公开(公告)号：WO2005113555A8

公开(公告)日：2006-12-14

申请号：PCT/EP2005005270

申请日：2005-05-13

Applicant: BASF AG ,  BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to novel triazolopyrimidine compounds of general formula (I), to their use for controlling pathogenic fungi and to agricultural pesticides containing compounds of this type as active constituents. In formula (I), X, Y, L, m, Ar and A are defined as follows: X represents halogen, cyano, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy or C 1 -C 4 haloalkoxy; Y represents halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl; L represents independently of one another halogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, nitro, amino, NHR, NR 2 , cyano, S(=O) n A 1 or C(=O)A 2 ; m represents 0, 1, 2, 3 or 4; A stands for a chemical bond or a CR 4 R 5 group; Ar represents phenyl or a 5- or 6-membered heteroaromatic group comprising 1, 2 or 3 heteroatoms selected from O, S and N as ring members, whereby the phenyl and the heteroaromatic group can comprise a fused benzole ring and can have 1, 2, 3, 4 or 5 R a substituents. R 1 to R 3 are defined as cited in claim 1.

Abstract translation: 本发明涉及如下通式的新型三唑并嘧啶化合物I和它们在防治有害真菌中的用途，以及植物保护剂，这样的化合物作为活性成分enthalten.In式I，X，Y，L，M，Ar和A具有下列含义：X 卤素，氰基，C _{1 -C 4 烷基，C 1 -C 4 卤代烷基，C < SUB> 1 -C 4 - 烷氧基或C 1 -C 4 卤代烷氧基; Y是卤素，C 1 -C 4 烷基或C 1 -C 4 卤代烷基; 独立地为卤素，C 1 -C 6 烷基，C 2 -C 6 烯基，C 1 -C ç 6 卤代烷基，C 1 -C 6 烷氧基，C 1 -C 6 < / SUB>卤代烷氧基，硝基，氨基，NHR，NR 2 ，氰基，S（= O）名词 A“或C（= O）A ^{2 ; m是0，1，2，3或4; A是一个化学键或基团CR 4 - [R 5 是; Ar是苯基或5-或6-元杂芳基具有1个，选自O，S和N的杂原子作为环成员，其中苯基和杂芳基可以具有一个稠合的苯环和1，2，3 2或3 ，4或5个取代基R 一可以包括;. R“至R 3 具有权利要求1中给出的含义。}}

公开(公告)号：WO2006066818A3

公开(公告)日：2006-11-02

申请号：PCT/EP2005013577

申请日：2005-12-16

Applicant: BASF AG ,  WAGNER OLIVER ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  NAVE BARBARA ,  STIERL REINHARD

Inventor： WAGNER OLIVER ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  NAVE BARBARA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D213/55 ,  C07D237/14 ,  C07D487/04

Abstract: The invention relates to novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds and the salts thereof that can be used in agriculture, the use of the same for controlling pathogenic fungi, and plant protection agents containing at least one such compound as an active constituent. Said novel 7-amino-6-hetaryl-1,2,4-triazolo[1,5-a]pyrimidine compounds correspond to general formula (I) wherein the substituents R 1 , R 2 , Het, X and Y have the following designations: Het represents a six-membered heteroaromatic radical selected from pyridinyl, pyridazinyl, pyrazinyl, 1,2,4-triazinyl and 1,3,5-triazinyl, the six-membered heteroaromatic radical comprising 1, 2 or 3 substituents L which are the same or different, R 1 , R 2 independently represent hydrogen, C 1 -C 8 alkyl, C 1 -C 8 halogenalkyl, C 1 -C 8 alkoxy, C 3 -C 8 cycloalkyl, C 3 -C 8 cycloalkoxy, C 5 -C 10 bicycloalkyl, C 3 -C 8 halogencycloalkyl, C 2 -C 8 alkenyl, C 2 -C 8 alkenyloxy, C 4 -C 10 alkadienyl, C 2 -C 8 halogenalkenyl, C 3 -C 8 cycloalkenyl, C 3 -C 8 halogencycloalkenyl, C 2 -C 8 alkinyl, C 2 -C 8 alkinyloxy, C 2 -C 8 halogenalkinyl, NH 2, C 1 -C 8 alkylamino, Di-C 1 -C 8 -alkylamino, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle, X represents hydrogen, halogen, OH, cyano, C 1 -C 4 alkyl and the like, and Y represents hydrogen, halogen, cyano, C 1 -C 4 alkyl, and the like.

Abstract translation: 本发明涉及新颖的7-氨基-6-杂芳基-1,2,4-三唑并[1,5-a]嘧啶化合物及其农业上可接受的盐，以及它们在防治有害真菌中的用途，以及植物保护剂，这些化合物的至少一种作为 含有活性成分。 新的7-氨基-6-杂芳基-1,2,4-三唑并[1,5-a]嘧啶化合物可通过通式（I）所示，其中取代基R ^{1 来表示 ，R 2 ，（I）的Het，X和Y在式具有以下含义：Het是其选自吡啶基，哒嗪基，吡嗪基的6元杂芳基，1,2,4- 三嗪基和1,3,5-三嗪基，其中所述6元杂芳基1，2或3个相同或不同的取代基L可以包括，R 1 ，R 2 独立地 另一个氢，C _{1 -C 8 烷基，C 1 -C 8 卤代烷基，C 1 -C 8 烷氧基，C 3 -C 8 环烷基，C 3 -C 8 环烷氧基，C 5 -C 10 双环，C 3 -C 8 卤代环烷基，C 2 -C 8 烯基，C 2 -C 8 烯 ，C 4 -C 10 链二烯基，C 2 -C 8 卤代，C 3 -C 8 环烯基，C 3 -C 8 卤代环，C 2 -C 8 炔基，C 2 -C 8 炔氧基，C 2 -C 8 卤代炔基，NH 2 C 1 -C 8 烷基氨基，二-C 1 -C 8 烷基氨基，苯基，萘基或五 - 或六元饱和，部分不饱和或芳族的杂环，X是氢，卤素，OH，氰基，C < SUB> 1 -C 4 烷基等，Y是氢，卤素，氰基，C 1 -C 4 烷基， 等等。}}

公开(公告)号：WO2005121146A3

公开(公告)日：2006-02-16

申请号：PCT/EP2005006171

申请日：2005-06-08

Applicant: BASF AG ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  HUENGER UDO ,  MUELLER BERND ,  NIEDENBRUECK MATTHIAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  RACK MICHAEL ,  NAVE BARBARA ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/647 ,  A01N43/90 ,  C07D487/00

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to triazolopyrimidines of formula (I), wherein the index n and the substituents R, R

Abstract translation: 本发明涉及下式的三唑并嘧啶I，其中索引n和取代基R，R

公开(公告)号：WO2005010000A3

公开(公告)日：2005-05-19

申请号：PCT/EP2004007924

申请日：2004-07-15

Applicant: BASF AG ,  WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： WAGNER OLIVER ,  GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  TORMO I BLASCO JORDI ,  AKERS ALAN ,  SPEAKMAN JOHN-BRYAN ,  RACK MICHAEL ,  STIERL REINHARD ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  C07D471/04

CPC classification number: C07D471/04 ,  A01N43/90

Abstract: The invention relates to bicyclic compounds of general formula I, wherein X, Y independently represent N or C-R ; n stands for 1, 2, 3, 4 or 5; R represents halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-halogenalkyl, C1-C6-halogenalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8 cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R ; R denotes halogen, cyano, C1-C6-alkyl, C1-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl, optionally mono- or polysubstituted by alkyl and/or halogen, OR , SR or NR R , and R represents hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl or C3-C6-cycloalkyl, optionally mono- or polysubstituted by alkyl and/or halogen. Said invention also relates to the agriculturally-acceptable salts of said compounds (I), plant protection agents, containing at least one compound of general formula (I) and/or one agriculturally-acceptable salt of (I) and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.

Abstract translation: 本发明涉及通式I的双环化合物，其中X，Y彼此独立地是N或C-R 4; n是1,2,3,4或5; ř表示卤素，氰基，C1-C6烷基，C1-C6烷氧基，C1-C6卤代烷基，C1-C6卤代烷氧基，C2-C6链烯基，C2-C6链烯氧基或C （O）R 5代表; [R <1>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8-环烷基，其任选被烷基和/或卤素取代的或者 多取代，C5-C8环烯基，其任选与乘法烷基和/或卤素或单 - ，或<6>，SR <6>或NR <7> - [R <8>取代; [R <2>为卤素，氰基，C1-C6烷基，C1-C6卤代烷基，C2-C6链烯基，C2-C6炔基，C3-C8环烷基，任选地被烷基和/或卤素单取代的 或多取代的，C5-C8环烯基，其任选地被烷基和/或卤素取代基取代一次或多次，或<6>，SR <6>或NR <7> - [R <8>; R 3是任选被烷基和/或卤素单取代或多取代的氢，C 1 -C 6烷基，C 1 -C 6卤代烷基或C 3 -C 6环烷基; 和化合物（I），植物保护剂的农业上可接受的盐，其包含通式（I）和/或（I）的农业上可接受的盐和至少一种液体或固体载体和用于防治植物病原性有害真菌的方法中的至少一种化合物。

公开(公告)号：WO9955156A3

公开(公告)日：1999-12-23

申请号：PCT/EP9902469

申请日：1999-04-13

Applicant: BASF AG ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL OTTO ,  WALTER HELMUT

Inventor： WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: A01N43/653 ,  C07D249/14 ,  C07D401/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

CPC classification number: C07D401/12 ,  A01N43/653 ,  C07D249/14 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

Abstract: The invention relates to the use of iminotriazoles of general formula (I), wherein R represents aryl or heteroaryl and these radicals can carry one to five groups independently of each other or the aryl- or heteroaryl radical forms a bicyclic system together with a fused phenyl ring, a fused C3-C6 carbocyclic compound or a 5- or 6-membered heterocyclic compound; A is COOR or CONR R , R and R being independently of each other, hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C3-C7-cycloalkyl or C1-C6-alkyl-aryl which can optionally be partially or completely halogenised or can carry one to three substituents chosen from the following: C1-C4 alkoxy, C1-C4-halogenalkoxy, C1-C4-alkylthio, C3-C7-cycloalkyl and C5-C7-cycloalkenyl.

Abstract translation: 使用Iminotriazolen通式（I），其中R <1>为芳基或杂芳基，这些基团彼此独立地可以携带一至五个基团，或其中芳基或杂芳基与稠合的苯环，稠合的C-C6的碳环或 的5-或6-元环Heteroocyclus形成双环系统，一个是COOR <3>或CONR <3> [R <4>，其中R <3>和R <4>独立地是氢，C1-C6烷基，C2- 表示C6链烯基，C3-C7环烷基或C1-C6烷基 - 芳基，其可被部分或完全卤化，如有必要，或一至三个选自C 1 -C 4 - 烷硫基的取代基，可携带C 3 -C 7环烯基。

公开(公告)号：WO9926930A2

公开(公告)日：1999-06-03

申请号：PCT/EP9807099

申请日：1998-11-06

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  ENGEL STEFAN ,  BAUMANN ERNST ,  DEYN WOLFGANG VON ,  HILL REGINA LUISE ,  MAYER GUIDO ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL OTTO ,  WALTER HELMUT

Inventor： RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  ENGEL STEFAN ,  BAUMANN ERNST ,  VON DEYN WOLFGANG ,  HILL REGINA LUISE ,  MAYER GUIDO ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WESTPHALEN KARL-OTTO ,  WALTER HELMUT

IPC: A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  C07D231/16 ,  C07D231/20 ,  C07D401/10 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D413/06 ,  C07D413/10 ,  C07D417/10 ,  C07D231/18

CPC classification number: C07D413/06 ,  A01N43/56 ,  A01N43/78 ,  A01N43/80 ,  C07D231/16 ,  C07D231/20

Abstract: The invention relates to benzylidene pyrazolones of formula (I), wherein the substituents and index n have the following meanings: R = optionally substituted C1-C6 alkyl; R = optionally substituted C1-C6 alkyl, optionally substituted C1-C6 alkoxy, halogen, nitro, cyano; R = hydrogen, halogen, nitro, cyano, a group NR R , OCOR , NR COR ,CO2R , -COSR , -CONR R , C1-C4-alkoxyiminoalkyl, C1-C6 alkoxycarbonyl, optionally substituted C1-C6 alkyl, optionally substituted C1-C6 alkoxy, optionally substituted C1-C6 alkylthio, optionally substituted C2-C6 alkenyl, optionally substituted phenyl, optionally substituted phenoxy, an optionally substituted 5- or 6-membered saturated or unsaturated heterocycle which can contain up to 4 nitrogen atoms and/or up to 2 oxygen or sulphur atoms as ring members; R = C1-C6 alkyl, C1-C4 halogen alkyl; or R and R = an optionally substituted saturated or unsaturated 2- or 3-membered bridge which can contain one sulphur atom which can be oxidized into sulfoxide or sulfone, R = hydrogen or optionally substituted C1-C6 alkyl; R = hydrogen, C1-C6 alkyl or C1-C4 halogenalkyl; n = 0, 1 or 2; X = hydrogen, chlorine or bromine. The compounds to which claim is laid are available in both a trans and a cis form or can be a mixture of these isomers.

Abstract translation: 式（I）的Benzylidenpyrazolone其中取代基和指数n具有以下含义：R t <1>是未取代的或取代的。 C1-C6烷基; [R <2>是未取代的或取代的。 C1-C6烷基，未取代或取代的。 C1-C6烷氧基，卤素，硝基，氰基; [R <3>是氢，卤素，硝基，氰基，基团NR <5> - [R <6>，OCOR <5>，NR <5> COR <6>，CO 2 <5>，-COSR <5>，-CONR <5> - [R <6>，C1-C4-alkoxyiminoalkyl，C1-C6烷基羰基，未取代的或取代的。 C1-C6烷基，未取代或取代的。 C1-C6烷氧基，未取代的或取代的。 C1-C6烷硫基，未取代或取代的。 C2-C6链烯基，未取代的或取代的。 C2-C6炔基，未取代的或取代的。 苯基，未取代的或取代的。 苯氧基，未取代的或取代的。 5-或6-元饱和或可含有至多4个氮原子和/或至多2个氧或硫原子作为环成员的不饱和的杂环; [R <4> C1-C6-烷基，C1-C4卤代烷基; 或R <3>，R <4>为可以含有可被氧化为亚砜或砜硫原子的任选取代的饱和或不饱和2-或3-元桥; [R <5>为氢或未取代或取代的。 C1-C6烷基; [R <6>是未取代的或取代的。 C1-C6烷基; [R <7>是氢，C1-C6烷基或C1-C4卤代烷基; n为0.1或2; X是氢，氯或溴; 其中要求保护的化合物在跨及在所述顺式 - 形式两者呈现，或者可以是这些异构体的混合物。

公开(公告)号：BRPI0612809A2

公开(公告)日：2016-11-29

申请号：BRPI0612809

申请日：2006-07-06

Applicant: BASF AG

Inventor： WAGNER OLIVER ,  ULMSCHNEIDER SARAH ,  HÜNGER UDO

IPC: C07D487/04 ,  A01N43/90

公开(公告)号：EE05291B1

公开(公告)日：2010-04-15

申请号：EEP9900292

申请日：1998-01-08

Applicant: BASF AG

Inventor： HILL REGINA LUISE ,  DEYN WOLFGANG VON ,  BAUMANN ERNST ,  ENGEL STEFAN ,  MAYER GUIDO ,  RHEINHEIMER JOACHIM ,  WITSCHEL MATTHIAS ,  MISSLITZ ULF ,  WAGNER OLIVER ,  OTTEN MARTINA ,  WALTER HELMUT ,  WESTPHALEN KARL-OTTO

IPC: A01N43/48 ,  C07D277/10 ,  A01N43/18 ,  A01N43/56 ,  A01N43/72 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  C07D231/20 ,  C07D231/24 ,  C07D261/04 ,  C07D261/20 ,  C07D263/10 ,  C07D273/00 ,  C07D277/20 ,  C07D277/34 ,  C07D291/04 ,  C07D401/10 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D411/10 ,  C07D413/10 ,  C07D417/10 ,  C07D419/10 ,  C07D498/10

Abstract: 4-(3-Heterocyclyl-benzoyl)-pyrazole derivatives (I) and their salts are new: R1, R3 = H; NO2; halo; CN; 1-6C alkyl, 1-6C alkoxy, 1-6C alkylthio, 1-6C alkylsulphinyl or 1-6C alkylsulphonyl optionally substituted by halo; H2NSO2; (1-6C alkyl)NHSO2; (1-6C alkyl)2NSO2; (1-6C alkyl)SO2NH-; (1-6C haloalkyl-SO2)NH-; (1-6C alkyl)(1-6C alkyl-SO2)N-; or (1-6C haloalkyl)(1-6C alkyl-SO2)N-; R2 = optionally substituted 5- or 6-membered heterocycle containing 1-4 O, S and/or N atoms; R6 = 1-6C alkyl; R7 = 1-6C alkyl; 3-6C alkenyl or 3-6C alkynyl optionally substituted by halo; 3-6C cycloalkyl; 1-6C alkylcarbonyl; 2-6C alkenylcarbonyl; 2-6C alkynylcarbonyl; 3-6C cycloalkylcarbonyl; 1-6C alkoxycarbonyl; 3-6C alkenyloxycarbonyl; 3-6C alkynyloxycarbonyl; 1-6C alkyl-NH-CO-; 3-6C alkenyl-NH-CO-; 3-6C alkynyl-NH-CO-; (1-6C alkyl)2N-CO-; (3-6C alkenyl)(1-6C alkyl)N-CO-carbonyl; (3-6C alkynyl)(1-6C alkyl)N-CO-; (1-6C alkoxy)(1-6C alkyl)N-CO-; (3-6C alkenyl)(1-6C alkoxy)N-CO-; (3-6C alkynyl)(1-6C alkoxy)N-CO-; (1-6C alkyl)2N-CS-; 1-6C alkoxyimino-1-6C alkyl; 1-6C alkylamino imino-1-6C alkyl; or di(1-6C alkylamino)imino-1-6C alkyl (alkyl, cycloalkyl and alkoxy groups are optionally substituted by 1 or more halo and/or by 1-3 CN, OH, 1-4C alkoxy, 1-4C alkylthio, di(1-4C alkyl)amino, 1-4C alkylcarbonyl, 1-4C alkoxycarbonyl, 1-4C alkoxy-1-4C alkoxycarbonyl, (1-4C alkyl)2N-1-4C alkoxycarbonyl, COOH, 1-4C alkyl-NH-CO-, (1-4C alkyl)2N-CO-, CONH2; 1-4C alkylcarbonyloxy or 3-6C cycloalkyl); or Ar; Ar-1-6C alkyl; Ar-CO-1-6C alkyl; Ar-CO-; Ar-O-CO-; Ar-NH-CO-; (1-6C alkyl)(Ar)N-CO-; or Ar-2-6C alkenylcarbonyl; Ar = phenyl or heterocyclyl optionally substituted by 1 or more halo and/or by 1-3 NO2, CN or 1-4C alkyl or 1-4C alkoxy (optionally substituted by halo), and R8 = H, 1-6C alkyl or 1-6C haloalkyl.

公开(公告)号：EA011360B1

公开(公告)日：2009-02-27

申请号：EA200601569

申请日：2005-03-08

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUCK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD ,  HUNGER UDO

IPC: C07D487/04

Abstract: 5,6-Диалкил-7-аминотриазолопиримидиныформулы Iвкоторойзаместителиимеютследующеезначение: Rозначаеталкил, алкоксиалкил, алкенилилиалкинил; Rозначаеталкил, алкоксилкил, алкенилилиалкинил; причем Rи/или Rзамещенысогласноописанию; способполученияэтихсоединенийи ихприменениедляборьбыс фитопатогеннымигрибами, атакжесредства, содержащиеэтисоединения.

公开(公告)号：NZ547363A

公开(公告)日：2009-01-31

申请号：NZ54736304

申请日：2004-12-17

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  WAGNER OLIVER ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

Abstract: Disclosed are triazolopyrimidines of formula (I), wherein the substituents have the following meaning: R1, R2 represent hydrogen, alkyl, alkyl halide, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl, or phenyl, naphthyl, or a five-membered to six-membered saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group comprising O, N, and S. R1 and R2 can also form a five-membered or six-membered heterocyclyl or heteroaryl along with the nitrogen atom to which the same are bonded, said heterocyclyl or heteroaryl being bonded via N, while optionally containing an additional heteroatom from the group comprising O, N, and S as a ring member and being optionally substituted according to the description; L represents halogen, cyano, alkyl, alkyl halide, alkoxy, alkenyloxy, or alkoxy carbonyl; m represents 1, 2, 3, or 4, the groups L being optionally different if m is greater than 1; X represents halogen, cyano, alkyl, alkyl halide, alkoxy, or haloalkoxy. Also disclosed are methods and intermediate products for producing said compounds, substances containing the same, and the use thereof for controlling plant-pathogenic fungi.