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公开(公告)号:ID24669A
公开(公告)日:2000-07-27
申请号:ID20000322
申请日:1998-07-07
Applicant: BASF AG
Inventor: BERND JANSSEN , TERESA BARLOZZARI , ANDREAS HAUPT , THOMAS ZIERKE , ANDREAS KLING
Abstract: Compounds of the present invention include cell growth inhibitors which are peptides of Formula I, A-B-D-E-F-(G)r-(K)s-L (I), and acid salts thereof, wherein A, B, D, E, F, G and K are α-amino acid residues, and s and r are each, independently, 0 or 1. L is a monovalent radical, such as, for example, an amino group, an N-substituted amino group, a &bgr;-hydroxylamino group, a hydrazido group, an alkoxy group, a thioalkoxy group, an aminoxy group, or an oximato group. The present invention also includes a method for treating cancer in a mammal, such as a human, comprising administering to the mammal an effective amount of a compound of Formula I in a pharmaceutically acceptable composition.
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公开(公告)号:AU2648292A
公开(公告)日:1993-05-21
申请号:AU2648292
申请日:1992-09-26
Applicant: BASF AG
Inventor: JUERGEN KAST , THOMAS ZIERKE , MATTHIAS BRATZ , ULF MISSLITZ , NORBERT MEYER , ANDREAS LANDES , WILHELM RADEMACHER , KARL-OTTO WESTPHALEN , HELMUT WALTER
IPC: A01N37/42 , A01N37/48 , A01N37/50 , A01N39/00 , C07C67/313 , C07C69/757 , C07C249/02 , C07C249/08 , C07C251/18 , C07C251/42 , C07C251/52 , C07C251/54 , C07C255/56 , C07C255/61 , C07C255/62 , C07C317/28 , C07D295/18 , C07D521/00
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公开(公告)号:ZA911021B
公开(公告)日:1992-10-28
申请号:ZA911021
申请日:1991-02-12
Applicant: BASF AG
Inventor: ZIERKE THOMAS , THOMAS ZIERKE , KUEKENHOEHNER THOMAS , THOMAS KUEKENHOEHNER , AMMERMAN EBERHARD , EBERHARD AMMERMAN , LORENZ GISELA , GISELA LORENZ
IPC: A01N43/40 , C07D213/30 , C07D213/42 , C07D213/57 , C07D213/89 , C07D , A01N , A01G
Abstract: Compounds of the formula 1 1 where R is unsubstituted or substituted cycloalkyl or cycloalkenyl, X, Y and Z are hydrogen, halogen, alkyl, alkoxy, alkoximino, haloalkyl, cyano, nitro or unsubstituted or substituted phenyl or phenoxy, W is -CH2- or -CH2CH2- and n is 0 or 1, and the plant-tolerated acid-addition salts thereof, and fungicides containing these compounds are described.
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4.
公开(公告)号:ZA907770B
公开(公告)日:1992-06-24
申请号:ZA907770
申请日:1990-09-28
Applicant: BASF AG
Inventor: SAUTER HUBERT , HUBERT SAUTER , ZIERKE THOMAS , THOMAS ZIERKE , REUTHER WOLFGANG , WOLFGANG REUTHER , BAUS ULF , ULF BAUS , LORENZ GISELA , GISELA LORENZ , AMMERMANN EBERHARD , EBERHARD AMMERMANN
IPC: A01N43/653 , C07D249/08 , C07D401/12 , C07D403/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D521/00 , C07D , A01N , B27N
Abstract: Compounds of the formula I I where Ar is unsubstituted or substituted phenyl, pyridyl, thienyl or napthyl, R1 is hydrogen or CN, R2 is unsubstituted or substituted aryl, hetaryl, alkyl or cycloalkyl, or is unsubstituted or substituted alkenyl or alkynyl, x is CH2, O or S and n is 0 or 1, their plant-tolerated acid addition salts and metal complexes, and fungicides and growth regulators containing these compounds.
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公开(公告)号:ZA200800026B
公开(公告)日:2009-08-26
申请号:ZA200800026
申请日:2008-01-02
Applicant: BASF AG
Inventor: CHRISTOPHER KORADIN , WOLFGANG VON DEYN , MICHAEL RACK , THOMAS ZIERKE , KUHN DAVID G , CULBERTSON DEBORAH L , ANSPAUGH DOUGLAS D , HASSAN OLOUMI-SADEGHI
IPC: A01N20090101 , C07D20090101
Abstract: Compounds of formula (I) wherein X is chloro or bromo; Y is chloro or trifluoromethyl; and A and B are hydrogen or methyl with the proviso that one of A or B must be methyl; or the enantiomers or salts thereof, use of compounds of formula I for combating insects or acarids and for treating, controlling, preventing or protecting animals against infestation or infection by parasites, and compositions comprising compounds of formula I.
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公开(公告)号:ZA200608604B
公开(公告)日:2008-05-28
申请号:ZA200608604
申请日:2006-10-16
Applicant: BASF AG
Inventor: THOMAS ZIERKE , ENGEL , STEFAN , PETER OTTO
IPC: C07C20090101
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7.
公开(公告)号:ZA9007770B
公开(公告)日:1992-06-24
申请号:ZA9007770
申请日:1990-09-28
Applicant: BASF AG
Inventor: SAUTER HUBERT , HUBERT SAUTER , ZIERKE THOMAS , THOMAS ZIERKE , REUTHER WOLFGANG , WOLFGANG REUTHER , BAUS ULF , ULF BAUS , LORENZ GISELA , GISELA LORENZ , AMMERMANN EBERHARD , EBERHARD AMMERMANN
IPC: A01N43/653 , C07D249/08 , C07D401/12 , C07D403/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D521/00 , C07D , A01N , B27N
CPC classification number: C07D231/12 , A01N43/653 , C07D233/56 , C07D249/08
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公开(公告)号:UA37239C2
公开(公告)日:2001-05-15
申请号:UA5010137
申请日:1991-11-26
Applicant: BASF AG
Inventor: REINER KOBER , REINER SEELE , HEINZ ISAK , ECKHARD HICKMANN , NORBERT GOETZ , THOMAS ZIERKE
IPC: C07B53/00 , C07C17/00 , C07C17/35 , C07C17/357 , C07C22/04 , C07C25/24 , C07C41/18 , C07C41/48 , C07C43/225 , C07C43/29 , C07D233/56 , C07D233/58 , C07D249/08 , C07D301/16 , C07D303/08 , C07D405/06 , C07D521/00
Abstract: Хлорметилдіарилоксиранизагальноїформули (I) де R1 і R2 незалежноодинвідодногоозначаютьводеньабогалоген, а n і m означають 1,2 або 3. Цейвинахідвідноситьсядоновихпорметилдіарилоксиранівзагальноїформули I (I) де R1 і R2 незалежноодинвідодногоозначаютьводень, галоген, n і m означають 1, 2 або 3 якіє проміжнимипродуктами, дляотриманняазолиілметилоксираіов, щомаютьфунгіциднуактивністьі щоє такожосновоюфунгіциднихкомпозицій.
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公开(公告)号:MD419C2
公开(公告)日:1996-07-31
申请号:MD950220
申请日:1994-12-13
Applicant: BASF AG
Inventor: SEELE RAINER , REINER KOBER , HEINZ ISAK , ECKHARD HICKMANN , NOBERT GOTZ , THOMAS ZIERKE
IPC: C07C25/24 , C07C17/04 , C07C17/35 , C07C17/357 , C07C43/225 , C07C43/29 , C07D233/56 , C07D233/58 , C07D249/08 , C07D303/08 , C07D521/00
Abstract: Sarcina prezentei invenţii constă în elaborarea procedeului, conform căruia este posibilă obţinerea unui randament sporit al Z-1,2-diarilalilclorurilor cu formula generalăutilizate în calitate de produse intermediare la obţinerea agenţilor activi farmacologici,fungicizi şi antimicotici.Procedeul de obţinere stereoselectivă a substanţelor cu formula generală (1) constă în aceea că clorhidrinele cu formula IIîn care radicalii R1 şi R2, independent unul de altul, semnifică hidrogen, halogen, alchil, halogenalchil, alcoxi, halogenalcoxi sau radical aromatic nesubstituit sau substituit, iar n şi m semnifică 1, 2 sau 3, se deshidratează în eter inert sau ester al acidului carbonic în calitate de dizolvant în prezenţa anhidridei acidului carbonic sau cetenei respective şi acidului organic sau anorganic sau oleum la temperatura până la 50°C.Revendicări:9
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公开(公告)号:ZA9101021B
公开(公告)日:1992-10-28
申请号:ZA9101021
申请日:1991-02-12
Applicant: BASF AG
Inventor: ZIERKE THOMAS , THOMAS ZIERKE , KUEKENHOEHNER THOMAS , THOMAS KUEKENHOEHNER , AMMERMAN EBERHARD , EBERHARD AMMERMAN , LORENZ GISELA , GISELA LORENZ
IPC: A01N43/40 , C07D213/30 , C07D213/42 , C07D213/57 , C07D213/89 , C07D , A01G , A01N
CPC classification number: C07D213/30 , A01N43/40
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