公开(公告)号：WO2005095405A3

公开(公告)日：2005-12-22

申请号：PCT/EP2005004187

申请日：2005-03-29

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 6-(2,6-dichlorophenyl)-triazolopyrimidines of formula (I) wherein the substituents have the following designations: R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, halogencycloalkenyl, alkinyl, halogenalkinyl or phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group containing O, N or S; R and R can also form, together with the nitrogen atom to which they are bound, a five-membered or six-membered heterocycle or heteroaryl which is bound by N and contains between one and three other heteroatoms from the group containing O, N and S as a cyclic member and is substituted according to the description; and X represents alkyl, cyano, alkoxy, halogenalkoxy, alkenyloxy or halogenalkenyloxy, but does not represent C1-C4 alkyl when R and R together represent piperidin-1-yl or 4-methylpiperidin-1-yl. The invention also relates to a method for producing said compounds, agents containing the same, and the use thereof for controlling plant pathogenic fungi.

Abstract translation: 6-（2,6-二氯苯基） - 三唑并嘧啶的式（I）的其中取代基具有以下含义：R t <1>，R <2>是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基 基，炔基，卤代炔基，或苯基，萘基，或含有选自O，N，或S，R <1>和R <2>也可以，一起一至四个杂原子的五元或六元饱和，部分不饱和或芳族杂环 形成一个五元或六元杂环基或杂芳基的氮原子与它们所连接，这是经N个附接和选自O，N和S的一至三个另外的杂原子作为环成员，并且可以根据该描述被取代; X为烷基，氰基，烷氧基，卤代烷氧基，烯氧基或卤代链烯氧基，其中X不为C1-C4烷基，当R <1>和R <2>是常见的哌啶-1-基或4-甲基 - 哌啶-1-基; 一种用于制备这些化合物，含有它们和它们在防治植物病原性有害真菌的用途的组合物的过程。

公开(公告)号：WO2005110080A2

公开(公告)日：2005-11-24

申请号：PCT/EP2005005070

申请日：2005-05-11

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N20060101 ,  A01N43/90 ,  A01N

CPC classification number: A01N43/90 ,  A01N59/06 ,  A01N59/02 ,  A01N57/12 ,  A01N47/38 ,  A01N47/34 ,  A01N47/24 ,  A01N47/04 ,  A01N43/50 ,  A01N43/76 ,  A01N43/653 ,  A01N43/36 ,  A01N43/40 ,  A01N43/32 ,  A01N37/48 ,  A01N37/46 ,  A01N37/38 ,  A01N37/34 ,  A01N2300/00

Abstract: The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R is alkyl, halogenalkyl, alkenyl or cyclopentyl, R is hydrogen or alkyl, R and R together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L is fluorine or chlorine, L , L are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (I) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.

Abstract translation: 一种杀真菌混合物，其包含作为活性组分：1）式（I）的5-甲基-7-氨基三唑并嘧啶，其中R <1>是烷基，卤代烷基，链烯基或环戊基; [R <2>是氢或烷基; [R <1>和R <2>也可以与氮原子一起与它们所连接的形式，其可以由甲基取代的哌啶环; →<1>是氟或氯; →<2>，L <3>独立地是氢，氟或氯; 和2）选自组A）唑类中的至少一种活性化合物; B）嗜球果伞素; C）酰基丙氨酸类; D）胺衍生物; E）苯胺基嘧啶; F）二甲酰亚胺; G）肉桂酸和类似物; 1H）抗生素; K）二硫代氨基甲酸酯; L）杂环化合物; M）硫和铜杀真菌剂; N）硝基苯基衍生物; O）苯基吡咯; P）Sulfensäurederivate; Q）其他杀菌剂; R）Wachstumsretardantien; 根据描述; 在协同有效量; 新的三唑并嘧啶，用于控制使用I化合物的混合物与基团A），以R的活性成分）包含这些混合物的有害真菌及其制造这样的混合物使用I化合物与基团A）至R）的活性成分和组合物的方法 ，

公开(公告)号：WO9959982A3

公开(公告)日：2000-03-16

申请号：PCT/EP9903003

申请日：1999-05-04

Applicant: BASF AG ,  BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

Inventor： BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

IPC: C07C251/38 ,  A01N37/40 ,  C07C49/303 ,  C07C251/42 ,  C07C251/50 ,  C07C251/52 ,  C07C251/60 ,  A01N37/50 ,  C07C49/35

CPC classification number: C07C251/60 ,  C07C2601/14

Abstract: The invention relates to bisoximether derivatives of formula (I) in which the variables have the following meanings: R represents halogen, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy or C1-C4 alkoxy halide; n is 1 to 5, whereby the radicals R can be different if n is not equal to 1; R represents C1-C4 alkyl, C3-C6 alkenyl or C3-C6 alkynyl, whereby these groups can be partially or completely halogenated; Q represents C(=CHOCH3)-COOCH3, C(=CHCH3)-COOCH3, C(=NOCH3)-COOCH3 or C(=NOCH3)-CONHCH3. The invention also relates to the salts of the bisoximether derivatives, to methods and intermediate products for the production of these compounds and to their use for combating animal pests and fungicidal pests.

Abstract translation: 式（I），其中各变量具有以下含义的双肟醚衍生物，R <1>为卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基; n为1至5，其中基团可以是与R <1>不同的，当n不为1; [R <2> C1-C4烷基，C3-C6链烯基或C3-C6炔基，其中这些基团可以部分或完全被卤代; Q为C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C（= NOCH 3）-COOCH 3或C（= NOCH 3）-CONHCH 3; 和它们的盐，方法和中间体制备这些化合物和它们用于控制动物害虫和有害真菌中的用途。

公开(公告)号：BRPI0607498A2

公开(公告)日：2016-11-01

申请号：BRPI0607498

申请日：2006-03-01

Applicant: BASF AG

Inventor： SCHWÖGLER ANJA ,  MÜLLER BERND ,  SCHIEWECK FRANK ,  KÖHLE HARALD ,  SCHIFFER HELMUT ,  LOHMANN JAN KLAAS ,  RHEINHEIMER JOACHIM ,  DIETZ JOCHEN ,  SCHERER MARIA ,  SCHÄFER PETER ,  GROTE THOMAS ,  HÜNGER UDO ,  GRAMMENOS WASSILIOS

IPC: C07D487/04 ,  A01N43/90

公开(公告)号：AU2005266555B2

公开(公告)日：2011-09-08

申请号：AU2005266555

申请日：2005-07-22

Applicant: BASF AG

Inventor： GROTE THOMAS ,  MULLER BERND ,  STIERL REINHARD ,  RHEINHEIMER JOACHIM ,  SCHWOGLER ANJA ,  GRAMMENOS WASSILIOS ,  SCHERER MARIA ,  SCHOFL ULRICH ,  GEWEHR MARKUS ,  SCHAFER PETER ,  STRATHMANN SIEGFRIED ,  RETHER JAN ,  BLETTNER CARSTEN ,  HUNGER UDO ,  SCHIEWECK FRANK ,  KOHLE HARALD

IPC: C07D401/04 ,  A01N43/54

Abstract: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type, whereby: k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R, independent of one another, represents halogen, OH, CN, NO C-C alkyl, C-C alkyl halide, C-C alkoxy, C-C alkoxy halide, C-C alkenyl, C-C alkynyl, C-C cycloalkyl, C-C alkoxy-C-C alkyl, amino, phenoxy, which is optionally substituted by halogen or C-C alkyl, NHR, NR, C(R)=N-OR, S(=O)A or C(=O)A, or two radicals R bound to adjacent carbon atoms can, together, also represent a group -O-Alk-O-, wherein Alk represents a linear or branched C-C alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R represents C-C alkyl halide, C-C alkoxy, C-C alkoxy halide, hydroxy, halogen, CN or NO; whereby R can also represent hydrogen or C-C alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R represents a radical that differs from halogen, C-C alkyl, C-C alkoxy and C-C alkyl halide, and; R represents C-C alkyl.

公开(公告)号：BRPI0608411A2

公开(公告)日：2009-12-29

申请号：BRPI0608411

申请日：2006-03-08

Applicant: BASF AG

Inventor： GROTE THOMAS ,  HUENGER UDO ,  SCHOFER PETER ,  SCHWOEGLER ANJA ,  RHEINHEIMER JOACHIM ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  SCHIEWECK FRANK

IPC: A01N43/54 ,  A01P3/00 ,  C07D239/00

Abstract: The invention relates to the use of 4-aminopyrimidines of formula (I), in which R 1 -H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkinyl, R 2 -H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, whereby the hydrocarbon chain in R 1 and/or R 2 can be substituted as given in the description, R 1 and R 2 can form, together with the carbon atom to which they are bonded, a 5-7-membered ring which can contain one to three same or different heteroatoms selected from the group O, N or S, R 3 -H, halogen, cyano, hydroxy, mercapto, azido, alkyl, alkenyl, alkinyl, alkylhalide, -O-D, -S(O) m -D, ON-CR a R b , CR c -NOR a , NR c N-CR a R b , NR a R b , NR c NR a R b , NOR a , NR c C(-NR c )NR a R b , NR c C(-O)NR a R b , NR a CN, -NR a C(-O)R c , NR a C(-NOR c )R c' , OC(-O)R a , C(-NOR c )NR a R b , CR c (-NNR a R b ), C(-O)NR a R b , C(-O)R a , CO 2 R a , C(-O)NR z R b , C(-O)-N-OR b , C(-S)-NR z R b , C(-O)NR a -NR z R b , C(-N-NR z R c )NR a R b , C(-NOR b )R a , C(-N-NR z R b )R a , CR a R b -OR z , CR a R b -NR z R c , ON(-CR a R b ), NR a (C(-O)R b ), NR a (C(-O)OR b ), C(-NR a )NR z R b , C(-0)-NR z R b ) NR a (C(-O)-NR z R b ), NR a (C(-NR c )R b ), NR a (N-CR c R b ), NR a -NR z R b , -NR z -OR a , NR a (C(-NR c )-NR z R b ), NR a (C(-NOR c )R b ) D=alkyl, alkenyl, alkinyl, alkylhalide, cycloalkyl, five- or six-membered saturated, partly-unsaturated or aromatic mono- or bicyclic heterocycles, containing one to four heteroatoms from the group O, N or S, one of the groups G1 or G2, whereby m, x, R a , R b , R c , R d , R e , R z , Y, Z are as defined in the description and the aliphatic, alicyclic or aromatic groups R 3 , R a , R b , R c , R d or R e can be substituted as given in the description for the prevention of fungal pests, novel 4-aminopyridines, method for production of said compounds and agents comprising the same.

公开(公告)号：PE20081170A1

公开(公告)日：2008-10-31

申请号：PE2007001625

申请日：2007-11-22

Applicant: BASF AG

Inventor： LOHMANN JAN KLAAS ,  GRAMMENOS WASSILIOS ,  PUHL MICHAEL ,  DIETZ JOCHEN ,  MULLER BERND ,  RHEINHEIMER JOACHIM ,  RENNER JENS ,  VRETTOU MARIANNA ,  ULMSCHNEIDER SARAH ,  GROTE THOMAS

IPC: A01N43/48 ,  A01N43/54 ,  C07D239/20 ,  C07D239/22 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

Abstract: SE REFIERE A COMPUESTOS DERIVADOS DE PIRIMIDILMETIL-SULFONAMIDAS DE FORMULA (I) DONDE n ES DE 0 A 3; R1 ES HALOGENO, ALQUILO(C1-C4), HALOALQUILO(C1-C4), ALCOXI(C1-C4); ENTRE OTROS; R2 ES H, ALQUILO(C1-C4), HALOALQUILO(C1-C4), ALQUENILO(C2-C4), ENTRE OTROS; A ES FENILENO, HETEROARENDIILO DE 5 O 6 MIEMBROS, ALCANDIILO(C1-C8), ENTRE OTROS; R3 ES H, ALCOXI(C1-C4), HALOALCOXI(C1-C4), CICLOALQUILO(C3-C8), ENTRE OTROS. SON COMPUESTOS PREFERIDOS: (PIRIMIDIN-4-ILMETIL)-AMIDA DEL ACIDO 4'-CLOROBIFENIL-4-SULFONICO, 4-YODO-N-PIRIMIDIN-4-ILMETILBENCENSULFONAMIDA, ESTER TER-BUTILICO DEL ACIDO (2-CLORO-PIRIMIDIN-4-ILMETIL)CARBAMICO, ENTRE OTROS. SE REFIERE TAMBIEN A COMPOSICIONES Y A UN PROCEDIMIENTO DE PREPARACION. DICHOS COMPUESTOS SON UTILES PARA EL CONTROL DE HONGOS FITOPATOGENOS DANINOS Y PLAGAS DE ARTROPODOS TALES COMO INSECTOS O ARACNIDOS

公开(公告)号：NZ546218A

公开(公告)日：2008-07-31

申请号：NZ54621804

申请日：2004-09-10

Applicant: BASF AG

Inventor： GRAMMENOS WASSILIOS ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  WAGNER OLIVER ,  GOTZ NORBERT ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

IPC: C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12 ,  C07C311/18 ,  A01N41/06

Abstract: Disclosed are 4-piridinylmethylsulfonamide derivatives of the formula I wherein the substituents are defined within the specification. Also disclosed is a method of controlling phytopathogenic harmful fungi, which comprises treating the fungi or the materials, plants, the soil or seeds to be protected against fungal attack with an effective amount of the above compounds of formula I.

公开(公告)号：BRPI0514924A

公开(公告)日：2008-06-24

申请号：BRPI0514924

申请日：2005-09-05

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  MUELLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  SCHWOEGLER ANJA ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVER ,  RETHER JAN ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD ,  SCHERER MARIA

IPC: C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07D231/14 ,  C07D277/56

Abstract: The invention relates to (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I) and to salts of said anilides that can be used for agricultural purposes for controlling pathogenic fungi. In said formula, the variables are defined as follows: A represents a phenyl or at least a monounsaturated 5- or 6-membered heterocycle comprising 1, 2 or 3 heteroatoms, selected from N, O, S, S(-O) and S(-O) 2 as ring members, whereby phenyl and the monounsaturated 5- or 6-membered heterocycle can be unsubstituted or can be substituted according to the description; B represents a group of general formula (II), in which the variables R 3 , R 4 , R 5 and the index m are defined as cited in the claims and the description; Y represents oxygen or sulphur, R 1 represents H, OH, alkyl, cycloalkyl, alkoxy, haloalkyl, halocycloalkyl or haloalkoxy; R 2 represents halogen, nitro, CN, alkyl, cycloalkyl, alkenyl, alkynyl, alkoxy, haloalkyl, halocycloalkyl, haloalkenyl, haloalkynyl or haloalkoxy; and n represents 0, 1, 2, 3 or 4; and salts that can be used for agricultural purposes. The invention also relates to the use of the (hetero)cyclyl(thio)carboxylic acid anilides of general formula (I), to a method for controlling pathogenic fungi and to a crop protection agent containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound.

公开(公告)号：BRPI0514067A

公开(公告)日：2008-05-27

申请号：BRPI0514067

申请日：2005-07-28

Applicant: BASF AG

Inventor： BLETTNER CARSTEN ,  DIETZ JOCHEN ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHAMANN SIEGFRIED ,  STIERL REINHARD ,  SCHWOEGLER ANJA ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  A01N20060101 ,  A01N43/50 ,  A01N43/54 ,  A01N43/653 ,  A01N43/84 ,  A01N47/04 ,  A01N47/14 ,  A01N47/24 ,  A01N47/38 ,  A01N57/12 ,  A01N59/20

Abstract: Fungicidal mixtures, comprising as active components 1) a 5-chloro-6-phenyl-7-heterocyclylaminotriazolopyrimidine of the formula I, in which D together with the nitrogen atom forms a pyrrolidine, piperidine or azepine ring, which rings are unsubstituted or substituted by one or two methyl groups or by an ethyl, propyl or butyl group; and L is methyl, fluorine or chlorine; and 2) at least one active compound II selected from the following groups: A) azoles; B) strobilurins; C) acylalanines; D) amine derivatives; E) anilinopyrimidines; F) dicarboximides; G) cinnamides and analogs; H) antibiotics; K) dithiocarbamates; L) heterocyclic compounds according to the description; M) sulfur and copper fungicides; N) nitrophenyl derivatives; O) phenylpyrroles; P) sulfenic acid derivatives; Q) other fungicides according to the description; or R) growth retardants; in a synergistically effective amount, novel triazolopyrimidines, methods for controlling harmful fungi using compounds or mixtures of a compound I with an active compound of groups A) to R) and the use of the compounds I with the active compounds of groups A) to R) for preparing such mixtures, and also compositions comprising these compounds or mixtures.