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公开(公告)号:AT195722T
公开(公告)日:2000-09-15
申请号:AT96934490
申请日:1996-09-30
Applicant: BASF AG
Inventor: MUELLER BERND , SAUTER HUBERT , BAYER HERBERT , GRAMMENOS WASSILIOS , GROTE THOMAS , KIRSTGEN REINHARD , OBERDORF KLAUS , ROEHL FRANZ , GOETZ NORBERT , RACK MICHAEL , MUELLER RUTH , LORENZ GISELA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , HARRIES VOLKER
IPC: C07C249/16 , A01N35/10 , A01N37/50 , A01N43/40 , A01N43/80 , A01N59/12 , C07C251/88 , C07D213/53 , C07D261/08
Abstract: Phenylacetic acid derivatives of the formula Iwhere the substituents and the indexes have the meanings given in the specification, their salts, their preparation and their use.
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公开(公告)号:ZA99866B
公开(公告)日:2000-08-04
申请号:ZA99866
申请日:1999-02-04
Applicant: BASF AG
Inventor: PTOCK ARNE , SAUTER HUBERT , KIRSTGEN REINHARD , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , BAYER HERBERT , GEWEHR MARKUS , CULLMANN OLIVER , MUELLER BERND , GOETZ ROLAND , ROEHL FRANZ , AMMERMANN EBERHARD , LORENZ GISELA , HARRIES VOLKER , STRATHMANN SIEGFRIED
IPC: A01N43/48 , A01N43/56 , C07D401/12 , C07D401/14 , C07D , A01N , A61K
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公开(公告)号:DK0873313T3
公开(公告)日:2000-06-05
申请号:DK96934777
申请日:1996-10-22
Applicant: BASF AG
Inventor: BAYER HERBERT , GRAMMENOS WASSILIOS , GROTE THOMAS , OBERDORF KLAUS , HARRIES VOLKER , M LLER BERND , SAUTER HUBERT , RIHL FRANZ , GITZ NORBERT , RACK MICHAEL , M LLER RUTH , LORENZ GISELA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , KIRSTGEN REINHARD
IPC: A01N43/40 , C07D213/54
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公开(公告)号:CZ2000194A3
公开(公告)日:2000-05-17
申请号:CZ2000194
申请日:1998-07-02
Applicant: BASF AG
Inventor: MUELLER BERND , SAUTER HUBERT , BAYER HERBERT , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , PTOCK ARNE , KIRSTGEN REINHARD , GOETZ NORBERT , GOETZ ROLAND , ROEHL FRANZ , AMMERMANN EBERHARD , HARRIES VOLKER , LORENZ GISELA , STRATHMANN SIEGFRIED
IPC: C07D243/14 , A61K31/55 , A61K31/551 , A61K31/5517 , A61K31/553 , A61K31/554 , A61P1/08 , A61P9/00 , A61P9/10 , A61P25/00 , A61P25/04 , A61P25/06 , A61P25/08 , A61P25/14 , A61P25/16 , A61P25/28 , A61P43/00 , C07D20060101 , C07D223/14 , C07D223/16 , C07D267/14 , C07D281/10 , C07D293/10 , C07D513/06 , C07D517/06 , C07D403/12 , C07D413/12 , A01N43/647 , A01N43/713 , C07D401/14
Abstract: Disclosed are thiazolobenzoheterocycles of the general formulaIncluding their isomers, racemates, enantioners and salts thereof, as well as processes for preparing these compounds and medicaments containing them. Also disclosed are novel intermediates for preparing the foregoing compounds, these intermediates having the formula
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公开(公告)号:AU5982699A
公开(公告)日:2000-05-01
申请号:AU5982699
申请日:1999-10-01
Applicant: BASF AG
Inventor: GEWEHR MARKUS , GRAMMENOS WASSILIOS , SAUTER HUBERT , BAYER HERBERT , GYPSER ANDREAS , MULLER BERND , PTOCK ARNE , CULLMANN OLIVER , GROTE THOMAS , AMMERMANN EBERHARD , LORENZ GISELA , STRATHMANN SIEGFRIED , HARRIES VOLKER
IPC: A01N25/02 , A01N25/08 , A01N43/72 , A01N43/88 , A61K31/539 , A61P31/10 , C07D273/00 , C07D273/01
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公开(公告)号:ZA9806752B
公开(公告)日:2000-01-31
申请号:ZA9806752
申请日:1998-07-29
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS , BAYER HERBERT , SAUTER HUBERT , GROTE THOMAS , GYPSER ANDREAS , MUELLER BERND , PTOCK ARNE , ROEHL FRANZ , GOETZ NORBERT , AMMERMANN EBERHARD , HARRIES VOLKER , LORENZ GISELA , STRATHMANN SIEGRIED
IPC: A01N43/653 , A01N43/80 , C07D249/12 , C07D261/12 , C07D401/12 , C07D403/12 , C07D , A01N
CPC classification number: A01N43/80 , A01N43/653 , C07D249/12
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237.
公开(公告)号:DE19822576A1
公开(公告)日:1999-11-25
申请号:DE19822576
申请日:1998-05-20
Applicant: BASF AG
Inventor: GYPSER ANDREAS , GROTE THOMAS , SAUTER HUBERT , BAYER HERBERT , CULLMANN OLIVER , GEWEHR MARKUS , GRAMMENOS WASSILIOS , PTOCK ARNE , MUELLER BERND , GOETZ ROLAND , GOETZ NORBERT , AMMERMANN EBERHARD , LORENZ GISELA , STRATHMANN SIEGFRIED , HARRIES VOLKER
IPC: C07D231/12 , C07D231/16 , C07D233/54 , C07D233/68 , C07D249/08 , C07D249/10 , C07D249/12 , C07D261/08 , C07D261/10 , C07D261/12 , C07D263/32 , C07D263/34 , C07D403/12 , C07D413/12 , C07D521/00 , A01N43/00 , A61K31/33 , C07D257/04 , C07D261/06 , C07D263/30 , C07D273/00 , C07D285/00
Abstract: Heteroaryl substituted benzyl phenyl ethers (I) are new. Heteroaryl substituted benzyl phenyl ethers (I) and their salts are new: Q = C(CHOMe)-COOMe, C(CHMe)-COOMe, C(NOMe)-COOMe, C(CHOMe)-CONHMe, N(OMe)-COOMe, or group of formula (a)-(d): RA = H, CN, halo, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, cycloalkoxy, alkenyloxy, alkynyloxy, alkylthio, alkenylthio, alkynylthio, alkylsulfinyl, alkenylsulfinyl, alkynylsulfinyl, alkylsulfonyl, alkenylsulfonyl or alkynylsulfonyl (each optionally substituted with halo), acetoxy, cycloalkylthio, cycloalkylsulfinyl, cycloalkylsulfonyl, NH2, NH(alkyl), N(alkyl)2, NH(alkoxy), N(alkyl)(alkoxy), or heterocyclyl optionally substituted with 29 groups; RB = H; alkyl, alkenyl or alkynyl (each optionally substituted with halo); or cycloalkyl; RC = H, alkyl, cycloalkyl, alkenyl or alkynyl (each optionally substituted with alkyl), OH, OMe, OEt, acetoxy, alkylcarbonyl, or alkoxycarbonyl; X = Y p-substituted heteroaryl; Y and Y = halo; CN; NO2; alkyl or alkenyl (each optionally substituted with halo); or alkoxy; Y = halo; CN; NO2; alkyl or alkenyl (each optionally substituted with halo); alkynyl; alkoxy; or Ph, PhO or PhCH2; Ph = phenyl optionally substituted with halo and/or 40 groups; m and n = 0-2; p = 0-3. The full definitions are given in the DEFINITIONS (Full Definitions) Field.
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公开(公告)号:AU712768B2
公开(公告)日:1999-11-18
申请号:AU5895696
申请日:1996-05-13
Applicant: BASF AG
Inventor: MULLER BERND , KIRSTGEN REINHARD , KONIG HARTMANN , RACK MICHAEL , OBERDORF KLAUS , ROHL FRANZ , SAUTER HUBERT , LORENZ GISELA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , HARRIES VOLKER
IPC: A01N43/56 , A01N43/653 , C07D231/18 , C07D231/20 , C07D231/22 , C07D249/12 , C07D401/04 , C07D401/12 , C07D403/04 , C07D403/12
Abstract: Substd. 2-phenyl-3-alkoxy-acrylate ester cpds. of formula (I) are new: n = 0-4; R = alkyl, alkenyl, alkynyl, etc.; or R+R on adjacent C = 3-4 membered bridge contg. 0-2 N, O and/or S, and the rest C (where the ring formed is opt. unsatd. or aromatic); R1, R2 = 1-4C alkyl; R3 = a pyrazolyl or triazolyl gp. of e.g. formula (a1): R4 = alkyl, alkenyl, alkynyl, etc.; Het = N, O or S; m = 0-2; R5 = CN, NO2, halo, etc..
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公开(公告)号:HU216890B
公开(公告)日:1999-10-28
申请号:HU9502454
申请日:1994-02-12
Applicant: BASF AG
Inventor: AMMERMANN EBERHARD , BAYER HERBERT , DOETZER REINHARD , GRAMMENOS WASSILIOS , HARRIES VOLKER , KIRSTGEN REINHARD , KOENIG HARTMANN , LORENZ GISELA , OBERDORF KLAUS , SAUTER HUBERT , WINGERT HORST
IPC: C07C251/48 , A01N37/50 , A01N43/50 , A01N43/56 , A01N43/647 , A01N43/653 , A01N43/74 , A01N43/76 , A01N43/78 , A01N43/80 , A01N43/82 , A01N43/824 , A01N43/828 , A01N43/836 , A01P3/00 , A01P7/02 , A01P7/04 , C07D207/00 , C07D231/18 , C07D231/20 , C07D231/22 , C07D233/70 , C07D233/84 , C07D249/04 , C07D249/08 , C07D249/12 , C07D261/12 , C07D263/20 , C07D263/38 , C07D263/40 , C07D263/46 , C07D271/06 , C07D271/07 , C07D271/10 , C07D271/113 , C07D277/20 , C07D277/28 , C07D277/34 , C07D277/36 , C07D285/08 , C07D285/125 , C07D401/04 , C07D403/04 , C07D405/04 , C07D409/04 , C07D413/04 , C07D417/04 , C07D417/14 , C07C231/18 , C07C231/22
Abstract: Ortho-substd. 2-methoxyiminophenyl ethanoic acid methyl amide derivs. of formula (I) are new. In (I), n = 0-4, X = O or S, Y = 5-membered heteroaromatic ring, which in addn. to R2 can also contain up to 3 gps. chosen from Cl, Me, CF3 or OMe, each R1 is NO2, CN, halogen, 1-4C alkyl, 1-4C haloalkyl, 1-4C alkoxy, 1-4C haloalkoxy, 1-4C alkylthio opt. substd. Ph or PhO. R2 = H, opt. substd. alkyl, alkenyl or alkynyl, on opt. substd. satd. or mono- or di-unsatd. ring contg. in addn. to C, 1-3 heteroatoms as ring members chosen from O, S and N or an opt. substd. mono- or di-nuclear aromatic ring contg. in addn. to C, 1-4 N or 1-2 N and 1 O or S heteroatoms as ring members.
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公开(公告)号:ZA9803231B
公开(公告)日:1999-10-18
申请号:ZA9803231
申请日:1998-04-17
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS , SAUTER HUBERT , BAYER HERBERT , GYPSER THOMAS GROTE ANDREAS , KIRSTGEN REINHARD , MUELLER BERND , PTOCK ARNE , ROEHL FRANZ , GOETZ ROLAND , LORENZ GISELA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , HARRIES VOLKER
IPC: A01N37/10 , A01N37/18 , A01N37/50 , A01N43/20 , A01N43/44 , A01N47/20 , C07C251/42 , C07C251/60 , C07C255/64 , C07C271/28 , C07D203/08 , C07D303/36 , C07D , A01N , C07C
CPC classification number: C07D203/08 , A01N37/50 , A01N43/20 , C07C251/60 , C07C255/64 , C07C2601/02 , C07D303/36
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