公开(公告)号：WO9955156A3

公开(公告)日：1999-12-23

申请号：PCT/EP9902469

申请日：1999-04-13

Applicant: BASF AG ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL OTTO ,  WALTER HELMUT

Inventor： WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: A01N43/653 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

CPC classification number: C07D401/12 ,  A01N43/653 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

Abstract: The invention relates to the use of iminotriazoles of general formula (I), wherein R represents aryl or heteroaryl and these radicals can carry one to five groups independently of each other or the aryl- or heteroaryl radical forms a bicyclic system together with a fused phenyl ring, a fused C3-C6 carbocyclic compound or a 5- or 6-membered heterocyclic compound; A is COOR or CONR R , R and R being independently of each other, hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C3-C7-cycloalkyl or C1-C6-alkyl-aryl which can optionally be partially or completely halogenised or can carry one to three substituents chosen from the following: C1-C4 alkoxy, C1-C4-halogenalkoxy, C1-C4-alkylthio, C3-C7-cycloalkyl and C5-C7-cycloalkenyl.

Abstract translation: 使用Iminotriazolen通式（I），其中R <1>为芳基或杂芳基，这些基团彼此独立地可以携带一至五个基团，或其中芳基或杂芳基与稠合的苯环，稠合的C-C6的碳环或 的5-或6-元环Heteroocyclus形成双环系统，一个是COOR <3>或CONR <3> [R <4>，其中R <3>和R <4>独立地是氢，C1-C6烷基，C2- 表示C6链烯基，C3-C7环烷基或C1-C6烷基 - 芳基，其可被部分或完全卤化，如有必要，或一至三个选自C 1 -C 4 - 烷硫基的取代基，可携带C 3 -C 7环烯基。

公开(公告)号：WO9926930A2

公开(公告)日：1999-06-03

申请号：PCT/EP9807099

申请日：1998-11-06

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  ENGEL STEFAN ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  HILL REGINA LUISE ,  MAYER GUIDO ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL OTTO ,  WALTER HELMUT

Inventor： RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  ENGEL STEFAN ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  HILL REGINA LUISE ,  MAYER GUIDO ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  C07D231/16 ,  C07D231/20 ,  C07D401/10 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D413/06 ,  C07D413/10 ,  C07D417/10 ,  C07D231/18

CPC classification number: C07D413/06 ,  A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  C07D231/16 ,  C07D231/20

Abstract: The invention relates to benzylidene pyrazolones of formula (I), wherein the substituents and index n have the following meanings: R = optionally substituted C1-C6 alkyl; R = optionally substituted C1-C6 alkyl, optionally substituted C1-C6 alkoxy, halogen, nitro, cyano; R = hydrogen, halogen, nitro, cyano, a group NR R , OCOR , NR COR ,CO2R , -COSR , -CONR R , C1-C4-alkoxyiminoalkyl, C1-C6 alkoxycarbonyl, optionally substituted C1-C6 alkyl, optionally substituted C1-C6 alkoxy, optionally substituted C1-C6 alkylthio, optionally substituted C2-C6 alkenyl, optionally substituted phenyl, optionally substituted phenoxy, an optionally substituted 5- or 6-membered saturated or unsaturated heterocycle which can contain up to 4 nitrogen atoms and/or up to 2 oxygen or sulphur atoms as ring members; R = C1-C6 alkyl, C1-C4 halogen alkyl; or R and R = an optionally substituted saturated or unsaturated 2- or 3-membered bridge which can contain one sulphur atom which can be oxidized into sulfoxide or sulfone, R = hydrogen or optionally substituted C1-C6 alkyl; R = hydrogen, C1-C6 alkyl or C1-C4 halogenalkyl; n = 0, 1 or 2; X = hydrogen, chlorine or bromine. The compounds to which claim is laid are available in both a trans and a cis form or can be a mixture of these isomers.

Abstract translation: 式（I）的Benzylidenpyrazolone其中取代基和指数n具有以下含义：R t <1>是未取代的或取代的。 C1-C6烷基; [R <2>是未取代的或取代的。 C1-C6烷基，未取代或取代的。 C1-C6烷氧基，卤素，硝基，氰基; [R <3>是氢，卤素，硝基，氰基，基团NR <5> - [R <6>，OCOR <5>，NR <5> COR <6>，CO 2 <5>，-COSR <5>，-CONR <5> - [R <6>，C1-C4-alkoxyiminoalkyl，C1-C6烷基羰基，未取代的或取代的。 C1-C6烷基，未取代或取代的。 C1-C6烷氧基，未取代的或取代的。 C1-C6烷硫基，未取代或取代的。 C2-C6链烯基，未取代的或取代的。 C2-C6炔基，未取代的或取代的。 苯基，未取代的或取代的。 苯氧基，未取代的或取代的。 5-或6-元饱和或可含有至多4个氮原子和/或至多2个氧或硫原子作为环成员的不饱和的杂环; [R <4> C1-C6-烷基，C1-C4卤代烷基; 或R <3>，R <4>为可以含有可被氧化为亚砜或砜硫原子的任选取代的饱和或不饱和2-或3-元桥; [R <5>为氢或未取代或取代的。 C1-C6烷基; [R <6>是未取代的或取代的。 C1-C6烷基; [R <7>是氢，C1-C6烷基或C1-C4卤代烷基; n为0.1或2; X是氢，氯或溴; 其中要求保护的化合物在跨及在所述顺式 - 形式两者呈现，或者可以是这些异构体的混合物。

公开(公告)号：WO9820000A2

公开(公告)日：1998-05-14

申请号：PCT/EP9706057

申请日：1997-11-03

Applicant: BASF AG ,  ZAGAR CYRILL ,  HAMPRECHT GERHARD ,  MENGES MARKUS ,  MENKE OLAF ,  SHAEFER PETER ,  WESTPHALEN KARL OTTO ,  MISSLITZ ULF ,  WALTER HELMUT ,  REINHARD ROBERT ,  JONES ROBERT BRIAN

Inventor： ZAGAR CYRILL ,  HAMPRECHT GERHARD ,  MENGES MARKUS ,  MENKE OLAF ,  SHAEFER PETER ,  WESTPHALEN KARL-OTTO ,  MISSLITZ ULF ,  WALTER HELMUT ,  REINHARD ROBERT ,  JONES ROBERT BRIAN

IPC: A01N43/56 ,  A61K31/415 ,  A61K31/4152 ,  A61K31/4155 ,  A61K31/454 ,  A61K31/5377 ,  A61P3/10 ,  C07D231/20 ,  C07D401/10 ,  C07D401/12 ,  C07D403/10 ,  C07D403/12 ,  C07D405/12

CPC classification number: C07D401/10 ,  C07D231/20 ,  C07D401/12 ,  C07D403/10 ,  C07D403/12 ,  C07D405/12

Abstract: The invention relates to substituted 3-benzylpyrazoles of formula (I), their precursors of formulas (IIa), (IIb), (IIc), their byproducts of formula (III) as well as their salts, wherein R stands for H, C1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkyl sulfonyl, C1-C4 halogen alkyl sulfonyl; R stands for C1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkoxy, C1-C4 halogen alkoxy, C1-C4 alkyl thio, C1-C4 halogen alkyl thio, C1-C4 alkyl sulfinyl, C1-C4 halogen alkyl sulfinyl, C1-C4 alkyl sulfonyl, C1-C4 halogen alkyl sulfonyl; R stands for H, CN, NO2, halogen, C1-C4 alkyl, C1-C4 halogen alkyl; X -X stands for chemical bond, optionally substituted methylene-, ethylene-, ethene-1,2-diyl or oxymethylene or thiamethylene chain linked through the heteroatom to the phenyl ring; R -R stands for H, CN, NO2, halogen -O-Y -R , -O-CO-Y -R , -N(Y -R ) (Y -R ), -N(Y -R )-SO2-Y -R , -N(SO2-Y -R ) (SO2-Y -R ), -N(Y -R )-CO-Y -R , -N(Y -R ) (O-Y -R ), -S-Y -R , -SO-Y -R , -SO2-Y -R , -SO2-O-Y -R , -SO2-N(Y -R ) (Y -R ), -CO-Y -R , -C(=NOR )-Y -R , -C(=NOR )-O-Y -R , -C(=NOR )-CO-O-Y -R , -CO-O-Y -R , -CO-S-Y -R , -CO-N(Y -R ) (Y -R ), -CO-N(Y -R ) (O-Y -R ); R stands C1-C4 alkyl, C1-C4 halogen alkyl. The invention further relates to the use of (I) as herbicide, for the desiccation/defoliation of plants, and of (I), (IIa), (IIb), (IIc) and (III) for lowering the sugar content in blood.

Abstract translation: 式的取代的3- benzylpyrazoles（I），它们在Formuln（IIA），（IIB），（IIC）的前体，和式（III）中，副产物和它们的盐，其中R <1> = H，C1-C4烷基 ，C1-C4卤代烷基，C1-C4烷基磺酰基，C1-C4卤代烷基磺酰基; [R <2> = C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，C1-C4烷硫基，C1-C4卤代烷硫基，C1-C4烷基亚磺酰基，C1-C4 卤代烷，C1-C4烷基磺酰基，C1-C4卤代烷基磺酰基; [R <3> = H，CN，NO 2，卤素，C1-C4烷基，C1-C4卤代烷基; X <1> - X <5> =化学键，任选取代的亚甲基，亚乙基，乙烯-1,2-二基，或通过结合到苯环或甲醛蒂亚姆乙烯链中的杂原子; [R <4> - R的<8> = H，CN，NO 2，卤素，-OY <1> -R <9> -O-CO-Y <1> -R <9> -N（Y <1 > -R <9>）（Y <2> -R <10>）， - N（Y <1> -R <9>） - SO2-Y <2> -R <10>，-N（SO 2 Y'> -R <9>）（SO 2-Y <2> -R <10>）， - N（Y <1> -R <9>） - CO-Y <2> -R <10>， -N（Y <1> -R <9>）（OY <2> -R <10>），-SY <1> -R <9>，-SO-Y <1> -R <9>， - SO2-Y <1> -R <9>，-SO 2 OY <1> -R <9>，-SO2-N（Y <1> -R <9>）（Y <2> -R <10> ）， - CO-Y <1> -R <9>，-C（= NOR <11>） - Y'> -R <9>，-C（= NOR <11>） - OY <1> - [R <9>，-C（= NOR <11>） - CO-OY <1> -R <9> -CO-OY <1> -R <9> -CO-SY <1> -R < 9>，-CO-N（Y <1> -R <9>）（Y <2> -R <10>），-CO-N（Y <1> [R <9>）（OY <2> - [R <10>）; [R <12> = C1-C4烷基，C1-C4卤代烷基; 使用：（Ⅰ）作为除草剂：用于植物干燥/落叶; （I），（IIA），（IIB），（IIC）和（III）用于降低血糖含量。

公开(公告)号：WO9605182A3

公开(公告)日：1996-07-04

申请号：PCT/EP9502973

申请日：1995-07-27

Applicant: BASF AG ,  PLATH PETER ,  KARDORFF UWE ,  DEYN WOLFGANG VON ,  ENGEL STEFAN ,  KAST JUERGEN ,  RANG HARALD ,  KOENIG HARTMANN ,  GERBER MATTHIAS ,  WALTER HELMUT ,  WESTPHALEN KARL-OTTO

Inventor： PLATH PETER ,  KARDORFF UEW ,  VON DEYN WOLFANG ,  ENGEL STEFAN ,  KAST JUERGEN ,  RANG HARALD ,  KOENIG HARTMANN ,  GERBER MATTHIAS ,  WALTER HELMUT ,  WESTPHALEN KARL-OTTO

IPC: C07D275/04 ,  A01N43/80 ,  A01P13/00 ,  C07D275/06 ,  C07D417/10

CPC classification number: C07D275/06 ,  A01N43/80 ,  C07D417/10

Abstract: Saccharin derivatives of formula (I) are disclosed, wherein the substituents have the following meanings: L, M stand for hydrogen, alkyl, alkoxy, alkylthio, chlorine, cyano, methylsulphonyl, nitro or trifluoromethyl; Z stands for hydrogen, alkyl, cycloalkyl, alkenyl, alkinyl, acyl, benzyl (optionally substituted by halogen, alkyl), or phenyl; J stands for an optionally substituted cyclohexane-1,3-dione ring linked at position 2.

公开(公告)号：CA2334955C

公开(公告)日：2011-10-11

申请号：CA2334955

申请日：1999-06-12

Applicant: BASF AG

Inventor： SIEVERNICH BERND ,  LANDES MAX ,  KIBLER ELMAR ,  VON DEYN WOLFGANG ,  WALTER HELMUT ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  VANTIEGHEM HERVE

IPC: A01N43/80 ,  A01N43/40 ,  A01N43/56 ,  A01N43/72 ,  A01N43/78 ,  A01N57/00 ,  A01N61/00

Abstract: The invention relates to synergistic herbicidal mixtures containing A) at least one 3-heterocyclyl-substituted benzoyl derivative of formula (I) in which the variables have the following meaning: R1, R3 represent hydrogen, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkyl sulfinyl, or alkyl sulfonyl; R2 represents a heterocyclic radical selected from the group: thiazole-2-yl, thiazole-4-yl, thiazole-5-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, 4,5-dihydroisoxazol-3-yl, 4,5-dihydroisoxazol-4-yl and 4,5-dihydroisoxazol-5-yl, whereby these can be optionally substituted one time or a multiple number of times by halogen, alkyl, alkoxy, alkyl halide, alkoxy halide, alkylthio; R4 represents hydrogen, halogen or alkyl; R5 represents alkyl; R6 represents hydrogen or alkyl; or one of the environmentally compatible salts thereof; and B) a synergistically effective quantity of at least one herbicidal compound from the group of acetyl CoA carboxylase inhibitors (ACC), acetolactate synthase inhibitors (ALS), amides, auxin herbicides, auxin transport inhibitors, carotinoid biosynthesis inhibitors, enolpyruvyl-shikimat-3-phosphate synthase inhibitors (ESPS), glutamine synthetase inhibitors, lipid biosynthesis inhibitors, mitosis inhibitors, protophorphyrinogen-IX-oxidase inhibitors, photosynthesis inhibitors, synergistic agents, growth substances, cell wall biosynthesis inhibitors and various other herbicides. The invention also relates to agents which contain these mixtures, to methods for producing these agents, and to the use thereof for controlling unwanted plants.

公开(公告)号：EE05455B1

公开(公告)日：2011-08-15

申请号：EEP9900290

申请日：1998-01-08

Applicant: BASF AG

Inventor： HILL REGINA LUISE ,  DEYN WOLFGANG VON ,  KARDORFF UWE ,  BAUMANN ERNST ,  ENGEL STEFAN ,  MAYER GUIDO ,  WITSCHEL MATTHIAS ,  RACK MICHAEL ,  GOETZ NORBERT ,  GEBHARDT JOACHIM ,  MISSLITZ ULF ,  WALTER HELMUT ,  WESTPHALEN KARL-OTTO ,  OTTEN MARTINA ,  RHEINHEIMER JOACHIM

IPC: A01N43/72 ,  C07D277/10 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  C07D231/20 ,  C07D237/00 ,  C07D261/00 ,  C07D261/04 ,  C07D261/20 ,  C07D263/10 ,  C07D273/00 ,  C07D277/20 ,  C07D277/34 ,  C07D291/04 ,  C07D311/00 ,  C07D403/10 ,  C07D413/10 ,  C07D417/10 ,  C07D419/10 ,  C07D498/10

Abstract: Benzoyl derivatives of the formula I where the variables have the following meanings: R1, R2 are hydrogen, nitro, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl or C1-C6-haloalkylsulfonyl; R3 is hydrogen, halogen or alkyl; R4, R5 are hydrogen, halogen, cyano, nitro, alkyl, alkoxy, alkylthio, dialkylamino, phenyl or carbonyl, it being possible for the 6 last-mentioned radicals to be substituted; X is O, S, NR9, CO or CR10R11; Y is O, S, NR12, CO or CR13R14; R15 is pyrazole which is unsubstituted or substituted, linked in the 4-position and has attached to it in the 5-position a hydroxyl or sulfonyloxy radical; and the agriculturally useful salts thereof; processes and intermediates for the preparation of the 3-heterocyclyl-substituted benzoyl derivatives; compositions comprising them; and the use of these derivatives or compositions comprising them for controlling undesirable plants.

公开(公告)号：CA2393996C

公开(公告)日：2010-05-11

申请号：CA2393996

申请日：2000-11-27

Applicant: BASF AG

Inventor： KUDIS STEFFEN ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  LANGEMANN KLAUS ,  MAYER GUIDO ,  MISSLITZ ULF ,  NEIDLEIN ULF ,  WITSCHEL MATTHIAS ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: C07D413/10 ,  A01N43/80 ,  A01P13/00 ,  C07B61/00 ,  C07D261/20

Abstract: The invention relates to cyclopropyl-anellated 3-(4,5-dihydroisoxazol-3-yl)-substituted benzoylpyrazoles of formula (I), wherein the variables have the meanings given in the description, and to the agriculturally usable salts. Said compounds have a herbicidal effect.

公开(公告)号：CA2277893C

公开(公告)日：2008-03-18

申请号：CA2277893

申请日：1998-01-08

Applicant: BASF AG

Inventor： WESTPHALEN KARL-OTTO ,  BAUMANN ERNST ,  ENGEL STEFAN ,  MAYER GUIDO ,  RHEINHEIMER JOACHIM ,  VON DEYN WOLFGANG ,  WAGNER OLIVER ,  MISSLITZ ULF ,  HILL REGINA LUISE ,  OTTEN MARTINA ,  WITSCHEL MATTHIAS ,  WALTER HELMUT

IPC: C07D277/10 ,  C07D413/10 ,  A01N43/18 ,  A01N43/48 ,  A01N43/56 ,  A01N43/72 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01P13/00 ,  C07D231/20 ,  C07D231/24 ,  C07D261/04 ,  C07D261/20 ,  C07D263/10 ,  C07D273/00 ,  C07D277/20 ,  C07D277/34 ,  C07D291/04 ,  C07D401/10 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D411/10 ,  C07D417/10 ,  C07D419/10 ,  C07D498/10

Abstract: The invention concerns 4-(3-hete-rocyclyl-1-benzoyl) pyrazoles of formula (I) in which the variables have the following meanings: R1, R3: hydrogen, nitro, halogen, cyano, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylthio halide, alkylsulphinyl, alkylsulphinyl halide, alkylsulphonyl, alkylsulphonyl halide, aminosulphonyl, N-alkylaminosulphonyl, N,N-dialkylaminosulphonyl, N-alkylsulphonylamino, N-alkylsulphonylamino halide, N-alkyl-N-alkylsulphonylamino or N-alkyl-N-alkylsulphonylamino halide; R2: an optionally substituted 5- or 6- member heterocyclyl group containing between 1 and 4 identical or different heteroatoms selected from the group comprising oxygen , sulphur or nitrogen; R4: hydrogen, halogen or alkyl; R5: substituted pyrazole bonded in position 4. The invention also concerns: the salts of these 4-(3-heterocyclyl-1-benzoyl)pyrazoles which can be used for agricultural purposes; processes for preparing these substances; agents containing them; and the use as herbicides of these derivatives or agents containing them.

公开(公告)号：SI0958292T1

公开(公告)日：2007-06-30

申请号：SI9830875

申请日：1998-01-08

Applicant: BASF AG

Inventor： VON DEYN WOLFGANG ,  HILL REGINA LUISE ,  BAUMANN ERNST ,  ENGEL STEFAN ,  MAYER GUIDO ,  RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WALTER HELMUT ,  WESTPHALEN KARL-OTTO

IPC: C07D277/10 ,  A01N43/18 ,  C07D413/00 ,  A01N43/48 ,  A01N43/56 ,  A01N43/72 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  C07D231/20 ,  C07D231/24 ,  C07D261/04 ,  C07D261/20 ,  C07D263/10 ,  C07D273/00 ,  C07D277/20 ,  C07D277/34 ,  C07D291/04 ,  C07D401/10 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D411/10 ,  C07D413/10 ,  C07D417/10 ,  C07D419/10 ,  C07D498/10

公开(公告)号：DE50014162D1

公开(公告)日：2007-04-26

申请号：DE50014162

申请日：2000-03-08

Applicant: BASF AG

Inventor： WITSCHEL MATTHIAS ,  KUDIS STEFFEN ,  LANGEMANN KLAUS ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  MAYER GUIDO ,  MISSLITZ ULF ,  NEIDLEIN ULF ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: C07D413/06 ,  C07D491/052 ,  A01N43/80 ,  A01N43/90 ,  C07B61/00 ,  C07D261/20 ,  C07D491/04 ,  C07D495/04 ,  C07D498/04

Abstract: Tricyclic benzoylpyrazole derivatives of the formula I wherein X, Y, R 1 , R 2 , R 6 , R 7 , R 3 , R 4 , R 5 , l, R 8 and R 9 are as defined in the disclosure and their agriculturally useful salts; processes and intermediates for preparing the tricyclic benzoylpyrazole derivatives; compositions comprising them and the use of these derivatives or of the compositions comprising them for controlling undesirable plants are described.