公开(公告)号：ES2128375T3

公开(公告)日：1999-05-16

申请号：ES93113815

申请日：1993-08-30

Applicant: BAYER AG

Inventor： FISCHER REINER DR ,  KREBS ANDREAS DR ,  LIEB FOLKER DR ,  RUTHER MICHAEL DR ,  STETTER JORG DR ,  ERDELEN CHRISTOPH DR

IPC: A01N43/16 ,  A01N43/40 ,  A01N43/90 ,  A01N47/06 ,  A01N57/24 ,  A61K31/35 ,  A61K31/351 ,  A61K31/365 ,  A61K31/44 ,  A61K31/443 ,  A61K31/4433 ,  A61P33/00 ,  C07D309/36 ,  C07D309/38 ,  C07D311/74 ,  C07D311/94 ,  C07D405/04 ,  C07D405/06 ,  C07D407/04 ,  C07D407/06 ,  C07D407/12 ,  C07D409/04 ,  C07D413/06 ,  C07D493/04 ,  C07D495/04 ,  C07F9/655

Abstract: The invention relates to 3-arylpyrone derivatives of the general formula (I) in which A represents hydrogen, halogen, optionally substituted radicals from the series comprising alkyl, cycloalkyl, alkenyl, alkynyl, arylalkyl, aryl, hetarylalkyl and hetaryl, or the groups -COR , -COR2R , -CN, -CONR R , -SO2R and -P(O)(OR )(OR ) in which R and R independently of one another represent hydrogen or optionally substituted radicals from the series comprising alkyl, alkenyl, arylalkyl, aryl, hetarylalkyl and hetaryl or R and R together represent an optionally substituted alkylene group which can be interrupted by one or more hetero atoms; B represents hydrogen or optionally substituted radicals from the series comprising alkyl, cycloalkyl, alkenyl, alkynyl, arylalkyl, aryl, hetarylalkyl and hetaryl; A and B together form an optionally substituted alkylene or alkenylene group which can be interrupted by, or contain, one or more hetero atoms or hetero groups; X represents halogen, alkyl or alkoxy; Y represents hydrogen, halogen, alkyl, haloalkyl or alkoxy; Z represents hydrogen, halogen, alkyl or alkoxy; n represents an integer 1, 2 or 3; and G represents hydrogen, a metal ion equivalent and an ammonium ion or a group -COR -SO2-R and -CONR R , in which R represents optionally substituted radicals from the series comprising alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl, alkylthioalkyl, or cycloalkyl, arylalkyl, aryl, hetarylalkyl, hetaryl, aryloxyalkyl and hetaryloxyalkyl, it being possible for each of the seven last-mentioned radicals to be interrupted by one or more hetero atoms; R represents optionally substituted radicals from the series comprising alkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl, aryl and arylalkyl; R , R and R independently of one another represent optionally substituted radicals from the series comprising alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, alkenylthio, alkynylthio, cycloalkylthio, aryl, aryloxy and arylthio; R and R independently of one another represent hydrogen or optionally substituted radicals from the series comprising alkyl, alkenyl, alkoxy, cycloalkyl, alkoxyalkyl, aryl or arylalkyl, or together form an optionally substituted alkylene group which can be interrupted by one or more hetero atoms or hetero groups; L represents oxygen or sulphur; and M represents oxygen or sulphur, which can be used as pesticides.t

公开(公告)号：AU2067088A

公开(公告)日：1989-02-16

申请号：AU2067088

申请日：1988-08-10

Applicant: BAYER AG

Inventor： GEHRING REINHOLD DR ,  KORTE UTA JENSEN DR ,  SCHALLNER OTTO DR ,  STETTER JORG DR ,  WROBLOWSKY HEINZ-JURGEN DR ,  MARHOLD ALBRECHT DR ,  BECKER BENEDIKT DR ,  BEHRENZ WOLFGANG DR ,  HOMEYER BERNHARD DR ,  STENDEL WILHELM DR ,  ANDREWS PETER DR

IPC: A01N43/56 ,  A01N47/02 ,  C07D231/18 ,  C07D231/44 ,  C07D231/38

Abstract: There are provided novel 1-arylpyrazoles of the formula (I) in which R represents hydrogen or alkyl, R represents alkyl or haloalkyl, R represents hydrogen, halogen, or a radical where R and R independently of one another in each case represent hydrogen, alkyl, alkenyl or alkynyl, Ar represents one of the radicals where A represents hydrogen, fluorine or chlorine, A represents fluorine or chlorine and A represents hydrogen or fluorine and n represents a number 0, 1 or 2, with the exception of the compound 5-amino-1-(2,5-difluoro- 4-trifluoromethyl-phenyl)-4-dichlorofluoromethylthio-pyrazole. The novel compounds of the formula (I) are outstandingly effective against insects and/or nematodes and can be employed as active substance in pesticides.

公开(公告)号：AU1764588A

公开(公告)日：1988-12-15

申请号：AU1764588

申请日：1988-06-14

Applicant: BAYER AG

Inventor： JENSEN-KORTE UTA DR ,  BEHRENZ WOLFGANG DR ,  STENDEL WILHELM DR ,  HOMEYER BERNHARD DR ,  SCHALINER OTTO DR ,  STETTER JORG DR ,  ANDREWS PETER DR ,  BECKER BENEDIKT DR

IPC: A01N43/56 ,  C07D231/44 ,  C07D231/38

Abstract: There are provided novel substituted 5-ethylamino-1-arylpyrazoles of the formula in which R represents hydrogen or alkyl, R represents haloalkyl and n represents a number 0, 1 or 2, with the exception of the compound of the formula (I) in which R represents hydrogen, R represents dichlorofluoromethyl and n simultaneously represents 0. The compounds of the formula (I) show a highly pronounced activity against animal pests, in particular against insects and nematodes, and are outstandingly suitable as active substances in pesticides.

公开(公告)号：DE3271363D1

公开(公告)日：1986-07-03

申请号：DE3271363

申请日：1982-08-05

Applicant: BAYER AG

Inventor： STETTER JORG DR ,  BUCHEL KARL HEINZ PROF DR ,  FROHBERGER PAUL-ERNST DR ,  REINECKE PAUL DR ,  BRANDES WILHELM DR

IPC: A01N43/50 ,  A01N43/64 ,  A01N43/653 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

Abstract: A substituted azolyl-phenoxy derivative of the formula in which A is a nitrogen atom or a CH group, B is a keto group or a CH(OH) grouping, R1 is an alkyl or halogenoalkyl group of an optionally substituted aryl group, R2 is a hydrogen atom, an alkyl group or an optionally substituted phenyl group, R3 is a hydrogen atom, an alkyl, alkenyl or alkinyl group, m is 1 or 2, X is a halogen atom, or an alkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy or halogenoalkylthio group, and n is 0, 1 or 2, or an addition product thereof with an acid or metal salt, which possesses fungicidal activity particularly for combating cereal diseases as well as rust and scab diseases.

公开(公告)号：GR77953B

公开(公告)日：1984-09-25

申请号：GR830170676

申请日：1983-03-04

Applicant: BAYER AG

Inventor： STETTER JORG DR ,  BUCHEL KARL HEINZ PROF DR ,  REINICKE PAUL DR ,  BRANDES WILHELM DR ,  FROHBERGER PAUL ERNST DR

IPC: A01N43/50 ,  A01N43/64 ,  A01N43/653 ,  C07D233/54 ,  C07D233/60 ,  C07D233/61 ,  C07D249/08 ,  C07D521/00

Abstract: Fungicidally active novel substituted azolylethyl oximinoalkyl ethers of the formula in which A is a nitrogen atom or the CH group, R1 is optionally substituted phenyl, R2, R3 and R4 each independently is hydrogen, alkyl or optionally substituted phenyl, and R5 is hydrogen, alkyl, alkenyl, alkinyl, optionally substituted phenyl or optionally substituted phenylalkyl, or addition products thereof with acids or metal salts.

公开(公告)号：DE2965415D1

公开(公告)日：1983-06-16

申请号：DE2965415

申请日：1979-10-22

Applicant: BAYER AG

Inventor： STETTER JORG DR ,  DRABER WILFRIED DR ,  REGEL ERIK ING GRAD ,  EUE LUDWIG DR ,  SCHMIDT ROBERT RUDOLF DR

IPC: A01N37/22 ,  A01N37/24 ,  A01N37/36 ,  A01N43/72 ,  A01N43/80 ,  C07C233/88 ,  C07D261/04 ,  C07D265/02 ,  C07C131/00

公开(公告)号：DE3060826D1

公开(公告)日：1982-10-28

申请号：DE3060826

申请日：1980-07-23

Applicant: BAYER AG

Inventor： LUNKENHEIMER WINFRIED DR ,  STETTER JORG DR ,  BRANDES WILHELM DR

IPC: A01N37/22 ,  A01N53/00 ,  C07C67/00 ,  C07C231/00 ,  C07C231/02 ,  C07C231/08 ,  C07C231/12 ,  C07C233/38 ,  C07C233/59 ,  C07C103/737

公开(公告)号：DE3060646D1

公开(公告)日：1982-08-26

申请号：DE3060646

申请日：1980-04-28

Applicant: BAYER AG

Inventor： KRAMER WOLFGANG DR ,  BUCHEL KARL HEINZ DR ,  STETTER JORG DR ,  PLEMPEL MANFRED DR ,  HALLER INGO DR

IPC: A01N43/64 ,  A01N43/653 ,  A61K31/41 ,  A61P31/04 ,  C07C45/63 ,  C07C45/67 ,  C07C45/71 ,  C07C49/16 ,  C07C49/167 ,  C07C49/245 ,  C07C49/255 ,  C07D233/60 ,  C07D249/08 ,  C07D521/00

公开(公告)号：DE2960238D1

公开(公告)日：1981-04-30

申请号：DE2960238

申请日：1979-01-29

Applicant: BAYER AG

Inventor： STETTER JORG DR ,  DRABER WILFRIED DR ,  THOMAS RUDOLF DR ,  EUE LUDWIG DR ,  SCHMIDT ROBERT RUDOLF DR ,  LUNKENHEIMER WINFRIED DR

IPC: A01N43/647 ,  A01N43/653 ,  A01N43/70 ,  A01N43/82 ,  A01N43/824 ,  C07D249/08 ,  C07D249/10 ,  C07D249/12 ,  C07D249/14 ,  C07D271/10 ,  C07D271/113 ,  C07D285/12 ,  C07D285/125

公开(公告)号：AU688401B2

公开(公告)日：1998-03-12

申请号：AU8043894

申请日：1994-12-14

Applicant: BAYER AG

Inventor： STETTER JORG DR ,  MENCKE NORBERT DR ,  TURBERG ANDREAS DR ,  WACHENDORFF ULRIKE DR ,  HARTWIG JURGEN DR ,  ERDELEN CHRISTOPH DR ,  OOMS PIETER DR ,  BERTSCH ACHIM DR ,  BOHM STEFAN DR ,  ALIG BERND DR

IPC: C07D231/46 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01P7/04 ,  C07C255/30 ,  C07D231/18 ,  C07D231/38 ,  C07D231/44 ,  C07D401/04 ,  C07D403/04 ,  C07C255/26

Abstract: 1-(Phenyl or pyridyl)-4-(trifluoroethylthio, -sulfinyl or -sulfonyl)-pyrazole derivatives (I) are new. Pyrazole derivatives of formula (I) are new. R1 = H, CN, 1-6C alkyl, (1-4C) alkoxy-(1-4C) alkyl, 1-4C haloalkyl or cyano-(1-2C) alkyl; R2 = trifluoroethyl; R3 = H, NH2, halo, -NHCOR4, -N=C(R5)-NR5R6, 1H-pyrrol-1-yl, -N=CR5R6 or -N=C(R5)-OR7; R4 = 1-6C alkyl (optionally substituted by 1-3 halo), (1-6C) alkoxy-(1-6C) alkyl or phenyl (optionally mono-, di- or trisubstituted); R5 = H or 1-6C alkyl; R6 = H, 1-6C alkyl or phenyl (optionally mono-, di- or trisubstituted); or CR5R6 = optionally substituted pyridyl; R7 = 1-6C alkyl; Ar = phenyl or pyridyl (both optionally substituted by 1-3 of halo, 1-6C haloalkyl, 1-6C haloalkylthio, 1-6C haloalkoxy, alkoxy, hydrazino, di-(1-6C alkyl)-hydrazino, NH2, 1-6C mono- or diaminoalkyl, 1-6C iminoalkyl, CN, 1-6C alkylthio or -CONR9R10); R9, R10 = H or alkyl; and n = 0-2. AN Independent claim is also included for the preparation of (I).