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    Sulfonyl derivatives of erythromycin
    2.
    发明授权
    Sulfonyl derivatives of erythromycin 失效
    红霉素的磺酰衍生物

    公开(公告)号：US3836519A

    公开(公告)日：1974-09-17

    申请号：US35712173

    申请日：1973-05-04

    Applicant: ABBOTT LAB

    Inventor： HALLAS R ,  MARTIN J ,  TADANIER J

    IPC: A61K31/335 ,  A61K31/70 ,  A61K31/7042 ,  A61K31/7048 ,  A61P31/04 ,  C07H17/08 ,  C07C129/18

    CPC classification number: C07H17/08

    Abstract: COVERS SULFONYL DERIVATIVES OF ERHYTHROMYCIN A, B AND C FALLING WITHIN THE FOLLOWING STRUCTURAL FORMULA:

    3,5,7,9,11,13-HEXA(H3C-),4-((2,4-DI(H3C-),3-(R-SO2-O-),

    4-(R1O-)-TETRAHYDROPYRAN-6-YL)-O-),6-((2-(H3C-),

    4-(N(-CH3)2-),5-(R2O-)-TETRAHYDROPYRAN-6-YL)-O-),7,12-

    DI(HO-),13-R3,14-(H5C2-)-OXACYCLOTETRADECANE-2,10-DIONE

    WHERE R IS SELECTED FROM THE ROUP CONSISTING OF LOWERALKYL, LOWERALKENYL, ARYL, SUBSTITUTED ARYL, BENZYL, SUBSTITUTED BENZYL, AROXYALKYL, AND SUBSTITUTED AROXYALKYL; R1 IS HYDROGEN OR METHYL; R2 IS HYDROGEN OR LOWERAKNANOYL AND R3 IS HYDROGEN OR HYDROXYL SAID ERYTHROMYCIN DERIVATIVES BEING USEFUL FOR THIER ANTIBIOTIC ACTIVITY.

    4{41 -o-sulfonyl erythromycin-9-o-oxime derivatives
    3.
    发明授权
    4{41 -o-sulfonyl erythromycin-9-o-oxime derivatives 失效
    4 {41-邻 - 亚甲基红霉素-9-O-氧化衍生物

    公开(公告)号：US3855203A

    公开(公告)日：1974-12-17

    申请号：US35698773

    申请日：1973-05-03

    Applicant: ABBOTT LAB

    Inventor： HALLAS R ,  TADANIER J ,  VON ESCH A

    IPC: A61K31/335 ,  A61K31/70 ,  A61K31/7042 ,  A61K31/7048 ,  A61P31/04 ,  C07H17/08 ,  C07C129/18

    CPC classification number: C07H17/08

    Abstract: Covers 4''''-O-sulfonyl erythromycin-9-O-oxime derivatives falling within the following structural formula: WHERE R is selected from the group consisting of loweralkyl, loweralkenyl, aryl, substituted aryl, benzyl and substituted benzyl, R1 is hydrogen or methyl, R2 is hydrogen or loweralkanoyl, R3 is hydrogen or hydroxyl, and R4 is selected from the group consisting of loweralkyl, cycloalkyl, substituted cycloalkyl, aryl, substituted aryl, benzyl and substituted benzyl. These 9-O-oxime derivative compounds are useful as antibiotics.

    Abstract translation: 涵盖落在以下结构式中的4“-O-磺酰基红霉素-9-O-肟衍生物：

    "> 4
    4.
    发明授权
    4"-deoxy-4"-oxoerythromycin b derivatives 失效
    4“-DEOXY-4” - 紫罗兰霉素B衍生物

    公开(公告)号：US3842069A

    公开(公告)日：1974-10-15

    申请号：US37238773

    申请日：1973-06-21

    Applicant: ABBOTT LAB

    Inventor： JONES P ,  MARTIN J ,  TADANIER J ,  MCALPINE J ,  PAUVLIK J

    IPC: C07H17/08 ,  C07C129/18

    CPC classification number: C07H17/08

    Abstract: 1. A 4"-DEOXY-4"-OXOERYTHROMYCIN COMPOUND SELECTED FROM THE GROUP CONSISTING OF

    2,10-DI(O=),4,5,7,9,11,13,-HEXA(H3C-),4-((4,6-DI(H3C-),

    4-(H3C-O-),5-(O=),6-(H3C-)-TETRAHYDROPYR-2-YL)-O-),6-

    ((3-(R1-O-),4-((H3C)2-N-),6-(H3C-)-TETRAHYDROPYR-2-YL)-

    O-),7-(HO-),12-(R-O-),14-(H5C2-)-OXACYCLOTETRADECANE

    WHERE R IS -CHR2SR3 WHERE R'' IS HYDROGEN OR LOWERALKYL, R3 IS LOWERALKYL AND R1 IS HYDROGEN OR LOWERALKANOYL AND;

    2-(O=),3,5,7,9,11,13-HEXA(H3C-),4-((4,6-DI(H3C-),

    4-(H3C-O-),5-(O=),6-(H3C-)-TETRAHYDROPYR-2-YL)-O-),6-

    ((3-(R1-O-),4-((H3C)2-N-),6-(H3C-)-TETRAHYDROPYR-2-YL)-

    O-),7,10-(-O-),10,12-(-O-CH(-R2)-O-),12-(H5C2-)-

    OXACYCLOTETRADECANE

    WHERE R1 AND R2 ARE AS BEFORE DEFINED.

    8-epi-erythromycins
    5.
    发明授权
    8-epi-erythromycins 失效
    8-EPI-ERYTHROMYCINS

    公开(公告)号：US3842068A

    公开(公告)日：1974-10-15

    申请号：US26308872

    申请日：1972-06-15

    Applicant: ABBOTT LAB

    Inventor： TADANIER J ,  MARTIN J

    IPC: C07H17/08 ,  C07C47/18

    CPC classification number: C07H17/08

    Abstract: 1. AN ERYTHROMYCIN DERIVATIVE SELECTED FROM THE GROUP CONSISTING OF 8-EPI-10,11-ANHYDROETHYTHROMYCN B, 8-EPI11, 12-EPOXYERYTHROMYCIN A 6,9-HEMIACETAL, 8-EPI-ERYTHROMYCIN B AND 8-EPI-10,11-ANHYDROERYTHROMYCIN A.

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