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公开(公告)号:FI971529A0
公开(公告)日:1997-04-11
申请号:FI971529
申请日:1997-04-11
Applicant: BASF AG
Inventor: RIECHERS HARTMUT , KLINGE DAGMAR , AMBERG WILHELM , KLING ANDREAS , MUELLER STEFAN , BAUMANN ERNST , RHEINHEIMER JOACHIM , VOGELBACHER UWE JOSEF , WERNET WOLFGANG , UNGER LILIANE , RASCHACK MANFRED
IPC: C07D251/30 , A61K31/505 , A61P9/00 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/08 , A61P13/02 , A61P15/00 , A61P25/04 , C07D239/00 , C07D239/26 , C07D239/28 , C07D239/34 , C07D239/38 , C07D239/60 , C07D239/70 , C07D239/96 , C07D251/12 , C07D251/52 , C07D257/02 , C07D309/00 , C07D403/06 , C07D403/12 , C07D405/12 , C07D417/12 , C07D487/04 , C07D491/04 , C07D491/044 , C07D491/048 , C07D
Abstract: Heterocyclyl-substd. propanoic acids and their derivs., of formula (I), are new. R = formyl, tetrazolyl, nitrile, COOH or a gp. that can be hydrolysed to COOH; X = N or CR14; R2 = H, OH, NH2, alkylamino, dialkylamino, halo, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; R14 = H or 1-5 C alkyl; R3 = R2 or alkoxyimino; or CR3 + CR14 = 5 or 6 membered alkylene or alkenyl ring (opt. substd. by 1-2 alkyl) in which a methylene can be replaced by O, S, NH or alkylamino; R4, R5 = phenyl or naphthyl (both opt. substd. by one or more halo, NO2, CN, OH, alkyl, haloalkyl, alkoxy, haloalkyloxy, phenoxy, alkylthio, NH2, alkylamine or dialkylamino) or 3-7 C cycloalkyl; or the phenyl or naphthyl gps. are opt. bonded at the O- position (by a bond, CH2, O, S, SO2, ethylene, ethenylene or opt. alkylated amino); R6 = H, 1-8 C alkyl, 2-6 C alkenyl, 3-6 C alkynyl, 3-8 C cycloalkyl (all opt. substd. by 1 or more halo, NO2, CN, alkoxy 3-6 C alkenyloxy, 3-6 C alkynyloxy, alkylthio, haloalkoxy, alkylcarbonyl, alkoxycarbonyl, 3-8 C alkylcarbonylalkyl, alkylamino, dialkylamino, phenyl, Ph or OPh), Ar or Het; Y = S, O or bond; Q = S, O, SO, SO2 or bond; Ph = substd. phenyl, where substits. are halo, NO2, CN, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; Ar = phenyl or naphthyl (both opt. substd. by 1 or more halo, NO2, CN, OH, NH2, alkylamino, dialkylamino or OCH2CH2O); Het = 5 or 6 membered heteroaromatic with 1-3 N atoms and/or one S or O (opt. substd. by 1-4 halo and/or 1 or 2 alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, phenyl, phenoxy or phenyl carbonyl (where the phenyl is opt. substd. by 1-5 halo and/or 1-3 alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkylthio)); alkyl and alkoxy have 1-4 C unless otherwise stated; provided that R6 is not H when Q = bond.
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公开(公告)号:FI971529A
公开(公告)日:1997-04-11
申请号:FI971529
申请日:1997-04-11
Applicant: BASF AG
Inventor: RIECHERS HARTMUT , KLINGE DAGMAR , AMBERG WILHELM , KLING ANDREAS , MUELLER STEFAN , BAUMANN ERNST , RHEINHEIMER JOACHIM , VOGELBACHER UWE JOSEF , WERNET WOLFGANG , UNGER LILIANE , RASCHACK MANFRED
IPC: C07D251/30 , A61K31/505 , A61P9/00 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/08 , A61P13/02 , A61P15/00 , A61P25/04 , C07D239/00 , C07D239/26 , C07D239/28 , C07D239/34 , C07D239/38 , C07D239/60 , C07D239/70 , C07D239/96 , C07D251/12 , C07D251/52 , C07D257/02 , C07D309/00 , C07D403/06 , C07D403/12 , C07D405/12 , C07D417/12 , C07D487/04 , C07D491/04 , C07D491/044 , C07D491/048 , C07D
Abstract: Heterocyclyl-substd. propanoic acids and their derivs., of formula (I), are new. R = formyl, tetrazolyl, nitrile, COOH or a gp. that can be hydrolysed to COOH; X = N or CR14; R2 = H, OH, NH2, alkylamino, dialkylamino, halo, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; R14 = H or 1-5 C alkyl; R3 = R2 or alkoxyimino; or CR3 + CR14 = 5 or 6 membered alkylene or alkenyl ring (opt. substd. by 1-2 alkyl) in which a methylene can be replaced by O, S, NH or alkylamino; R4, R5 = phenyl or naphthyl (both opt. substd. by one or more halo, NO2, CN, OH, alkyl, haloalkyl, alkoxy, haloalkyloxy, phenoxy, alkylthio, NH2, alkylamine or dialkylamino) or 3-7 C cycloalkyl; or the phenyl or naphthyl gps. are opt. bonded at the O- position (by a bond, CH2, O, S, SO2, ethylene, ethenylene or opt. alkylated amino); R6 = H, 1-8 C alkyl, 2-6 C alkenyl, 3-6 C alkynyl, 3-8 C cycloalkyl (all opt. substd. by 1 or more halo, NO2, CN, alkoxy 3-6 C alkenyloxy, 3-6 C alkynyloxy, alkylthio, haloalkoxy, alkylcarbonyl, alkoxycarbonyl, 3-8 C alkylcarbonylalkyl, alkylamino, dialkylamino, phenyl, Ph or OPh), Ar or Het; Y = S, O or bond; Q = S, O, SO, SO2 or bond; Ph = substd. phenyl, where substits. are halo, NO2, CN, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; Ar = phenyl or naphthyl (both opt. substd. by 1 or more halo, NO2, CN, OH, NH2, alkylamino, dialkylamino or OCH2CH2O); Het = 5 or 6 membered heteroaromatic with 1-3 N atoms and/or one S or O (opt. substd. by 1-4 halo and/or 1 or 2 alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, phenyl, phenoxy or phenyl carbonyl (where the phenyl is opt. substd. by 1-5 halo and/or 1-3 alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkylthio)); alkyl and alkoxy have 1-4 C unless otherwise stated; provided that R6 is not H when Q = bond.
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公开(公告)号:CA2231493A1
公开(公告)日:1997-04-10
申请号:CA2231493
申请日:1996-09-26
Applicant: BASF AG
Inventor: VOGELBACHER UWE JOSEF , BAUMANN ERNST , WALTER HELMUT , MISSLITZ ULF , RHEINHEIMER JOACHIM , WESTPHALEN KARL-OTTO
IPC: C07D251/34 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/66 , A01N43/76 , A01N43/78 , A01N43/80 , C07D239/60 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D401/14 , C07D403/14 , A01N43/48 , A01N43/64 , A01N43/713 , A01N43/72
Abstract: The invention relates to salicylic acid derivatives of formula I, in which the substituents have the following meaning: A is a five membered heteroaromatic with a oxygen atom, nitrogen atom or sulphur atom or with one to four nitrogen atoms or with one to two nitrogen atoms and additionally a sulphur atom or an oxygen atom in the ring which can carry at least one -B-R5 group and additionally one or a plurality of the following substituents: nitro, halogen, cyano, optionally substituted alkyl, alkyl thio, alkyl sulfonyl, alkyl sulfinyl, formyl or a R5 group; a six membered hereroaromatic with two to three nitrogen atoms in the ring which can carry at least one -B-R5 group and additionally one or a plurality of the following substituents: nitro, halogen, cyano, optionally substituted alkyl, alkyl thio, alkyl sulfonyl, alkyl sulfinyl, formyl or a R5 group; B is oxygen, sulphur, SO, SO2; X is oxygen or sulphur; Y is nitrogen or C-H; Z is nitrogen or a C-R4 grouping, the substituents R1, R2, and R3 having the meaning given in claim 1. The invention also relates to a process for the preparation of these derivatives, herbicidal agents and a method of controlling undesirable vegetation.
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公开(公告)号:SI9520048A
公开(公告)日:1997-02-28
申请号:SI9520048
申请日:1995-03-23
Applicant: BASF AG
Inventor: BAUMANN ERNST , VOGELBACHER UWE JOSEF , RHEINHEIMER JOACHIM , KLINGE DAGMAR , RIECHERS HARTMUT , KROEGER BURKHARD , BIALOJAN SIEGFRIED , BOLLSCHWEILER CLAUS , WERNET WOLFGANG , UNGER LILIANE , RASCHACK MANFRED
IPC: A61K31/00 , A61K31/505 , A61K31/506 , C07D251/26 , A61K31/53 , A61P9/00 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/08 , A61P13/02 , A61P15/00 , A61P25/04 , A61P39/02 , C07D239/26 , C07D239/34 , C07D239/38 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12
Abstract: PCT No. PCT/EP95/01099 Sec. 371 Date Sep. 30, 1996 Sec. 102(e) Date Sep. 30, 1996 PCT Filed Mar. 23, 1995 PCT Pub. No. WO95/26716 PCT Pub. Date Oct. 12, 1995A method of inhibiting endothelin receptors by administering to a patient a compound of the formula I I
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公开(公告)号:NZ283333A
公开(公告)日:1997-02-24
申请号:NZ28333395
申请日:1995-03-23
Applicant: BASF AG
Inventor: BAUMANN ERNST , VOGELBACHER UWE JOSEF , RHEINHEIMER JOACHIM , KLINGE DAGMAR , RIECHERS HARTMUT , KROGER BURKHARD , BIALOJAN SIEGFRIED , BOLLSCHWEILER CLAUS , WERNET WOLFGANG , UNGER LILIANE , RASCHACK MANFRED
IPC: A61K31/00 , A61K31/505 , A61K31/506 , A61K31/53 , C07D251/26 , A61P9/00 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/08 , A61P13/02 , A61P15/00 , A61P25/04 , A61P39/02 , C07D239/26 , C07D239/34 , C07D239/38 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D239/00 , C07D251/00
Abstract: PCT No. PCT/EP95/01099 Sec. 371 Date Sep. 30, 1996 Sec. 102(e) Date Sep. 30, 1996 PCT Filed Mar. 23, 1995 PCT Pub. No. WO95/26716 PCT Pub. Date Oct. 12, 1995A method of inhibiting endothelin receptors by administering to a patient a compound of the formula I I
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公开(公告)号:NO964121A
公开(公告)日:1996-11-26
申请号:NO964121
申请日:1996-09-27
Applicant: BASF AG
Inventor: BAUMANN ERNST , VOGELBACHER UWE JOSEF , RHEINHEIMER JOACHIM , KLINGE DAGMAR , RIECHERS HARTMUT , KROGER BURKHARD , BIALOJAN SIEGFRIED , BOLLSCHWEILER CLAUS , WERNET WOLFGANG , UNGER LILIANE , RASCHACK MANFRED
IPC: C07D251/26 , A61K31/505 , A61K31/506 , A61K31/53 , A61P9/00 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/08 , A61P13/02 , A61P15/00 , A61P25/04 , A61P39/02 , C07D239/26 , C07D239/34 , C07D239/38 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , A61K
CPC classification number: A61K31/505 , A61K31/506 , A61K31/53
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公开(公告)号:FI963885A0
公开(公告)日:1996-09-27
申请号:FI963885
申请日:1996-09-27
Applicant: BASF AG
Inventor: BAUMANN ERNST , VOGELBACHER UWE JOSEF , RHEINHEIMER JOACHIM , KLINGE DAGMAR , RIECHERS HARTMUT , KROEGER BURKHARD , BIALOJAN SIEGFRIED , BOLLSCHWEILER CLAUS , WERNET WOLFGANG , UNGER LILIANE , RASCHACK MANFRED
IPC: C07D251/26 , A61K31/00 , A61K31/505 , A61K31/506 , A61K31/53 , A61P9/00 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/08 , A61P13/02 , A61P15/00 , A61P25/04 , A61P39/02 , C07D239/26 , C07D239/34 , C07D239/38 , C07D401/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , A61K
Abstract: PCT No. PCT/EP95/01099 Sec. 371 Date Sep. 30, 1996 Sec. 102(e) Date Sep. 30, 1996 PCT Filed Mar. 23, 1995 PCT Pub. No. WO95/26716 PCT Pub. Date Oct. 12, 1995A method of inhibiting endothelin receptors by administering to a patient a compound of the formula I I
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公开(公告)号:HUT73559A
公开(公告)日:1996-08-28
申请号:HU9503037
申请日:1994-04-13
Applicant: BASF AG
Inventor: BAUMANN ERNST , BRATZ MATTHIAS , GERBER MATTHIAS , HARREUS ALBRECHT , RADEMACHER WILHELM , RHEINHEIMER JOACHIM , THEOBALD HANS , VOGELBACHER UWE JOSEF , WALTER HELMUT , WESTPHALEN KARL-OTTO
IPC: C07D233/64 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/66 , A01N43/713 , A01N43/76 , A01N43/80 , A01P13/00 , C07D207/333 , C07D207/335 , C07D213/55 , C07D231/12 , C07D239/34 , C07D239/38 , C07D239/56 , C07D239/60 , C07D261/08 , C07D263/32 , C07D275/02 , C07D277/14 , C07D307/28 , C07D333/16 , C07D333/24 , C07D333/28 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D491/04 , C07D491/048
Abstract: PCT No. PCT/EP94/01140 Sec. 371 Date Dec. 1, 1995 Sec. 102(e) Date Dec. 1, 1995 PCT Filed Apr. 13, 1994 PCT Pub. No. WO94/25455 PCT Pub. Date Nov. 10, 19943-Halo-3-hetarylcarboxylic acid derivatives having the formula I I in which R is a formyl group, a group CO2H or a radical which can be hydrolyzed to COOH, and the remaining substituents have the following meanings: R2 and R3 are halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy or C1-C4-alkylthio; X is nitrogen or CR13, where R13 is hydrogen or together with R3 forms an alkylene or alkenylene chain in which in each case one methylene group is replaced by oxygen; R4 is an unsubstituted or substituted five- or six-membered heteroaromatic ring which contains one to three nitrogen atoms and/or one sulfur or oxygen atom; R5 is hydrogen, substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl or phenyl; Y is sulfur, oxygen or a single bond; and Z is halogen. The derivatives I having herbicidal and plant-growth regulating properties.
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公开(公告)号:CZ276795A3
公开(公告)日:1996-02-14
申请号:CZ276795
申请日:1994-04-14
Applicant: BASF AG
Inventor: BAUMANN ERNST , RHEINHEIMER JOACHIM , VOGELBACHER JOSEF , BRATZ MATTHIAS , MEYER NORBERT , GERBER MATTHIAS , WESTPHALEN KARL OTTO , WALTER HELMUT , RADEMACHER WILHELM
IPC: C07D251/34 , A01N43/54 , A01N43/60 , A01N43/66 , A01P13/00 , C07C69/22 , C07C69/712 , C07C69/734 , C07D239/26 , C07D239/30 , C07D239/34 , C07D239/38 , C07D239/52 , C07D239/60 , C07D251/30 , C07D307/46 , C07D307/54 , C07D333/24 , C07D405/12 , C07D409/12 , C07D491/048
Abstract: PCT No. PCT/EP94/01156 Sec. 371 Date Oct. 19, 1995 Sec. 102(e) Date Oct. 19, 1995 PCT Filed Apr. 14, 1994 PCT Pub. No. WO94/25443 PCT Pub. Date Nov. 10, 19943-(Het)aryloxy(thio)carboxylic acid derivatives of the formula I I where R1 is hydrogen, COOH or a radical which can be hydrolyzed to give COOH; R2 and R3 are each halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; X is nitrogen or CR14, where R14 is hydrogen or, together with R3, forms a 3-membered or 4-membered alkylene or alkenylene chain, in each of which a methylene group is replaced by oxygen; R4 is alkyl, cycloalkyl, cycloalkenyl, alkenyl or alkynyl, each of which is unsubstituted or substituted; an unsubstituted or substituted five-membered or six-membered heteroaromatic structure containing one to three nitrogen atoms or one sulfur or oxygen atom; unsubstituted or substituted phenyl or naphthyl; R4 and R5, together with the neighboring carbon atom, form a 3-membered to 8-membered ring which may contain an oxygen or sulfur atom and which is unsubstituted or substituted; R5 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl or phenyl, each of which is unsubstituted or substituted; R6 is unsubstituted or substituted phenyl or naphthyl or an unsubstituted or substituted five-membered or six-membered heteroaromatic structure containing one to three nitrogen atoms or one sulfur or oxygen atom; Y is sulfur or oxygen or a single bond; and Z is sulfur or oxygen.
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公开(公告)号:BR9406358A
公开(公告)日:1996-02-13
申请号:BR9406358
申请日:1994-04-13
Applicant: BASF AG
Inventor: BAUMANN ERNST , HARREUS ALBRECHT , BRATZ MATTHIAS , RHEINHEIMER JOACHIM , VOGELBACHER UWE JOSEF , THEOBALD HANS , GERBER MATTHIAS , WALTER HELMUT , WESTPHALEN KARL-OTTO , RADEMACHER WILHELM
IPC: C07D233/64 , A01N43/50 , A01N43/54 , A01N43/56 , A01N43/653 , A01N43/66 , A01N43/713 , A01N43/76 , A01N43/80 , A01P13/00 , C07D207/333 , C07D207/335 , C07D213/55 , C07D231/12 , C07D239/34 , C07D239/38 , C07D239/56 , C07D239/60 , C07D261/08 , C07D263/32 , C07D275/02 , C07D277/14 , C07D307/28 , C07D333/16 , C07D333/24 , C07D333/28 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D413/12 , C07D417/12 , C07D491/04 , C07D491/048
Abstract: PCT No. PCT/EP94/01140 Sec. 371 Date Dec. 1, 1995 Sec. 102(e) Date Dec. 1, 1995 PCT Filed Apr. 13, 1994 PCT Pub. No. WO94/25455 PCT Pub. Date Nov. 10, 19943-Halo-3-hetarylcarboxylic acid derivatives having the formula I I in which R is a formyl group, a group CO2H or a radical which can be hydrolyzed to COOH, and the remaining substituents have the following meanings: R2 and R3 are halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy or C1-C4-alkylthio; X is nitrogen or CR13, where R13 is hydrogen or together with R3 forms an alkylene or alkenylene chain in which in each case one methylene group is replaced by oxygen; R4 is an unsubstituted or substituted five- or six-membered heteroaromatic ring which contains one to three nitrogen atoms and/or one sulfur or oxygen atom; R5 is hydrogen, substituted or unsubstituted alkyl, alkenyl, alkynyl, cycloalkyl or phenyl; Y is sulfur, oxygen or a single bond; and Z is halogen. The derivatives I having herbicidal and plant-growth regulating properties.
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