公开(公告)号：CZ292229B6

公开(公告)日：2003-08-13

申请号：CZ8998

申请日：1996-07-12

Applicant: BASF AG

Inventor： BUSCHMANN ERNST DR ,  ZIERKE THOMAS DR

IPC: C07C231/02 ,  C07C237/02 ,  C07K1/06 ,  C07K1/08 ,  C07K7/06

Abstract: The present invention relates to a process for preparing {alpha}-(N,N-dialkylamino)-carboxamides of the general formula I, in which the symbols Re1 through Ri5 have specific meanings. The novel preparation process is characterized by bringing into reaction corresponding free acids with primary or secondary amines in the presence of alkanephosphonic acid anhydrides, whereby amino acid or peptide derivatives are used as the primary or secondary amines.

公开(公告)号：CZ9801846A3

公开(公告)日：1998-09-16

申请号：CZ184698

申请日：1996-12-11

Applicant: BASF AG

Inventor： AMBERG WILHELM DR ,  BARLOZZARI TERESA ,  BERNARD HARALD DR ,  BUSCHMANN ERNST DR ,  HAUPT ANDREAS DR ,  HEGE HANS-GUENTHER DR ,  JANSSEN BERND DR ,  KLING ANDREAS DR ,  LIETZ HELMUT ,  RITTER KURT DR ,  ULRICH MARTINA DR ,  WEYMANN JURGEN DR ,  ZIERKE THOMAS DR

IPC: A61K38/00 ,  A61K31/00 ,  A61K38/08 ,  A61P35/00 ,  A61P35/02 ,  C07K1/00 ,  C07K7/06

CPC classification number: A61K38/08

公开(公告)号：CZ9800089A3

公开(公告)日：1998-06-17

申请号：CZ8998

申请日：1996-07-12

Applicant: BASF AG

Inventor： BUSCHMANN ERNST DR ,  ZIERKE THOMAS DR

IPC: C07C231/02 ,  C07C237/02 ,  C07K1/06 ,  C07K1/08 ,  C07K7/06

CPC classification number: C07K7/06 ,  C07C231/02 ,  C07K1/082 ,  Y02P20/55

公开(公告)号：CZ245797A3

公开(公告)日：1998-06-17

申请号：CZ245797

申请日：1996-02-12

Applicant: BASF AG

Inventor： BOHM HANS-JOACHIM DR ,  HOFFKEN HANS WOLFGANG DR ,  HORNBERGER WILFRIED DR ,  KOSER STEFAN DR ,  MACK HELMUT DR ,  PFEIFFER THOMAS DR ,  SEITZ WERNER DR ,  ZIERKE THOMAS DR

IPC: A61K31/00 ,  A61K38/55 ,  A61P7/02 ,  C07D205/04 ,  C07D207/16 ,  C07D213/53 ,  C07D213/63 ,  C07D213/72 ,  C07D213/78 ,  C07D213/79 ,  C07D239/28 ,  C07D241/14 ,  C07D241/24 ,  C07D401/12 ,  C07K5/06 ,  C07K5/062 ,  C07K5/078 ,  A61K31/40 ,  A61K31/445 ,  A61K31/495

Abstract: The invention relates to a compound of the formula I: or a salt thereof with a physiologically tolerated acid, or stereoisomers thereof, wherein R 1 , R 2 , A, B, C and D have the meanings described in the specification.

公开(公告)号：CZ9702376A3

公开(公告)日：1998-04-15

申请号：CZ237697

申请日：1996-02-06

Applicant: BASF AG

Inventor： SEITZ WERNER DR ,  MACK HELMUT DR ,  ZIERKE THOMAS DR ,  BOHM HANS-JOACHIM DR ,  HOFFKEN HANS WOLFGANG DR ,  KOSER STEFAN DR ,  PFEIFFER THOMAS DR ,  HORNBERGER WILFRIED DR

IPC: A61K38/55 ,  A61K38/00 ,  A61P7/02 ,  C07K5/06 ,  C07K5/065 ,  C07K5/072 ,  C07K5/087

CPC classification number: C07K5/0812 ,  A61K38/00 ,  C07K5/06026 ,  C07K5/06034 ,  C07K5/0606 ,  C07K5/06078 ,  C07K5/06113 ,  C07K5/06191

公开(公告)号：CZ237697A3

公开(公告)日：1998-04-15

申请号：CZ237697

申请日：1996-02-06

Applicant: BASF AG

Inventor： SEITZ WERNER DR ,  MACK HELMUT DR ,  ZIERKE THOMAS DR ,  BOHM HANS-JOACHIM DR ,  HOFFKEN HANS WOLFGANG DR ,  KOSER STEFAN DR ,  PFEIFFER THOMAS DR ,  HORNBERGER WILFRIED DR

IPC: A61K38/55 ,  A61K38/00 ,  A61P7/02 ,  C07K5/06 ,  C07K5/065 ,  C07K5/072 ,  C07K5/087

Abstract: PCT No. PCT/EP96/00472 Sec. 371 Date Jul. 30, 1997 Sec. 102(e) Date Jul. 30, 1997 PCT Filed Feb. 6, 1996 PCT Pub. No. WO96/24609 PCT Pub. Date Aug. 15, 1996Thrombin inhibitors of the formula where R1, A, B and D have the meaning indicated in the description, and intermediates for the preparation thereof are described. The compounds I are suitable for controlling diseases.

公开(公告)号：ES2055465T3

公开(公告)日：1994-08-16

申请号：ES91101436

申请日：1991-02-04

Applicant: BASF AG

Inventor： ZIERKE THOMAS DR ,  KUEKENHOEHNER THOMAS DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N43/40 ,  C07D213/30 ,  C07D213/42 ,  C07D213/57 ,  C07D213/89

Abstract: Compounds of the formula 1 1 where R is unsubstituted or substituted cycloalkyl or cycloalkenyl, X, Y and Z are hydrogen, halogen, alkyl, alkoxy, alkoximino, haloalkyl, cyano, nitro or unsubstituted or substituted phenyl or phenoxy, W is -CH2- or -CH2CH2- and n is 0 or 1, and the plant-tolerated acid-addition salts thereof, and fungicides containing these compounds are described.

公开(公告)号：AT109143T

公开(公告)日：1994-08-15

申请号：AT91106178

申请日：1991-04-18

Applicant: BASF AG

Inventor： ZIERKE THOMAS DR ,  KUEKENHOEHNER THOMAS DR ,  FRANK JUERGEN DR ,  AMMERMANN EBERHARD DR ,  LORENZ GISELA DR

IPC: A01N43/80 ,  A61K31/42 ,  A61P31/04 ,  C07D249/08 ,  C07D413/06 ,  C07D413/14 ,  C07D521/00

Abstract: 5-(1,2,4-Triazol-1-yl-methyl)-isoxazolines I I where R1 and R2 are each H, alkoxyalkyl, haloalkyl, alkyl, cycloalkylalkyl, phenylalkyl, naphthylalkyl, cycloalkyl, phenyl, naphthyl or hetaryl, where the aryl and hetaryl moieties of the stated substituents may furthermore carry an unsubstituted or halogen-substituted phenyl or phenoxy radical or up to 3 of the following radicals: halogen, CN, NO2, alkyl, haloalkyl or alkoxy, and the salts and metal complexes of I are suitable as fungicides and for regulating plant growth.

公开(公告)号：ES2054165T3

公开(公告)日：1994-08-01

申请号：ES90113144

申请日：1990-07-10

Applicant: BASF AG

Inventor： KOBER REINER DR ,  SEELE RAINER DR ,  ISAK HEINZ DR ,  HICKMANN ECKHARD DR ,  GOETZ NORBERT DR ,  ZIERKE THOMAS DR

IPC: C07B53/00 ,  C07C17/00 ,  C07C17/35 ,  C07C17/357 ,  C07C22/04 ,  C07C25/24 ,  C07C41/18 ,  C07C41/48 ,  C07C43/225 ,  C07C43/29 ,  C07D233/56 ,  C07D233/58 ,  C07D249/08 ,  C07D301/16 ,  C07D303/08 ,  C07D405/06 ,  C07D521/00

Abstract: Preparation of Z-1,2-diarylallyl chlorides of the general formula I in which the radicals R and R independently of one another are hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or a substituted aromatic radical, and n and m represent 1, 2 or 3, by dehydrating chlorohydrins of the formula II in which the radicals have the abovementioned meanings, at temperatures of up to 50 DEG C in the presence of a carboxylic anhydride and of an organic or inorganic acid, in an inert ether or carboxylate as the solvent, the reaction of these products to give azolylmethyloxiranes, and novel intermediates.

公开(公告)号：DE59006126D1

公开(公告)日：1994-07-21

申请号：DE59006126

申请日：1990-09-24

Applicant: BASF AG

Inventor： SAUTER HUBERT DR ,  ZIERKE THOMAS DR ,  REUTHER WOLFGANG DR ,  BAUS ULF DR ,  LORENZ GISELA DR ,  AMMERMANN EBERHARD DR

IPC: A01N43/653 ,  C07D249/08 ,  C07D401/12 ,  C07D403/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  C07D521/00

Abstract: Compounds of the formula I I where Ar is unsubstituted or substituted phenyl, pyridyl, thienyl or napthyl, R1 is hydrogen or CN, R2 is unsubstituted or substituted aryl, hetaryl, alkyl or cycloalkyl, or is unsubstituted or substituted alkenyl or alkynyl, x is CH2, O or S and n is 0 or 1, their plant-tolerated acid addition salts and metal complexes, and fungicides and growth regulators containing these compounds.