公开(公告)号：CA2489394A1

公开(公告)日：2004-01-15

申请号：CA2489394

申请日：2003-06-30

Applicant: BASF AG

Inventor： GOLD RANDALL EVEN ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  SCHELBERGER KLAUS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  HENNINGSEN MICHAEL

IPC: A01N43/32 ,  A01N43/54

Abstract: The invention relates to fungicidal mixtures that contain A) the compound of formula (I), and B) a pyrimidine derivative of formula (II), wherein R represents methyl, cyclopropyl or 1-propinyl, in a synergistically effective amount. The invention also relates to a method for controlling parasitic fun gi using mixtures of the compounds (I) and (II) and the use of compounds (I) an d (II) in the production of such mixtures.

公开(公告)号：AU2003242638A1

公开(公告)日：2004-01-06

申请号：AU2003242638

申请日：2003-06-06

Applicant: BASF AG

Inventor： SANDER MICHAEL ,  HENNINGSEN MICHAEL ,  NOACK RAINER

IPC: C07D405/06 ,  C07D521/00

Abstract: The present invention relates to a process for the preparation of 1,2,4-triazol-1-ylmethyloxiranes of the formula I in which A and B are identical or different and, independently of one another, are C 1 -C 4 -alkyl, phenyl-C 1 -C 2 -alkyl, C 3 -C 6 -cycloalkyl, C 3 -C 6 -cycloalkenyl, tetrahydropyranyl, tetrahydrofuranyl, dioxanyl or phenyl, where the phenyl radical can carry one to three substituents chosen from the group: halogen, nitro, C 1 -C 4 -alkyl, C l -C 4 -alkyloxy, phenoxy, amino, C 1 -C 2 -haloalkyl or phenylsulfonyl, which comprises reacting a) an oxirane of the formula II in which A and B have the meanings given above and L is a nucleophilically substitutable leaving group, with 4-amino-1,2,4-triazole of the formula III to give 4-amino-1,2,4-triazolium salts of the formula IV and b) deaminating the 4-amino-1,2,4-triazolium salts IV with alkali metal nitrites and acid or organic nitrites to give 1,2,4-triazol-1-ylmethyloxiranes of the formula I, and to 4-aminotriazolium salts of the formula IV as intermediates.

公开(公告)号：BR0112167A

公开(公告)日：2003-05-06

申请号：BR0112167

申请日：2001-07-04

Applicant: BASF AG

Inventor： KRAMER ANDREAS ,  KIEFER MATTHIAS ,  HENNINGSEN MICHAEL ,  SIEGEL WOLFGANG ,  DER JOCHEN SCHR

IPC: C07B61/00 ,  C07C249/06 ,  C07C249/08 ,  C07C251/40 ,  C07C251/58 ,  C07C251/60 ,  C07C49/12

Abstract: The present invention relates to a process for preparing trioxime derivatives of the formula I in which the substituents R 1 and R 2 are identical or different and each is cyano, alkyl, haloalkyl or cycloalkyl, and R 3 and R 4 are identical or different and each is alkyl, haloalkyl, cycloalkyl, alkylcarbonyl or arylalkyl, by the following reaction steps in water without isolation of the intermediates: A) nitrosation of 1,3-diketones of the formula II to give monooximes of the formula III, B) oximation of III with hydroxylamine derivatives of the formula IV H 2 N-OR 3' IV in which R 3' is hydrogen or a group R 3 to give bisoximes of the formula V, C) alkylation of V with alkylating agents or acylation of V with acylating agents to give compounds of the formula VI and D) subsequent oximation of VI with hydroxylamine to give compounds of the formula I.

公开(公告)号：CA2440518A1

公开(公告)日：2002-09-26

申请号：CA2440518

申请日：2002-03-15

Applicant: BASF AG

Inventor： KUSCHE ANDREAS ,  GERLACH TILL ,  HULLMANN MICHAEL ,  HENNINGSEN MICHAEL ,  RUB LOTHAR ,  KASHAMMER STEFAN

IPC: C07D265/30 ,  C07B61/00 ,  C07D295/02 ,  C07D295/023 ,  C07D295/03 ,  C07D295/033 ,  A01N43/84

Abstract: The invention relates to a method of producing the N-substituted 2,6-dialkyl morpholines of general formula (I), wherein R1 and R2 independently represen t hydrogen, alkyl or cycloalkyl, or R1 and R2, together with the carbon atom t o which they are bound, represent a 5 to 14 membered carbocyclic compound, and R3 and R4 independently represent alkyl or cycloalkyl. The inventive substances are produced by reacting at least one carbonyl compound of genera l formula (II), wherein R1 and R2 are defined as above, with at least one morpholine of general formula (III), wherein R3 and R4 are defined as above, in the presence of hydrogen and at least one metal-containing catalyst, the active component of said catalyst substantially consisting of platinum group metals.

公开(公告)号：NO20011822L

公开(公告)日：2001-04-20

申请号：NO20011822

申请日：2001-04-10

Applicant: BASF AG

Inventor： BISCHOF NORBERT ,  BUSCHMANN ERNST ,  HENNINGSEN MICHAEL ,  KREI GEORG ARNOLD ,  MUNSCHAUER RAINER ,  PFEIFFER THOMAS ,  STEINER GERD ,  VIERGUTZ WOLFGANG

IPC: A61K31/40 ,  C07D209/52 ,  C07B37/10 ,  C07D20060101

Abstract: A process for preparing (+)-exo-6-phenyl-3-azabicyclo[3.2.0]heptanes of the formula Iwhere R is hydrogen, chlorine, bromine, fluorine or methoxy, which comprises photocyclizing a bisallylammonium salt of the formula IIwhere R has the meanings given above and X- is an anion, in an inert solvent in a glass apparatus with addition of sensitizer and precipitating using (-)-ditoluoyltartaric acid the desired (+)-exo-isomer I as ditoluoyltartrate from the resulting mixture, with or without recrystallization of this tartrate from an alcohol/water mixture.

公开(公告)号：AU1036500A

公开(公告)日：2000-05-08

申请号：AU1036500

申请日：1999-10-13

Applicant: BASF AG

Inventor： BISCHOF NORBERT ,  BUSCHMANN ERNST ,  HENNINGSEN MICHAEL ,  KREI GEORG ARNOLD ,  MUNSCHAUER RAINER ,  PFEIFFER THOMAS ,  STEINER GERD ,  VIERGUTZ WOLFGANG

IPC: C07D209/52 ,  A61K31/40 ,  C07B37/10 ,  C07D20060101

Abstract: A process for preparing (+)-exo-6-phenyl-3-azabicyclo[3.2.0]heptanes of the formula Iwhere R is hydrogen, chlorine, bromine, fluorine or methoxy, which comprises photocyclizing a bisallylammonium salt of the formula IIwhere R has the meanings given above and X- is an anion, in an inert solvent in a glass apparatus with addition of sensitizer and precipitating using (-)-ditoluoyltartaric acid the desired (+)-exo-isomer I as ditoluoyltartrate from the resulting mixture, with or without recrystallization of this tartrate from an alcohol/water mixture.

公开(公告)号：PL210307B1

公开(公告)日：2011-12-30

申请号：PL39057203

申请日：2003-06-30

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  SCHELBERGER KLAUS ,  SCHERER MARIA ,  HENNINGSEN MICHAEL ,  GOLD RANDALL EVEN

IPC: A01N37/34 ,  A01N25/04 ,  A01N43/32 ,  A01N43/653 ,  A01P3/00

公开(公告)号：PL208860B1

公开(公告)日：2011-06-30

申请号：PL37481603

申请日：2003-06-30

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  SCHELBERGER KLAUS ,  SCHERER MARIA ,  HENNINGSEN MICHAEL ,  GOLD RANDALL EVEN

IPC: A01N43/32 ,  A01N25/06 ,  A01N43/18 ,  A01N43/40 ,  A01P3/00

公开(公告)号：CA2440518C

公开(公告)日：2010-05-25

申请号：CA2440518

申请日：2002-03-15

Applicant: BASF AG

Inventor： HENNINGSEN MICHAEL ,  KUSCHE ANDREAS ,  HULLMANN MICHAEL ,  RUB LOTHAR ,  KASHAMMER STEFAN ,  GERLACH TILL

IPC: C07D265/30 ,  C07D295/02 ,  A01N43/84 ,  C07B61/00 ,  C07D295/023 ,  C07D295/03 ,  C07D295/033

Abstract: The invention relates to a method of producing the N-substituted 2,6-dialkyl morpholines of general formula (I), wherein R1 and R2 independently represent hydrogen, alkyl or cycloalkyl, or R1 and R2, together with the carbon atom to which they are bound, represent a 5 to 14 membered carbocyclic compound, and R3 and R4 independently represent alkyl or cycloalkyl. The inventive substances are produced by reacting at least one carbonyl compound of general formula (II), wherein R1 and R2 are defined as above, with at least one morpholine of general formula (III), wherein R3 and R4 are defined as above, in the presence of hydrogen and at least one metal-containing catalyst, the active component of said catalyst substantially consisting of platinum group metals.

公开(公告)号：AT375722T

公开(公告)日：2007-11-15

申请号：AT05016044

申请日：2003-06-30

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  STIERL REINHARD ,  SCHOEFL ULRICH ,  SCHELBERGER KLAUS ,  SCHERER MARIA ,  HENNINGSEN MICHAEL ,  EVAN GOLD RANDALL

IPC: A01N43/32 ,  A01N25/04 ,  A01N43/653

Abstract: New fungicidal mixtures contain dithianon (I) and at least one 1,2,4-triazole derivative (II) in synergistic amounts, where (II) is metconazole, epoxiconazole, fluquinconazole, tebuconazole (IIa), tetraconazole, difenconazole and/or prothioconazole (preferably metconazole, epoxiconazole or (IIa)). Independent claims are included for: (1) a fungicidal composition comprising the (I)/(II) mixture plus a solid or liquid carrier; and (2) a method for controlling harmful fungi, by applying (I) and (II) to the fungi, their habitat or plants, seeds, soil, surfaces, materials or regions to be protected. ACTIVITY : Fungicide. In tests against Botrytis cinerea in paprika seedlings, (I) at 16 ppm or (IIa) at 4 ppm gave no control, whereas a combination of 16 ppm (I) and 4 ppm (IIa) gave 59% control. MECHANISM OF ACTION : Synergist.