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公开(公告)号:HRP20241163T1
公开(公告)日:2024-11-22
申请号:HRP20241163
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: KULKARNI SHASHANK , YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON MAC ARTHUR JR , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
IPC: C07D413/14 , A61K31/553 , A61P35/00 , C07D403/04 , C07D409/14 , C07D413/04
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公开(公告)号:HRP20220710T1
公开(公告)日:2022-07-22
申请号:HRP20220710
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON MAC ARTHUR JR , KULKARNI SHASHANK , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
IPC: C07D413/14 , A61K31/553 , A61P35/00 , C07D403/04 , C07D409/14 , C07D413/04
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公开(公告)号:DK3784666T3
公开(公告)日:2022-06-20
申请号:DK19726792
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON MAC ARTHUR JR , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN , KULKARNI SHASHANK
IPC: C07D413/14 , A61K31/553 , A61P35/00 , C07D403/04 , C07D409/14 , C07D413/04
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公开(公告)号:DK4043460T3
公开(公告)日:2024-08-26
申请号:DK22161962
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: KULKARNI SHASHANK , YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON MAC ARTHUR JR , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
IPC: C07D413/14 , A61K31/553 , A61P35/00 , C07D403/04 , C07D409/14 , C07D413/04
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公开(公告)号:PL3784666T3
公开(公告)日:2022-07-18
申请号:PL19726792
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON MAC ARTHUR JR , KULKARNI SHASHANK , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
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公开(公告)号:AU2019261308A1
公开(公告)日:2020-10-22
申请号:AU2019261308
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON JR MAC ARTHUR , KUKAMI SHASHANK , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
IPC: C07D413/14 , A61K31/553 , A61P35/00 , C07D403/04 , C07D409/14 , C07D413/04
Abstract: The present invention provides compounds of Formula (I'), or pharmaceutically acceptable salts thereof, pharmaceutical compositions thereof, and methods of use thereof for treating cellular proliferative disorders (e.g. cancer).
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公开(公告)号:AU2019257651A1
公开(公告)日:2020-10-15
申请号:AU2019257651
申请日:2019-04-23
Applicant: VERTEX PHARMA
Inventor: LAUFFER DAVID J , BEMIS GUY , BOYD MICHAEL , DEININGER DAVID , DENG HONGBO , DORSCH WARREN , GU WENXIN , HOOVER RUSSELL R , JOHNSON JR MAC ARTHUR , LEDEBOER MARK WILLEM , LEDFORD BRIAN , MALTAIS FRANCOIS , PENNEY MARINA , TAKEMOTO DARIN , WAAL NATHAN D , WENG TIANSHENG , LI PAN
IPC: C07D471/04 , A61K31/505 , A61P35/00 , C07D475/04
Abstract: The present invention provides compounds of Formula (I), or pharmaceutically acceptable salts thereof, pharmaceutical compositions thereof, and methods of use thereof for reating cellular proliferate disorders (e.g. cancer).
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公开(公告)号:SI3784666T1
公开(公告)日:2022-07-29
申请号:SI201930251
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON MAC ARTHUR JR , KULKARNI SHASHANK , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
IPC: C07D413/00 , A61K31/00 , A61P35/00 , C07D403/00 , C07D409/00
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公开(公告)号:ES2919572T3
公开(公告)日:2022-07-27
申请号:ES19726792
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL , JOHNSON MAC , KULKARNI SHASHANK , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
IPC: C07D413/14 , A61K31/553 , A61P35/00 , C07D403/04 , C07D409/14 , C07D413/04
Abstract: La presente invención proporciona compuestos de fórmula (i'), o sales farmacéuticamente aceptables de las mismas, composiciones farmacéuticas de las mismas y los métodos de uso de los mismos para tratar los trastornos proliferativos celulares (por ejemplo, cáncer). (Traducción automática con Google Translate, sin valor legal)
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公开(公告)号:CA3098335A1
公开(公告)日:2019-10-31
申请号:CA3098335
申请日:2019-04-23
Applicant: MERCK PATENT GMBH , VERTEX PHARMA
Inventor: YU HENRY , CLARK MICHAEL , BEMIS GUY , BOYD MICHAEL , CHANDUPATLA KISHAN , COLLIER PHILIP , DENG HONGBO , DONG HUIJUN , DORSCH WARREN , HOOVER RUSSELL R , JOHNSON MAC ARTHUR , KUKAMI SHASHANK , PENNEY MARINA , RONKIN STEVEN , TAKEMOTO DARIN , TANG QING , WAAL NATHAN D , WANG TIANSHENG , LAUFFER DAVID J , LI PAN
IPC: C07D413/14 , A61K31/553 , A61P35/00 , C07D403/04 , C07D409/14 , C07D413/04
Abstract: The present invention provides compounds of Formula (I'), or pharmaceutically acceptable salts thereof, pharmaceutical compositions thereof, and methods of use thereof for treating cellular proliferative disorders (e.g. cancer).
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