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    1.
    发明专利
    未知

    公开(公告)号：DE19645313A1

    公开(公告)日：1998-05-07

    申请号：DE19645313

    申请日：1996-11-04

    Applicant: BASF AG

    Inventor： ZAGAR CYRILL DR ,  HAMPRECHT GERHARD DR ,  MENGES MARKUS DR ,  MENKE OLAF DR ,  SCHAEFER PETER DR ,  WESTPHALEN KARL-OTTO DR ,  MISLITZ ULF DR ,  WALTER HELMUT DR

    IPC: A01N43/56 ,  A61K31/415 ,  A61K31/4152 ,  A61K31/4155 ,  A61K31/454 ,  A61K31/5377 ,  A61P3/10 ,  C07D231/20 ,  C07D401/10 ,  C07D401/12 ,  C07D403/10 ,  C07D403/12 ,  C07D405/12 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18

    Abstract: The invention relates to substituted 3-benzylpyrazoles of formula (I), their precursors of formulas (IIa), (IIb), (IIc), their byproducts of formula (III) as well as their salts, wherein R stands for H, C1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkyl sulfonyl, C1-C4 halogen alkyl sulfonyl; R stands for C1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkoxy, C1-C4 halogen alkoxy, C1-C4 alkyl thio, C1-C4 halogen alkyl thio, C1-C4 alkyl sulfinyl, C1-C4 halogen alkyl sulfinyl, C1-C4 alkyl sulfonyl, C1-C4 halogen alkyl sulfonyl; R stands for H, CN, NO2, halogen, C1-C4 alkyl, C1-C4 halogen alkyl; X -X stands for chemical bond, optionally substituted methylene-, ethylene-, ethene-1,2-diyl or oxymethylene or thiamethylene chain linked through the heteroatom to the phenyl ring; R -R stands for H, CN, NO2, halogen -O-Y -R , -O-CO-Y -R , -N(Y -R ) (Y -R ), -N(Y -R )-SO2-Y -R , -N(SO2-Y -R ) (SO2-Y -R ), -N(Y -R )-CO-Y -R , -N(Y -R ) (O-Y -R ), -S-Y -R , -SO-Y -R , -SO2-Y -R , -SO2-O-Y -R , -SO2-N(Y -R ) (Y -R ), -CO-Y -R , -C(=NOR )-Y -R , -C(=NOR )-O-Y -R , -C(=NOR )-CO-O-Y -R , -CO-O-Y -R , -CO-S-Y -R , -CO-N(Y -R ) (Y -R ), -CO-N(Y -R ) (O-Y -R ); R stands C1-C4 alkyl, C1-C4 halogen alkyl. The invention further relates to the use of (I) as herbicide, for the desiccation/defoliation of plants, and of (I), (IIa), (IIb), (IIc) and (III) for lowering the sugar content in blood.

    New 3-pyrimidinyl:benzyl-hydroxylamine derivs.
    2.
    发明专利
    New 3-pyrimidinyl:benzyl-hydroxylamine derivs. 未知

    公开(公告)号：DE19616719A1

    公开(公告)日：1997-10-30

    申请号：DE19616719

    申请日：1996-04-26

    Applicant: BASF AG

    Inventor： MENKE OLAF DR ,  HAMPRECHT GERHARD DR ,  HEISTRACHER ELISABETH DR ,  MENGES MARKUS DR ,  SCHAEFER PETER DR ,  ZAGAR CYRILL DR ,  WESTPHALEN KARL-OTTO DR ,  MISLITZ ULF DR ,  WALTER HELMUT DR

    IPC: A01N43/54 ,  A01N47/12 ,  A01N47/30 ,  A01N53/00 ,  C07D239/46 ,  C07C239/10 ,  C07C239/16 ,  C07C239/20 ,  C07C265/12 ,  C07C271/06 ,  C07C275/40

    Abstract: N- or O-(3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-3-yl)benzyl)-hydroxylamine derivs. of formula (I) and salts of (I; R , R and/or R = H) are new. X = -N(R )-O-, with R bonded to O or N; Y = O or S ; R = halo, CN, NO2 or CF3; R = H or halo; R = H, NH2 or Me; R = H, halo, alkyl, haloalkyl, alkylthio, alkylsulphinyl or alkylsulphonyl; R = H, halo or alkyl; R = H, alkyl, haloalkyl, 3-6C cycloalkyl or 2-6C alkenyl; R = (i) H; (ii) alkyl, cycloalkyl, haloalkyl, alkenyl, alkynyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, alkoxycarbonyl, (2-6C)alkenyloxycarbonyl, (2-6C)alkynyloxycarbonyl, alkylthiocarbonyl, alkylsulphonyl or alkylcarbamoyl (all opt. substd. by 1-3 of NO2, CN, cycloalkyl, OH, alkoxy, cycloalkoxy, alkenyloxy, alkynyloxy, alkoxyalkoxy, alkylthio, alkylcarbonyl, alkylcarbonyloxy, alkylsulphinyl, alkylsulphonyl, 1-6C alkylideneaminoxy, alkylcarbamoyl, Ar, OAr, SO2Ar, Het, OHet, COZ R , OCOZ R and NR R ); or (iii) cycloa lkylcarbonyl, benzoyl, phenylsulphonyl or phenylcarbamoyl (all opt. substd. by 1-3 of halo, NO2, CN, alkyl, alkoxy and haloalkyl); R = H ; or alkyl, cycloalkyl, haloalkyl, alkenyl or alkynyl (all opt. substd. by 1-3 of NO2, CN, halo, cycloalkyl, OH, alkoxy, cycloalkoxy, alkenyloxy, alkynyloxy, alkoxyalkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, 1-6C alkylideneaminoxy, Ar, OAr, SO2Ar, Het, OHet, COZ R , OCOZ R and NR R ); Z = a bond, O, S or NR ; Z = a bond, O, S or NR ; Ar = phenyl (opt. substd. by 1-3 of halo, NO2, CN, alkyl, haloalkyl and alkoxy); Het = 3-7 membered satd., partially or completely unsatd. or aromatic heterocycle contg. 1-3 heteroatoms selected from 2 O, 2 S and 3 N (opt. substd. by 1-3 of halo, NO2, CN, alkyl, alkoxy, haloalkyl and alkylcarbonyl); R , R = H, alkyl, haloalkyl, cycloalkyl, alkenyl, alkynyl, alkoxyalkyl or alkoxycarbonylalkyl, or phenyl or phenylalkyl (both opt. ring-substd. by 1-3 of NO2, CN, halo, alkyl, haloalkyl, alkoxy or alkylcarbonyl); or Z + R and/or Z + R may complete an N-bonded heterocycle as defined for Het (except that the optional substituents do not include alkylcarbonyl); R , R = H, OH, alkyl, cycloalkyl or alkoxy; unless specified otherwise, alkyl moieties have 1-6C, alkenyl or alkynyl moieties 3-6C and cycloalkyl moieties 3-8C.

    3.
    发明专利
    未知

    公开(公告)号：DE19532048A1

    公开(公告)日：1997-03-06

    申请号：DE19532048

    申请日：1995-08-31

    Applicant: BASF AG

    Inventor： HEISTRACHER ELISABETH DR ,  HAMPRECHT GERHARD DR ,  MENKE OLAF DR ,  SCHAEFER PETER DR ,  ZAGAR CYRILL DR ,  WESTPHALEN KARL-OTTO DR ,  MISLITZ ULF DR ,  WALTER HELMUT DR

    IPC: C07D277/64 ,  A01N43/78 ,  C07D277/68 ,  C07D277/76 ,  C07D417/04 ,  A01N43/54

    Abstract: The invention concerns substituted benzothiazols of general formula (I) and their salts. In the formula: X , X = O or S; R = H, NH2, C1-C6 alkyl or C1-C6 alkyl halide; R = H, halogen, C1-C6 alkyl, C1-C6 alkyl halide, C1-C6 alkythio, C1-C6 alkylsulphinyl or C1-C6 alkylsulphonyl; R = H, halogen or C1-C6 alkyl; R = H or halogen; R = CN, halogen, C1-C6 alkyl, C1-C6 alkyl halide, C1-C6 alkoxy or C1-C6 alkoxy halide; Y = a chemical bond, -O-, -S-, -SO- or -SO2-; R = hydrogen, CN, halogen, C3-C6 cycloalkyl, C1-C6 alkyl halide, C3-C6 alkenyl, C3-C6 alkyl halide, C3-C6 alkinyl or C1-C6 alkyl, wherein the said cycloalkyl, alkyl, alkenyl and alkinyl groups can be substituted by CN, C1-C6 alkoxy, C1-C6 alkylthio, C1-C6 alkoxycarbonyl, C1-C6 alkylaminocarbonyl, di(C1-C6 alkyl)aminocarbonyl, C1-C6 alkylcarbonyloxy, C1-C6 alkoxy halide, C1-C6 alkylthio halide or C3-C6 cycloalkyl, provided that R can mean cyano only when Y stands for a chemical bond, oxygen or sulphur, and R can mean halogen only when Y stands for a chemical bond. The invention further concerns the use of these substances as herbicides and for the desiccation and abscission of plants.

    4.
    发明专利
    未知

    公开(公告)号：DE19523372A1

    公开(公告)日：1997-01-09

    申请号：DE19523372

    申请日：1995-06-29

    Applicant: BASF AG

    Inventor： MENKE OLAF DR ,  KLINTZ RALF DR ,  HAMPRECHT GERHARD DR ,  HEISTRACHER ELISABETH DR ,  SCHAEFER PETER DR ,  ZAGAR CYRILL DR ,  GOETZ NORBERT DR ,  WESTPHALEN KARL-OTTO DR ,  WALTER HELMUT DR ,  MISLITZ ULF DR

    IPC: A01N43/54 ,  C07C275/24 ,  C07C281/02 ,  C07C281/06 ,  C07D239/54 ,  C07D413/12 ,  C07D419/12 ,  C07D239/545 ,  C07C271/22

    Abstract: The invention concerns 1-amino-3-benzyluracils of formula (I) and their salts. In said formula (I), R = halogen; R , R = H, CN, SCN, halogen, C1-C4-alkyl halide, C1-C4-alkoxy halide, C1-C4-alkylthio halide; R = R + C1-C4-alkyl, C1-C4-alkoxy, C1-C6-alkyl-NH-CO-; R = H, CN, NO2, OH, halogen, optionally substituted NH2, optionally substituted C1-C6-alkoxy halide, C1-C6-alkylthio halide, C1-C6-alkoxy, C1-C6-alkylthio, C3-C8-cycloalkoxy, C3-C8-cycloalkylthio, C3-C6-alkenyloxy, C3-C6-alkenylthio, C3-C6-alkinyloxy, C3-C6-alkinylthio, C1-C6-alkyl-COO-, C1-C6-alkyl-COS-, C3-C6-alkenyl-COO-, C3-C6-alkenyl-COS-, C3-C6-alkinyl-COO-, C3-C6-alkinyl-COS-, C1-C6-alkyl-SO2-O- or C1-C6-alkyl-SO2-; R = 1) H, OH, SH, halogen, C1-C6-alkoxy halide, C1C6-alkylthio halide, C1-C6-alkylthio-(C1-C6-alkyl)carbonyl, C1-C6-alkyliminooxy-CO-, 2) optionally substituted C1C6-alkoxy, C1-C6-alkylthio, C3-C8-cycloalkoxy, C3-C8-cycloalkylthio, C2-C6-alkenyloxy, C2-C6-alkenylthio, C2-C6-alkinyloxy, C2-C6-alkinylthio, C1-C6-alkyl-COO-, C2-C6-alkyl-COS-, C1-C6-alkoxy-COO-, C2-C6-alkenyl-COO-, C2-C6-alkenyl-COS-, C2-C6-alkinyl-COO-, C2-C6-alkinyl-COS-, C1-C6-alkyl-SO2-O-, C1-C6-alkyl-SO2-, 3) -CY-R {Y = -O-, -S-, optionally substituted -NH-}, -C(R )(Z R )(Z R ) {Z , Z = -O-, -S-}, -C(R )=C(R )-CN, -C(R )=C(R )-CO-R , -CH(R )-CH(R )-CO-R , -C(R )=C(R )-CH2-CO-R , -C(R )=C(R )-C(R )=C(R )-CO-R , -C(R )=C(R )-CH2-CH(R )-CO-R , -CO-OR , -CO-SR , -CO-N(R )-OR , -C=C-CO-NH-OR , -C=C-CO-N(R )-OR , -C=C-CS-NH-OR , -C=C-CS-N(R )-OR , -C(R )=C(R )-CO-NH-OR , -C(R )=C(R )-CO-N(R )-OR ,-C(R )=C(R )-CS-NH-OR , -C(R )=C(R )-CS-N(R )-OR , -C(R )=C(R )-C(R )=N-OR , -C(R )=N-OR , -C=C-C(R )=N-OR , -C(Z R )(Z R )-OR , -C(Z R )(Z R )-SR , -C(Z R )(Z R )-N(R )R , optionally substituted amino or -CONH2, azaheterocyclyl, -CO-azaheterocyclyl, or a chain comprising (N + O or N + O + S) heterocyclyl. These compounds can be used as herbicides for desiccating/defoliating plants.

    New (tetra:hydro)phthalimido-cinnamic acid derivatives
    9.
    发明专利
    New (tetra:hydro)phthalimido-cinnamic acid derivatives 未知

    公开(公告)号：DE19610701A1

    公开(公告)日：1997-09-25

    申请号：DE19610701

    申请日：1996-03-19

    Applicant: BASF AG

    Inventor： HEISTRACHER ELISABETH DR ,  HAMPRECHT GERHARD DR ,  MENGES MARKUS DR ,  MENKE OLAF DR ,  SCHAEFER PETER DR ,  ZAGAR CYRILL DR ,  WESTPHALEN KARL-OTTO DR ,  MISLITZ ULF DR ,  WALTER HELMUT DR

    IPC: A01N37/46 ,  C07D209/48 ,  A01N43/38 ,  C07C205/07 ,  C07C211/46

    Abstract: Tetrahydrophthalimido-cinnamic acid derivatives of formula (I) and their salts are new. R1 = H or 1-6C alkyl; R2 = CN, halo, 1-6C alkyl, 1-6C haloalkyl, 1-6C alkoxy or 1-6C haloalkoxy; R3 = NO2, CN or halo; R4 = OR5, SR5, NR6R7 or NR6OR7; R5 = H, 1-6C alkyl (optionally substituted by halo, cyano, 1-6C alkoxy, 1-6C alkylthio,(1-6C alkyl)carbonyl, (1-6C alkyl)aminocarbonyl, di(1-6C alkyl)aminocarbonyl or 1-6C alkyloxyimino), 3-6C alkenyl, 3-6C alkynyl, 3-6C cycloalkyl, di(1-6C alkoxy)-2-6C alkyl, di(1-6C alkylthio)-2-6C alkyl, 3-6C haloalkenyl, or phenyl or benzyl (both optionally ring-substituted by 1-3 of CN, NO2, halo, 1-6C alkyl, 1-6C haloalkyl, 1-6C alkoxy, 1-6C haloalkoxy, 1-6C alkylthio, 1-6C haloalkylthio and (1-6C alkyl)carbonyl); R6-R8 = (1-6C alkyl)carbonyl, (1-6C haloalkyl)carbonyl or as for R5; or R6+R7 = 4-6-membered hydrocarbon chain, optionally with a non-terminal CH2 replaced by O or 1-4C alkylimino. Also claimed are (1) the preparation of substituted anilines (amino-cinnamic acid derivatives) of formula (X) by reduction of the corresponding nitro compound of formula (XI); and (2) the preparation of the nitro compounds (XI) (a) from 4-chloro-5-nitro-2-R2-aniline by the Meerwein reaction, using an alkyne of formula H-C?=C-COR4 (III), or (b) from 4-chloro-5-nitro-2-R2-benzaldehyde by reaction with an ylide of formula (Ar)3P=CX-COR4 (V), or an acidic CH compound of formula CH2Y-COR4 (VI). X = F, Cl or Br; Y = NO2 or CN; Ar = optionally substituted aromatic residue.

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