-
公开(公告)号:DE50309134D1
公开(公告)日:2008-03-20
申请号:DE50309134
申请日:2003-12-16
Applicant: BASF AG
Inventor: MUELLER BERND , TORMO I BLASCO JORDI , GROTE THOMAS , BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A01N43/653
Abstract: Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R 1 is C 1 -C 10 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -alkynyl, C 3 -C 10 -cycloalkyl, C 3 -C 10 -cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R 2 is C 1 -C 4 -alkyl which may be substituted by halogen, cyano, nitro or C 1 -C 2 -alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SO m -R x , NR x R y or NR x -(C-O)-R y ; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
-
公开(公告)号:BRPI0512332A
公开(公告)日:2008-03-04
申请号:BRPI0512332
申请日:2005-06-14
Applicant: BASF AG
Inventor: BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , MUELLER BERND , NIEDENBRUECK MATTHIAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , NAVE BARBARA , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A01N43/653 , A01N43/90
Abstract: The use of substituted triazolopyrimidines of the formula I in which R 1 is alkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen or a group R 1 , where R 1 and/or R 2 may be substituted according to the description, and X is halogen; as fungicides, novel 6-(2-tolyl)triazolopyrimidines, processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
-
公开(公告)号:BRPI0512306A
公开(公告)日:2008-02-26
申请号:BRPI0512306
申请日:2005-06-18
Applicant: BASF AG
Inventor: REINHEIMER JOACHIM , SCHIEWECK FRANK , GROTE THOMAS , BLETTNER CARSTEN , SCHWOEGLER ANJA , GEWEHR MARKUS , GRAMMENOS WASSILIOS , HUENGER UDO , MUELLER BERND , SCHOFER PETER , SPEAKMAN JOHN BRYAN , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D401/04 , A01N43/40 , C07D213/61 , C07D213/70 , C07D213/78 , C07D213/84 , C07D213/86 , C07D417/04
Abstract: The invention relates to 2-substituted pyridines of the formula I in which the index n and the substituents R1 to R4 and L are as defined in the description and in each case one of the two ring members X1, X2 is N, the other is C—H or C-halogen; Y is a group —CH—R1—, —N—R1—, —O— or —S— and is five- or six-membered hetaryl comprising 1 to 3 heteroatoms selected from the group consisting of O, N and S or is phenyl, and to processes for their preparation, intermediates for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.
-
公开(公告)号:AT385499T
公开(公告)日:2008-02-15
申请号:AT03789291
申请日:2003-12-16
Applicant: BASF AG
Inventor: MUELLER BERND , TORMO I BLASCO JORDI , GROTE THOMAS , BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A01N43/653
Abstract: Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R 1 is C 1 -C 10 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -alkynyl, C 3 -C 10 -cycloalkyl, C 3 -C 10 -cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R 2 is C 1 -C 4 -alkyl which may be substituted by halogen, cyano, nitro or C 1 -C 2 -alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SO m -R x , NR x R y or NR x -(C-O)-R y ; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.
-
公开(公告)号:BRPI0511884A
公开(公告)日:2008-01-15
申请号:BRPI0511884
申请日:2005-06-08
Applicant: BASF AG
Inventor: BLETTNER CARSTEN , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , HUENGER UDO , MUELLER BERND , NIEDENBRUECK MATTHIAS , RHEINHEIMER JOACHIM , SCHOFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , RACK MICHAEL , NAVE BARBARA , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A01N43/647 , A01N43/90 , C07D487/00
Abstract: The invention relates to triazolopyrimidines of the formula I in which the index n and the substituents R, R 1 , R 2 and X are as defined below: X is nitro, a group -C(S)NR 3 R 4 , a group -C(-N-OR 5 )(NR 6 R 7 ) or a group -C(-N-NR 8 R 9 )(NR 10 R 11 ), R is halogen, cyano, hydroxyl, cyanato, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one, two, three or four heteroatoms from the group consisting of O, N or S; R 1 is alkyl in which one carbon atom may be replaced by a silicon atom, alkenyl, alkynyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via a carbon atom and which contains one, two, three or four heteroatoms, independently of one another selected from the group consisting of O, N and S, as ring members; where R 1 may be substituted as defined in the description; R 2 is alkyl, alkenyl or alkynyl which may be substituted as defined in the description; R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , R 9 , R 10 and R 11 are, independently of one another, selected from the group consisting of hydrogen, alkyl, cycloalkyl, alkenyl or alkynyl, where the 4 lastmentioned radicals may be substituted as defined in the description; or R 3 and R 4 , R 6 and R 7 , R 8 and R 9 and/or R 10 and R 11 together with the nitrogen atom to which they are attached form a four-, five- or six-membered saturated or partially unsaturated ring which may be substituted as defined in the description; and n is 0 or an integer 1, 2, 3 or 4; and the agriculturally acceptable salts thereof, to crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt thereof and at least one liquid or solid carrier and to a method for controlling phytopathogenic harmful fungi.
-
公开(公告)号:CR9335A
公开(公告)日:2007-10-04
申请号:CR9335
申请日:2007-08-24
Applicant: BASF AG
Inventor: GEWEHR MARKUS , DIETZ JOCHEN , GROTE THOMAS , BLETTNER CARSTEN , GRAMMENOS WASSILIOS , HUNGER UDO , MULLER BERND , SCHIEWECK FRANK , SCHWOGLER ANJA , LOHMANN JAN KLAAS , RHEINHEIMER JOACHIM , SCHAFER PETER , STRATHMANN SIEGFRIED , STIERL REINHARD
IPC: A01N43/56 , C07D231/14
Abstract: La presente invencion se refiere a anilidas de acido pirazolcarboxilico de la formula I.
-
公开(公告)号:AT373004T
公开(公告)日:2007-09-15
申请号:AT04803894
申请日:2004-12-15
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A01N43/90
Abstract: Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is hydrogen, chlorine or bromine; R 1 , R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and/or may be substituted as defined in the description; R 3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, cycloalkyl, halocycloalkyl or phenylalkyl; R 1 , R 2 and/or R 3 may be substituted as defined in the description; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.
-
公开(公告)号:DE502005001146D1
公开(公告)日:2007-09-13
申请号:DE502005001146
申请日:2005-01-15
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , BLETTNER CARSTEN , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , RHEINHEIMER JOACHIM , SCHAEFER PETER , SCHIEWECK FRANK , SCHWOEGLER ANJA , WAGNER OLIVER , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOEFL ULRICH , STIERL REINHARD
IPC: C07D487/04 , A01N43/90
Abstract: The invention relates to substituted triazolopyrimidines of formula (I), with the substituents as follows: R 1 , R 2 =H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, comprising one to four heteroatoms of the group O, N or S, R 1 and R 2 can, together with the nitrogen atom to which it is attached, form a five- or six-membered heterocycle or heteroaryl, bonded via N and containing one to three further heteroatoms from the group O, N and S as ring members, substituted as per the description, L 1 =fluorine, chlorine or bromine, L 2 =H, alkyl or alkoxy and X=halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy. The invention further relates to methods and intermediates for production of said compounds, agents comprising the same and use thereof for controlling fungal pests harmful to plants.
-
公开(公告)号:MX2007008397A
公开(公告)日:2007-09-07
申请号:MX2007008397
申请日:2006-01-30
Applicant: BASF AG
Inventor: MULLER BERND , GROTE THOMAS , JABS THORSTEN , RHEINHEIMER JOACHIM , SCHIEWECK FRANK , BLETTNER CARSTEN , NAVE BARBARA , SCHWOEGLER ANJA
IPC: A61K31/506 , A61K31/505 , C07D239/42 , C07D239/48 , C07D401/04 , C07D403/04 , C07D417/04
Abstract: La presente invencion se refiere a 5-fenilpirimidinas I sustituidas que llevan un radical X en la posicion 4 del anillo pirimidina, un radical Y en la posicion 6 del anillo pirimidina, el radical X que designa un grupo de la formula NR1R2, OR1a o SR1a, en donde R1, R2, de modo independiente entre si, designan hidrogeno, alquilo C1-C10, alquenilo C2-C6, alquinilo C2-C6, haloalquilo C1-C10, cicloalquilo C3-C8, halocicloalquilo C3-C8, fenilo, o heteroarilo de 5 o 6 miembros o heterociclilo de 5 o 6 miembros, que contiene 1, 2, 3 o 4 atomos de nitrogeno o 1, 2 o 3 atomos de nitrogeno y un atomo de azufre u oxigeno como miembros del anillo, cuyos radicales pueden no estar sustituidos o pueden llevar 1, 2, 3 o 4 radicales Ra1; o el radical NR1R2 tambien puede formar un anillo heterociclico opcionalmente sustituido de 5 o 6 miembros, que contiene 1, 2, 3 o 4 atomos de nitrogeno o 1, 2 o 3 atomos de nitrogeno y un atomo de azufre u oxigeno como miembros del anillo, que son no adyacentes al nitrogeno de NR1R2, en donde dos atomos de C adyacentes o un atomo de N y un atomo de C adyacente pueden unirse por una cadena alquileno C1-C4 y en donde el anillo heterociclico puede no estar sustituido o puede llevar 1, 2, 3 o 4 radicales Ra1 tal como se definio en la reivindicacion 1 R1a tiene uno de los significados dados para R1 salvo para hidrogeno; el radical Y esta seleccionado del grupo que consiste en halogeno, ciano, alquilo C1-C4, alquenilo C2-C4, alquinilo C2-C4, cicloalquilo C3-C6, alcoxi C1-C4, alqueniloxi C3-C4, alquiniloxi C3-C4, alquiltio C1-C6, di-(alquil C1-C6)amino o alquil C1-C6-amino, en donde los radicales alquilo, alquenilo y alquinilo de Y pueden estar sustituidos con halogeno, ciano, nitro, alcoxi C1-C2 o alcoxi C1-C4-carbonilo; y en donde el radical pirimidina tambien puede llevar un radical diferente de hidrogeno en la posicion 2 y en donde el anillo fenilo en la posicion 5 del anillo pirimidina puede no estar sustituido o puede llevar 1, 2, 3, 4 o 5 radicales L que son diferentes de hidrogeno, y las sales farmaceuticamente aceptables de 5-fenilpirimidinas sustituidas para usar en terapeutica, en particular en terapeutica o tratamiento de enfermedades cancerosas.
-
公开(公告)号:EA008920B1
公开(公告)日:2007-08-31
申请号:EA200501533
申请日:2004-03-30
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , BLETTNER CARSTEN , MULLER BERND , GEWEHR MARCUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , SCHAFER PETER , SCHIEWECK FRANK , SCHWOGLER ANJA , SCHERER MARIA , STRATHMANN SIEGFRIED , SCHOFL ULRICH , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: Предложены 7-алкиламинотриазолопиримидиныформулы Iвкоторойзаместителиимеютследующиезначения: L означаетнезависимодруготдругагалоген, С-С-алкил, C-C-галогеналкил, S(O)A, Аозначает C-C-алкил, n равно 0, m равно 1, 2, 3, 4 или 5, причемпоменьшеймереоднагруппа L находитсяв орто-положениик связис триазолопиримидиновымскелетом; X означаетгалоген, циано, С-С-алкил, илиС-С-алкокси; R- водородилиС-С-алкил; R- С-C-алкинил, которыйможетбытьнезамещеннымиличастичноилиполностьюгалогенированным; способихполучения, атакжесодержащееихсредствои способборьбыс фитопатогеннымигрибами.
-
-
-
-
-
-
-
-
-