公开(公告)号：CZ472890A3

公开(公告)日：1994-12-15

申请号：CS472890

申请日：1990-09-28

Applicant: BASF AG

Inventor： SAUTER HUBERT DR ,  ZIERKE THOMAS DR ,  REUTHER WOLFGANG DR ,  BAUS ULF DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR

IPC: A01N43/653 ,  C07D249/08 ,  C07D401/12 ,  C07D403/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  C07D521/00

Abstract: Compounds of the formula I I where Ar is unsubstituted or substituted phenyl, pyridyl, thienyl or napthyl, R1 is hydrogen or CN, R2 is unsubstituted or substituted aryl, hetaryl, alkyl or cycloalkyl, or is unsubstituted or substituted alkenyl or alkynyl, x is CH2, O or S and n is 0 or 1, their plant-tolerated acid addition salts and metal complexes, and fungicides and growth regulators containing these compounds.

公开(公告)号：ES2055262T3

公开(公告)日：1994-08-16

申请号：ES90118281

申请日：1990-09-24

Applicant: BASF AG

Inventor： SAUTER HUBERT DR ,  ZIERKE THOMAS DR ,  REUTHER WOLFGANG DR ,  BAUS ULF DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR

IPC: A01N43/653 ,  C07D249/08 ,  C07D401/12 ,  C07D403/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  C07D521/00

Abstract: Compounds of the formula I I where Ar is unsubstituted or substituted phenyl, pyridyl, thienyl or napthyl, R1 is hydrogen or CN, R2 is unsubstituted or substituted aryl, hetaryl, alkyl or cycloalkyl, or is unsubstituted or substituted alkenyl or alkynyl, x is CH2, O or S and n is 0 or 1, their plant-tolerated acid addition salts and metal complexes, and fungicides and growth regulators containing these compounds.

公开(公告)号：DK0442339T3

公开(公告)日：1994-07-25

申请号：DK91101436

申请日：1991-02-04

Applicant: BASF AG

Inventor： ZIERKE THOMAS DR ,  KUEKENHOEHNER THOMAS DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N43/40 ,  C07D213/30 ,  C07D213/42 ,  C07D213/57 ,  C07D213/89

Abstract: Compounds of the formula 1 1 where R is unsubstituted or substituted cycloalkyl or cycloalkenyl, X, Y and Z are hydrogen, halogen, alkyl, alkoxy, alkoximino, haloalkyl, cyano, nitro or unsubstituted or substituted phenyl or phenoxy, W is -CH2- or -CH2CH2- and n is 0 or 1, and the plant-tolerated acid-addition salts thereof, and fungicides containing these compounds are described.

公开(公告)号：AT103595T

公开(公告)日：1994-04-15

申请号：AT91101013

申请日：1991-01-26

Applicant: BASF AG

Inventor： ZIPPERER BERNHARD DR ,  LAUER MANFRED DR ,  GOETZ NORBERT DR ,  ZIERKE THOMAS DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  C07D213/30 ,  C07D213/50 ,  C07D401/06 ,  C07D405/06 ,  C07D407/06 ,  C07D409/06

公开(公告)号：DE4027139A1

公开(公告)日：1992-03-05

申请号：DE4027139

申请日：1990-08-28

Applicant: BASF AG

Inventor： ZIERKE THOMAS DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N43/40 ,  C07D213/30 ,  C07D213/50 ,  C07D405/04

Abstract: (A) Pyridine derivs. of formula (I) and their N-oxides, mineral acid salts and metal complexes are new: X = OH; Y = OCHO, OCOW3R3 or OSO2W3R3; or X+Y = O, OCH(W3R3)O, OCH(OW3R4)O or OC(W3R3)(OW4R4)O; W1-W4 = direct bonds, CH2, CH2CH2, CHMe, CH2O or CH2S; R1-R4 = (a) 1-6C alkyl opt. substd. by halogen or 3-8C cycloalkyl, (b) 3-8C cycloalkyl opt. substd. by 1-3 of 1-6C alkyl, (c) 1-4C alkyl substd. by 1-4C alkoxy or alkylthio, (d) 2-6C alkenyl, etc., or R2 may be H when X+Y = OCH(W3R3)O, or OC(W3R3)(OW4R4)O and W2 is a direct bond; except for: cis-1-(2,4-dichlorophenyl) -2-(3-pyridyl)-1,2 -epoxypropane; trans-1-(2,4 -dichlorophenyl) -2-(3-pyridyl) -1,2-epoxypropane; etc.. Intermediates of formula (II) are also new provided that: (a) R1W1 is not H (sic), vinyl, phenyl or 3-pyridyl when R2W2 = H; (b) R1W1 is not 2,4-dichlorophenyl when R2W2 = Me; (c) R2W2 is not phenyl or 4-methoxyphenyl when R1W1 = phenyl; (d) W2 is not CH2 or CHMe when R1 = H (sic) or 1-5C alkyl, R2 = opt. substd. phenyl and W1 is a direct bond.

公开(公告)号：CS35991A2

公开(公告)日：1991-09-15

申请号：CS35991

申请日：1991-02-13

Applicant: BASF AG

Inventor： ZIERKE THOMAS DR ,  KUEKENHOEHNER THOMAS DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N43/40 ,  C07D213/30 ,  C07D213/42 ,  C07D213/57 ,  C07D213/89

Abstract: Compounds of the formula 1 1 where R is unsubstituted or substituted cycloalkyl or cycloalkenyl, X, Y and Z are hydrogen, halogen, alkyl, alkoxy, alkoximino, haloalkyl, cyano, nitro or unsubstituted or substituted phenyl or phenoxy, W is -CH2- or -CH2CH2- and n is 0 or 1, and the plant-tolerated acid-addition salts thereof, and fungicides containing these compounds are described.

公开(公告)号：DE4003919A1

公开(公告)日：1991-08-14

申请号：DE4003919

申请日：1990-02-09

Applicant: BASF AG

Inventor： ZIPPERER BERNHARD DR ,  LAUER MANFRED DR ,  GOETZ NORBERT DR ,  ZIERKE THOMAS DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N43/40 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  C07D213/30 ,  C07D213/50 ,  C07D401/06 ,  C07D405/06 ,  C07D407/06 ,  C07D409/06

Abstract: Heteroarylalkenes of the general formula I … …… … (Ar = heteroaryl, … A = C1-C6-alkyl, C2-C6-alkenyl, C3-C8-cycloalkyl, (C3-C8)-cycloalkyl-(C1-C3)-alkyl, mono-, di- or tricyclic substituted or unsubstituted aryl or aralkyl; … Z = … … where …… R = hydrogen, C2-C4-acyl, optionally substituted benzoyl, C1-C4-alkylsulphonyl, phenylsulphonyl which is unsubstituted or substituted by C1-C4-alkyl, or the radical R , … R is C1-C4-alkyl, substituted or unsubstituted phenyl or benzyl and … Hal is fluorine, chlorine, bromine or iodine; …… B is substituted or unsubstituted mono- or dicyclic aryl, aralkyl or heteroaryl) … and their N-oxides and acid addition salts; furthermore the preparation of these substances, intermediates therefor and their preparation, heteroarylalkene-containing fungicidal agents, and a suitable method for controlling fungal pests.

公开(公告)号：CZ288448B6

公开(公告)日：2001-06-13

申请号：CZ326096

申请日：1995-04-26

Applicant: BASF AG

Inventor： AMBERG WILHELM DR ,  BERNARD HARALD DR ,  BUSCHMANN ERNST DR ,  HAUPT ANDREAS DR ,  JANITSCHKE LOTHAR DR ,  MUELLER STEFAN DR ,  DE POTZOLLI BERND DR ,  RITTER KURT DR ,  THYES MARCO DR ,  ZIERKE THOMAS DR ,  JANSSEN BERND DR ,  KARL ULRICH DR ,  KLING ANDREAS DR

IPC: A61K38/00 ,  A61K38/08 ,  A61P35/00 ,  C07K1/08 ,  C07K5/10 ,  C07K5/103 ,  C07K7/06 ,  C07K14/52

Abstract: In the present invention, there is described pentapeptide hydrochloride of the formula Mei2Val-Val-MeVal-Pro-Pro-NHBz1.HCl, which is present in crystalline form. It is prepared from the compound of the formula Z-Val-Val-MeVal-Pro-ORe1, in which Z represents a benzyloxycarbonyl protecting group, which might be optionally substituted on the phenyl ring and Re1 represents alkyl containing 1 to 5 carbon atoms. In the present invention, there are also described intermediates for preparing the above indicated pentapeptide hydrochloride. The above-described compound exhibits antineoplastic activity.

公开(公告)号：CZ9800243A3

公开(公告)日：1998-07-15

申请号：CZ24398

申请日：1996-07-12

Applicant: BASF AG

Inventor： AMBERG WILHELM DR ,  BERNARD HARALD DR ,  BUSCHMANN ERNST DR ,  HAUPT ANDREAS DR ,  JANSSEN BERND DR ,  KARL ULRICH DR ,  KLING ANDREAS DR ,  MULLER STEFAN DR ,  RITTER KURT DR ,  ZIERKE THOMAS DR

IPC: C07K1/02 ,  C07K1/12 ,  C07K5/078 ,  C07K5/083 ,  C07K5/103 ,  C07K7/06 ,  C07K5/06 ,  C07K5/08 ,  C07K5/10

CPC classification number: C07K7/06 ,  C07K5/06165 ,  C07K5/0808 ,  C07K5/101

公开(公告)号：CZ8998A3

公开(公告)日：1998-06-17

申请号：CZ8998

申请日：1996-07-12

Applicant: BASF AG

Inventor： BUSCHMANN ERNST DR ,  ZIERKE THOMAS DR

IPC: C07C231/02 ,  C07C237/02 ,  C07K1/06 ,  C07K1/08 ,  C07K7/06

Abstract: PCT No. PCT/EP96/03075 Sec. 371 Date Jan. 20, 1998 Sec. 102(e) Date Jan. 20, 1998 PCT Filed Jul. 12, 1996 PCT Pub. No. WO97/05096 PCT Pub. Date Feb. 13, 1997A process for preparing alpha -(N,N-dialkylamino) carboxamides of the formula I where the substituents have the stated meanings, comprises reacting the corresponding free acids with primary or secondary amines in the presence of anhydrides of an alkanephosphonic acid.