25.
    发明专利
    未知

    公开(公告)号:BRPI0511884A

    公开(公告)日:2008-01-15

    申请号:BRPI0511884

    申请日:2005-06-08

    Applicant: BASF AG

    Abstract: The invention relates to triazolopyrimidines of the formula I in which the index n and the substituents R, R 1 , R 2 and X are as defined below: X is nitro, a group -C(S)NR 3 R 4 , a group -C(-N-OR 5 )(NR 6 R 7 ) or a group -C(-N-NR 8 R 9 )(NR 10 R 11 ), R is halogen, cyano, hydroxyl, cyanato, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N or S; R 1 is alkyl in which one carbon atom may be replaced by a silicon atom, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via a carbon atom and which contains one, two, three or four heteroatoms, independently of one another selected from the group consisting of O, N and S, as ring members; where R 1 may be substituted as defined in the description; R 2 is alkyl, alkenyl or alkynyl which may be substituted as defined in the description; R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 and R 11 are, independently of one another, selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl or alkynyl, where the 4 lastmentioned radicals may be substituted as defined in the description; or R 3 and R 4 , R 6 and R 7 , R 8 and R 9 and/or R 10 and R 11 together with the nitrogen atom to which they are attached form a four-, five- or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; and n is 0 or an integer 1, 2, 3 or 4; and the agriculturally acceptable salts thereof, to crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt thereof and at least one liquid or solid carrier and to a method for controlling phytopathogenic harmful fungi.

    27.
    发明专利
    未知

    公开(公告)号:AT373004T

    公开(公告)日:2007-09-15

    申请号:AT04803894

    申请日:2004-12-15

    Applicant: BASF AG

    Abstract: Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is hydrogen, chlorine or bromine; R 1 , R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and/or may be substituted as defined in the description; R 3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, cycloalkyl, halocycloalkyl or phenylalkyl; R 1 , R 2 and/or R 3 may be substituted as defined in the description; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

    28.
    发明专利
    未知

    公开(公告)号:DE502005001146D1

    公开(公告)日:2007-09-13

    申请号:DE502005001146

    申请日:2005-01-15

    Applicant: BASF AG

    Abstract: The invention relates to substituted triazolopyrimidines of formula (I), with the substituents as follows: R 1 , R 2 =H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, comprising one to four heteroatoms of the group O, N or S, R 1 and R 2 can, together with the nitrogen atom to which it is attached, form a five- or six-membered heterocycle or heteroaryl, bonded via N and containing one to three further heteroatoms from the group O, N and S as ring members, substituted as per the description, L 1 =fluorine, chlorine or bromine, L 2 =H, alkyl or alkoxy and X=halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy. The invention further relates to methods and intermediates for production of said compounds, agents comprising the same and use thereof for controlling fungal pests harmful to plants.

    5-FENILPIRIMIDINAS I EN TERAPEUTICA.

    公开(公告)号:MX2007008397A

    公开(公告)日:2007-09-07

    申请号:MX2007008397

    申请日:2006-01-30

    Applicant: BASF AG

    Abstract: La presente invencion se refiere a 5-fenilpirimidinas I sustituidas que llevan un radical X en la posicion 4 del anillo pirimidina, un radical Y en la posicion 6 del anillo pirimidina, el radical X que designa un grupo de la formula NR1R2, OR1a o SR1a, en donde R1, R2, de modo independiente entre si, designan hidrogeno, alquilo C1-C10, alquenilo C2-C6, alquinilo C2-C6, haloalquilo C1-C10, cicloalquilo C3-C8, halocicloalquilo C3-C8, fenilo, o heteroarilo de 5 o 6 miembros o heterociclilo de 5 o 6 miembros, que contiene 1, 2, 3 o 4 atomos de nitrogeno o 1, 2 o 3 atomos de nitrogeno y un atomo de azufre u oxigeno como miembros del anillo, cuyos radicales pueden no estar sustituidos o pueden llevar 1, 2, 3 o 4 radicales Ra1; o el radical NR1R2 tambien puede formar un anillo heterociclico opcionalmente sustituido de 5 o 6 miembros, que contiene 1, 2, 3 o 4 atomos de nitrogeno o 1, 2 o 3 atomos de nitrogeno y un atomo de azufre u oxigeno como miembros del anillo, que son no adyacentes al nitrogeno de NR1R2, en donde dos atomos de C adyacentes o un atomo de N y un atomo de C adyacente pueden unirse por una cadena alquileno C1-C4 y en donde el anillo heterociclico puede no estar sustituido o puede llevar 1, 2, 3 o 4 radicales Ra1 tal como se definio en la reivindicacion 1 R1a tiene uno de los significados dados para R1 salvo para hidrogeno; el radical Y esta seleccionado del grupo que consiste en halogeno, ciano, alquilo C1-C4, alquenilo C2-C4, alquinilo C2-C4, cicloalquilo C3-C6, alcoxi C1-C4, alqueniloxi C3-C4, alquiniloxi C3-C4, alquiltio C1-C6, di-(alquil C1-C6)amino o alquil C1-C6-amino, en donde los radicales alquilo, alquenilo y alquinilo de Y pueden estar sustituidos con halogeno, ciano, nitro, alcoxi C1-C2 o alcoxi C1-C4-carbonilo; y en donde el radical pirimidina tambien puede llevar un radical diferente de hidrogeno en la posicion 2 y en donde el anillo fenilo en la posicion 5 del anillo pirimidina puede no estar sustituido o puede llevar 1, 2, 3, 4 o 5 radicales L que son diferentes de hidrogeno, y las sales farmaceuticamente aceptables de 5-fenilpirimidinas sustituidas para usar en terapeutica, en particular en terapeutica o tratamiento de enfermedades cancerosas.

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