公开(公告)号：AU2005256507A1

公开(公告)日：2006-01-05

申请号：AU2005256507

申请日：2005-06-24

Applicant: BASF AG

Inventor： BLETTNER CARSTEN ,  GEWEHR MARKUS ,  SCHWOGLER ANJA ,  SCHOFL ULRICH ,  MULLER BERND ,  WAGNER OLIVER ,  GROTE THOMAS ,  SPEAKMAN JOHN-BRYAN ,  RHEINHEIMER JOACHIM ,  JABS THORSTEN ,  BLASCO JORDI TORMO I ,  SCHIEWECK FRANK ,  STIERL REINHARD ,  GRAMMENOS WASSILIOS ,  SCHERER MARIA ,  SCHAFER PETER ,  STRATHMANN SIEGFRIED

IPC: C07D487/04 ,  A01N43/90

Abstract: The present invention relates to novel triazolopyrimidine compounds of the formula I in which: X is halogen, cyano, C 1 -C 4 -alkyl, C 1 -C 4 -haloalkyl, C 1 -C 4 -alkoxy or C 1 -C 2 -haloalkoxy; W is oxygen or sulfur; Y is O-R 4 or a group NR 5 R 6 ; A is a chemical bond or a group CR 7 R 8 ; and the variables L, R 1 to R 7 are as defined in claim 1. The present invention furthermore provides the use of the triazolopyrimidine compounds of the formula I, their tautomers and their agriculturally acceptable salts for controlling phytopathogenic fungi (=harmful fungi) and a method for controlling phytopathogenic harmful fungi, which method comprises treating the fungi or the materials, plants, the soil or seed to be protected against fungal attack with an effective amount of a compound of the formula I, a tautomer of I and/or an agriculturally acceptable salt of I or a tautomer thereof.

公开(公告)号：PE20050812A1

公开(公告)日：2005-11-03

申请号：PE2005000008

申请日：2005-01-03

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  WAGNER OLIVIER ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD

IPC: A01N43/653 ,  C07D487/04

Abstract: SE REFIERE A TRIAZOLOPIRIMIDINAS DE FORMULA (I), DONDE L ES H, CLORO O BROMO; R1 Y R2 SON INDEPENDIENTEMENTE ALQUILO C1-C8, HALOGENOALQUILO C1-C8. CICLOALQUILO C3-C8 o FENILO, NAFTILO o UN HETEROCICLO SATURADO, PARCIALMENTE INSATURADO O AROMATICO, CON 5 o 6 MIEMBROS, QUE CONTIENEN UNO A CUATRO HETEROATOMOS DEL GRUPO: O, N o S; R3 ES ALQUILO C1-C8, HALOGENOALQUILO C1-C8, ALQUENILO C3-C8, HALOGENOALQUILO C-C8, ALQUINILO C3-C8, ENTRE OTROS; DONDE R1 Y/O R2 PUEDEN LLEVAR 1 A 4 GRUPOS Ra, SIENDO Ra HALOGENO, CIANO, NITRO, HIDROXI, ALQUILO C1-C6, HALOGENOALQUILO, FENILO, NAFTILO, HETEROCICLO SATURADO, PARCIALMENTE INSATURADO O AROMATICO DE CINCO o DIEZ MIEMBROS, QUE CONTIENE UNO A CUATRO HETEROATOMOS DE: O, N o S, PUDIENDO ESTOS GRUPOS ALIFATICOS, ALICICLICOS o AROMATICOS POR SU PARTE ESTAR PARCIAL O COMPLETAMENTE HALOGENADOS O LLEVAR UNO A TRES GRUPOS Rb; DONDE Rb ES HALOGENO, CIANO, NITRO, MERCAPTO, AMINO, ALCOXI, FORMILO, ALQUILCARBONILO, ALQUILCARBONILOXI, DIALQUILAMINOTIOCARBONILO, ENTRE OTROS, CONTENIENDO LOS GRUPOS ALQUILO 1 A 6 ATOMOS DE CARBONO Y LOS GRUPOS ALQUENILO O ALQUINILO MENCIONADOS DE A 8 ATOMOS DE CARBONO; Y, UNO A TRES DE LOS RADICALES SIGUIENTES: CICLOALQUILO, CICLOALCOXI, DONDE, LOS SISTEMAS CICLICOS PUEDEN CONTENER 3 A 10 MIEMBROS ANULARES, ARILO, ARILOXI, ARILTIO, ARIL-ALCOXI C1-C6, HETARILOXI, ENTRE OTROS; Y, X ES HALOGENO, CIANO, ALQUILO C1-C4, HALOGENOALQUILO C1-C4, ALCOXI C1-C4, ENTRE OTROS. TIENE APLICACION PARA COMBATIR HONGOS NOCIVOS

公开(公告)号：PE20050823A1

公开(公告)日：2005-10-27

申请号：PE2005000004

申请日：2005-01-03

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  MULLER BERND ,  GROTE THOMAS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  SCHWOGLER ANJA ,  RHEINHEIMER JOACHIM ,  BLETTNER CARSTEN ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  WAGNER OLIVIER ,  SPEAKMAN JOHN-BRYAN ,  RETHER JAN ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD

IPC: A01N43/10 ,  A01N43/40 ,  A01N43/56 ,  A01N43/74 ,  A01N43/78 ,  A01N47/48 ,  C07C251/38 ,  C07D207/34 ,  C07D213/82 ,  C07D231/14 ,  C07D263/34 ,  C07D277/56 ,  C07D279/12 ,  C07D307/30 ,  C07D307/54 ,  C07D307/71 ,  C07D333/38

Abstract: SE REFIERE A LAS (HETERO)CICLILCARBOXANILIDAS DE FORMULA GENERAL (I) EN LAS QUE "n" REPRESENTA 0,1,2,3 o 4; "m" REPRESENTA 1,2 o 3; Y ES A OXIGENO o AZUFRE; A ES FENILO o UN HETEROCICLO DE 5 o 6 MIEMBROS QUE ESTA INSATURADO POR LO MENOS EN FORMA SIMPLE, CON 1, 2, o 3 HETEROATOMOS SELECCIONADOS DE ENTRE N, O, S, S(=O) Y S(=O)2, COMO MIEMBROS DEL ANILLO, ENTRE OTROS, R1 ES H, OH, ALQUILO-C1-C4, CICLOALQUILO C3-C6, ALCOXI C1-C4, ENTRE OTROS; R2 ES HALOGENO, NITRO, CN, ALQUILO C1-C4, ALQUINILO C2-C4, ENTRE OTROS; R3m Y R4m SON INDEPENDIENTEMENTE EL UNO DEL OTRO, HALOGENO, HIDROGENO, ALQUILO-C1-C6, FENILHALOALQUILO C2-C4, ENTRE OTROS; R5 ES HIDROGENO, ALQUILO-C1-C6, CICLOALQUILO-C3-C6, ALQUENILO-C2-C6, ALQUINILO C2-C6, FENILO, FENILALQUILO-C1-C4, FENILALQUENILO-C2-C4, ENTRE OTROS; R6 ES H, ALQUILO-C1-C8, CICLOALQUILO-C3-C6, ALQUENILO C2-C8, ALQUINILO C2-C8, NAFTILALQUILO-C1-C6, ENTRE OTROS; Y, LAS SALES DE LAS MISMAS, QUE PUEDEN USARSE EN LA AGRICULTURA COMO FUNGICIDA o FITOPROTECTOR

公开(公告)号：EA006133B1

公开(公告)日：2005-10-27

申请号：EA200400111

申请日：2002-07-16

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MULLER BERND ,  GEWEHR MARCUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

Abstract: Изобретениеотноситсяк 7-аминотриазолопиримидинамформулы Iгдезаместителиимеютследующиезначения:R, Rозначаетводород, алкил, алкенил, алкинил, циклоалкил, фенил, нафтил; или5- или 6-членныйгетероциклил, содержащийотодногодочетырехатомовазотаилиотодногодотрехатомовазотаи одинатомсерыиликислорода; или5- или 6-членныйгетероарил, содержащийотодногодочетырехатомовазотаилиотодногодотрехатомовазотаи одинатомсерыиликислорода; илиRи Rвместес атомомазота, которыйихсоединяет, могутобразовывать 5- или 6-членныйцикл, которыйсодержитотодногодочетырехатомовазотаи отодногодотрехатомовазотаи одинатомсерыиликислорода;Rозначаеталкил, алкенил, алкинил, циклоалкил, фенилалкилилигалогеналкил,причем Rможетбытьнезамещеннымиличастичноилиполностьюзамещеннымсогласноописанию;X означаетгалоген, циано, С-Салкокси, С-Сгалогеналкил, фенилилизамещенныйостатком Rфенил;кспособуи промежуточнымпродуктамдляихполучения, содержащимихсредствам, атакжек ихприменению.

公开(公告)号：NZ531066A

公开(公告)日：2005-04-29

申请号：NZ53106602

申请日：2002-07-08

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N25/04 ,  A01N43/90 ,  C07D487/04 ,  C07D249/00 ,  C07D239/00

Abstract: Disclosed are 6-(2,6-difluoro-phenyl)-triazolopyrimidines of formula I, wherein: R1 and R2 are independently H, alkyl, alkenyl, alkynyl, alkadineyl, cycloalkyl, phenyl, naphthyl, heterocyclyl, or heteroaryl, and are optionally substituted, R1 and R2 may together form an optionally substituted heterocyclic ring, X is halogen, cyano, alkoxy, haloalkoxy or alkenyloxy. The compounds are used in a method for controlling phytopathogenic fungi, comprising treating the fungi, materials, plants, soil or seed with an effective amount of the compounds.

公开(公告)号：AU2004278095A1

公开(公告)日：2005-04-14

申请号：AU2004278095

申请日：2004-09-10

Applicant: BASF AG

Inventor： MULLER BERND ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GOTZ NORBERT ,  SCHOFL ULRICH ,  GEWEHR MARKUS ,  STIERL REINHARD ,  SCHIEWECK FRANK ,  BLASCO JORDI TORMO I ,  SCHERER MARIA ,  WAGNER OLIVER ,  STRATHMANN SIEGFRIED ,  SCHWOGLER ANJA ,  SCHAFER PETER ,  BLETTNER CARSTEN ,  RHEINHEIMER JOACHIM

IPC: C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

Abstract: Sulfonamides of the formula I where the substituents are as follows: R 1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R 2 , R 3 , R 4 , R 5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R 2 and R 3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R 2 ' and R 3 ', R 2 ', R 3 ' are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R 2 , R 3 , R 4 and R 5 are hydrogen: X is phenyl substituted by a group C(R 6 )-NOR 7 , where R 6 is alkyl and R 7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R 2 , R 3 , R 4 and R 5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

公开(公告)号：AU2004266783A1

公开(公告)日：2005-03-03

申请号：AU2004266783

申请日：2004-07-03

Applicant: BASF AG

Inventor： SCHWOGLER ANJA ,  GRAMMENOS WASSILIOS ,  SCHOFL ULRICH ,  WAGNER OLIVER ,  SCHAFER PETER ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED ,  BLASCO JORDI TORMO I ,  MULLER BERND ,  BLETTNER CARSTEN ,  RHEINHEIMER JOACHIM ,  STIERL REINHARD ,  SCHIEWECK FRANK ,  GEWEHR MARKUS ,  GYPSER ANDREAS ,  SCHERER MARIA

IPC: C07D239/42

Abstract: The invention relates to 2-substituted pyrimidines of the formula I in which the index n and these substituents R 1 , R 2 and R 3 are as defined in the description and R 4 is as defined below: R 4 corresponds to one of the formulae where R a is hydrogen, C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 3 -C 6 -cycloalkyl or C 1 -C 4 -alkoxy and R 5 is hydrogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 1 -C 4 -alkyloxy-C 1 -C 2 -alkyl, phenyl-C 1 -C 2 -alkyl or phenyloxy-C 1 -C 2 -alkyl, to processes for preparing these compounds, to compositions comprising these compounds and to their use as pesticides.

公开(公告)号：CZ294102B6

公开(公告)日：2004-10-13

申请号：CZ287698

申请日：1997-03-06

Applicant: BASF AG

Inventor： EICKEN KARL ,  GEBHARDT JOACHIM ,  RANG HARALD ,  RACK MICHAEL ,  SCHAFER PETER

IPC: B01J31/24 ,  C07B37/04 ,  C07B61/00 ,  C07C201/12 ,  C07C205/06 ,  C07C205/11 ,  C07C205/12 ,  C07C205/35 ,  C07C253/30

Abstract: The present invention relates to a process for preparing nitrobiphenylene of the general formula I wherein m stands for 1 or 2, R represents a halogen or R' whereby R' is selected from the group consisting of a cyano group, formyl, a formyloxy group and optionally a substituted alkyl, alkenyl, alkoxy group, alkenyloxy group, alkylcarbonyl, alkoxycarbonyl, alkylcarbonyloxy group, cycloalkyl, cycloalkoxy group, phenyl or phenoxy group, n stands for 0, 1, 2 or 3 and, if n is 2 or 3. According to the invention, a chloronitrobenzene of the general formula II is reacted in the presence of a base and a palladium catalyst being selected from the group consisting of (a) triarylphosphane complex containing in zero oxidation stage, (b) a palladium salt in the presence of triphenylphosphane and (c) optionally a supported metallic palladium, in the presence of triarylphosphane with a phenyl boric acid of the general formula IIIa, or of alkyl ester thereof of the general formula IIIb or with anhydride thereof.

公开(公告)号：AU2003293894A1

公开(公告)日：2004-07-09

申请号：AU2003293894

申请日：2003-12-16

Applicant: BASF AG

Inventor： GROTE THOMAS ,  BLETTNER CARSTEN ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD ,  MULLER BERND ,  BLASCO JORDI TORMO I

IPC: C07D487/04 ,  A01N43/653

Abstract: Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R 1 is C 1 -C 10 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -alkynyl, C 3 -C 10 -cycloalkyl, C 3 -C 10 -cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R 2 is C 1 -C 4 -alkyl which may be substituted by halogen, cyano, nitro or C 1 -C 2 -alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SO m -R x , NR x R y or NR x -(C-O)-R y ; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

公开(公告)号：AU2003283348A1

公开(公告)日：2004-06-07

申请号：AU2003283348

申请日：2003-11-04

Applicant: BASF AG

Inventor： BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  STIERL REINHARD

IPC: C07D487/04

Abstract: The invention relates to 5-alkyl-7-aminotriazolopyrimidines of the formula (I) and to the salts thereof. In said formula substituents have the following meanings: R1 and R2 each is a hydrogen atom or a group of alkyl, alcenyl, haloalkyl, cycloalky, phenyl or naphtyle, saturated, unstaturated or aromatic heterocycle having from five to six members which contain from one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can from together with a connecting them nitrogen atom a cycle of 5 to 6 members containing from one to four nitrogen atoms or from one to three nitrogen atoms and one sulfur or oxygen atom, R3 is a cycloalkyl or bicycloalkyl group, R1, R2 and R3 can be substituted in conformity with a description, and X is an alkyl or alkyl halide group. The inventive methods and intermediary products necessary for producing said compounds, agents containing them and the use therefore for fighting against harmful mushroom are also disclosed.