公开(公告)号：DE59509541D1

公开(公告)日：2001-09-27

申请号：DE59509541

申请日：1995-10-07

Applicant: BASF AG

Inventor： RIECHERS HARTMUT ,  KLINGE DAGMAR ,  AMBERG WILHELM ,  KLING ANDREAS ,  MUELLER STEFAN ,  BAUMANN ERNST ,  RHEINHEIMER JOACHIM ,  VOGELBACHER JOSEF ,  WERNET WOLFGANG ,  UNGER LILIANE ,  RASCHACK MANFRED

IPC: C07D251/30 ,  A61K31/505 ,  A61P9/00 ,  A61P9/08 ,  A61P9/10 ,  A61P9/12 ,  A61P11/08 ,  A61P13/02 ,  A61P15/00 ,  A61P25/04 ,  C07D239/00 ,  C07D239/26 ,  C07D239/28 ,  C07D239/34 ,  C07D239/38 ,  C07D239/60 ,  C07D239/70 ,  C07D239/96 ,  C07D251/12 ,  C07D251/52 ,  C07D257/02 ,  C07D309/00 ,  C07D403/06 ,  C07D403/12 ,  C07D405/12 ,  C07D417/12 ,  C07D487/04 ,  C07D491/04 ,  C07D491/044 ,  C07D491/048

Abstract: Heterocyclyl-substd. propanoic acids and their derivs., of formula (I), are new. R = formyl, tetrazolyl, nitrile, COOH or a gp. that can be hydrolysed to COOH; X = N or CR14; R2 = H, OH, NH2, alkylamino, dialkylamino, halo, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; R14 = H or 1-5 C alkyl; R3 = R2 or alkoxyimino; or CR3 + CR14 = 5 or 6 membered alkylene or alkenyl ring (opt. substd. by 1-2 alkyl) in which a methylene can be replaced by O, S, NH or alkylamino; R4, R5 = phenyl or naphthyl (both opt. substd. by one or more halo, NO2, CN, OH, alkyl, haloalkyl, alkoxy, haloalkyloxy, phenoxy, alkylthio, NH2, alkylamine or dialkylamino) or 3-7 C cycloalkyl; or the phenyl or naphthyl gps. are opt. bonded at the O- position (by a bond, CH2, O, S, SO2, ethylene, ethenylene or opt. alkylated amino); R6 = H, 1-8 C alkyl, 2-6 C alkenyl, 3-6 C alkynyl, 3-8 C cycloalkyl (all opt. substd. by 1 or more halo, NO2, CN, alkoxy 3-6 C alkenyloxy, 3-6 C alkynyloxy, alkylthio, haloalkoxy, alkylcarbonyl, alkoxycarbonyl, 3-8 C alkylcarbonylalkyl, alkylamino, dialkylamino, phenyl, Ph or OPh), Ar or Het; Y = S, O or bond; Q = S, O, SO, SO2 or bond; Ph = substd. phenyl, where substits. are halo, NO2, CN, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; Ar = phenyl or naphthyl (both opt. substd. by 1 or more halo, NO2, CN, OH, NH2, alkylamino, dialkylamino or OCH2CH2O); Het = 5 or 6 membered heteroaromatic with 1-3 N atoms and/or one S or O (opt. substd. by 1-4 halo and/or 1 or 2 alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, phenyl, phenoxy or phenyl carbonyl (where the phenyl is opt. substd. by 1-5 halo and/or 1-3 alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkylthio)); alkyl and alkoxy have 1-4 C unless otherwise stated; provided that R6 is not H when Q = bond.

公开(公告)号：DE59709989D1

公开(公告)日：2003-06-05

申请号：DE59709989

申请日：1997-12-04

Applicant: BASF AG

Inventor： VOGELBACHER JOSEF ,  KEIL MICHAEL ,  KLINTZ RALF ,  WAHL JOSEPH ,  WINGERT HORST ,  KOENIG HARTMANN ,  RACK MICHAEL ,  GOETZ ROLAND ,  TELES HENRIQUE

IPC: C07D231/20 ,  C07D231/22

Abstract: PCT No. PCT/EP97/06780 Sec. 371 Date Jun. 14, 1999 Sec. 102(e) Date Jun. 14, 1999 PCT Filed Dec. 4, 1997 PCT Pub. No. WO98/27062 PCT Pub. Date Jun. 25, 1998A process is described for preparing N-substituted 3-hydroxypyrazoles of the formula I where R1 is unsubstituted or substituted alkyl, alkenyl, alkynyl, cycloalkyl, aryl or heteroaryl and R2, R3 are hydrogen, cyano, halogen and unsubstituted or substituted alkyl, alkenyl, alkynyl, cycloalkyl, aryl or heteroaryl, by oxidizing a corresponding pyrazolidin-3-one.

公开(公告)号：CZ9502767A3

公开(公告)日：1996-02-14

申请号：CZ276795

申请日：1994-04-14

Applicant: BASF AG

Inventor： BAUMANN ERNST ,  RHEINHEIMER JOACHIM ,  VOGELBACHER JOSEF ,  BRATZ MATTHIAS ,  MEYER NORBERT ,  GERBER MATTHIAS ,  WESTPHALEN KARL OTTO ,  WALTER HELMUT ,  RADEMACHER WILHELM

IPC: C07D251/34 ,  A01N43/54 ,  A01N43/60 ,  A01N43/66 ,  A01P13/00 ,  C07C69/712 ,  C07C69/734 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D239/60 ,  C07D251/30 ,  C07D307/54 ,  C07D333/24 ,  C07D491/048 ,  C07C69/22 ,  C07D239/52 ,  C07D307/46 ,  C07D405/12 ,  C07D409/12

CPC classification number: C07C69/734 ,  A01N43/54 ,  C07C69/712 ,  C07D239/60 ,  C07D251/30

公开(公告)号：CZ291719B6

公开(公告)日：2003-05-14

申请号：CZ276795

申请日：1994-04-14

Applicant: BASF AG

Inventor： BAUMANN ERNST ,  RHEINHEIMER JOACHIM ,  VOGELBACHER JOSEF ,  BRATZ MATTHIAS ,  MEYER NORBERT ,  GERBER MATTHIAS ,  WESTPHALEN KARL OTTO ,  WALTER HELMUT ,  RADEMACHER WILHELM

IPC: C07D251/34 ,  A01N43/54 ,  A01N43/60 ,  A01N43/66 ,  A01P13/00 ,  C07C69/22 ,  C07C69/712 ,  C07C69/734 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D239/52 ,  C07D239/60 ,  C07D251/30 ,  C07D307/46 ,  C07D307/54 ,  C07D333/24 ,  C07D405/12 ,  C07D409/12 ,  C07D491/048

Abstract: In the present invention there are described 3-aryloxycarboxylic acid derivatives of the general formula I, process of their preparation based on synthesis of corresponding starting compounds, further intermediates serving for their preparation, a herbicidal agent containing as active substance the derivative of the general formula I, composition for influencing growth of plants and containing the same active substance, method of suppressing undesired plant growth, based on action of the aforementioned active substance as well as method for regulating plant growth, based on use of the same active substance.

公开(公告)号：DE59807486D1

公开(公告)日：2003-04-17

申请号：DE59807486

申请日：1998-08-21

Applicant: BASF AG

Inventor： KLINTZ RALF ,  GOETZ NORBERT ,  KEIL MICHAEL ,  HEILIG MANFRED ,  WINGERT HORST ,  VOGELBACHER JOSEF ,  WAHL JOSEF ,  WETTERICH FRANK ,  DAUN GREGOR

IPC: C07C239/10 ,  C07C239/12 ,  C07C251/48 ,  C07C251/58 ,  C07C259/04 ,  C07D213/76 ,  C07D215/38 ,  C07D215/40 ,  C07D231/20 ,  C07D231/22 ,  C07D239/54 ,  C07D249/12 ,  C07D401/04 ,  C07D471/04

Abstract: The invention relates to a method for producing N-acylated (hetero)aromatic hydroxylamine derivatives of formula (I), wherein the substituents, the ring atom and the index have the meanings give in the Description, by hydrogenating a (hetero)aromatic nitro-compound of general formula (II) in the presence of a hydrogenation catalyst.

公开(公告)号：DE59410072D1

公开(公告)日：2002-04-11

申请号：DE59410072

申请日：1994-04-13

Applicant: BASF AG

Inventor： BAUMANN ERNST ,  RHEINHEIMER JOACHIM ,  VOGELBACHER JOSEF ,  BRATZ MATTHIAS ,  THEOBALD HANS ,  GERBER MATTHIAS ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT ,  RADEMACHER WILHELM

IPC: C07D251/22 ,  A01N43/54 ,  A01N43/64 ,  A01N43/66 ,  A01N43/72 ,  A01P13/00 ,  A01P21/00 ,  C07C45/58 ,  C07C47/198 ,  C07C47/277 ,  C07C59/125 ,  C07C67/31 ,  C07C69/708 ,  C07C69/734 ,  C07C205/28 ,  C07C323/22 ,  C07C323/50 ,  C07D239/26 ,  C07D239/30 ,  C07D239/34 ,  C07D239/38 ,  C07D239/60 ,  C07D251/24 ,  C07D251/30 ,  C07D251/34 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D411/12 ,  C07D413/12 ,  C07D477/12 ,  C07D491/048

Abstract: PCT No. PCT/EP94/01141 Sec. 371 Date Oct. 19, 1995 Sec. 102(e) Date Oct. 19, 1995 PCT Filed Apr. 13, 1994 PCT Pub. No. WO94/25442 PCT Pub. Date Nov. 10, 19943-(Het)arylcarboxylic acid derivatives of the formula I I where R is formyl, CO2H or a radical hydrolyzable to COOH and the other substituents have the following meanings: R2 and R3 are each halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkylthio; X is nitrogen or CR14, where R14 is hydrogen or, together with R3, forms an alkylene or alkenylene chain, in each of which a methylene group is replaced by oxygen; R4 is phenyl or naphthyl, each of which is unsubstituted or substituted or an unsubstituted or substituted five-membered or six-membered heteroaromatic structure containing one to three nitrogen atoms or one sulfur or oxygen atom; R5 is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl or phenyl; R6 is C1-C8-alkyl, C3-C6-alkenyl, C3-C6-alkynyl or C3-C4-cyclo-alkyl, each of which may be mono- or polysubstituted; Y is sulfur, oxygen or a single bond; and Z is sulfur or oxygen; with the proviso that R6 is not unsubstituted C1-C4-alkyl when R4 is unsubstituted phenyl, Z is oxygen and simultaneously R5 is methyl or hydrogen.

公开(公告)号：DE59509537D1

公开(公告)日：2001-09-27

申请号：DE59509537

申请日：1995-03-23

Applicant: BASF AG

Inventor： BAUMANN ERNST ,  VOGELBACHER JOSEF ,  RHEINHEIMER JOACHIM ,  KLINGE DAGMAR ,  RIECHERS HARTMUT ,  KROEGER BURKHARD ,  BIALOJAN SIEGFRIED ,  BOLLSCHWEILER CLAUS ,  WERNET WOLFGANG ,  UNGER LILIANE ,  RASCHACK MANFRED

IPC: C07D251/26 ,  A61K31/00 ,  A61K31/505 ,  A61K31/506 ,  A61K31/53 ,  A61P9/00 ,  A61P9/08 ,  A61P9/10 ,  A61P9/12 ,  A61P11/08 ,  A61P13/02 ,  A61P15/00 ,  A61P25/04 ,  A61P39/02 ,  C07D239/26 ,  C07D239/34 ,  C07D239/38 ,  C07D401/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

Abstract: PCT No. PCT/EP95/01099 Sec. 371 Date Sep. 30, 1996 Sec. 102(e) Date Sep. 30, 1996 PCT Filed Mar. 23, 1995 PCT Pub. No. WO95/26716 PCT Pub. Date Oct. 12, 1995A method of inhibiting endothelin receptors by administering to a patient a compound of the formula I I

公开(公告)号：UA79182C2

公开(公告)日：2007-05-25

申请号：UA2005006791

申请日：2003-12-01

Applicant: BASF AG

Inventor： VOGELBACHER JOSEF ,  WEVERS HENDRIK

IPC: C07C45/46 ,  C07C45/81 ,  C07C49/84 ,  C07C51/347 ,  C07C51/363 ,  C07C51/58 ,  C07C51/60

Abstract: Disclosed is a method for producing benzophenones of formula I, wherein X can represent chlorine, hydroxy, methoxy, or C1-C6 alkylcarbonyloxy while Y represents chlorine or bromine, by reacting an acid chloride of formula II, wherein X and Y have the meaning mentioned above, with 3,4,5-trimethoxytoluene. The inventive method is characterized by that the reaction is carried out in the presence of a) an aromatic hydrocarbon as a thinner, and b) 0.01 to 0.2 mole percent of an iron catalyst, the percentage being in relation to the acid chloride, c)at a temperature ranging between 60 DEGREE C and the boiling point of the respective thinner. , I , II

公开(公告)号：DE50304687D1

公开(公告)日：2006-09-28

申请号：DE50304687

申请日：2003-12-01

Applicant: BASF AG

Inventor： MAYWALD VOLKER ,  HOFFMANN NICO ,  KEIL MICHAEL ,  VOGELBACHER JOSEF ,  WEVERS HENDRIK

IPC: C07C45/46 ,  C07C45/81 ,  C07C49/84 ,  C07C51/363 ,  C07C51/60

Abstract: A process for preparing benzophenones of the formula I, where X may be chlorine, hydroxyl, methoxy or C 1 -C 6 -alkylcarbonyloxy, and Y may be chlorine or bromine, by reacting an acid chloride of the formula II where X and Y are as defined above with 3,4,5-trimethoxytoluene, which comprises carrying out the reaction in the presence of a) an aromatic hydrocarbon as a diluent and b) from 0.01 to 0.2 mol % of an iron catalyst, based on the acid chloride, c) at a temperature between 60° C. and the boiling point of the particular diluent.

公开(公告)号：DE59808710D1

公开(公告)日：2003-07-17

申请号：DE59808710

申请日：1998-07-20

Applicant: BASF AG

Inventor： WINGERT HORST ,  GOETZ NORBERT ,  KEIL MICHAEL ,  KLINTZ RALF ,  VOGELBACHER JOSEF ,  WAHL JOSEF

IPC: C07D231/20 ,  C07B39/00 ,  C07C205/11 ,  C07D231/08 ,  C07D231/22

Abstract: PCT No. PCT/EP98/04490 Sec. 371 Date Jan. 27, 2000 Sec. 102(e) Date Jan. 27, 2000 PCT Filed Jul. 20, 1998 PCT Pub. No. WO99/06373 PCT Pub. Date Feb. 11, 19992-(3-Pyrazolyloxymethylene)nitrobenzene [sic] derivatives of the formula I where the substituents and indices have the meanings given in the description, are prepared by bromination of an o-nitrotoluene of the formula II and subsequent reaction with a 3-hydroxypyrazole of the formula IV