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公开(公告)号：KR101074212B1
公开(公告)日：2011-10-14
申请号：KR1020090042909
申请日：2009-05-18
Applicant: 원광대학교산학협력단 , 한국화학연구원
Abstract: 본발명은 4-퀴놀린온유도체화합물을포함하는수목용살충제조성물및 이를이용한살충방법에관한것으로서, 상세하게는본 발명의 4-퀴놀린온유도체화합물이소나무재선충에대해높은살충효과를나타냄을확인함으로써, 이화합물을함유하는조성물은소나무재선충에대한수목용살충제조성물로유용하게이용될수 있다.
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公开(公告)号：KR100916160B1
公开(公告)日：2009-09-08
申请号：KR1020070061580
申请日：2007-06-22
Applicant: 주식회사 앤씨비아이티 , 한국화학연구원
Abstract: 본 발명은 하기 화학식 1로 표시되는 화합물을 유효성분으로 포함하는 약제학적 항암 조성물에 관한 것이다. 본 발명의 조성물은 종양세포의 증식에 대하여 IC
50 값이 0.16 μM 이하까지 나타내어 매우 효율적으로 종양세포의 증식을 억제함으로써, 암에 대하여 치료 또는 예방 효능을 나타낸다.
화학식 1
암, 종양-
公开(公告)号：KR1020040095550A
公开(公告)日：2004-11-15
申请号：KR1020030029497
申请日：2003-05-09
Applicant: 한국화학연구원
IPC: A01N43/90
Abstract: PURPOSE: Provided is a triazole derivative which has selective antibacterial effect on plant pathogenic bacteria, excellent invasion upon them and preventing and treating effect on them. Also, provided are a method for preparing the triazole derivative and antibacterial composition for agriculture comprising it. CONSTITUTION: The triazole derivative is represented by the formula(1), as defined in the specification. The triazole derivative is manufactured by reacting 1 equivalent weight of 1-phenacyl 5-bromotriazole of the formula(2) and 1-1.2 equivalent weight of a compound of the formula(3) of R2(NH)nNH2 in an organic solvent at 50-180 deg.C. The antibacterial composition for agriculture contains 0.01-90 wt.% of the triazole derivative of the formula(1).
Abstract translation: 目的：提供对植物病原菌具有选择性抗菌作用的三唑衍生物，对其具有优异的侵袭性，对其具有预防和治疗作用。 此外，提供了制备用于农业的三唑衍生物和抗菌组合物的方法。 构成：三唑衍生物由说明书中定义的式（1）表示。 该三唑衍生物通过在有机溶剂中使1当量的式（2）的1-苯甲酰甲基5-溴三唑与1-1.2当量的式（3）的R2（NH）nNH2的化合物在有机溶剂中反应来制备， -180摄氏度 用于农业的抗菌组合物含有0.01-90重量％的式（1）的三唑衍生物。
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公开(公告)号：KR100434814B1
公开(公告)日：2004-06-07
申请号：KR1020020021507
申请日：2002-04-19
Applicant: 한국화학연구원
IPC: A01N43/38
Abstract: PURPOSE: Provided is a fungicidal composition for agriculture and horticulture having as an active ingredient a 3-alkoxyindole-2-carboxylate derivative, and pharmaceutically acceptable carrier. It has selectively high fungicidal activity to resistant bacteria and plant pathogenic bacteria. CONSTITUTION: A fungicidal composition for agriculture and horticulture is characterized by containing a 3-alkoxyindole-2-carboxylate derivative, and pharmaceutically acceptable carrier, wherein the 3-alkoxyindole-2-carboxylate derivative is represented by the formula(1) as defined in the specification.
Abstract translation: 目的：提供一种以3-烷氧基吲哚-2-羧酸衍生物和药学上可接受的载体为活性成分的农业和园艺用杀菌组合物。 它对抗药性细菌和植物致病菌具有选择性高的杀菌活性。 组成：用于农业和园艺的杀真菌组合物的特征在于含有3-烷氧基吲哚-2-羧酸酯衍生物和药学上可接受的载体，其中3-烷氧基吲哚-2-羧酸酯衍生物由式（1）表示，如 规范。
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公开(公告)号：KR100419846B1
公开(公告)日：2004-02-25
申请号：KR1020010051413
申请日：2001-08-24
Applicant: 한국화학연구원
IPC: A01N37/10
Abstract: PURPOSE: A new methoxy acrylate compound introduced by an unsaturated carbonylthioenol group is provided which exhibits excellent germicidal activity against various plant pathogenic bacteria and is useful as an agricultural or horticultural fungicide. CONSTITUTION: The agricultural or horticultural fungicide contains a methoxy acrylate derivative represented by the formula(1). In formula, R1 represents a phenyl, substituted phenyl, naphthyl, substituted naphthyl, pyridyl, substituted pyridyl, furanyl, substituted furanyl, pyrrolyl, substituted pyrrolyl, thiopheneyl, substituted thiophenyl, indolinyl or substituted indolinyl group, in which the substituted group is selected from halogen, cyclo, C1-3 alkyl, C1-3 haloalkyl and C1-3 alkoxy group and can be substituted in the range of 1 to 4, two adjacent substituted groups can combine to form -OCH2CH2O-; R2 represents H or C1-3 alkyl; R3 represents C1-3 alkyl; X represents S or NH; Y represents CH or N.
Abstract translation: 目的：提供一种由不饱和羰基硫醇基引入的新型甲氧基丙烯酸酯化合物，它对各种植物病原菌表现出优异的杀菌活性，并可用作农业或园艺杀真菌剂。 组成：农业或园艺杀真菌剂含有由式（1）表示的甲氧基丙烯酸酯衍生物。 在通式中，R1表示取代的苯基，萘基，取代的萘基，吡啶基，取代的吡啶基，呋喃基，取代的呋喃基，吡咯基，取代的吡咯基，噻吩基，取代的噻吩基，吲哚啉基或取代的吲哚啉基， 卤素，环，C1-3烷基，C1-3卤代烷基和C1-3烷氧基并且可以在1至4范围内取代，两个相邻的取代基可以结合形成-OCH2CH2O-; R2代表H或C1-3烷基; R3代表C1-3烷基; X代表S或NH; Y代表CH或N.
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Patent Agency Ranking
公开(公告)号：KR1020030083103A
公开(公告)日：2003-10-30
申请号：KR1020020021507
申请日：2002-04-19
Applicant: 한국화학연구원
IPC: A01N43/38
Abstract: PURPOSE: Provided is a fungicidal composition for agriculture and horticulture having as an active ingredient a 3-alkoxyindole-2-carboxylate derivative, and pharmaceutically acceptable carrier. It has selectively high fungicidal activity to resistant bacteria and plant pathogenic bacteria. CONSTITUTION: A fungicidal composition for agriculture and horticulture is characterized by containing a 3-alkoxyindole-2-carboxylate derivative, and pharmaceutically acceptable carrier, wherein the 3-alkoxyindole-2-carboxylate derivative is represented by the formula(1) as defined in the specification.
Abstract translation: 目的：提供作为活性成分的3-烷氧基吲哚-2-羧酸酯衍生物和药学上可接受的载体的用于农业和园艺的杀真菌组合物。 它对抗性细菌和植物病原菌具有高选择性的杀真菌活性。 构成：用于农业和园艺的杀真菌组合物的特征在于含有3-烷氧基吲哚-2-羧酸酯衍生物和药学上可接受的载体，其中3-烷氧基吲哚-2-羧酸酯衍生物由式（1）表示，如 规范。
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公开(公告)号：KR1020030009821A
公开(公告)日：2003-02-05
申请号：KR1020010044459
申请日：2001-07-24
Applicant: 한국화학연구원
IPC: A01N43/42
CPC classification number: A01N43/42 , A01N43/50 , A01N43/653
Abstract: PURPOSE: An agricultural or horticultural fungicide composition containing a 4-azoyl-2-quinolinone derivative is provided which exhibits a preventive effect and treating effect against various fungi, in particular, excellent selective bactericidal activity against any plant pathogenic bacteria. CONSTITUTION: The titled composition contains a 4-azoyl-2-quinolinone derivative of formula(1) as an active component. In formula, X is O or S, Y is CH or N, R1 is C1-5 alkyl, R2, R3, R4 and R5 are the same or different, each differently H, H, C1-3 alkyl, C1-3 alkoxy, phenyl or NO2.
Abstract translation: 目的：提供含有4-偶氮基-2-喹啉酮衍生物的农业或园艺杀菌剂组合物，其具有对各种真菌的预防作用和治疗效果，特别是对任何植物病原菌的优异的选择性杀菌活性。 构成：标题化合物含有作为活性成分的式（1）的4-偶氮基-2-喹啉酮衍生物。 在式中，X是O或S，Y是CH或N，R 1是C 1-5烷基，R 2，R 3，R 4和R 5相同或不同，各自不同的是H，H，C 1-3烷基，C 1-3烷氧基 ，苯基或NO2。
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公开(公告)号：KR100342383B1
公开(公告)日：2002-12-06
申请号：KR1019990022778
申请日：1999-06-17
Applicant: 한국화학연구원
IPC: C07D413/06
Abstract: 본발명은이소옥사졸리딘유도체에관한것으로서, 이이소옥사졸리딘유도체는하기화학식 1을갖는다. 이화합물은흰가루병에대한살균효과가매우우수하다. [화학식 1] (상기식에서, R은수소원자, C알킬, 시클로헥실, 티오알킬, 티오페닐, 페닐술폰닐, 트리플루오로메틸또는펜타플루오로에틸기이며, R는 C알킬, 페닐, 치환된페닐, 나프틸또는티오펜기이며, 여기서치환된페닐은할로겐원자, 알킬, 알콕시또는트리플루오로메틸기가 1 내지 3개가치환된페닐기를나타내며, X, Y는수소원자, 할로겐원자, C알킬기, 알콕시기이고, Z는질소원자또는메틸렌기이다.)
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公开(公告)号：KR1020020024488A
公开(公告)日：2002-03-30
申请号：KR1020000056264
申请日：2000-09-25
Applicant: 한국화학연구원
IPC: A01N43/76
CPC classification number: A01N43/76 , C07D413/04
Abstract: PURPOSE: A new oxazole derivative obtained by using amide as a starting material is provided which has a strong antibacterial effect on plant pathogenic bacteria with a small amount, for example Pyricularia oryzae Cavera, Rhizoctonia SolaniAG-1, Botrytis cinerea KCI, Phytophthora infestans or the like. CONSTITUTION: An amid compound(formula II) is refluxed in a solvent of dichloroacetone and ethanol to give chloromethyl oxazole(formula III). A chlorine atom of the chloromethyl oxazole is substituted to an iodine atom by use of sodium iodide and then reacted with 2-(2-hydroxyphenyl)-3-methoxy acrylic acid methylester(formula IV)(in case of A=C) or 2-methoxyimino-(2-hydroxyphenyl)-acetic acid methylester(formula IV)(in case of A=N) to produce an oxazole derivative(formula I).
Abstract translation: 目的：提供通过使用酰胺作为起始原料得到的新的恶唑衍生物，其对少量的植物致病菌具有强烈的抗菌作用，例如稻瘟霉，丝核菌属（Rhricoctonia SolaniAG-1），灰葡萄孢（Botrytis cinerea KCI），致病疫霉（Phytophthora infestans）或 喜欢。 构成：将化合物（式II）在二氯丙酮和乙醇的溶剂中回流，得到氯甲基恶唑（式III）。 氯甲基恶唑的氯原子用碘化钠代替碘原子，然后与2-（2-羟基苯基）-3-甲氧基丙烯酸甲酯（式IV）（在A = C）或2 （2-羟基亚苯基） - 乙酸甲酯（式IV）（在A = N的情况下），得到恶唑衍生物（式I）。
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公开(公告)号：KR1020010101593A
公开(公告)日：2001-11-14
申请号：KR1020017009074
申请日：2000-01-18
Applicant: 한국화학연구원
IPC: C07D407/14
CPC classification number: C07D231/12 , C07D233/56 , C07D249/08 , C07D405/06
Abstract: 하기 일반식 (I)의 항진균제 화합물 또는 그의 약제학적으로 허용 가능한 염:
상기 식에서, X는 CH 또는 N이고; Y는 O, 또는 이고;
R
1 및 R
2 는 각각 F 또는 Cl이고;
R
3 는 티오페닐, 나프틸, 또는 페닐(phenyl)기이고, 상기 페닐기는 C
1-4 알킬, C
1-4 할로알킬, C
1-4 알콕시, 메틸렌디옥시 및 할로겐으로 이루어진 군으로부터 선택된 하나 이상의 치환체로 선택적으로 치환되며, R
4 는 H 또는 트리플루오로메틸기이다.
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