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公开(公告)号:BRPI0417628A
公开(公告)日:2007-03-27
申请号:BRPI0417628
申请日:2004-12-14
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SHIEWECK FRANK , GLER ANJA SCHW , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , FL ULRICH SCH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R 1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen or one of the groups mentioned under R 1 , R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R 1 and/or R 2 may be substituted as defined in the description; L 1 , L 2 , L 3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
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公开(公告)号:BRPI0416849A
公开(公告)日:2007-02-27
申请号:BRPI0416849
申请日:2004-11-18
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOELER ANJA , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A61K31/519
Abstract: 6-(2,4,6-Trifluorophenyl)triazolopyrimidines of the formula I in which the substituents have the following meanings: R 1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl, cycloalkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen or one of the groups mentioned in R 1 , R 1 and R 2 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered ring which is interrupted by an atom from the group consisting of O, N and S, and/or R 1 and/or R 2 can be substituted according to the description; X is cyano, C 1 -C 4 -alkoxy, C 3 -C 4 -alkenyloxy, C 1 -C 2 -haloalkoxy or C 3 -C 4 -halo-alkenyloxy; process for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.
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公开(公告)号:BRPI0414410A
公开(公告)日:2006-11-14
申请号:BRPI0414410
申请日:2004-09-10
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , BLASCO JORDI TORMO I , GROTE THOMAS , RHEINHEIMER JOAQUIM , SCHOFER PETER , SCHIEWECK FRANK , GLER ANJA SWCHW , WAGNER OLIVER , TZ NORBERT G , STRATHMANN SIEGFRIED , FL ULRICH SCH , SCHERER MARIA , STIERL REINHARD
IPC: C07D213/42 , C07D215/12 , C07D401/12 , C07D409/12
Abstract: Sulfonamides of the formula I where the substituents are as follows: R 1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R 2 , R 3 , R 4 , R 5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R 2 and R 3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R 2 ' and R 3 ', R 2 ', R 3 ' are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R 2 , R 3 , R 4 and R 5 are hydrogen: X is phenyl substituted by a group C(R 6 )-NOR 7 , where R 6 is alkyl and R 7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R 2 , R 3 , R 4 and R 5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
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公开(公告)号:BRPI0409159A
公开(公告)日:2006-05-02
申请号:BRPI0409159
申请日:2004-03-30
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEL ULRICH , STIERL REINHARD
IPC: A01N43/54 , C07D239/28 , C07D239/30 , C07D239/34 , C07D239/42 , C07D239/46 , C07D239/52
Abstract: 2-Substituted pyrimidines of the formula I in which the index n and the substituents L, Ra, Rb, Rc, Rz, Ru, Rv, A', A'' and A''' are as defined in the description and: R1 is C3-C10-alkyl, C3-C10-alkenyl, C3-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S, R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl, and R3 is cyano, CO2Ra, C(-O)NRzRb, C(-O)-N-ORb, C(-S)-NRaRb, C(-NORa)NRzRb, C(-NRa)NRzRb, C(-O)NRa-NRzRb, C(-N-NRzRc)NRaRb, C(-O)Ra, C(-NORb)Ra, C(-N-NRzRb)Ra, CRaRb-ORz, CRaRb-NRzRc, ON(-CRaRb), O-C(-O)Ra, NRaRb', NRa(C(-O)Rb), NRa(C(-O)ORb), NRa(C(-O)-NRzRb), NRa(C(-NRc)Rb), NRa(N-CRcRb), NRa-NRzRb, NRz-ORa, NRa(C(-NRc)-NRzRb), NRa(C(-NORc)Rb), processes for preparing these compounds, compositions comprising these compounds and their pesticidal use are described.
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公开(公告)号:BRPI0409431A
公开(公告)日:2006-04-25
申请号:BRPI0409431
申请日:2004-04-16
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , GLER ANJA SCHW , WAGNER OLIVER , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , SCHERER MARIA , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: Bicyclic compounds of the formula I in which A 1 or A 5 is C and the other of the two variables A 1 , A 5 is N, C or C-R 3 ; A 2 , A 3 , A 4 independently of one another are N or C-R 3a , where one of the variables A 2 , A 3 or A 4 may also be S or a group N-R 4 if A 1 and A 5 are both C, and where A 4 is not N or C-R 3a if A 1 is N, A 3 is C-R 3a and A 5 is C, and where A 1 is attached to A 2 and A 3 to A 4 or A 2 is attached to A 3 and A 4 to A 5 or A 1 is attached to A 5 and A 2 to A 3 or A 1 is attached to A 5 and A 3 to A 4 or A 1 is attached to A 2 and A 4 to A 5 by double bonds; n is 0, 1, 2, 3, 4 or 5; R a is halogen, cyano, C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkyl, C 1 -C 6 -haloalkoxy, C 2 -C 6 -alkenyl, C 2 -C 6 -alkenyloxy or C(O)R 5 ; R 1 is halogen, cyano, C 1 -C 10 -alkyl, where a carbon atom of the C 1 -C 10 -alkyl radical may be replaced by a silicium atom, C 1 -C 6 -haloalkyl, C 2 -C 10 -alkenyl, C 2 -C 6 -haloalkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 -cycloalkyl, C 3 -C 8 -cycloalkyl-C 1 -C 4 -alkyl, where the cycloalkyl moiety of the two last-mentioned groups may be unsubstituted or contain 1, 2, 3, 4, 5, or 6 radicals selected from the group consisting of C 1 -C 4 -alkylidene, C 1 -C 4 -alkyl, halogen, C 1 -C 4 -haloalkyl and hydroxy and the alkyl moiety of C 3 -C 8 -cycloalkyl-C 1 -C 4 -alkyl may be unsubstituted or contain 1, 2, 3, or 4 radicals selected from the group consisting of halogen, C 1 -C 4 -haloalkyl and hydroxy, C 5 -C 8 -cycloalkenyl which may be unsubstituted or contain 1, 2, 3 or 4 radicals selected from the group consisting of C 1 -C 4 -alkyl, halogen, C 1 -C 4 -haloalkyl and hydroxy, OR 6 , SR 6 , NR 7 R 8 , a radical of the formula -C(R 11 )(R 12 )C(-NOR 13 )(R 14 ) or a radical of the formula -C(-NOR 15 )C(-NOR 16 )(R 17 ); R 2 is halogen, cyano, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -haloalkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 -cycloalkyl, C 5 -C 8 -cycloalkenyl, OR 6 , SR 6 or NR 7 R 8 ; and the agriculturally acceptable salts of the compounds I, crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt of I and at least one solid or liquid carrier and a method for controlling phytopathogenic harmful fungi are described.
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公开(公告)号:BRPI0408754A
公开(公告)日:2006-03-28
申请号:BRPI0408754
申请日:2004-03-24
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , GLER ANJA SCHW , SCHERER MARIA , STRATHMANN SIEGFRIED , FL ULRICH SCH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: 7-(Alkenylamino)triazolopyrimidines of the formula I wherein the substituents have the following meanings: L is halogen, alkyl, haloalkyl, alkoxy, amino, NHR or NR 2 ; R is alkyl or alkyl-carbonyl; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl or alkoxy; R 1 is alkyl or haloalkyl; R 2 is hydrogen, alkyl or haloalkyl; R 3 is alkenyl, which can be unsubstituted or partially or completely halogenated or can be substituted according to the Description; R 4 is hydrogen or alkyl, R 3 and R 4 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered unsaturated ring which can be interrupted by an atom from the group consisting of O, N and S and/or can carry one or more sub-stituents. Processes for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.
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公开(公告)号:BRPI0406757A
公开(公告)日:2005-12-20
申请号:BRPI0406757
申请日:2004-01-28
Applicant: BASF AG
Inventor: MUELLER BERND , GROTE THOMAS , BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , BLASCO JORDI TORMO I , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/653 , A01N43/707 , A01N43/78 , A01N43/82 , C07D239/56 , C07D403/04 , C07D521/00 , A01N43/90
Abstract: Pyrimidines of the formula I
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公开(公告)号:HRP20040985A2
公开(公告)日:2004-12-31
申请号:HRP20040985
申请日:2004-10-20
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD , SCHOEFL ULRICH
IPC: A01N43/90 , C07C255/57 , C07D487/04 , C07C323/62
Abstract: The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L 1 represents cyano, S(-O) n A 1 or C(-O)A 2 , wherein A 1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A 2 stands for C 1 -C 8 alkoxy, C 1 -C 6 haloalkoxy or one of the groups named in A 1 ; and n stands for 0, 1 or 2; L 2 , L 3 represent hydrogen or halogen; L 4 , L 5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R 1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R 2 represents hydrogen or R 1 ; R 1 and R 2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R 1 and/or R 2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.
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公开(公告)号:BR9915370A
公开(公告)日:2001-08-14
申请号:BR9915370
申请日:1999-11-06
Applicant: BASF AG
Inventor: REINHARD ROBERT , HAMPRECHT GERHARD , SCHOFER PETER , ZAGAR CYRILL , OTTEN MARTINA , WESTPHALEN KARL-OTTO , WALTER HELMUT , MENKE OLAF
IPC: C07D239/56 , A01N43/54 , A01N43/76 , A01N43/78 , C07C271/22 , C07C271/54 , C07C275/30 , C07D239/54 , C07D413/04 , C07D413/14 , C07D417/04 , C07D417/14
Abstract: The invention relates to herbicidally effective 3-{benz(ox/thi)azol-7-yl}-1H-pyrimidine-2,4-diones of formula (I) wherein X=oxygen or sulphur, Y=oxygen or sulphur; Z=chemical bond, C1-C4-alkylene, O, S, SO, SO2; R =H, NH2, C1-C6-alkyl, C1-C6-alkyl halide; R =H, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkylthio, C1-C6-alkylsulfinyl or C1C6-alkylsulfonyl; R =H, halogen, C1-C6-alkyl; R =H, halogen; R =CN, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkoxy or C1-C6-halogenalkoxy; R =H, C3-C7-cycloalkyl containing a 3 to 7-membered saturated heterocyclyl and one or more oxygen and/or sulphur atoms, whereby each heterocyclic ring may contain a carbonyl or thiocarbonyl ring member. The invention also relates to the agriculturally usable salts of the compounds of formula (I).
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公开(公告)号:BR9911812A
公开(公告)日:2001-03-27
申请号:BR9911812
申请日:1999-06-29
Applicant: BASF AG
Inventor: HAMPRECHT GERHARD , MENKE OLAF , REINHARD ROBERT , SCHOFER PETER , ZAGAR CYRILL , OTTEN MARTINA , WESTPHALEN KARL-OTTO , WALTER HELMUT
IPC: C07D487/04 , A01N43/90 , C07C275/34 , C07C275/40 , C07C281/08 , C07C337/08 , C07D498/04 , C07D513/04
Abstract: A process for preparing fused triazoles of formula Iwhere:X-X is C-O, C-S, C-SO, C-SO2, or C-NR1;V is C=W2, R1R2C-C(=W2)- or C(=V2)-C(=W2);W1, W2 are oxygen or sulfur;which comprises reacting substituted N-aminoureas are reacted with formaldehyde or paraformaldehyde to give the corresponding methyleneimino ureas; cyclizing these in the presence of catalytic amounts of acid or metal oxide to give tetrahydro-4H-1,3,4-oxa(or thia)diazines, and cyclizing the fused triazoles using phosgene or a phosgene substitute. Also disclosed are novel fused triazoles of the formula I'
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