公开(公告)号：WO03008417A9

公开(公告)日：2003-10-30

申请号：PCT/EP0207578

申请日：2002-07-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 式（I）的取代的6-（2-甲苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基，炔基或链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5-或6-元杂环基，或者含有1-4个氮原子或1-3个氮原子的5-或6-元杂芳基， 硫或氧原子，或者其中R 1和R 2基团可以如说明书中所定义的那样未被取代或被取代，或者R 1和R 2与中间的氮原子一起表示5或6 - 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的可被取代的 - 元杂环; R 3是卤素，氰基，烷基，烷氧基，卤代烷基或C（= O）A，其中A是氢，羟基，烷基，氨基或单或二烷基氨基; n是1至4的整数; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基; 它们的制备方法，含有它们的组合物以及它们用于防治植物病原性真菌的用途。

公开(公告)号：WO02074753A3

公开(公告)日：2002-12-27

申请号：PCT/EP0202739

申请日：2002-03-13

Applicant: BASF AG ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00 ,  C07D473/00

CPC classification number: C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04 ,  C07D473/06 ,  C07D487/04

Abstract: The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: R represents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group 0, N or S, and which can be substituted as defined in the description; R represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, R and R can also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; R and R represent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; R and R represent hydrogen, halogen, alkyl or halogenalkyl; and R represents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi.

Abstract translation: 式（I）其中取代基具有以下Begende含义的5-苯基嘧啶，R <1> 5〜10元饱和，部分不饱和或芳族单环或双环杂环，选自下组0含有一至四个杂原子，N或 如说明书中所定义的可被取代的S，R <2>为氢，卤素，氰基，烷基，卤代烷基或烷氧基; [R <3>，R <4>是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R <3>和R <4>可与氮原子一起他们 连接，形成可以被杂原子中断并且可以携带一个或多个取代基的五元或六元环; [R <5> - [R <6>是氢，卤素，烷基，卤代烷基或烷氧基; [R <7> - [R <8>是氢，卤素，烷基或卤代烷基; [R <9>是氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧基羰，卤代烷氧基或烷氧羰，涉及用于制备这些化合物和它们在防治有害真菌中的用途的方法和中间体。

公开(公告)号：WO0248146A2

公开(公告)日：2002-06-20

申请号：PCT/EP0114577

申请日：2001-12-12

Applicant: BASF AG ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D471/04 ,  C07D487/04

CPC classification number: C07D471/04 ,  A01N43/90 ,  C07D487/04

Abstract: The invention relates to the use of substituted imidazoazines of formula (I), in which the variables have the following meanings: R represents alkyl, phenyl, phenylalkyl, naphthyl, anthracenyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, containing one to three N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, or condensed 8-membered to 12-membered hetaryl or condensed 8-membered to 12-membered heterocyclyl, containing one to four N atoms and/or one O atom or S atom or one or two O atoms and/or S atoms, whereby R can be unsubstituted or can be substituted as cited in the description; R and R represent hydrogen, alkyl, alkenyl, alkynyl, alkyl halide, alkenyl halide, alkynyl halide, trialkyl silylalkyl, phenyl, phenylalkyl or R and R , together with the bridging N atom, form a 5-membered or 6-membered heterocyclic or heteroaromatic ring, which can be interrupted by one to three N atoms and/or one O atom or S atom or by one or two O atoms and/or S atoms, and which can be substituted; A and B represent N or CR ; R , R and R represent hydrogen, halogen, cyano, nitro, hydroxy, alkyl, alkyl halide, cycloalkyl, alkoxy, alkoxy halide, alkylthio, amino, alkyl amino, dialkylamino, alkenyl, alkenyloxy, alkynyl or alkynyloxy. The inventive compounds are used for controlling phytopathogenic harmful fungi. The invention further relates to agents containing the inventive compounds, to novel imidazoazines, and to methods for the production thereof.

Abstract translation: 使用式（I）的取代的Imidazoazinen的，其中各变量具有以下含义：R t <1>是烷基，苯基，苯基烷基，萘基，蒽基，环烷基，5-或6-员杂芳基或5-或6-元杂环基 含有1至3个N原子和/或一个O或S原子或一个或两个O和/或S原子，或稠合8-12 gliederiges杂芳基或稠合的8-12 gliederiges杂环基， 含有一至四个N原子和/或一个O或S原子或一个或两个O和/或O原子，其中R是未取代的<1>或作为可在本说明书中被取代; [R <2>，R <3>是氢，烷基，烯基，炔基，卤代烷基，卤代烯基，卤代炔基，三烷基甲硅烷基，苯基，苯基烷基或R <2>，R <3>连同桥接氮原子的5-或6- 形成 - 元杂环基或可被一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子被中断杂芳族环; A，B，N或CR <4>; [R <4>，R <5> - [R <6>为氢，卤素，氰基，硝基，羟基，烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，烷硫基，氨基，烷基氨基，二烷基氨基，烯基，烯氧基，炔氧基或炔氧基; 防治植物病原性有害真菌的，含有它们，它们的制备新imidazoazines和方法的组合物。

公开(公告)号：WO0020399A3

公开(公告)日：2000-07-27

申请号：PCT/EP9907125

申请日：1999-09-24

Applicant: BASF AG ,  GYPSER ANDREAS ,  KIRSTGEN REINHARD ,  SAUTER HUBERT ,  BAYER HERBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  PTOCK ARNE ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

Inventor： GYPSER ANDREAS ,  KIRSTGEN REINHARD ,  SAUTER HUBERT ,  BAYER HERBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  PTOCK ARNE ,  TORMO I BLASCO JORDI ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/56 ,  C07D231/08 ,  C07D401/04 ,  C07D401/06 ,  C07D405/04 ,  C07D409/04

CPC classification number: C07D401/04 ,  C07D231/08 ,  C07D401/06 ,  C07D405/04 ,  C07D409/04

Abstract: The invention relates to the use of substituted 5-hydroxypyrazoles of formula (I) in which the substituents have the following meanings: B represents aryl or heteroaryl; A represents C=O, C=S or SO2; R represents alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, cycloalkyl, C3-C10-cycloalkenyl, cycloalkynyl, or aryl, heterocyclyl or heteroaryl; R represents hydrogen; R represents hydrogen, nitro, cyano, N(R')2, alkyl, alkyl halide, alkoxy, alkoxy halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide, whereby R', independent of one another, represents hydrogen or alkyl; or R and R , together, represent a group =O, =S or =N-O-R , whereby R represents hydrogen, alkyl, alkyl halide, alkenyl, alkenyl halide, alkynyl or alkynyl halide; R represents hydrogen, halogen, nitro, cyano N(R')2, alkyl, alkyl halide, COOR', heteroaryl or heterocyclyl. The invention also relates to the use of said compounds for combating harmful fungi, to agents containing the compounds, to novel 5-hydroxypyrazoles and to methods for the production thereof.

Abstract translation: 本发明涉及式（I）的5-羟基吡唑啉的用途，其中取代基具有以下含义：B芳基或杂芳基; A C = O，C = S或SO 2; R 1是烷基，卤代烷基，烯基，卤代烯基，炔基或卤代炔基，环烷基，C 3 -C 10 - 环烯基，环炔基或芳基，杂环基或杂芳基; R 2氢; [R <3>为氢，硝基，氰基，N（R '）2，烷基，卤代烷基，烷氧基，卤代烷氧基，链烯基，卤代烯基，炔基或卤代炔基，其中R' 独立地为氢或烷基; 或R <2>和R <3>一起表示基团= O，= S或= N-O-R <5>，其中R <5>是氢，烷基，卤代烷基，链烯基，卤代烯基，炔基或卤代炔基; R 4是氢，卤素，硝基，氰基，N（R'）2，烷基，卤代烷基，COOR'，杂芳基或杂环基; 用于控制有害真菌，含有它们的试剂和新的5-羟基吡唑及其制备方法。

公开(公告)号：BRPI0610576A2

公开(公告)日：2016-11-16

申请号：BRPI0610576

申请日：2006-05-24

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  DIETZ JOCHEN ,  GEWEHR MARKUS ,  NIEDENBRÜCK MATTHIAS ,  GROTE THOMAS

IPC: C07D231/00 ,  A01N43/56 ,  A01P3/00

公开(公告)号：BRPI0608802A2

公开(公告)日：2016-08-23

申请号：BRPI0608802

申请日：2006-05-10

Applicant: BASF AG

Inventor： SCHWOGLER ANJA ,  MULLER BERND ,  SCHIEWECK FRANK ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  RHEINHEIMER JOACHIM ,  DIETZ JOCHEN ,  GEWEHR MARKUS ,  SCHÄFER PETER ,  GROTE THOMAS ,  HÜNGER UDO ,  GRAMMENOS WASSILIOS

IPC: C07D231/14 ,  A01N43/56

公开(公告)号：BRPI0508281B1

公开(公告)日：2015-04-14

申请号：BRPI0508281

申请日：2005-03-08

Applicant: BASF AG

Inventor： BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MÜLLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHÄFER PETER ,  SCHIEWECK FRANK ,  SCHWÖGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRÜCK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHÖFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

公开(公告)号：CA2617503C

公开(公告)日：2014-07-15

申请号：CA2617503

申请日：2006-08-01

Applicant: BASF AG

Inventor： DIETZ JOCHEN ,  GEWEHR MARKUS ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD ,  WERNER FRANK ,  SCHERER MARIA

IPC: A01N43/56 ,  A01N35/04 ,  A01N37/34 ,  A01N37/38 ,  A01N43/653 ,  A01N43/90 ,  A01N47/14 ,  A01N47/24 ,  A01N47/38 ,  A01P3/00

Abstract: The invention relates to fungicidal mixtures containing the following as active components: 1) at least one 1-methyl pyrazol-4-yl carboxylic acid anilide of formula (I), in which X = O or S, R1 = C1-C4 alkyl or C1-C4 haloalkyl, R2 = hydrogen or halogen, R3, R4 and R5 = independently of one another cyano, nitro, halogen, C1-C4 alkyl, C1-C4 haloalkyl, C1-C4 alkoxy, C1-C4 haloalkoxy or C1-C4 alkylthio; and 2) at least one active ingredient II, selected from the active ingredient groups A) to F) in a synergistically active quantity: A) azoles; B) strobilurins; C) carboxamides; D) heterocyclic compounds; E) carbamates; F) other fungicides. The invention also relates to a method for controlling pathogenic fungi using mixtures of at least one compound I and at least one active ingredient II, to the use of the compound(s) I and active ingredients II for producing mixtures of this type and to agents and seeds containing said mixtures.

公开(公告)号：CA2597022C

公开(公告)日：2013-05-07

申请号：CA2597022

申请日：2006-02-15

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  DIETZ JOCHEN ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GRAMMENOS WASSILIOS ,  HUENGER UDO ,  MUELLER BERND ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  LOHMANN JAN KLAAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD

IPC: C07D231/14 ,  A01N43/56

Abstract: The invention relates to pyrazole carboxylic acid anilides of formula (I), in which the variables have the following meanings: n is zero or 2; m is 2 or 3; X1 represents fluorine or chlorine; X2 represents halogen, Y represents CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, methoxy or methylthio; p is 0 or 1; R1 represents fluorine, chlorine, bromine, C1-C4 alkyl and C1-C4 alkyl halide; R2 represents hydrogen or halogen; R3 represents hydrogen, methyl or ethyl, and; W represents O or S; with the provision that if: a) W = O, R1 = methyl, and R3 represents hydrogen, R2 does not represent fluorine or; b) W = O, n = 0, m = 2, p = 0, and R2 and R3 represent hydrogen, R1 does not represent trifluoromethyl or difluoromethyl. The invention also relates to a method for producing these compounds, to agents containing them, and to a method for using them for controlling pathogenic fungi.

公开(公告)号：CA2557781C

公开(公告)日：2012-01-10

申请号：CA2557781

申请日：2005-03-08

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90 ,  C07D239/00 ,  C07D249/00

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl or alkoxyalkyl, whereby the aliphatic groups can be substituted according to the description; R2 represents CHR3CH3, cyclopropyl, CH=CH2 or CH2CH=CH2 and R3 represents hydrogen, CH3 or CH2CH3. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.