3 = Me, or (c) R11 all R2 and R4 = H and R3 = Me.
-
公开(公告)号:AT77089T
公开(公告)日:1992-06-15
申请号:AT87118929
申请日:1987-12-21
Applicant: HOECHST AG
Inventor: HAMMANN PETER DR , GRABLEY SUSANNE DR , VOELSKOW HARTMUT DR , SACHSE BURKHARD DR , RAETHER WOLFGANG DR , GIANI CARLO DR , SEIBERT GERHARD PROF DR
IPC: C12P17/08 , A01N47/44 , A01N63/02 , A61K20060101 , A61K31/365 , A61P31/00 , A61P31/10 , C07D313/00 , C07D493/04 , C07D493/08 , C12N20060101 , C12P20060101 , C12P1/02 , C12P1/06 , C12P17/16 , C12P17/18 , C12R1/465
-
公开(公告)号:DE4029648A1
公开(公告)日:1992-03-26
申请号:DE4029648
申请日:1990-09-19
Applicant: HOECHST AG
Inventor: MINN KLEMENS DR , BRAUN PETER DR , SACHSE BURKHARD DR , WICKE HEINRICH DR
IPC: A01N43/54 , C07D239/46 , C07D401/12 , C07D405/12 , C07D409/12 , C07D491/048
Abstract: Compounds have the formula (I), in which R , R represent independently from each other hydrogen or (C1-C4)alkyl; R and R if necessary form together a saturated or partially unsaturated carbocyclic or heterocyclic moiety with the heteroatoms O, N or S and 5 or 6 cyclic members; R represents hydrogen or halogen; R , R , R represent independently from each other hydrogen, halogen, (C1-C4)alkyl, (C1-C4)alkoxy or phenoxy eventually substituted in the phenyl moiety by halogen, (C1-C4)alkyl or (C1-C4)alkoxy; R , R and R form together a saturated, partially insaturated or aromatic carbocyclic or heterocyclic moiety with the heteroatoms O, N or S and 5 to 7 cyclic members; R is hydrogen or (C1-C4)alkyl; R is hydrogen, (C1-C4)alkyl, (C1-C4)alkoxy, phenyl-(C1-C4)alkoxy or halogen; R is hydrogen, (C1-C4)alkyl, perhalo-(C1-C4)alkyl, (C1-C4)alkoxy-(C1-C4)alkyl or phenyl-(C1-C4)alkyl; R and R if necessary form together a saturated or partially unsaturated carbocycle or heterocycle with the heteroatoms O, N or S and 5 to 6 cyclic members; X is oxygen or sulphur and n equals 0 or 1. These compounds have advantageous pesticide properties, in particular against fungus pests. A process for producing compounds having formula (I) is also disclosed.
-
公开(公告)号:DE3935277A1
公开(公告)日:1991-05-02
申请号:DE3935277
申请日:1989-10-24
Applicant: HOECHST AG
Inventor: ORT OSWALD DR , WILLMS LOTHAR DR , BAUER KLAUS DR , BIERINGER HERMANN DR , SCHULZ ARNO DR , SACHSE BURKHARD DR , BRAUN PETER DR
IPC: A01N43/54 , A01N43/824 , A01N55/10 , C07D213/34 , C07D239/30 , C07D239/34 , C07D239/52 , C07D239/54 , C07D239/557 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12
Abstract: Compounds of formula (I) or their salts, where R to R , W, X, a and b are as defined in claim 1 and L is a heterocyclic or isocyclic aromatic residue with 5 to 6 ring atoms which can be condensed with an aromatic or non-aromatic 5- or 6-membered ring and which may be substituted or unsubstituted, and a, b and c independently stand for 0 or 1, are suitable for use as herbicides, plant growth regulators and fungicides. They can be produced by the process defined in claim 5, and some new intermediate products (see claims 14 and 15) can be used.
-
公开(公告)号:CS269997B2
公开(公告)日:1990-05-14
申请号:CS872487
申请日:1987-12-01
Applicant: HOECHST AG
Inventor: EHRHARDT HEINZ DR , MILDENBERGER HILMAR DR , MAIER THOMAS DR , SCHALLER RAINER DR , SACHSE BURKHARD DR , BRAUN PETER DR
IPC: C07D401/04 , A01N47/38 , A61K31/415 , A61K31/4427 , A61K31/443 , A61K31/445 , A61P31/04 , C07D401/14 , C07D405/14 , C07D521/00
Abstract: Compounds of the formula (I) (I) in which n denotes a number from 2 to 6, m denotes 1 or 2, R denotes +TR CH2CH2CH2OR1, R1 denotes (substituted) alkyl, (substituted) alkenyl, C3-alkynyl, cycloalkyl, cycloalkenyl or an aromatic or heteroaromatic radical, R2 denotes H or alkyl and Y denotes H, alkyl, phenyl or halophenyl, and the metal-salt complexes thereof have advantageous fungicidal actions and are highly suitable for use in plant protection or in the industrial sector.
-
公开(公告)号:DE3733220A1
公开(公告)日:1989-04-13
申请号:DE3733220
申请日:1987-10-01
Applicant: HOECHST AG
Inventor: SALBECK GERHARD DR , LUEDERS WALTER DR , KNAUF WERNER DR , WALTERSDORFER ANNA DR , KERN MANFRED DR , SACHSE BURKHARD DR , WICKE HEINRICH DR
IPC: A01N43/58 , C07D237/16 , C07D237/18
Abstract: Compounds of the formula I in which R1 denotes hydrogen or (C1-C6)-alkyl, optionally substituted by halogen or a hydroxyl group, R2 denotes hydrogen, (C1-C6)-alkyl, or halogen, X denotes oxygen or sulphur and R3 denotes (C1-C20)-alkyl, which can be mono- or polysubstituted by hydroxyl, halogen, amino, (di)-(C1-C4)-alkylamino, (C1-C4)-alkoxy, (C1-C4)-haloalkoxy, (C1-C4)-alkoxy-(C1-C4)-alkyleneoxy, (C1-C4)-alkylthio which can be substituted by (C1-C3)-alkyl, halogen or (C1-C3)-haloalkyl, or can be substituted by (C1-C4)-alkylsulphinyl, (C1-C4)-alkylsulphonyl, trimethoxysilyl, amidocarbonyl, (C1-C4)-alkylsulphonyloxy, (C1-C6)-alkylcarbonyl, (C1-C6)-alkoxycarbonyl, (C1-C6)-alkylcarbonyloxy, cyano, thiocyano, (C3-C8)-cycloalkyl, which can be substituted by hydroxyl or (C1-C4)-alkylcarbonyloxy, aryl, aryloxy, arylthio, arylsulphinyl, arylsulphonyl, arylsulphonyloxy or arylcarbonyl, all of which can be substituted by (C1-C4)-alkyl, (C1-C4)-alkoxy or halogen, with the proviso that if the (C1-C20)-alkyl radical is substituted by substituted or unsubstituted aryl or aryloxy, hydroxyl additionally substitutes this alkylene moiety, have advantageous insecticidal, acaricidal, nematocidal or fungicidal properties.
-
公开(公告)号:DE3508398A1
公开(公告)日:1986-11-06
申请号:DE3508398
申请日:1985-03-08
Applicant: HOECHST AG
Inventor: TAMMER THOMAS DR , SACHSE BURKHARD DR , HARTZ PETER DR
IPC: A01N33/08 , A01N33/20 , A01N35/04 , A01N35/10 , A01N37/40 , A01N37/42 , A01N37/44 , A01N41/10 , A01N43/00 , A01N43/06 , A01N43/24 , A01N43/28 , A01N43/40 , A01N43/46 , A01N43/60 , A01N43/62 , A01N45/00 , C07D207/08 , C07D209/02 , C07D211/08 , C07D211/14 , C07D211/22 , C07D211/42 , C07D211/46 , C07D211/58 , C07D211/62 , C07D211/70 , C07D211/74 , C07D213/50 , C07D213/64 , C07D213/643 , C07D213/74 , C07D215/22 , C07D215/227 , C07D217/04 , C07D223/04 , C07D241/44 , C07D243/08 , C07D263/04 , C07D265/30 , C07D279/12 , C07D295/04 , C07D295/084 , C07D295/10 , C07D295/108 , C07D295/125 , C07D307/52 , C07D307/81 , C07D307/91 , C07D319/18 , C07D333/22 , C07D333/28 , C07D333/32 , C07D333/34 , C07D333/44 , C07D333/58 , C07D333/76 , C07D405/06 , C07D491/10 , C07F9/38 , A01N47/34 , C07C97/10 , C07C101/12
-
60.
公开(公告)号:DE3503981A1
公开(公告)日:1986-08-07
申请号:DE3503981
申请日:1985-02-06
Applicant: HOECHST AG
Inventor: EHRHARDT HEINZ DR , MILDENBERGER HILMAR DR , HANDTE REINHARD DR , SACHSE BURKHARD DR , HARTZ PETER DR
IPC: C07D211/44 , C07D217/04 , C07D295/092 , C07D265/30 , A01N35/00 , A01N43/00 , C07C93/04 , C07D295/10
Abstract: Compounds of the formula I in which X denotes O, S, SO or SO2, R denotes alkyl, cycloalkyl, (subst.) alkenyl, (subst.) cycloalkenyl, (subst.) phenyl, (subst.) naphthyl, (subst.) tetrahydronaphthyl or a (subst.) heterocycle having up to 3 O, N or S atoms, R denotes (subst.) alkyl, (subst.) phenyl, R and R denote (subst.) alkyl, or R and R , together with the adjacent nitrogen atom, denote a saturated (subst.) heterocycle, in which 1 CH2 group can be replaced by CO and which additionally can contain a fused benzo ring or alicycle, m denotes 0, 1 or 2 and n denotes a number from 0 to 8, with the proviso that m + n = 2, and their salts and quaternisation products have useful fungicidal properties. They are particularly suitable for use in useful plant crops.
-
-
-
-
-
-
-
-
-