公开(公告)号：AT146475T

公开(公告)日：1997-01-15

申请号：AT91111462

申请日：1991-07-10

Applicant: BASF AG

Inventor： MUENSTER PETER DR ,  FREUND WOLFGANG DR ,  STEINER GERD DR ,  WALTER HELMUT DR ,  WESTPHALEN KARL-OTTO DR ,  GERBER MATTHIAS DR

IPC: A01N43/36 ,  A01N43/90 ,  C07D307/68 ,  C07D333/38 ,  C07D333/40 ,  C07D409/04 ,  C07D409/12 ,  C07D491/04 ,  C07D491/048 ,  C07D495/04 ,  C07D333/00 ,  C07D209/00 ,  C07D307/00

Abstract: Dicarboximides of the general formula Ia and Ib ulfur, R1 is hydrogen, cycloalkyl, alkyl, hydroxyl, alkoxy, cyanoalkyl, alkenyl, alkynyl, phenyl, naphthyl or a 5-membered or 6-membered heterocyclic structure, where the stated radicals may be substituted, and R2 and R3 are each nitro, cyano, halogen, amino, mono- or dialkylamino, alkylcarbonylamino, unsubstituted or halogen-substituted alkoxy or alkylthio, alkylsulfonyl, haloalkylsulfonyl, alkenyl, alkynyl, phenyl, phenoxy or phenylthio or one of the radicals R1, with the proviso that specific compounds named in the description are excluded. Processes for the preparation of the compounds Ia and Ib and herbicides containing them.

公开(公告)号：CZ323794A3

公开(公告)日：1995-05-17

申请号：CZ323794

申请日：1993-06-08

Applicant: BASF AG

Inventor： STEINER GERD DR ,  UNGER LILIANE DR ,  BEHL BERTHOLD DR ,  TESCHENDORF HANS-JUERGEN DR ,  MUNSCHAUER RAINER DR

IPC: C07D513/04 ,  A61K20060101 ,  A61K31/33 ,  A61K31/395 ,  A61K31/40 ,  A61K31/4045 ,  A61K31/4184 ,  A61K31/505 ,  A61K31/506 ,  A61K31/513 ,  A61K31/517 ,  A61K31/519 ,  A61K31/54 ,  A61K31/542 ,  A61P25/00 ,  A61P25/20 ,  A61P25/22 ,  A61P25/24 ,  A61P43/00 ,  C07D20060101 ,  C07D207/00 ,  C07D209/02 ,  C07D209/52 ,  C07D221/00 ,  C07D239/00 ,  C07D401/04 ,  C07D401/06 ,  C07D401/14 ,  C07D403/00 ,  C07D403/04 ,  C07D403/06 ,  C07D403/14 ,  C07D409/04 ,  C07D409/06 ,  C07D409/14 ,  C07D417/14 ,  C07D471/04 ,  C07D487/04 ,  C07D495/04

Abstract: PCT No. PCT/EP93/01438 Sec. 371 Date Dec. 16, 1994 Sec. 102(e) Date Dec. 16, 1994 PCT Filed Jun. 8, 1993 PCT Pub. No. WO94/00458 PCT Pub. Date Jan. 6, 1994.Abstract of the Disclosure: Compounds of the formula I I where R1, R2, n , R3, A, X, Y and Z have the meanings stated in the description, and the preparation thereof are described. The novel compounds are suitable for controlling diseases , i.e., as neuroleptics, antidepressants, sedatives, hypnotics, CNS protectives or muscle relaxants.

公开(公告)号：DE4112353A1

公开(公告)日：1992-10-22

申请号：DE4112353

申请日：1991-04-16

Applicant: BASF AG

Inventor： STEINER GERD DR ,  UNGER LILIANE DR ,  HOFMANN HANS PETER DR ,  TESCHENDORF HANS-JUERGEN DR ME ,  BEHL BERTHOLD DR ,  BINDER RUDOLF DR

IPC: A61K31/445 ,  A61K31/4433 ,  A61K31/451 ,  A61P25/20 ,  A61P25/24 ,  A61P25/26 ,  C07D211/22 ,  C07D211/46 ,  C07D211/48 ,  C07D211/52 ,  C07D211/70 ,  C07D409/04

Abstract: The description relates to compounds of formula (I) in which A-B-D, R , R , R and n have the meanings given in the specification, and their production. The compounds are suitable for the treatment of diseases.

公开(公告)号：DE4023048A1

公开(公告)日：1992-01-23

申请号：DE4023048

申请日：1990-07-20

Applicant: BASF AG

Inventor： MUENSTER PETER DR ,  FREUND WOLFGANG DR ,  STEINER GERD DR ,  WALTER HELMUT DR ,  WESTPHALEN KARL-OTTO DR ,  GERBER MATTHIAS DR

IPC: A01N43/36 ,  A01N43/90 ,  C07D307/68 ,  C07D333/38 ,  C07D333/40 ,  C07D409/04 ,  C07D409/12 ,  C07D491/04 ,  C07D491/048 ,  C07D495/04

Abstract: Dicarboximides of the general formula Ia and Ib ulfur, R1 is hydrogen, cycloalkyl, alkyl, hydroxyl, alkoxy, cyanoalkyl, alkenyl, alkynyl, phenyl, naphthyl or a 5-membered or 6-membered heterocyclic structure, where the stated radicals may be substituted, and R2 and R3 are each nitro, cyano, halogen, amino, mono- or dialkylamino, alkylcarbonylamino, unsubstituted or halogen-substituted alkoxy or alkylthio, alkylsulfonyl, haloalkylsulfonyl, alkenyl, alkynyl, phenyl, phenoxy or phenylthio or one of the radicals R1, with the proviso that specific compounds named in the description are excluded. Processes for the preparation of the compounds Ia and Ib and herbicides containing them.

公开(公告)号：DE3717395A1

公开(公告)日：1988-12-08

申请号：DE3717395

申请日：1987-05-23

Applicant: BASF AG

Inventor： STEINER GERD DR ,  HIMMELE WALTER DR ,  BUSCHMANN ERNST DR ,  TESCHENDORF HANS-JUERGEN DR ME ,  WEIFENBACH HARALD DR

IPC: A61K31/40 ,  A61K31/403 ,  A61P25/08 ,  A61P25/18 ,  A61P25/20 ,  A61P25/24 ,  A61P25/26 ,  C07D209/60

Abstract: A 5-phenyl-1,3,3a,4,5,9b-hexahydro-3H-benz(e)indole compound of the formula I: I wherein R1 is hydrogen or C1-6 alkyl, R2 is hydrogen or C1-3 alkyl in the 3a- or 4-position, R3 and R4 are each hydrogen, hydroxyl, halogen, C1-3 alkyl, C1-3 alkoxy, C1-3 alkylthio or trifluoromethyl, acetylamino or amino and R5 is hydrogen or C1-3 alkyl, or a salt thereof with a physiologically tolerated acid. The compounds and compositions are useful for treating depression or trating convulsions and which exhibit a sedative and tranquilizing effect when administered to a patient.

公开(公告)号：DE3717394A1

公开(公告)日：1988-12-01

申请号：DE3717394

申请日：1987-05-23

Applicant: BASF AG

Inventor： HIMMELE WALTER DR ,  STEINER GERD DR ,  TESCHENDORF HANS-JUERGEN DR ME ,  WEIFENBACH HARALD DR

IPC: A61K31/40 ,  A61P25/20 ,  C07D207/06 ,  C07D207/08

公开(公告)号：DE3524743A1

公开(公告)日：1987-01-15

申请号：DE3524743

申请日：1985-07-11

Applicant: BASF AG

Inventor： STEINER GERD DR ,  THYES MARCO DR

IPC: C07D333/00 ,  C07D409/14 ,  C07D495/14 ,  C07D495/12

公开(公告)号：AT20349T

公开(公告)日：1986-06-15

申请号：AT83111277

申请日：1983-11-11

Applicant: BASF AG

Inventor： FRANKE ALBRECHT DR ,  STEINER GERD DR ,  HOFMANN HANS-PETER DR ,  MUELLER CLAUS-DIETER DR ,  TESCHENDORF HANS-JUERGEN DR

IPC: A61K31/40 ,  A61K31/403 ,  A61K31/4035 ,  A61K31/425 ,  A61K31/428 ,  A61P25/20 ,  A61P25/24 ,  A61P25/26 ,  C07D209/46 ,  C07D209/48 ,  C07D275/04 ,  C07D275/06 ,  C07D495/04 ,  C07D513/04

公开(公告)号：AT16384T

公开(公告)日：1985-11-15

申请号：AT81110718

申请日：1981-12-23

Applicant: BASF AG

Inventor： FRANKE ALBRECHT DR ,  STEINER GERD DR ,  THIEME PETER C DR ,  LENKE DIETER DR ,  GRIES JOSEF DR ,  TESCHENDORF HANS-JUERGEN DR

IPC: C07D249/08 ,  A61K31/41 ,  A61K31/415 ,  A61K31/42 ,  A61K31/495 ,  A61K31/496 ,  A61K31/505 ,  A61P9/02 ,  A61P11/08 ,  A61P25/08 ,  A61P25/20 ,  C07D231/12 ,  C07D231/38 ,  C07D233/60 ,  C07D233/88 ,  C07D239/42 ,  C07D261/08 ,  C07D295/06 ,  C07D295/092 ,  C07D521/00

公开(公告)号：GR75401B

公开(公告)日：1984-07-13

申请号：GR810166900

申请日：1981-12-23

Applicant: BASF AG

Inventor： FRANKE ALBRECHT DR ,  STEINER GERD DR ,  THIEME PETER C DR ,  LENKE DIETER DR ,  GRIES JOSEF DR ,  TESCHENDORF HANS-JUERGEN DR

IPC: C07D249/08 ,  A61K31/41 ,  A61K31/415 ,  A61K31/42 ,  A61K31/495 ,  A61K31/496 ,  A61K31/505 ,  A61P9/02 ,  A61P11/08 ,  A61P25/08 ,  A61P25/20 ,  C07D231/12 ,  C07D231/38 ,  C07D233/60 ,  C07D233/88 ,  C07D239/42 ,  C07D261/08 ,  C07D295/06 ,  C07D295/092 ,  C07D521/00

Abstract: Novel (hetarylphenoxy)-(phenylpiperazinyl)-propanols of the formula I where R1 is hydrogen, amino or alkyl of 1 to 4 carbon atoms, R2 is hydrogen, halogen, alkyl of 1 to 4 carbon atoms or alkoxy where alkyl is of 1 to 3 carbon atoms, the phenyl ring can be monosubstituted or disubstituted by R2, and the heterocyclic structure Het. is pyrimidinyl, triazol-1-yl, imidazol-1-yl, pyrazol-3-yl or isoxazol-3-yl, and their physiologically tolerated addition salts with acids, processes for their preparation, and pharmaceutical formulations which contain these compounds and exhibit predominantly hypotensive, sedative, neuroleptic and broncholytic properties.