公开(公告)号：ZA8703879B

公开(公告)日：1988-02-24

申请号：ZA8703879

申请日：1987-05-29

Applicant: HOECHST AG

Inventor： GIENCKE WOLFGANG ,  WOLFGANG GIENCKE ,  MILDENBERGER HILMAR ,  HILMAR MILDENBERGER ,  HEUBACH GUENTHER ,  GUENTHER HEUBACH ,  SACHSE BURKHARD ,  BURKHARD SACHSE ,  FUSS ANDREAS ,  ANDREAS FUSS ,  WALTERSDORFER ANNA ,  ANNA WALTERSDORFER ,  KNAUF WERNER ,  WERNER KNAUF ,  KERN MANFRED ,  MANFRED KERN ,  BONIN WERNER ,  WERNER BONIN

IPC: A01N43/54 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48 ,  A01N ,  C07D

CPC classification number: C07D239/42 ,  A01N43/54 ,  C07D239/47

公开(公告)号：PT86271A

公开(公告)日：1988-01-01

申请号：PT8627187

申请日：1987-12-02

Applicant: HOECHST AG

Inventor： EHRHARDT HEINZ ,  MILDENBERGER HILMAR ,  MAIER THOMAS ,  SACHSE BURKHARD ,  SCHALLER RAINER ,  BRAUN PETER

IPC: A01N47/38 ,  A61K31/415 ,  A61K31/4427 ,  C07D401/04 ,  A61K31/443 ,  A61K31/445 ,  A61P31/04 ,  C07D401/14 ,  C07D405/14 ,  C07D521/00 ,  C07D403/00 ,  C07D401/00 ,  A01N43/50

Abstract: Compounds of the formula (I) (I) in which n denotes a number from 2 to 6, m denotes 1 or 2, R denotes +TR CH2CH2CH2OR1, R1 denotes (substituted) alkyl, (substituted) alkenyl, C3-alkynyl, cycloalkyl, cycloalkenyl or an aromatic or heteroaromatic radical, R2 denotes H or alkyl and Y denotes H, alkyl, phenyl or halophenyl, and the metal-salt complexes thereof have advantageous fungicidal actions and are highly suitable for use in plant protection or in the industrial sector.

公开(公告)号：AU7219287A

公开(公告)日：1987-11-05

申请号：AU7219287

申请日：1987-04-29

Applicant: HOECHST AG

Inventor： HEUBACH GUNTHER ,  MATTERSTOCK KARL ,  MILDENBERGER HILMAR ,  SACHSE BURKHARD

IPC: A01N43/74 ,  C07D263/58 ,  C07D277/82 ,  A01N43/76 ,  A01N43/78

公开(公告)号：DK144387A

公开(公告)日：1987-09-22

申请号：DK144387

申请日：1987-03-20

Applicant: HOECHST AG

Inventor： SACHSE BURKHARD ,  SCHREIBER BERNHARD

IPC: A01N43/653 ,  A01N47/44 ,  A01N55/00 ,  A01N55/04 ,  A01N55/10 ,  A01N57/16 ,  A01N59/02 ,  A01N57/24

公开(公告)号：AU6998987A

公开(公告)日：1987-09-17

申请号：AU6998987

申请日：1987-03-13

Applicant: HOECHST AG

Inventor： BLUME ERNST ,  EHRHARDT HEINZ ,  RAETHER WOLFGANG ,  DITTMAR WALTER ,  HANEL HEINZ ,  SACHSE BURKHARD ,  SCHAPER WOLFGANG

IPC: C07D247/00 ,  A01N43/50 ,  A01N43/653 ,  C07C41/00 ,  C07C43/18 ,  C07C67/00 ,  C07C201/00 ,  C07C213/00 ,  C07C215/42 ,  C07C217/48 ,  C07C217/74 ,  C07C253/00 ,  C07C255/54 ,  C07C313/00 ,  C07C317/12 ,  C07C317/14 ,  C07C317/18 ,  C07C317/20 ,  C07C323/22 ,  C07D233/56 ,  C07D233/60 ,  C07D233/61 ,  C07D249/08 ,  C07D307/38 ,  C07D333/00 ,  C07D401/12 ,  C07D403/12 ,  C07D405/06 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D417/12 ,  C07D521/00 ,  A61K31/41 ,  A61K31/495 ,  A61K31/445 ,  A61K31/425 ,  A61K31/44 ,  A61K31/505 ,  A61K31/415 ,  C07D403/08 ,  C07D409/06 ,  C07D413/12

Abstract: Compounds I I where A equals t-butyl or a large number of (substituted) aromatics; Y equals azolyl; or Y equals -X-R1 where X=oxygen or sulfur and R1 equals (cyclo)alkyl or (heterocyclic) aryl; or Y equals where R2 equals (cyclo)alkyl, acetyl or aryl; or Y equals -NR3R4 where R3/R4 is alkyl; or Y equals several nitrogen-containing heterocyclic rings; Z equals OH, alkylcarbonyloxy, hal, alkoxy or benzyloxy; and the salts thereof are effective antimycotics or fungicides. They are obtained by reaction of II II with (CH3)2 III and further reaction of the compound IV obtained from this with a nucleophile YM (M=hydrogen or a metal equivalent). The compounds I (where Z=OH) resulting from this can be acylated or alkylated, or converted into I where Z=hal.

公开(公告)号：DK125187A

公开(公告)日：1987-09-13

申请号：DK125187

申请日：1987-03-11

Applicant: HOECHST AG

Inventor： SCHAPER WOLFGANG ,  FUSS ANDREAS ,  RAETHER WOLFGANG ,  DITTMAR WALTER ,  HAENEL HEINZ ,  GERHARDS HERMANN JOSEF ,  SACHSE BURKHARD

IPC: A61K31/415 ,  A01N43/50 ,  A01N43/653 ,  A61P25/08 ,  A61P31/04 ,  A61P31/10 ,  A61P33/02 ,  C07D233/56 ,  C07D233/58 ,  C07D233/60 ,  C07D233/61 ,  C07D247/00 ,  C07D249/08 ,  C07D335/00 ,  C07D405/06 ,  C07D409/06 ,  C07D521/00

Abstract: Azole compounds of the formula (I) in which A denotes CH or N, n = 1, 2 or 3, k = 1 or 2, Ar denotes a (subst.) aromatic radical or (subst.) thienyl, W denotes the atoms necessary to complete a benzene, naphthalene or thiophene ring system, X denotes a radical C(R )2 and in the case in which W denotes the atoms necessary to complete a benzene or naphthalene ring system, also denotes oxygen or sulphur, R and R denote H, halogen, (subst.) alkyl, cycloalkyl, alkoxy, alkylthio, cyano or nitro, and in the case in which W simultaneously denotes the atoms necessary to complete a benzene ring, R also denotes phenyl, phenoxy, phenylthio, phenylsulfinyl, phenylsulphonyl, benzyl, benzyloxy or hydroxyl, where the phenyl groups can be substituted or R and R together, if they are o-orientated, denote an alkylene chain; R denotes H or alkyl or two radicals R together, if they are bonded to the same C-atom, denote an alkylene chain, and their stereoisomers and salts have advantageous fungicidal, antimycotic and anticonvulsive effects.

公开(公告)号：AU562814B2

公开(公告)日：1987-06-18

申请号：AU8433082

申请日：1982-05-31

Applicant: HOECHST AG

Inventor： HERTENSTEIN ULRICH ,  MILDENBERGER HILMAR ,  SACHSE BURKHARD ,  HARTZ PETER

IPC: A01N43/653 ,  A01P3/00 ,  A61K31/41 ,  A61K31/415 ,  C07D231/12 ,  C07D233/56 ,  C07D233/58 ,  C07D233/60 ,  C07D233/64 ,  C07D233/68 ,  C07D233/91 ,  C07D235/06 ,  C07D249/08 ,  C07D521/00 ,  A01N27/00 ,  A01N43/52 ,  A01N43/56 ,  A01N43/50 ,  A01N43/64

Abstract: Substituted ethanols of the general formula in which Ar1 is a carbocyclic or heterocyclic ring and Az is a triazolyl, benzimidazolyl, pyrazolyl or imidazolyl radical, are reacted with aryl hydrocarbons Ar2-H, in which Ar2 has the same meaning as Ar1, in the presence of an acidic catalyst, to give 1,1-diaryl-2-azolylethanes. The substances, which, apart from the imidazolyl derivatives, are new, can be used as biocides, in particular fungicides.

公开(公告)号：ZA866529B

公开(公告)日：1987-04-29

申请号：ZA866529

申请日：1986-08-28

Applicant: HOECHST AG

Inventor： SCHAPER WOLFGANG ,  HARTZ PETER ,  RAETHER WOLFGANG ,  DITTMAR WALTER ,  SACHSE BURKHARD

IPC: C07D409/06 ,  A01N43/50 ,  A01N43/653 ,  A61K31/41 ,  A61K31/415 ,  A61P31/00 ,  A61P31/04 ,  C07D233/60 ,  C07D249/08 ,  C07D333/00 ,  C07D409/08 ,  C07D521/00 ,  C07D ,  A61K ,  A01N

Abstract: Azole derivatives of the formula I where A equals CH or N and R /R equals substituted or unsubstituted phenyl, biphenylyl, phenoxyphenyl, benzylphenyl, benzyloxyphenyl, naphthyl, thienyl, furyl or pyridyl and their salts and esters have outstanding antimycotic and fungicidal activity in all stereoisomeric forms. They are obtained by reaction of a compound II with a sulphur ylide of the formula III to give the compound IV which is reacted with the corresponding compound V to give I. Compound VI can also be used as a starting material and is reacted with 2 equivalents of IIIa compound IV being formed; or compound VI is first reacted with an equivalent of IIIa to give II, and II is then reacted, without working up, with the sulphur ylide IIIb (CH3)2SCH2 to give IV and this is reacted with V to give I.

公开(公告)号：DK217987D0

公开(公告)日：1987-04-29

申请号：DK217987

申请日：1987-04-29

Applicant: HOECHST AG

Inventor： HEUBACH GUENTHER ,  MATTERSTOCK KARL ,  MILDENBERGER HILMAR ,  SACHSE BURKHARD

IPC: A01N43/74 ,  C07D263/58 ,  C07D277/82

公开(公告)号：PT84466A

公开(公告)日：1987-04-01

申请号：PT8446687

申请日：1987-03-12

Applicant: HOECHST AG

Inventor： SCHAPER WOLFGANG ,  FUSS ANDREAS ,  RAETHER WOLFGANG ,  DITTMAR WALTER ,  HAENEL HEINZ ,  GERHARDS HERMANN JOSEF ,  SACHSE BURKHARD

IPC: A61K31/415 ,  A01N43/50 ,  A01N43/653 ,  A61P25/08 ,  A61P31/04 ,  A61P31/10 ,  A61P33/02 ,  C07D233/56 ,  C07D233/58 ,  C07D233/60 ,  C07D233/61 ,  C07D247/00 ,  C07D249/08 ,  C07D335/00 ,  C07D405/06 ,  C07D409/06 ,  C07D521/00 ,  C07D233/00 ,  C07D249/00

Abstract: Azole compounds of the formula (I) in which A denotes CH or N, n = 1, 2 or 3, k = 1 or 2, Ar denotes a (subst.) aromatic radical or (subst.) thienyl, W denotes the atoms necessary to complete a benzene, naphthalene or thiophene ring system, X denotes a radical C(R )2 and in the case in which W denotes the atoms necessary to complete a benzene or naphthalene ring system, also denotes oxygen or sulphur, R and R denote H, halogen, (subst.) alkyl, cycloalkyl, alkoxy, alkylthio, cyano or nitro, and in the case in which W simultaneously denotes the atoms necessary to complete a benzene ring, R also denotes phenyl, phenoxy, phenylthio, phenylsulfinyl, phenylsulphonyl, benzyl, benzyloxy or hydroxyl, where the phenyl groups can be substituted or R and R together, if they are o-orientated, denote an alkylene chain; R denotes H or alkyl or two radicals R together, if they are bonded to the same C-atom, denote an alkylene chain, and their stereoisomers and salts have advantageous fungicidal, antimycotic and anticonvulsive effects.