公开(公告)号：PT85000B

公开(公告)日：1990-03-08

申请号：PT8500087

申请日：1987-06-03

Applicant: HOECHST AG

Inventor： GIENCKE WOLFGANG ,  SACHSE BURKHARD ,  MILDENBERGER HILMAR ,  KNAUF WERNER ,  KERN MANFRED ,  WALTERSDORFER ANNA ,  HEUBACH GUNTHER ,  FUSS ANDREAS

IPC: A01N43/54 ,  C07D239/34 ,  C07D239/42 ,  C07D239/46 ,  C07D239/26

公开(公告)号：PH24050A

公开(公告)日：1990-03-05

申请号：PH34277

申请日：1986-09-22

Applicant: HOECHST AG

Inventor： SIEGEL HERBERT ,  GERHARDS HERMANN JOSEF ,  SCHACHT ULRICH ,  DITTMAR WALTER ,  KAMPE KLAUS-DIETER ,  USINGER PATRICIA ,  LEVEN MARGARET ,  RAETHER WOLFGANG ,  SACHSE BURKHARD ,  ALPERMANN HANS GEORG

IPC: A61K31/41 ,  A61K31/415 ,  C07D233/60 ,  C07D233/64 ,  C07D249/08 ,  C07D521/00

Abstract: Arylmethylazoles of the formula I I in which Aryl is (substituted) phenyl or naphthyl; Z is CH or N; R1 and Q are H or alkyl; R2 is H, alk(en)yl or alkynyl; R3 and R4 are H, alkyl or other hydrocarbons; or R3 and R4 together are a -(CH2)2-11 chain or a bridged -(CH2)4-5 chain, and their acid addition salts, stereoisomers and optically active enantiomers possess outstanding antimycotic and antidepressant activity. They are obtained, inter alia, from arylmethylazoles II II which are reacted with a strong base and then with a carbonyl compound III O=CR3R4; thereafter, the product is reacted with the protic acid or with an alkyl halide IV R2Hal. If desired, the products are converted to the acid addition salts, or the stereoisomers or optically active enantiomers are resolved.

公开(公告)号：PT89542A

公开(公告)日：1989-10-04

申请号：PT8954289

申请日：1989-01-26

Applicant: HOECHST AG

Inventor： SACHSE BURKHARD ,  WICKE HEINRICH ,  SCHMIDT ERNST ,  KNAUF WERNER ,  KERN MANFRED ,  WALTERSDORFER ANNA ,  MATTERSTOCK KARL ,  SCHUCK ERNST

IPC: A01N33/26 ,  A01N37/22 ,  A01N37/24 ,  A01N37/28 ,  A01N37/30 ,  A01N37/34 ,  A01N37/40 ,  A01N37/42 ,  A01N37/44 ,  A01N37/46 ,  A01N37/48 ,  A01N37/52 ,  A01N47/48 ,  C07C67/00 ,  C07C233/66 ,  C07C233/75 ,  C07C233/81 ,  C07C235/56 ,  C07C235/64 ,  C07C235/84 ,  C07C241/00 ,  C07C243/38 ,  C07C253/30 ,  C07C255/57 ,  C07C255/60 ,  C07C259/18 ,  C07C313/28 ,  C07C313/36 ,  C07C319/20 ,  C07C323/62 ,  C07C327/48 ,  C07C327/56 ,  C07C331/08 ,  C07C331/14 ,  C07C103/00 ,  C07C143/00 ,  A01N37/00 ,  A01N47/00

Abstract: Compounds of the general formula I in which X represents O, S or NOR , R represents hydrogen, halogen, CN, SCN, NO2, OH, carbamoyl, alkyl, alkoxy, thioalkyl, it being possible for these to be entirely or partly substituted by halogen, or represents phenyl, thiophenyl or phenoxy, it being possible for these to be substituted by 1 or 2 halogen atoms or a CF3 group, or represents acyl, R represents hydrogen, alkyl, alkenyl, alkynyl, it being possible for these to be entirely or partly substituted by halogen, or represents acyl or cyanomethyl, R represents hydrogen, alkyl or S-CCl3, R and R in each case independently of one another represent NO2, halogen, CN, COOH, CONH2, alkyl or alkoxy, it being possible for these to be entirely or partly substituted by halogen, or represent alkoxycarbonyl or CONR R , R represents hydrogen or halogen, R represents hydrogen, halogen, alkoxy or phenoxy, R and R represent alkyl, m represents 0 or 1 and n represents 0-5, with the proviso that in the event where X = NOR m must be 0, and the salts thereof which can be used in agriculture, have advantageous insecticidal, acaricidal, fungicidal or nematocidal properties. There are furthermore described processes for the preparation of the compounds of the formula I.

公开(公告)号：DD269398A5

公开(公告)日：1989-06-28

申请号：DD31101387

申请日：1987-12-22

Applicant: HOECHST AG

Inventor： HAMMANN PETER ,  GRABLEY SUSANNE ,  VOELSKOW HARTMUT ,  SACHSE BURKHARD ,  RAETHER WOLFGANG ,  GIANI CARLO ,  SEIBERT GERHARD

IPC: C12P17/08 ,  A01N63/02 ,  A61K20060101 ,  A61K31/365 ,  A61P31/00 ,  A61P31/10 ,  C07D313/00 ,  C07D493/04 ,  C07D493/08 ,  C12N20060101 ,  C12P20060101 ,  C12P1/02 ,  C12P17/18 ,  C12R1/465

公开(公告)号：DD268852A5

公开(公告)日：1989-06-14

申请号：DD30063287

申请日：1987-03-10

Applicant: HOECHST AG

Inventor： SCHAPER WOLFGANG ,  FUSS ANDREAS ,  RAETHER WOLFGANG ,  DITTMAR WALTER ,  HAENEL HEINZ ,  GERHARDS HERMAN J ,  SACHSE BURKHARD

IPC: A61K31/415 ,  A01N43/50 ,  A01N43/653 ,  A61P25/08 ,  A61P31/04 ,  A61P31/10 ,  A61P33/02 ,  C07D233/56 ,  C07D233/58 ,  C07D233/60 ,  C07D233/61 ,  C07D247/00 ,  C07D249/08 ,  C07D335/00 ,  C07D405/06 ,  C07D409/06 ,  C07D521/00 ,  A01N43/18 ,  A01N43/16 ,  A01N43/10 ,  A01N31/14 ,  A01N27/00

Abstract: Azole compounds of the formula (I) in which A denotes CH or N, n = 1, 2 or 3, k = 1 or 2, Ar denotes a (subst.) aromatic radical or (subst.) thienyl, W denotes the atoms necessary to complete a benzene, naphthalene or thiophene ring system, X denotes a radical C(R )2 and in the case in which W denotes the atoms necessary to complete a benzene or naphthalene ring system, also denotes oxygen or sulphur, R and R denote H, halogen, (subst.) alkyl, cycloalkyl, alkoxy, alkylthio, cyano or nitro, and in the case in which W simultaneously denotes the atoms necessary to complete a benzene ring, R also denotes phenyl, phenoxy, phenylthio, phenylsulfinyl, phenylsulphonyl, benzyl, benzyloxy or hydroxyl, where the phenyl groups can be substituted or R and R together, if they are o-orientated, denote an alkylene chain; R denotes H or alkyl or two radicals R together, if they are bonded to the same C-atom, denote an alkylene chain, and their stereoisomers and salts have advantageous fungicidal, antimycotic and anticonvulsive effects.

公开(公告)号：DK684987A

公开(公告)日：1988-06-25

申请号：DK684987

申请日：1987-12-23

Applicant: HOECHST AG

Inventor： HAMMANN PETER ,  GRABLEY SUSANNE ,  VOELSKOW HARTMUT ,  SACHSE BURKHARD ,  RAETHER WOLFGANG ,  GIANI CARLO ,  SEIBERT GERHARD

IPC: C12P17/08 ,  A01N47/44 ,  A01N63/02 ,  A61K20060101 ,  A61K31/365 ,  A61P31/00 ,  A61P31/10 ,  C07D313/00 ,  C07D493/04 ,  C07D493/08 ,  C12N20060101 ,  C12P20060101 ,  C12P1/02 ,  C12P1/06 ,  C12P17/16 ,  C12P17/18 ,  C12R1/465 ,  C07H19/01 ,  C12N1/20 ,  C12P19/02

Abstract: Streptomyces parvullus, DSM 3816, produces on aerobic fermentation new antibiotics which are distinguished by antimicrobial activity even after derivatization.

公开(公告)号：ZA873879B

公开(公告)日：1988-02-24

申请号：ZA873879

申请日：1987-05-29

Applicant: HOECHST AG

Inventor： GIENCKE WOLFGANG ,  WOLFGANG GIENCKE ,  MILDENBERGER HILMAR ,  HILMAR MILDENBERGER ,  HEUBACH GUENTHER ,  GUENTHER HEUBACH ,  SACHSE BURKHARD ,  BURKHARD SACHSE ,  FUSS ANDREAS ,  ANDREAS FUSS ,  WALTERSDORFER ANNA ,  ANNA WALTERSDORFER ,  KNAUF WERNER ,  WERNER KNAUF ,  KERN MANFRED ,  MANFRED KERN ,  BONIN WERNER ,  WERNER BONIN

IPC: A01N43/54 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48 ,  A01N ,  C07D

公开(公告)号：DD253755A5

公开(公告)日：1988-02-03

申请号：DD28930886

申请日：1986-04-17

Applicant: HOECHST AG

Inventor： SCHMIERER ROLAND ,  MILDENBERGER HILMAR ,  HANDTE REINHARD ,  BUERSTELL HELMUT ,  SACHSE BURKHARD ,  BAUER KLAUS ,  BIERINGER HERMANN

IPC: C07D413/04 ,  A01N43/50 ,  A01N43/82 ,  A01N43/836 ,  A01N55/10 ,  A01N57/24 ,  C07D233/54 ,  C07D233/64 ,  C07D233/66 ,  C07D233/90 ,  C07D403/04 ,  C07D403/06 ,  C07D403/12 ,  C07D521/00 ,  A01N37/00 ,  A01N43/84 ,  A01N43/40 ,  A01N43/76 ,  A01N43/653

Abstract: The new compounds of the formula I or salts thereof I in which R denotes a (substituted) cyclohexyl radical or a (substituted) cyclohexenyl radical; and Y denotes cyano, a (substituted) (di)(thio)carboxylic acid (ester), carboxamide or acetal radical, a keto or oxime radical or a heterocyclic radical, possess an advantageous action as plant growth-regulators and, in addition, have favorable herbicidal and fungicidal properties.

公开(公告)号：DK633287D0

公开(公告)日：1987-12-02

申请号：DK633287

申请日：1987-12-02

Applicant: HOECHST AG

Inventor： EHRHARDT HEINZ ,  MILDENBERGER HILMAR ,  MAIER THOMAS ,  SCHALLER RAINER ,  SACHSE BURKHARD ,  BRAUN PETER

IPC: A01N47/38 ,  A61K31/415 ,  A61K31/4427 ,  C07D401/04 ,  A61K31/443 ,  A61K31/445 ,  A61P31/04 ,  C07D401/14 ,  C07D405/14 ,  C07D521/00 ,  C07D401/06

Abstract: Compounds of the formula (I) (I) in which n denotes a number from 2 to 6, m denotes 1 or 2, R denotes +TR CH2CH2CH2OR1, R1 denotes (substituted) alkyl, (substituted) alkenyl, C3-alkynyl, cycloalkyl, cycloalkenyl or an aromatic or heteroaromatic radical, R2 denotes H or alkyl and Y denotes H, alkyl, phenyl or halophenyl, and the metal-salt complexes thereof have advantageous fungicidal actions and are highly suitable for use in plant protection or in the industrial sector.

公开(公告)号：DK275087A

公开(公告)日：1987-12-01

申请号：DK275087

申请日：1987-05-29

Applicant: HOECHST AG

Inventor： GIENCKE WOLFGANG ,  MILDENBERGER HILMAR ,  HEUBACH GUENTHER ,  SACHSE BURKHARD ,  FUSS ANDREAS ,  WALTERSDORFER ANNA ,  KNAUF WERNER ,  KERN MANFRED ,  BONIN WERNER

IPC: A01N43/54 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48