公开(公告)号：ES2104794T3

公开(公告)日：1997-10-16

申请号：ES92119064

申请日：1992-11-06

Applicant: BASF AG

Inventor： MUELLER STEFAN DR ,  THEOBALD HANS DR ,  RANG HARALD DR ,  HARRIES VOLKER DR

IPC: A01N55/00 ,  A01N55/10 ,  C07F7/08 ,  C07F7/10

Abstract: 3-isoxazolylphenyl compounds Ia and Ib, … … in which the substituents and the index have the following meaning: …… R represents halogen; alkyl; haloalkyl; alkoxy; haloalkoxy; alkenyl; haloalkenyl; optionally substituted phenylethenyl; alkynyl; cycloalkyl; aryl, hetaryl; CO2R or CONR R , … (R = hydrogen, alkyl, cycloalkyl and benzyl; R and R = hydrogen, alkyl, cycloalkyl and benzyl, or all together with the nitrogen atom to which they are bonded a heterocyclic radical), … n represents O, 1 or 2; … R represents halogen or alkyl; … R represents hydrogen; alkyl; alkenyl; alkynyl or cyano; … R and R independently of one another represent optionally substituted alkyl, alkenyl, cycloalkyl, phenyl, naphthyl, pyridyl or pyrimidyl; … or R and R together represent optionally substituted alkylene; … R represents hydrogen; … optionally substituted alkyl, or one of the groups mentioned in R ; … X represents a group CH2, O, S or NR … (R = hydrogen, alkyl, cycloalkyl, alkenyl, alkynyl or optionally substituted benzyl), … their preparation, compositions comprising them, and their use.

公开(公告)号：DE4027572A1

公开(公告)日：1992-03-05

申请号：DE4027572

申请日：1990-08-31

Applicant: BASF AG

Inventor： MUELLER STEFAN DR ,  WOLF BERND DR ,  THEOBALD HANS DR ,  HARREUS ALBRECHT DR ,  KARDORFF UWE DR ,  KUENAST CHRISTOPH DR

IPC: A01N53/00 ,  A01N53/04 ,  C07D307/79

Abstract: 2,3-Dihydrobenzofurylmethyl esters of the general formula I in which the substituents and index have the following meanings: R is hydrogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl or cyano; R and R are independently of one another hydrogen or C1-C4-alkyl and n is 0 or 1, their preparation, and pesticides containing them.>

公开(公告)号：DE4417478A1

公开(公告)日：1995-11-23

申请号：DE4417478

申请日：1994-05-19

Applicant: BASF AG

Inventor： KARL ULRICH DR ,  MUELLER STEFAN DR ,  POTZOLLI BERND DE DR

IPC: C07B61/00 ,  C07C227/18 ,  C07C229/12 ,  C07C269/06 ,  C07C271/22 ,  C07C323/59 ,  C07C269/04 ,  C07B51/00 ,  C07C291/02

Abstract: A process for producing N-protected N-alkylated amino acids of formula (I) is described in which the components have the meaning given in the description. In the process, to a compound of formula (II) is added a solution of potassium-tert.-butanolate in a non-proteinic organic solvent and then a C1-2-alkyl halide is added.

公开(公告)号：DE4016049A1

公开(公告)日：1991-11-21

申请号：DE4016049

申请日：1990-05-18

Applicant: BASF AG

Inventor： MUELLER STEFAN DR ,  THEOBALD HANS DR ,  WOLF BERND DR ,  HOFMEISTER PETER DR ,  KARDORFF UWE DR ,  KUENAST CHRISTOPH DR

IPC: A01N43/72 ,  A01N43/80 ,  A01N53/00 ,  A01N53/06 ,  C07D261/08 ,  C07D261/10 ,  C07D261/12 ,  C07D261/18 ,  C07D413/12

Abstract: 3-Isoxazolylbenzyl esters of the general formulae Ia and Ib Ia Ib where R is halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C2--C4-alkenyl, C2-C4-haloalkenyl, C2-C4-alkynyl, C2-C4-haloalkynyl, unsubstituted or substituted phenylethenyl, C3-C8-cycloalkyl, aryl, hetaryl, CO2R3 or CONR4R5, R3, R4 and R5 are each hydrogen or C1-C6-alkyl, n is 0, 1 or 2, and the radicals R may be different when n is 2, R1 is halogen or C1-C4-alkyl, R2 is hydrogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl or cyano and A is the carbonyl radical of an acid component usually found in pyrethroids, are contained in pesticides.

公开(公告)号：DE59208576D1

公开(公告)日：1997-07-10

申请号：DE59208576

申请日：1992-11-06

Applicant: BASF AG

Inventor： MUELLER STEFAN DR ,  THEOBALD HANS DR ,  RANG HARALD DR ,  HARRIES VOLKER DR

IPC: A01N55/00 ,  A01N55/10 ,  C07F7/08 ,  C07F7/10

Abstract: 3-isoxazolylphenyl compounds Ia and Ib, … … in which the substituents and the index have the following meaning: …… R represents halogen; alkyl; haloalkyl; alkoxy; haloalkoxy; alkenyl; haloalkenyl; optionally substituted phenylethenyl; alkynyl; cycloalkyl; aryl, hetaryl; CO2R or CONR R , … (R = hydrogen, alkyl, cycloalkyl and benzyl; R and R = hydrogen, alkyl, cycloalkyl and benzyl, or all together with the nitrogen atom to which they are bonded a heterocyclic radical), … n represents O, 1 or 2; … R represents halogen or alkyl; … R represents hydrogen; alkyl; alkenyl; alkynyl or cyano; … R and R independently of one another represent optionally substituted alkyl, alkenyl, cycloalkyl, phenyl, naphthyl, pyridyl or pyrimidyl; … or R and R together represent optionally substituted alkylene; … R represents hydrogen; … optionally substituted alkyl, or one of the groups mentioned in R ; … X represents a group CH2, O, S or NR … (R = hydrogen, alkyl, cycloalkyl, alkenyl, alkynyl or optionally substituted benzyl), … their preparation, compositions comprising them, and their use.

公开(公告)号：DE4337331A1

公开(公告)日：1995-05-04

申请号：DE4337331

申请日：1993-11-02

Applicant: BASF AG

Inventor： KARL ULRICH DR ,  MUELLER STEFAN DR ,  POTZOLLI BERND DE DR ,  KNUEHL KLAUS

IPC: C07C269/06 ,  C07C271/22 ,  C07C323/52 ,  C07C229/12 ,  C07C229/36 ,  C07C229/22 ,  C07C227/18

Abstract: PCT No. PCT/EP94/03480 Sec. 371 Date Sep. 6, 1995 Sec. 102(e) Date Sep. 6, 1995 PCT Filed Oct. 22, 1994 PCT Pub. No. WO95/12574 PCT Pub. Date May 11, 1995A process for preparing N-protected N-alkylated amino acids of the formula where Rs and R1-R3 have the meanings indicated in the description comprises adding a compound of the abovementioned formula where R3 is hydrogen to a solution of a base in a non-protic solvent and subsequently adding an alkylating agent.

公开(公告)号：ES2067083T3

公开(公告)日：1995-03-16

申请号：ES91107586

申请日：1991-05-10

Applicant: BASF AG

Inventor： MUELLER STEFAN DR ,  THEOBALD HANS DR ,  WOLF BERND DR ,  HOFMEISTER PETER DR ,  KARDORFF UWE DR ,  KUENAST CHRISTOPH DR

IPC: A01N43/72 ,  A01N43/80 ,  A01N53/00 ,  A01N53/06 ,  C07D261/08 ,  C07D261/10 ,  C07D261/12 ,  C07D261/18 ,  C07D413/12

Abstract: 3-Isoxazolylbenzyl esters of the general formulae Ia and Ib Ia Ib where R is halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C2--C4-alkenyl, C2-C4-haloalkenyl, C2-C4-alkynyl, C2-C4-haloalkynyl, unsubstituted or substituted phenylethenyl, C3-C8-cycloalkyl, aryl, hetaryl, CO2R3 or CONR4R5, R3, R4 and R5 are each hydrogen or C1-C6-alkyl, n is 0, 1 or 2, and the radicals R may be different when n is 2, R1 is halogen or C1-C4-alkyl, R2 is hydrogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl or cyano and A is the carbonyl radical of an acid component usually found in pyrethroids, are contained in pesticides.

公开(公告)号：DE4415998A1

公开(公告)日：1995-11-09

申请号：DE4415998

申请日：1994-05-06

Applicant: BASF AG

Inventor： AMBERG WILHELM DR ,  BERNARD HARALD DR ,  BUSCHMANN ERNST DR ,  HAUPT ANDREAS DR ,  JANITSCHKE LOTHAR DR ,  JANSSEN BERND DR ,  KARL ULRICH DR ,  KLING ANDREAS DR ,  MUELLER STEFAN DR ,  POTZOLLI BERND DE DR ,  RITTER KURT DR ,  ZIERKE THOMAS DR ,  THYES MARCO DR

IPC: A61K38/00 ,  A61P35/00 ,  C07K5/10 ,  C07K5/103 ,  C07K7/06

Abstract: Compounds of formula (I) are disclosed, wherein R , R , R , and R have the meanings indicated in the description, as well as a process for the production of these compounds. The compounds are suitable for use as starting material for the synthesis of substances which have anti-tumour properties.

公开(公告)号：DE4415997A1

公开(公告)日：1995-11-09

申请号：DE4415997

申请日：1994-05-06

Applicant: BASF AG

Inventor： AMBERG WILHELM DR ,  BERNARD HARALD DR ,  BUSCHMANN ERNST DR ,  HAUPT ANDREAS DR ,  JANITSCHKE LOTHAR DR ,  JANSSEN BERND DR ,  KARL ULRICH DR ,  KLING ANDREAS DR ,  MUELLER STEFAN DR ,  POTZOLLI BERND DE DR ,  RITTER KURT DR ,  ZIERKE THOMAS DR ,  THYES MARCO DR

IPC: A61K38/00 ,  A61K38/08 ,  A61P35/00 ,  C07K1/08 ,  C07K5/10 ,  C07K5/103 ,  C07K7/06 ,  C07K14/52

Abstract: Disclosed is the compound Me2Val-Val-MeVal-Pro-Pro-NHBzl. HCl. The compound is produced from Z-Val-Val-MeVal-Pro-OR , wherein Z and R have the meanings indicated in the description. The compound disclosed has anti-neoplastic properties.

公开(公告)号：AT115141T

公开(公告)日：1994-12-15

申请号：AT91107586

申请日：1991-05-10

Applicant: BASF AG

Inventor： MUELLER STEFAN DR ,  THEOBALD HANS DR ,  WOLF BERND DR ,  HOFMEISTER PETER DR ,  KARDORFF UWE DR ,  KUENAST CHRISTOPH DR

IPC: A01N43/72 ,  A01N43/80 ,  A01N53/00 ,  A01N53/06 ,  C07D261/08 ,  C07D261/10 ,  C07D261/12 ,  C07D261/18 ,  C07D413/12

Abstract: 3-Isoxazolylbenzyl esters of the general formulae Ia and Ib Ia Ib where R is halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C2--C4-alkenyl, C2-C4-haloalkenyl, C2-C4-alkynyl, C2-C4-haloalkynyl, unsubstituted or substituted phenylethenyl, C3-C8-cycloalkyl, aryl, hetaryl, CO2R3 or CONR4R5, R3, R4 and R5 are each hydrogen or C1-C6-alkyl, n is 0, 1 or 2, and the radicals R may be different when n is 2, R1 is halogen or C1-C4-alkyl, R2 is hydrogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl or cyano and A is the carbonyl radical of an acid component usually found in pyrethroids, are contained in pesticides.