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公开(公告)号:BRPI0608709A2
公开(公告)日:2010-01-26
申请号:BRPI0608709
申请日:2006-03-15
Applicant: BASF AG
Inventor: DIETZ JOCHEN , GROTE THOMAS , BLETTNER CARSTEN , HUENGER UDO , SCHOFER PETER , RETHER JAN , EICKEN KARL , GEWEHR MARKUS , GRAMMENOS WASSILIOS , MUELLER BERND , SCHIEWECK FRANK , SCHWOEGLER ANJA , LOHMANN JAN KLAAS , RHEINHEIMER JOACHIM , STRATHMANN SIEGFRIED , STIERL REINHARD
IPC: C07D213/82 , A01N43/40
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公开(公告)号:BRPI0514950A
公开(公告)日:2008-07-01
申请号:BRPI0514950
申请日:2005-09-05
Applicant: BASF AG
Inventor: GEWEHR MARKUS , GROTE THOMAS , MUELLER BERND , GRAMMENOS WASSILIOS , GLER ANJA SCHW , RHEINHEIMER JOACHIM , BLETTNER CARSTEN , SCHOFER PETER , SCHIEWECK FRANK , WAGNER OLIVER , RETHER JAN , STRATHMANN SIEGFRIED , STIERL REINHARD , SCHERER MARIA
IPC: A01N43/56 , A01N43/78 , C07D213/82 , C07D231/40 , C07D277/56 , C07D333/38 , C07D405/12 , C07D409/12 , C07D411/12 , C07D413/12 , C07D417/12
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公开(公告)号:BRPI0513720A
公开(公告)日:2008-05-13
申请号:BRPI0513720
申请日:2005-07-22
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS , GROTE THOMAS , BLETTNER CARSTEN , GEWEHR MARKUS , HUENGER UDO , MUELLER BERND , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , SCHOEFL ULRICH , KOELE HARALD , STRATHMANN SIEGFRIED , SCHERER MARIA , STIERL REINHARD , RETHER JAN
IPC: C07D401/04 , A01N43/54
Abstract: 2-Pyridyl pyrimidine derivatives (I) are new. 2-Pyridyl pyrimidine derivatives of formula (I) and their salts are new. k : 0-3; m : 0-5; n : 1-5; R 1>halo, OH, CN, NO 2, 1-4C (halo)alkyl, 104C (halo)alkoxy, 2-4C alkenyl, 2-4C alkynyl, 3-8C cycloalkyl, (1-4C)alkoxy(1-4C)alkyl, NH 2, phenoxy (optionally substituted with halo or 1-4C alkyl), NHR, NRR, C(Ra)=NORb, SO pA 1> or COA 2>; or R 1>+R 1>1-4C (halo)alkylenedioxy; R : 1-4C alkyl or 1-4C alkylcarbonyl; Ra : H or 1-4C alkyl; Rb : 1-4C alkyl, 3-4C alkenyl or 3-4C alkynyl; p : 0-2; A 1>1-4C alkyl, or also NH 2, 1-4C alkylamino or di(1-4C alkyl)amino when p = 2; A 2>H, OH, 1-4C alkyl, 1-4C alkylamino, di(1-4C alkyl)amino, 2-4C alkenyl or 1-4C (halo)alkoxy; R 2>1-4C haloalkyl, 1-4C (halo)alkoxy, OH, halo, CN or NO 2, or R 2> can be H or 1-4C alkyl if n = 3-5 and/or k = 1-3 and/or at least one R 1> is other than halo, 1-4C (halo)alkyl and 1-4C alkoxy; and R 3>1-4C alkyl. An independent claim is also included for controlling phytopathogenic fungi by treating the fungi, or materials, plants, soil or seeds to be protected from fungal attack, with a compound (I). [Image] ACTIVITY : Plant antifungal. In a protective test against Alternaria solani on tomato plants, plants treated with 2-(5-methyl-6-phenyl-2-pyridyl)-4,5-pentamethylene-pyrimidine (250 ppm) suffered no attack, whereas 90% of untreated plants were attacked. MECHANISM OF ACTION : None given.
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公开(公告)号:ZA200606942B
公开(公告)日:2008-04-30
申请号:ZA200606942
申请日:2006-08-21
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , BLETTNER CARSTEN , MULLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOGLER ANJA , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOFL ULRICH , STIERL REINHARD
IPC: A01N20090101 , C07D20090101
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公开(公告)号:BRPI0512557A
公开(公告)日:2008-03-25
申请号:BRPI0512557
申请日:2005-06-24
Applicant: BASF AG
Inventor: BLETTNER CARSTEN , SCHIEWECK FRANK , BLASCO JORDI TORMO I , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHWOEGLER ANJA , WAGNER OLIVER , SPEAKMAN JOHN-BRYAN , JABS THORSTEN , STRATHMANN SIEGFRIED , FL ULRICH SCH , SCHERER MARIA , STIERL REINHARD
IPC: C07D487/04 , A01N43/90
Abstract: The present invention relates to novel triazolopyrimidine compounds of the formula I in which: X is halogen, cyano, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy or C 1 -C 2 -haloalkoxy; W is oxygen or sulfur; Y is O-R 4 or a group NR 5 R 6 ; A is a chemical bond or a group CR 7 R 8 ; and the variables L, R 1 to R 7 are as defined in claim 1. The present invention furthermore provides the use of the triazolopyrimidine compounds of the formula I, their tautomers and their agriculturally acceptable salts for controlling phytopathogenic fungi (=harmful fungi) and a method for controlling phytopathogenic harmful fungi, which method comprises treating the fungi or the materials, plants, the soil or seed to be protected against fungal attack with an effective amount of a compound of the formula I, a tautomer of I and/or an agriculturally acceptable salt of I or a tautomer thereof.
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公开(公告)号:BRPI0512249A
公开(公告)日:2008-02-19
申请号:BRPI0512249
申请日:2005-06-14
Applicant: BASF AG
Inventor: BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , MUELLER BERND , NIEDENBRUECK MATTHIAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , WAGNER OLIVER , NAVE BARBARA , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD , SCHWOEGLER ANJA
IPC: A01N43/90 , C07D487/04
Abstract: Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R 1 is alkyl, halocycloalkyl, alkenyl, cycloalkyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen, alkyl or one of the groups mentioned under R 1 ; R 1 and/or R 2 may carry one to four identical or different groups R a : R a is chlorine, bromine, iodine, cyano, nitro, hydroxyl, alkyl, alkylcarbonyl, cycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, alkylthio, alkylamino, dialkyl-amino, alkenyl, cycloalkenyl, alkenyloxy, haloalkenyloxy, alkynyl, halo-alkynyl, alkynyloxy, haloalkynyloxy, cycloalkoxy, cycloalkenyloxy, oxyalkylenoxy, naphthyl, a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, where these aliphatic, alicyclic or aromatic groups for their part may be substituted according to the description; and X is halogen; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
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公开(公告)号:BRPI0511888A
公开(公告)日:2008-01-15
申请号:BRPI0511888
申请日:2005-06-08
Applicant: BASF AG
Inventor: BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , MUELLER BERND , NIEDENBRUECK MATTHIAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , GLER ANJA SCHW , WAGNER OLIVER , RAPADO LILIANA PARRA , RACK MICHAEL , NAVE BARBARA , SCHERER MARIA , STRATHMANN SIEGFRIED , FL ULRICH SCH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: The invention relates to the use of triazolopyrimidines of the formula I In which: R 1 , R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl, C 3 -C 6 -cycloalkynyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N and S, where R 1 , R 2 may be substituted as defined in the description or R 1 and R 2 together with the nitrogen atom to which they are attached may form five- to eight-membered heterocyclyl or heteroaryl which is attached via nitrogen and may contain one, two or three further heteroatoms from the group consisting of O, N and S as ring members and/or may be substituted as defined in the description; L independently of one another are halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyloxy, cyano, C(-O)A 1 , S(-O) m A 2 , NR c R d or NR c -(C-O)-R d , where A 1 , A 2 , R c , R d and m are as defined in the description; L 1 is halogen, alkyl or haloalkyl; L 2 is nitro, a group -C(S)NR 3 R 4 , a group -C(-N-OR 5 )(NR 6 R 7 ) or a group -C(-N-NR 8 R 9 )(NR 10 OR 11 ); X is halogen, cyano, alkyl, alkoxy, haloalkyl or haloalkoxy; R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 and R 11 are independently of one another selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl and alkynyl, where the 4 last-mentioned radicals may be substituted as defined in the description; or R 3 and R 4 , or R 6 and R 7 , or R 8 and R 9 or R 10 and R 11 together with the nitrogen atom to which they are attached form a four, five, or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; n is 0, 1, 2 or 3; and the agriculturally acceptable salts thereof, novel triazolopyrimidines, crop protection compositions comprising at least one compound of the formula I and at least one solid or liquid carrier, and a method for controlling phytopathogenic harmful fungi.
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公开(公告)号:BRPI0508976A
公开(公告)日:2007-08-28
申请号:BRPI0508976
申请日:2005-03-26
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , NIEDENBRUECK MATTHIAS , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: The invention relates to 5,6-cycloalkyl-7-aminotriazolopyrimidines of formula (I), where X=alkylene or alkenylene, whereby the carbon chain can be interrupted by one or two heteroatoms selected from S, O or NR 1 , R 1 -H, alkyl or C(-O)alkyl, L=halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, alkinyl or NR 2 R 3 ; R 2 ,R 3 =each one of the groups given for R 1 and m=a whole number from 0 to 5, whereby the aliphatic groups can be substituted by one to three of the following groups: halogen, cyano, nitro, hydroxy, alkoxy, alkylthio, or NR a R b , where R a , R b -H or alkyl in which the carbon chains can be halogenated. The invention further relates to methods for production of said compounds, agents comprising the same and use thereof for the prevention of fungal pests harmful to plants.
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公开(公告)号:BRPI0508337A
公开(公告)日:2007-07-24
申请号:BRPI0508337
申请日:2005-06-08
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , NIEDENBRUECK MATTHIAS , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A01N43/90
Abstract: 5,6-Dialkyl-7-aminotriazolopyrimidines of the formula I in which the substituents are as defined below: R 1 is alkyl, alkoxymethylene or alkoxyethylene, where the aliphatic groups may be substituted as defined in the description; R 2 is n-propyl or n-butyl; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
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公开(公告)号:BRPI0417765A
公开(公告)日:2007-04-17
申请号:BRPI0417765
申请日:2004-12-17
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , GLER ANJA SCHW , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , FL ULRINCH SCH , STIERL REINHARD , MUELLER BERND
IPC: C07D487/04 , A01N43/90
Abstract: Triazolopyrimidines of the formula I in which the substituents are as defined below: R 1 , R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and may be substituted as defined in the description; L is halogen, cyano, alkyl, haloalkyl, alkoxy, alkenyloxy or alkoxycarbonyl; m is 1, 2, 3 or 4, where the groups L may be different if m is greater than 1; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi
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