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公开(公告)号:CA2013432A1
公开(公告)日:1990-10-10
申请号:CA2013432
申请日:1990-03-29
Applicant: KIMURA MASAYASU , NAITO KENJI , SAKUMA OSAMU , MORITA TADASHI
Inventor: KIMURA MASAYASU , NAITO KENJI , SAKUMA OSAMU , MORITA TADASHI
IPC: A61K31/14 , A61K31/215 , A61P21/02 , C07C43/174 , C07C45/41 , C07C57/34 , C07C57/40 , C07C69/612 , C07C69/618 , C07C205/11 , C07C209/12 , C07C211/27 , C07C211/28 , C07C211/29 , C07C211/30 , C07C211/49 , C07C211/63 , C07C215/18 , C07C215/30 , C07C215/40 , C07C217/10 , C07C217/20 , C07C219/22 , C07C225/06 , C07C225/16 , C07C227/18 , C07C229/34 , C07C229/38 , C07C231/12 , C07C233/43 , C07C317/28 , C07C323/25 , C07C323/62 , C07D213/06 , C07D213/16 , C07D295/02 , C07D295/135 , C07D309/12 , C07D339/08 , A61K31/245 , C07C323/32 , C07C217/48 , C07C323/63
Abstract: A guaternary ammonium compound having a muscle relaxation activity represented by the formula (I): wherein R1 represents a methylene, a lower alkylenoxy, a lower alkenylene, a lower alkynylene, -CO-, -COO-, a lower alkylene carbonyloxy, -CH(OR5)-, a lower alkylenecarbonyl, a hydroxy lower alkylene, -O-, -S-, -SO-, or -SO2-; R2 represents a hydrogen atom, a hydroxy lower alkyl, an aldehyde, a lower alkyl carbonyl, -NO2 , or -NHR6; R3 represents a hydrogen atom of a group -R1,(CH2)a-¢CH(CH2A)-CH2!b-A; R4 represents an anion; R5 and R6 represent a hydrogen atom or a acetyl; A represents a quaternary ammonium group; a represents an integer of 1 to 8; b represents 0 or 1; m represents an integer of 1 to 4; and (Z) represents a trivalent benzene ring, a trivalent naphthalene ring, a trivalent diphenyl or a trivalent ethane radical.
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公开(公告)号:CA2005741A1
公开(公告)日:1990-06-26
申请号:CA2005741
申请日:1989-12-15
Applicant: HIDAKA HIROYOSHI , ISHIKAWA TOMOHIKO , HAGIWARA MASATOSHI , INOUE TSUTOMU , NAITOH KENJI , SAKUMA OSAMU , YUASA MASAYUKI , MORITA TADASHI , TOSHIOKA TADASHI , UMEZAWA ISAO , INABA TAKASHI
Inventor: HIDAKA HIROYOSHI , ISHIKAWA TOMOHIKO , HAGIWARA MASATOSHI , INOUE TSUTOMU , NAITOH KENJI , SAKUMA OSAMU , YUASA MASAYUKI , MORITA TADASHI , TOSHIOKA TADASHI , UMEZAWA ISAO , INABA TAKASHI
IPC: C07C311/16 , C07D217/02 , C07D217/10 , C07D401/12 , C07D401/14 , C07D405/12 , C07D409/12 , C07D491/10 , C07D401/00 , C07D413/00
Abstract: Novel quinoline sulfonamino derivatives having a vessel smooth muscle relaxation activity as well as a platelet agglutination inhibitory activity and inhibitory activity to protein kinase A, myosin light chain kinase, proteinkinase C, and calmodulindependent proteinkinase II, but having little action or cardio function; a process for the production of the derivatives, and a pharmaceutical composition containing the derivative.
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公开(公告)号:WO1995018060A1
公开(公告)日:1995-07-06
申请号:PCT/JP1994002045
申请日:1994-12-06
Applicant: KABUSHI KAISHA KOMATSU SEISAKUSHO , MORITA, Tadashi , MIZUI, Seiichi
Inventor: KABUSHI KAISHA KOMATSU SEISAKUSHO
IPC: B66C23/00
CPC classification number: B66C13/20 , B66C13/063
Abstract: An object of this invention is to improve the safety of a crane. A boom control signal alpha r and a winch control signal beta r are simultaneously outputted to, respectively, a boom driving portion and a winch driving portion of a driving portion (30) for obtaining, respectively, target values Xr, Yr with current working radius X and lift Y that vary according to the flexure amount of a boom (4) as feedback amounts, thereby a boom hoisting angle and a rope length being controlled simultaneously.
Abstract translation: 本发明的目的是提高起重机的安全性。 动臂控制信号αr和绞盘控制信号βr分别同时输出到驱动部分(30)的起重臂驱动部分和绞盘驱动部分,以分别获得具有当前工作半径的目标值Xr,Yr X和升降机Y根据作为反馈量的起重臂(4)的挠曲量而变化,从而同时控制起重臂提升角度和绳索长度。
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