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    63.
    发明专利
    未知

    公开(公告)号：DK443287A

    公开(公告)日：1988-02-27

    申请号：DK443287

    申请日：1987-08-25

    Applicant: CIBA GEIGY AG

    Inventor： STURM ELMAR ,  LANG ROBERT WERNER ,  KRISTIANSEN ODD

    IPC: A01N47/34 ,  C07D239/34

    Abstract: The invention relates to novel N-benzoyl-N,-4-(5-phenylpyrimid-2-yloxy)phenylureas of formula +TR wherein X1 is hydrogen, halogen, C1-C3alkoxy or C1-C3alkylthio, X2 is halogen, methyl, C1-C3alkoxy or C1-C3alkylthio, Y1, Y2, Y3 and Y4 are each independently hydrogen, halogen, methyl, trifluoromethyl or methoxy, Z is methyl, halomethyl containing 1 to 3 halogen atoms or pentafluoroethyl; and R1, R2 and R3 are each independently hydrogen, halogen, C1-C3alkyl, trifluoromethyl or C1-C3alkoxy, to the preparation thereof and to intermediates for the synthesis of these compounds, as well as to compositions containing them for use in pest control, especially for controlling representatives of the order Acarina that attack plants and animals and for controlling insects. The novel compounds exhibit especially pronounced activity against plant-destructive mites.

    1-FLURO-1-ARYLOXY-2-AZOLYLMETHYL-2-ALKANOLS
    64.
    发明专利
    1-FLURO-1-ARYLOXY-2-AZOLYLMETHYL-2-ALKANOLS 未知

    公开(公告)号：AU568828B2

    公开(公告)日：1988-01-14

    申请号：AU2231083

    申请日：1983-12-12

    Applicant: CIBA GEIGY AG

    Inventor： STURM ELMAR ,  MULLER URS ,  TOBLER HANS

    IPC: A01N43/50 ,  A01N43/64 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00

    Abstract: The compounds described are those of the general formula I (I) in which R1 is an azolyl group; R2 is C1-C12-alkyl; R3 is hydrogen, C1-C12-alkyl, C2-C4-alkenyl or C2-C4-alkinyl, or benzyl which is unsubstituted or substituted by C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, halogen and/or cyano; R4 is hydrogen, fluorine or C1-C6-alkyl; R5 is an unsubstituted or substituted radical chosen from the series comprising phenyl, naphthyl, biphenyl, benzylphenyl and benzyloxyphenyl, the substituents being chosen from the series comprising halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy C1-C6-haloalkyl, C1-C6-alkylthio, C1-C6-haloalkoxy, C1-C3-haloalkylthio, nitro and/or thiocyano; and X is oxygen or sulfur; including the acid addition salts, quaternary azolium salts and metal complexes. Methods for the preparation of these products are also disclosed, as well as agrochemical compositions containing one of these compounds as the active substance. A method of controlling phytopathogenic microorganisms and/or of regulating plant growth with the aid of these substances is furthermore described.

    5-ESTERS OF MILBEMYCINS FOR CONTROLLING PARASITIC PESTS
    65.
    发明专利
    5-ESTERS OF MILBEMYCINS FOR CONTROLLING PARASITIC PESTS 未知

    公开(公告)号：ZA866360B

    公开(公告)日：1987-05-27

    申请号：ZA866360

    申请日：1986-08-22

    Applicant: CIBA GEIGY AG

    Inventor： MAIENFISCH PETER ,  STURM ELMAR

    IPC: C07D493/22 ,  A01N43/90 ,  A23K20/195 ,  A61K31/365 ,  A61P33/10 ,  C07H19/01 ,  C07D ,  A01N

    Abstract: The invention relates to ecto- and endoparasitic milbemycins of formula I (I) wherein R is methyl, ethyl, isopropyl or sec-butyl; R1 is hydrogen, fluorine or C1-C4 alkyl; R2 is one of the groups in which formulae is a value from 2 to 6; X is oxygen or sulfur; R3 is halogen; and R4 is hydrogen, C1-C12 alkoxy, C3-C7cycloalkoxy or C2-C6alkenyloxy; or C1-C18alkyl which is unsubstituted or substituted by halogen, C1-C4alkoxy, hydroxy and/or COOG, G being hydrogen, an alkali metal cation or an alkaline earth metal cation; or R4 is C3-C7cycloalkyl which is unsubstituted or substituted by halogen and/or C1-C4alkyl; C2-C18alkenyl which is unsubstituted or substituted by halogen; C2-C18alkynyl which is unsubstituted or substituted by halogen; phenyl which is unsubstituted or substituted by halogen, C1-C4alkyl C1-C4alkoxy, nitro, cyano and/or C1-C4haloalkyl; or a 5- or 6-membered unsaturated or saturated heterocyclic ring system which contains one to three hetero atoms selected from the series consisting of nitrogen, oxygen and sulfur and which is unsubstituted or substituted by oxo and/or by one to three substituents selected from halogen, C1-C4alkyl, C1-C4alkoxy and/or C1-C4haloalkyl; to the use thereof in agriculture and to the preparation thereof by esterifying the 5-OH-milbemycins on which they are based.

    FUNGICIDE AND METHOD OF ITS EFFICIENT COMPONENT PRODUCTION
    66.
    发明专利
    FUNGICIDE AND METHOD OF ITS EFFICIENT COMPONENT PRODUCTION 未知

    公开(公告)号：CS250237B2

    公开(公告)日：1987-04-16

    申请号：CS932683

    申请日：1983-12-12

    Applicant: CIBA GEIGY

    Inventor： STURM ELMAR ,  MEYER ALFRED

    IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00

    Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.

    1-AZOLYL-2-ARYL-3-FLUOROALKAN-2-OLS AS MICROBICIDES
    69.
    发明专利
    1-AZOLYL-2-ARYL-3-FLUOROALKAN-2-OLS AS MICROBICIDES 未知

    公开(公告)号：CA1209152A

    公开(公告)日：1986-08-05

    申请号：CA443044

    申请日：1983-12-12

    Applicant: CIBA GEIGY AG

    Inventor： STURM ELMAR ,  MEYER ALFRED

    IPC: A01N43/50 ,  A01N43/653 ,  A01P3/00 ,  C07C39/00 ,  C07C45/63 ,  C07C45/71 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D303/08 ,  C07D303/22 ,  C07D303/34 ,  C07D521/00

    Abstract: 1-AzoLyL-2-aryL-3-fLuoroaLkan-2-oLs as microbicides 1-AzoLyL-2-aryL-3-fLuoro-aLkan-2-oLes of the generaL formuLa I (I) in which Az is 1H-1,2,4-triazoLe, 4H-1,2,4-triazoLe or 1HimidazoLe; Ar is an unsubstituted or substituted aromatic radicaL from the series comprising phenyL, biphenyL, phenoxyphenyL and naphthyL; R1 is hydrogen, C1-C4-aLkyL, C3-C5-aLkenyL or benzyL; Rz is hydrogen, fLuorine or C1-C6-aLkyL and R3 is hydrogen, fLuorine, C1-C6-aLkyL, C1-C6-haLoaLkyL, C1-C6-aLkoxy, C1-C6-aLkyLthio, phenyL, phenoxy, phenyLthio or C3-C7-cycLoaLkyL, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poLy-substituted by haLogen, C1-C4-aLkyL, C1-C4-aLkoxy, C1-C4-haLoaLkyL, nitro and/or cyano; incLuding the acid addition saLts, quaternary azoLium saLts and metaL compLexes, are described. Methods for the preparation of these products are aLso discLosed, as weLL as agrochemicaL compositions containing one of these compounds as the active substance. A method for controLLing phytopathogenic microorganisms with the aid of these substances is aLso described.

    5-AZOLYLACETOXYMILBEMYCINS AS ECTO-AND ENDOPARASITES
    70.
    发明专利
    5-AZOLYLACETOXYMILBEMYCINS AS ECTO-AND ENDOPARASITES 未知

    公开(公告)号：ZA858993B

    公开(公告)日：1986-07-30

    申请号：ZA858993

    申请日：1985-11-25

    Applicant: CIBA GEIGY AG

    Inventor： STURM ELMAR ,  MAIENFISCH PETER

    IPC: A61K31/365 ,  A61P33/10 ,  A01N43/90 ,  C07D493/22 ,  C07H19/01 ,  C07D ,  A01N

    Abstract: The present invention relates to milbemycin derivatives of the formula I (I) wherein X is hydrogen or beta -halogen, R is methyl, ethyl, isopropyl or sec-butyl and Az is a 5 membered heterocyclic aromatic ring which contains 2-4 nitrogen atoms and is attached in the 1-position and which is unsubstituted or substituted by one or two C1-C6alkyl groups. These compounds, and the acid addition salts and metal complexes thereof, are effective pesticides for controlling endo-and ectoparasites, especially for controlling neamatodes which are parasites of animals. The may be obtained by appropriate esterification in 5-position of milbemycin derivatives. The selective beta -halogenation of 14,15-epoxymilbemycin derivatives can be effected via the intermediate DELTA 13,14-15-hydroxymilbemycins with appropriate halogenating agents.

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